Page last updated: 2024-08-21

quinazolines and carbostyril

quinazolines has been researched along with carbostyril in 33 studies

Research

Studies (33)

TimeframeStudies, this research(%)All Research%
pre-19903 (9.09)18.7374
1990's3 (9.09)18.2507
2000's12 (36.36)29.6817
2010's12 (36.36)24.3611
2020's3 (9.09)2.80

Authors

AuthorsStudies
Kano, Y; Komatsu, K; Qine, Z1
Alvarez, R; Kenley, RA; Lin, LH; Venuti, MC; Visor, GC1
Alvarez, R; Berks, AH; Bruno, JJ; Jones, GH; Prince, A; Venuti, MC1
Beretz, A; Cazenave, JP; Corre, G; Lanza, F; Stierlé, A1
Dousa, TP; Grande, JP; Matousovic, K; Tsuboi, Y; Walker, H1
Daugschies, A; Gässlein, U; Rommel, M1
Aubry, AF; Gray, V; Hobson, T; Rabel, S; Sebastian, D; Xie, M; Xu, JQ1
Gras, S; Hill, BT; Perrin, D; van Hille, B1
Barrie, E; Kelland, LR; Rowlands, MG; Smith, V; Workman, P1
Sánchez De Cos Escuín, J1
Doherty, JB; Hop, CE; Hunt, JA; Ita, I; Kallashi, F; Kumar, S; McCormick, SX; O'Keefe, SJ; O'Neill, EA; Pivnichny, JV; Porter, G; Ruzek, RD; Sinclair, PJ; Thompson, JE; Wang, Z; Woods, A; Zaller, DM1
Angibaud, P; Bourdrez, X; Devine, A; End, DW; Freyne, E; Ligny, Y; Mannens, G; Muller, P; Pilatte, I; Poncelet, V; Skrzat, S; Smets, G; Van Dun, J; Van Remoortere, P; Venet, M; Wouters, W1
Khuri, FR1
Angibaud, P; Bourdrez, X; Damsch, S; End, DW; Freyne, E; Janicot, M; Lezouret, P; Ligny, Y; Mannens, G; Mevellec, L; Meyer, C; Muller, P; Pilatte, I; Poncelet, V; Roux, B; Smets, G; Van Dun, J; Van Remoortere, P; Venet, M; Wouters, W1
Blackburn, C; Brodjian, S; Brown, J; Che, JL; Collins, CA; Cullis, CA; Dayton, B; Doherty, C; Geddes, B; Govek, E; Kadambi, V; Kym, PR; Lai, S; LaMarche, MJ; Maguire, M; Marsh, KC; Marsilje, T1
Borner, MM1
Filov, VA; Gershanovich, ML; Imianitov, EN; Stukov, AN1
Agarwal, SK; Burman, AC; Jha, A; Mukherjee, R; Srivastava, SK1
Chen, JJ; Hwang, TL; Kuo, YH; Wang, TY; Wu, JB1
Doçi, CL; Hasina, R; Lingen, MW; Mankame, TP; Wroblewski, K; Zhou, G1
Boyett, JM; Geyer, R; Haas-Kogan, D; Kieran, MW; Kun, L; Ng, S; Pollack, IF; Poussaint, TY; Prabhu, SP; Vajapeyam, S1
Boyett, JM; Cha, S; Geyer, R; Haas-Kogan, D; Kocak, M; Kun, LE; Packer, RI; Patay, Z; Pollack, IF; Poussaint, TY; Robertson, RL; Vajapeyam, S; Vezina, G; Zimmerman, R1
Bear, CE; Kim Chiaw, P; Yu, W1
Belavic, JM1
Chaumais, MC; De Man, FS; Dorfmüller, P; Eddahibi, S; Fadel, E; François, C; Girerd, B; Guignabert, C; Huertas, A; Humbert, M; Lecerf, F; Montani, D; Perros, F; Tu, L1
Cho, NJ; Park, YS1
Cho, BC; Kim, HR; Lim, SM; Shim, HS; Soo, RA1
Erba, HP1
Bhakta, S; Bucar, F; Evangelopoulos, D; Guzman, JD; Hochfellner, C; Kunert, O; McHugh, TD; Wube, A; Zloh, M1
Guo, M; He, J; Jiang, X; Jiang, Y; Li, J; Liu, J; Ouyang, L; Wang, J; Zhang, J; Zhang, S1
Bagal, SK; Bickerton, S; Bodnarchuk, MS; Breed, J; Carbajo, RJ; Cassar, DJ; Chakraborty, A; Cosulich, S; Cumming, I; Davies, M; Eatherton, A; Evans, L; Feron, L; Fillery, S; Gleave, ES; Goldberg, FW; Hanson, L; Harlfinger, S; Howard, M; Howells, R; Jackson, A; Kemmitt, P; Kettle, JG; Kingston, JK; Lamont, S; Lewis, HJ; Li, S; Liu, L; Ogg, D; Phillips, C; Polanski, R; Robb, G; Robinson, D; Ross, S; Smith, JM; Tonge, M; Whiteley, R; Yang, J; Zhang, L; Zhao, X1
Kwon, M; Lee, DW; Lee, HN; Lee, W1
Jiang, X; Li, D; Li, Y; Liu, W; Zhao, Q1

