Page last updated: 2024-08-21

quinazolines and carbachol

quinazolines has been researched along with carbachol in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19905 (23.81)18.7374
1990's3 (14.29)18.2507
2000's9 (42.86)29.6817
2010's4 (19.05)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ebbert, M; Janssens, WJ; Leidig, A; Meuter, C; Peters, T; Wilffert, B; Wilhelm, D1
Gulati, OD; Gupta, AK; Makol, R; Raghunath, PR; Shah, DS1
Nott, MW; Winslow, E1
Abdel-Latif, AA; Akhtar, RA1
Aghajanian, GK; Gallager, DW; Menkes, DB; Reinhard, JF1
Aghajanian, GK; Rogawski, MA1
Boutkan, H; Breslau, PJ; Burger, DH; Kappetein, AP1
Barrett, KE; Keely, SJ; Uribe, JM1
Barrett, KE; Calandrella, SO; Keely, SJ1
Andersson, K; Fujiwara, M; Persson, K1
Barrett, KE; McCole, DF; Uribe, JM1
Dartt, DA; Hodges, RR; Tepavcevic, V; Zoukhri, D1
Bernardino, CR; Chang, EL; Dartt, DA; Hodges, RR; Horikawa, Y; Rios, JD; Rubin, PA; Shatos, MA; Zoukhri, D1
Azegami, Y; Kaneda, T; Nakajyo, S; Shimizu, K; Urakawa, N; Yamamoto, H1
Mattingly, RR; Menard, RE1
Akhtar, S; Benboubetra, M; Benter, IF; Griffiths, SM; Yousif, MH1
Blagbrough, IS; Farghaly, HS; Medina-Tato, DA; Watson, ML1
Alexandre, L; Behr-Roussel, D; Denoux, Y; Giuliano, F; Gorny, D; Lebret, T; Oger, S1
Donnellan, F; Geoghegan, P; Harvey, BJ; Keating, N; Keely, SJ; Murray, FE1
Gutkind, JS; Hoffman, MP; Knox, SM; Lombaert, IM; Reed, X; Vitale-Cross, L1
Cho, NJ; Park, YS1

Trials

1 trial(s) available for quinazolines and carbachol

ArticleYear
Prevention of urinary retention after general surgery: a controlled trial of carbachol/diazepam versus alfusozine.
    Journal of the American College of Surgeons, 1997, Volume: 185, Issue:3

    Topics: Adrenergic alpha-Antagonists; Aged; Carbachol; Diazepam; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Incidence; Male; Muscle Relaxants, Central; Parasympathomimetics; Postoperative Complications; Quinazolines; Treatment Failure; Urinary Retention; Urination

1997

Other Studies

20 other study(ies) available for quinazolines and carbachol

ArticleYear
In vitro pharmacology of R 80122, a novel phosphodiesterase inhibitor.
    Journal of cardiovascular pharmacology, 1992, Volume: 20, Issue:5

    Topics: Action Potentials; Animals; Benzimidazoles; Carbachol; Female; Guinea Pigs; Heart Rate; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Milrinone; Myocardial Contraction; Norepinephrine; Ouabain; Oxindoles; Papillary Muscles; Phosphodiesterase Inhibitors; Pyridones; Quinazolines; Stimulation, Chemical; Vasodilator Agents

1992
Neuromuscular blocking action of 2-(2-(3-pyridyl) vinyl)-3-0-tolyl-3, 4-dihydroquinazoline-4-one (SRC 909).
    Archives internationales de pharmacodynamie et de therapie, 1974, Volume: 209, Issue:2

    Topics: Abdominal Muscles; Acetylcholine; Animals; Anura; Atropine; Calcium; Carbachol; Cats; Choline; Cold Temperature; Dose-Response Relationship, Drug; Female; Gallamine Triethiodide; Glycols; In Vitro Techniques; Leg; Male; Methysergide; Morphine; Muscle Contraction; Muscles; Neuromuscular Blocking Agents; Pentolinium Tartrate; Phrenic Nerve; Physostigmine; Potassium Chloride; Pyridines; Quinazolines; Quinazolinones; Rats; Sciatic Nerve; Tubocurarine; Vinyl Compounds

1974
Effects of quazodine (MJ 1988) on contractions of the isolated hemidiaphragm of the rat and the biventer cervicis muscle of the chick.
    British journal of pharmacology, 1973, Volume: 48, Issue:3

    Topics: Acetylcholine; Animals; Calcium; Carbachol; Chickens; Diaphragm; Drug Synergism; Electric Stimulation; In Vitro Techniques; Methyl Ethers; Muscle Contraction; Muscles; Quinazolines; Rats; Theophylline; Tubocurarine

1973
Carbachol causes rapid phosphodiesteratic cleavage of phosphatidylinositol 4,5-bisphosphate and accumulation of inositol phosphates in rabbit iris smooth muscle; prazosin inhibits noradrenaline- and ionophore A23187-stimulated accumulation of inositol pho
    The Biochemical journal, 1984, Nov-15, Volume: 224, Issue:1

    Topics: Animals; Calcimycin; Carbachol; Cations; Female; In Vitro Techniques; Inositol Phosphates; Iris; Male; Muscle, Smooth; Norepinephrine; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositols; Prazosin; Quinazolines; Rabbits; Sugar Phosphates; Time Factors

1984
Alpha 1-adrenoceptor denervation supersensitivity in brain: physiological and receptor binding studies.
    Brain research, 1983, Aug-01, Volume: 272, Issue:1

