Page last updated: 2024-08-21

quinazolines and cp 465,022

quinazolines has been researched along with cp 465,022 in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (71.43)29.6817
2010's2 (28.57)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chenard, BL; Collins, MB; Ducat, MF; Elliott, ML; Ewing, FE; Huang, JI; Kelly, KA; Lazzaro, JT; Menniti, FS; Pagnozzi, MJ; Weeks, JL; Welch, WM; White, WF1
Chenard, BL; Ewing, FE; Ganong, AH; Huang, J; Lazzaro, JT; Lerma, J; Menniti, FS; Paternain, AV; Welch, WM1
Buchan, AM; Chenard, BL; Critchett, DJ; Ganong, AH; Guanowsky, V; Menniti, FS; Seymour, PA; Welch, WM1
Balannik, V; Lerma, J; Menniti, FS; Paternain, AV; Stern-Bach, Y1
Cokić, B; Stein, V1
Hajós, M; Hoffmann, WE; Kiss, T1
Kurnikova, M; Narangoda, C; Sampson, JM; Singh, AK; Sobolevsky, AI; Yelshanskaya, MV1

Other Studies

7 other study(ies) available for quinazolines and cp 465,022

ArticleYear
Characterization of the binding site for a novel class of noncompetitive alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor antagonists.
    Molecular pharmacology, 2000, Volume: 58, Issue:6

    Topics: Animals; Binding Sites; Calcium; In Vitro Techniques; Neurons; Quinazolines; Rats; Rats, Sprague-Dawley; Receptors, AMPA

2000
Functional characterization of CP-465,022, a selective, noncompetitive AMPA receptor antagonist.
    Neuropharmacology, 2002, Volume: 42, Issue:2

    Topics: Animals; Cell Differentiation; Cells, Cultured; Cerebellum; Cerebral Cortex; DNA, Complementary; Dose-Response Relationship, Drug; Ganglia, Spinal; Humans; Membrane Potentials; Neurons; Patch-Clamp Techniques; Quinazolines; Rats; Receptors, AMPA; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Transfection; Tumor Cells, Cultured

2002
CP-465,022, a selective noncompetitive AMPA receptor antagonist, blocks AMPA receptors but is not neuroprotective in vivo.
    Stroke, 2003, Volume: 34, Issue:1

    Topics: Animals; Brain Ischemia; Hippocampus; Male; Motor Activity; Neuroprotective Agents; Pentylenetetrazole; Quinazolines; Rats; Receptors, AMPA; Seizures; Synaptic Transmission

2003
Molecular mechanism of AMPA receptor noncompetitive antagonism.
    Neuron, 2005, Oct-20, Volume: 48, Issue:2

    Topics: Animals; Benzodiazepines; Binding Sites; Blotting, Western; Brain; Cell Line; Cloning, Molecular; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Gene Expression Regulation; Humans; Membrane Potentials; Models, Neurological; Mutagenesis; Patch-Clamp Techniques; Peptide Fragments; Protein Conformation; Quinazolines; Rats; Receptors, AMPA; Transfection; Tritium; Xenopus laevis

2005
Stargazin modulates AMPA receptor antagonism.
    Neuropharmacology, 2008, Volume: 54, Issue:7

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzodiazepines; Binding Sites; Calcium Channels; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Glutamic Acid; Membrane Potentials; Microinjections; Models, Molecular; Oocytes; Patch-Clamp Techniques; Protein Structure, Tertiary; Quinazolines; Receptors, AMPA; Synaptic Transmission; Transcription, Genetic; Xenopus laevis

2008
Delta oscillation and short-term plasticity in the rat medial prefrontal cortex: modelling NMDA hypofunction of schizophrenia.
    The international journal of neuropsychopharmacology, 2011, Volume: 14, Issue:1

    Topics: Animals; Biphenyl Compounds; Delta Rhythm; Disease Models, Animal; Dizocilpine Maleate; Electric Stimulation; Electroencephalography; Excitatory Postsynaptic Potentials; Hippocampus; Lidocaine; Male; N-Methylaspartate; Neuronal Plasticity; Prefrontal Cortex; Quinazolines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Schizophrenia; Sulfonamides; Synaptic Transmission; Time Factors

2011
Structural Bases of Noncompetitive Inhibition of AMPA-Subtype Ionotropic Glutamate Receptors by Antiepileptic Drugs.
    Neuron, 2016, Sep-21, Volume: 91, Issue:6

    Topics: Animals; Anticonvulsants; Benzodiazepines; Binding Sites; Crystallization; Molecular Docking Simulation; Nitriles; Pyridones; Quinazolines; Rats; Receptors, AMPA

2016