Reviews

9 review(s) available for quinazolines and carbostyril

ArticleYear
[New therapeutic targets and strategies in lung cancer].
    Archivos de bronconeumologia, 2002, Volume: 38, Issue:8

    Topics: Alkyl and Aryl Transferases; Angiogenesis Inhibitors; Antineoplastic Agents; Benzamides; Benzodiazepines; Clinical Trials as Topic; Clinical Trials, Phase I as Topic; Clinical Trials, Phase II as Topic; Clinical Trials, Phase III as Topic; Endothelial Growth Factors; Enzyme Inhibitors; Epidermal Growth Factor; ErbB Receptors; Erlotinib Hydrochloride; Farnesyltranstransferase; Gefitinib; Humans; Imatinib Mesylate; Imidazoles; Intercellular Signaling Peptides and Proteins; Lung Neoplasms; Lymphokines; Metalloendopeptidases; Multicenter Studies as Topic; Piperazines; Polyisoprenyl Phosphates; Protein-Tyrosine Kinases; Pyrimidines; Quinazolines; Quinolones; Randomized Controlled Trials as Topic; Receptor Protein-Tyrosine Kinases; Sesquiterpenes; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors

2002
Primary and secondary prevention of non-small-cell lung cancer: the SPORE Trials of Lung Cancer Prevention.
    Clinical lung cancer, 2003, Volume: 5 Suppl 1

    Topics: Antineoplastic Agents; Biomarkers, Tumor; Carcinoma, Non-Small-Cell Lung; Chemoprevention; Clinical Trials as Topic; Disease Progression; Epidermal Growth Factor; Gefitinib; Humans; Lung Neoplasms; Precancerous Conditions; Protein-Tyrosine Kinases; Quinazolines; Quinolones

2003
[Molecular targets in colon cancer].
    Therapeutische Umschau. Revue therapeutique, 2006, Volume: 63, Issue:4

    Topics: Angiogenesis Inhibitors; Antibiotics, Antineoplastic; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Antineoplastic Agents, Phytogenic; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Benzamides; Camptothecin; Cetuximab; Clinical Trials as Topic; Clinical Trials, Phase II as Topic; Colonic Neoplasms; Drug Delivery Systems; ErbB Receptors; Gefitinib; Humans; Imatinib Mesylate; Indoles; Irinotecan; Organoplatinum Compounds; Oxaliplatin; Phthalazines; Piperazines; Platelet-Derived Growth Factor; Protein Kinase Inhibitors; Pyridines; Pyrimidines; Pyrroles; Quinazolines; Quinolones; Receptors, Platelet-Derived Growth Factor; Receptors, Somatomedin; Signal Transduction; Sirolimus; Sunitinib

2006
[Problems in the current target therapy of malignancies].
    Voprosy onkologii, 2005, Volume: 51, Issue:5

    Topics: Alemtuzumab; Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antibodies, Monoclonal, Murine-Derived; Antibodies, Neoplasm; Antineoplastic Agents; Azathioprine; Benzamides; Bevacizumab; Cetuximab; Erlotinib Hydrochloride; Gefitinib; Humans; Imatinib Mesylate; Neoplasms; Phthalazines; Piperazines; Pyridines; Pyrimidines; Quinazolines; Quinolones; Rituximab; Sesquiterpenes; Sesquiterpenes, Guaiane; Trastuzumab

2005
Synthesis and structure-activity relationships of potent antitumor active quinoline and naphthyridine derivatives.
    Anti-cancer agents in medicinal chemistry, 2007, Volume: 7, Issue:6

    Topics: Antineoplastic Agents; Humans; Immunologic Factors; Naphthyridines; Quinazolines; Quinolines; Quinolones; Structure-Activity Relationship

2007
Role of FGF receptors as an emerging therapeutic target in lung squamous cell carcinoma.
    Future oncology (London, England), 2013, Volume: 9, Issue:3

    Topics: Alanine; Antineoplastic Agents; Benzimidazoles; Carcinoma, Squamous Cell; Gene Amplification; Humans; Lung Neoplasms; Molecular Targeted Therapy; Quinazolines; Quinolones; Receptors, Fibroblast Growth Factor; Signal Transduction; Triazines

2013
Finding the optimal combination therapy for the treatment of newly diagnosed AML in older patients unfit for intensive therapy.
    Leukemia research, 2015, Volume: 39, Issue:2

    Topics: Aminoglycosides; Antibodies, Monoclonal, Humanized; Antineoplastic Combined Chemotherapy Protocols; Azacitidine; Clinical Trials, Phase II as Topic; Clinical Trials, Phase III as Topic; Critical Care; Cytarabine; Decitabine; Female; Gemtuzumab; Humans; Leukemia, Myeloid, Acute; Male; Organophosphates; Quinazolines; Quinolones

2015
Recent advances in the development of dual VEGFR and c-Met small molecule inhibitors as anticancer drugs.
    European journal of medicinal chemistry, 2016, Jan-27, Volume: 108

    Topics: Antineoplastic Agents; Drug Discovery; Humans; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-met; Pyridines; Quinazolines; Quinolones; Receptors, Vascular Endothelial Growth Factor; Small Molecule Libraries

2016
Evodiamine: A Privileged Structure with Broad-ranging Biological Activities.
    Mini reviews in medicinal chemistry, 2022, Volume: 22, Issue:21

    Topics: Alkaloids; Butyrylcholinesterase; Cyclic Nucleotide Phosphodiesterases, Type 5; DNA Topoisomerases, Type I; DNA Topoisomerases, Type II; Female; Histone Deacetylases; Humans; Quinazolines; Quinolones; Sirtuins; Tubulin

2022

Other Studies

24 other study(ies) available for quinazolines and carbostyril

ArticleYear
[On the evaluation of the preparation of Chinese medicinal prescriptions. VI. The changes of the alkaloid contents by processing of Evodia fruit].
    Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan, 1991, Volume: 111, Issue:1

    Topics: Alkaloids; Chromatography, High Pressure Liquid; Drugs, Chinese Herbal; Humans; Indole Alkaloids; Plant Extracts; Quinazolines; Quinolones; Taste

1991
Electrochemical evaluation of the interaction between ascorbic acid and the cardiotonic drug RS-82856.
    Drug design and delivery, 1987, Volume: 2, Issue:2

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Ascorbic Acid; Cardiotonic Agents; Drug Interactions; Electrochemistry; Platelet Aggregation Inhibitors; Quinazolines; Quinolones; Solutions

1987
Inhibitors of cyclic AMP phosphodiesterase. 1. Analogues of cilostamide and anagrelide.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:2

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Blood Platelets; Humans; Indicators and Reagents; Magnetic Resonance Spectroscopy; Mass Spectrometry; Myocardium; Quinazolines; Quinolines; Quinolones; Rats; Spectrophotometry, Infrared; Structure-Activity Relationship

1987
Cyclic nucleotide phosphodiesterase inhibitors prevent aggregation of human platelets by raising cyclic AMP and reducing cytoplasmic free calcium mobilization.
    Thrombosis research, 1987, Mar-01, Volume: 45, Issue:5

    Topics: 2',3'-Cyclic-Nucleotide Phosphodiesterases; Alprostadil; Aminoquinolines; Blood Platelets; Calcium; Cyclic AMP; Cytoplasm; Humans; Isoquinolines; Phthalazines; Platelet Aggregation; Quercetin; Quinazolines; Quinolines; Quinolones; Tetrahydroisoquinolines

1987
Inhibitors of cyclic nucleotide phosphodiesterase isozymes block renal tubular cell proliferation induced by folic acid.
    The Journal of laboratory and clinical medicine, 1997, Volume: 130, Issue:5

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Cell Division; Cilostazol; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic Nucleotide Phosphodiesterases, Type 3; Down-Regulation; Folic Acid; Isoenzymes; Kidney Tubules; Male; Phosphodiesterase Inhibitors; Proliferating Cell Nuclear Antigen; Pyrrolidinones; Quinazolines; Quinolones; Rats; Rats, Sprague-Dawley; Rolipram; Signal Transduction; Tetrazoles

1997
Comparative efficacy of anticoccidials under the conditions of commercial broiler production and in battery trials.
    Veterinary parasitology, 1998, Apr-15, Volume: 76, Issue:3

    Topics: Animal Husbandry; Animals; Chickens; Clopidol; Coccidiosis; Coccidiostats; Drug Resistance; Eimeria; Feces; Food Industry; Ionophores; Monensin; Nicarbazin; Piperidines; Poultry Diseases; Predictive Value of Tests; Pyrans; Quinazolines; Quinazolinones; Quinolones

1998
In-use testing of extemporaneously prepared suspensions of second generation non-nucleoside reversed transcriptase inhibitors in support of phase I clinical studies.
    Journal of pharmaceutical and biomedical analysis, 2000, Aug-15, Volume: 23, Issue:2-3

    Topics: Anti-HIV Agents; Chromatography, High Pressure Liquid; Clinical Trials, Phase I as Topic; Pharmaceutical Preparations; Quinazolines; Quinazolinones; Quinolones; Reverse Transcriptase Inhibitors; Solubility; Spectrophotometry, Ultraviolet

2000
Expression in yeast and purification of functional recombinant human poly(ADP-ribose)polymerase (PARP). Comparative pharmacological profile with that of the rat enzyme.
    Journal of enzyme inhibition, 2000, Volume: 15, Issue:5

    Topics: 1-Naphthylamine; Animals; Benzamides; Electrophoresis, Polyacrylamide Gel; Enzyme Inhibitors; Gene Expression; Humans; Kinetics; Male; Naphthalimides; Phenanthrenes; Poly(ADP-ribose) Polymerase Inhibitors; Poly(ADP-ribose) Polymerases; Quinazolines; Quinolones; Rats; Recombinant Proteins; Saccharomyces; Sensitivity and Specificity; Testis

2000
Establishment and characterization of acquired resistance to the farnesyl protein transferase inhibitor R115777 in a human colon cancer cell line.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2002, Volume: 8, Issue:6

    Topics: Alkyl and Aryl Transferases; Antineoplastic Agents; Blotting, Western; Cell Division; Chromones; Colorectal Neoplasms; Drug Resistance, Neoplasm; ErbB Receptors; Farnesyltranstransferase; Humans; Morpholines; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Quinazolines; Quinolones; Transfection; Tumor Cells, Cultured

2002
p38 Inhibitors: piperidine- and 4-aminopiperidine-substituted naphthyridinones, quinolinones, and dihydroquinazolinones.
    Bioorganic & medicinal chemistry letters, 2003, Feb-10, Volume: 13, Issue:3

    Topics: Animals; Anti-Infective Agents; Area Under Curve; Biological Availability; Dogs; Enzyme Inhibitors; Half-Life; Macaca mulatta; Mitogen-Activated Protein Kinases; Naphthyridines; p38 Mitogen-Activated Protein Kinases; Piperidines; Quinazolines; Quinolones; Rats; Structure-Activity Relationship; Tumor Necrosis Factor-alpha

2003
5-imidazolyl-quinolinones, -quinazolinones and -benzo-azepinones as farnesyltransferase inhibitors.
    Bioorganic & medicinal chemistry letters, 2003, May-05, Volume: 13, Issue:9

    Topics: Alkyl and Aryl Transferases; Animals; Antineoplastic Agents; Azepines; Farnesyltranstransferase; Humans; In Vitro Techniques; Indicators and Reagents; Mice; Microsomes, Liver; Quinazolines; Quinolones; Structure-Activity Relationship; Xenograft Model Antitumor Assays

2003
Substituted azoloquinolines and -quinazolines as new potent farnesyl protein transferase inhibitors.
    Bioorganic & medicinal chemistry letters, 2003, Dec-15, Volume: 13, Issue:24

    Topics: Alkyl and Aryl Transferases; Animals; Cell Division; Drug Design; Enzyme Inhibitors; Farnesyltranstransferase; Kinetics; Molecular Conformation; Molecular Structure; Quinazolines; Quinolines; Quinolones; Structure-Activity Relationship

2003
Identification and characterization of amino-piperidinequinolones and quinazolinones as MCHr1 antagonists.
    Bioorganic & medicinal chemistry letters, 2006, May-15, Volume: 16, Issue:10

    Topics: Animals; Mice; Quinazolines; Quinolones; Receptors, Pituitary Hormone

2006
A new quinolone and other constituents from the fruits of Tetradium ruticarpum: effects on neutrophil pro-inflammatory responses.
    Chemistry & biodiversity, 2010, Volume: 7, Issue:7

    Topics: Anti-Inflammatory Agents; Evodia; Fruit; Humans; Indole Alkaloids; Molecular Structure; Neutrophils; Pancreatic Elastase; Plant Extracts; Quinazolines; Quinolines; Quinolones; Superoxides

2010
Dual inhibition of vascular endothelial growth factor receptor and epidermal growth factor receptor is an effective chemopreventive strategy in the mouse 4-NQO model of oral carcinogenesis.
    Cancer prevention research (Philadelphia, Pa.), 2010, Volume: 3, Issue:11

    Topics: 4-Nitroquinoline-1-oxide; Animals; Antineoplastic Agents; Carcinogens; Disease Models, Animal; Drug Resistance, Neoplasm; Epithelial-Mesenchymal Transition; ErbB Receptors; Immunohistochemistry; Mice; Mice, Inbred CBA; Mouth Neoplasms; Neovascularization, Pathologic; Piperidines; Quinazolines; Quinolones; Receptors, Vascular Endothelial Growth Factor

2010
DTI assessment of the brainstem white matter tracts in pediatric BSG before and after therapy: a report from the Pediatric Brain Tumor Consortium.
    Child's nervous system : ChNS : official journal of the International Society for Pediatric Neurosurgery, 2011, Volume: 27, Issue:1

    Topics: Adolescent; Anisotropy; Antineoplastic Agents; Brain Stem; Brain Stem Neoplasms; Child; Child, Preschool; Clinical Trials, Phase II as Topic; Combined Modality Therapy; Diffusion Tensor Imaging; Gefitinib; Glioma; Humans; Image Interpretation, Computer-Assisted; Male; Nerve Fibers, Myelinated; Quinazolines; Quinolones; Radiotherapy

2011
MRI as a central component of clinical trials analysis in brainstem glioma: a report from the Pediatric Brain Tumor Consortium (PBTC).
    Neuro-oncology, 2011, Volume: 13, Issue:4

    Topics: Adolescent; Antineoplastic Combined Chemotherapy Protocols; Brain Stem Neoplasms; Child; Child, Preschool; Combined Modality Therapy; Diffusion; Female; Gefitinib; Glioma; Humans; Magnetic Resonance Imaging; Male; Quinazolines; Quinolones; Radiotherapy Dosage; Research Design; Survival Rate; Treatment Outcome

2011
Probing conformational rescue induced by a chemical corrector of F508del-cystic fibrosis transmembrane conductance regulator (CFTR) mutant.
    The Journal of biological chemistry, 2011, Jul-15, Volume: 286, Issue:28

    Topics: Aminophenols; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; HEK293 Cells; Humans; Mutation; Piperazines; Protein Binding; Protein Folding; Protein Structure, Tertiary; Quinazolines; Quinolones

2011
Annual drug update: 2011 in review.
    The Nurse practitioner, 2012, Feb-12, Volume: 37, Issue:2

    Topics: Abatacept; Aminoglycosides; Carbamates; Drug Approval; Fentanyl; Fidaxomicin; Humans; Immunoconjugates; Indans; Linagliptin; Phenylenediamines; Proline; Purines; Quinazolines; Quinolones; United States; United States Food and Drug Administration

2012
A critical role for p130Cas in the progression of pulmonary hypertension in humans and rodents.
    American journal of respiratory and critical care medicine, 2012, Oct-01, Volume: 186, Issue:7

    Topics: Animals; Benzamides; Benzimidazoles; Case-Control Studies; Crk-Associated Substrate Protein; Disease Models, Animal; Endothelial Cells; Epidermal Growth Factor; Familial Primary Pulmonary Hypertension; Fibroblast Growth Factor 2; Gefitinib; Humans; Hypertension, Pulmonary; Imatinib Mesylate; Mice; Monocrotaline; Myocytes, Smooth Muscle; Piperazines; Platelet-Derived Growth Factor; Protein Kinase Inhibitors; Pulmonary Artery; Pyrimidines; Quinazolines; Quinolones; Rats; Signal Transduction

2012
EGFR and PKC are involved in the activation of ERK1/2 and p90 RSK and the subsequent proliferation of SNU-407 colon cancer cells by muscarinic acetylcholine receptors.
    Molecular and cellular biochemistry, 2012, Volume: 370, Issue:1-2

    Topics: Calcium; Carbachol; Cell Line, Tumor; Cell Proliferation; Colonic Neoplasms; Enzyme Activation; ErbB Receptors; Extracellular Signal-Regulated MAP Kinases; Humans; Indoles; Maleimides; Protein Kinase C; Quinazolines; Quinolones; Receptors, Muscarinic; Ribosomal Protein S6 Kinases, 90-kDa; Tyrphostins

2012
Antagonistic effects of indoloquinazoline alkaloids on antimycobacterial activity of evocarpine.
    Journal of applied microbiology, 2015, Volume: 118, Issue:4

    Topics: Alkaloids; Anti-Bacterial Agents; Drug Antagonism; Humans; Mycobacterium tuberculosis; Plant Extracts; Quinazolines; Quinolones; Tuberculosis

2015
Structure-Based Design and Pharmacokinetic Optimization of Covalent Allosteric Inhibitors of the Mutant GTPase KRAS
    Journal of medicinal chemistry, 2020, 05-14, Volume: 63, Issue:9

    Topics: Allosteric Regulation; Animals; Antineoplastic Agents; Caco-2 Cells; Cell Line, Tumor; Drug Design; Humans; Male; Mice, Nude; Molecular Conformation; Mutation; Neoplasms; Piperazines; Proto-Oncogene Proteins p21(ras); Quinazolines; Quinolones; Rats, Wistar; Structure-Activity Relationship; Xenograft Model Antitumor Assays

2020
Dual inhibition of FOXM1 and its compensatory signaling pathway decreased the survival of ovarian cancer cells.
    Oncology reports, 2021, Volume: 45, Issue:1

    Topics: Acetophenones; Benzopyrans; Cell Line, Tumor; Cell Survival; Female; Forkhead Box Protein M1; GTP Phosphohydrolases; Humans; Membrane Proteins; Ovarian Neoplasms; Pyridines; Quinazolines; Quinolones; Signal Transduction; Thiophenes

2021