    Topics: Animals; Carbachol; Denervation; Evoked Potentials; Geniculate Bodies; Hydroxydopamines; Male; Neurons; Norepinephrine; Oxidopamine; Prazosin; Quinazolines; Radioligand Assay; Rats; Receptors, Adrenergic; Serotonin

1983
Activation of lateral geniculate neurons by locus coeruleus or dorsal noradrenergic bundle stimulation: selective blockade by the alpha 1-adrenoceptor antagonist prazosin.
    Brain research, 1982, Oct-28, Volume: 250, Issue:1

    Topics: Action Potentials; Animals; Carbachol; Electric Stimulation; Geniculate Bodies; Locus Coeruleus; Male; Neurons; Norepinephrine; Prazosin; Quinazolines; Rats; Rats, Inbred Strains; Serotonin

1982
Carbachol stimulates transactivation of epidermal growth factor receptor and mitogen-activated protein kinase in T84 cells. Implications for carbachol-stimulated chloride secretion.
    The Journal of biological chemistry, 1998, Oct-16, Volume: 273, Issue:42

    Topics: Adaptor Proteins, Signal Transducing; Adaptor Proteins, Vesicular Transport; Biological Transport; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Chlorides; Colon; ErbB Receptors; GRB2 Adaptor Protein; Intestinal Mucosa; Phosphorylation; Protein Binding; Protein Kinase C; Proteins; Quinazolines; Receptor, Muscarinic M3; Receptors, Muscarinic; Shc Signaling Adaptor Proteins; Signal Transduction; Transcriptional Activation; Tyrphostins

1998
Carbachol-stimulated transactivation of epidermal growth factor receptor and mitogen-activated protein kinase in T(84) cells is mediated by intracellular Ca2+, PYK-2, and p60(src).
    The Journal of biological chemistry, 2000, Apr-28, Volume: 275, Issue:17

    Topics: Calcium; Carbachol; Cell Line; Chlorides; Colon; Enzyme Inhibitors; Epithelial Cells; ErbB Receptors; Flavonoids; Fluphenazine; Focal Adhesion Kinase 2; Humans; Mitogen-Activated Protein Kinases; Phosphorylation; Phosphotyrosine; Protein-Tyrosine Kinases; Proto-Oncogene Proteins pp60(c-src); Quinazolines; Signal Transduction; Thapsigargin; Time Factors; Transcriptional Activation; Tyrphostins

2000
Nitric oxide-induced cGMP accumulation in the mouse bladder is not related to smooth muscle relaxation.
    European journal of pharmacology, 2000, Aug-04, Volume: 401, Issue:2

    Topics: Animals; Arginine; Carbachol; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; Female; In Vitro Techniques; Mice; Mice, Inbred BALB C; Molsidomine; Muscle Relaxation; Muscle, Smooth; Nitric Oxide Donors; Nitric Oxide Synthase; Nitroarginine; Nitroprusside; Phosphodiesterase Inhibitors; Piperazines; Piperidines; Purines; Quinazolines; Sildenafil Citrate; Sulfones; Urethra; Urinary Bladder

2000
Interferon-gamma activates EGF receptor and increases TGF-alpha in T84 cells: implications for chloride secretion.
    American journal of physiology. Gastrointestinal and liver physiology, 2002, Volume: 283, Issue:4

    Topics: Antibodies; Blotting, Western; Carbachol; Cell Line; Cell Membrane; Chlorides; Colon; Enzyme Inhibitors; ErbB Receptors; Humans; Immunosorbent Techniques; Interferon-gamma; Intestinal Mucosa; Kinetics; Phosphorylation; Phosphotyrosine; Protein Tyrosine Phosphatases; Pyrimidines; Quinazolines; src-Family Kinases; Transforming Growth Factor alpha; Tyrphostins

2002
Signal transduction pathways used by EGF to stimulate protein secretion in rat lacrimal gland.
    Investigative ophthalmology & visual science, 2003, Volume: 44, Issue:3

    Topics: Animals; Blotting, Western; Calcium; Carbachol; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme-Linked Immunosorbent Assay; Epidermal Growth Factor; ErbB Receptors; Eye Proteins; Lacrimal Apparatus; Male; Peroxidase; Phenylephrine; Phospholipase C gamma; Phosphorylation; Protein Kinase C; Quinazolines; Rats; Rats, Sprague-Dawley; Signal Transduction; Tetradecanoylphorbol Acetate; Type C Phospholipases; Tyrphostins

2003
Activation of mitogen-activated protein kinase by cholinergic agonists and EGF in human compared with rat cultured conjunctival goblet cells.
    Investigative ophthalmology & visual science, 2003, Volume: 44, Issue:6

    Topics: Adult; Aged; Aged, 80 and over; Animals; Blotting, Western; Carbachol; Cells, Cultured; Cholinergic Agonists; Conjunctiva; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; ErbB Receptors; Goblet Cells; Humans; Male; Middle Aged; Mitogen-Activated Protein Kinases; Muscarinic Antagonists; Piperidines; Quinazolines; Rats; Rats, Sprague-Dawley; Time Factors; Tyrphostins

2003
Lack of cyclic nucleotide regulation of MBCQ-induced relaxation of rat ileal smooth muscle.
    Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi, 2003, Volume: 39, Issue:3

    Topics: 3',5'-Cyclic-GMP Phosphodiesterases; Animals; Carbachol; Cholinergic Agonists; Cyclic AMP; Cyclic GMP; Cyclic Nucleotide Phosphodiesterases, Type 5; Dipyridamole; Ileum; Male; Muscle Relaxation; Muscle, Smooth; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Potassium; Purinones; Quinazolines; Rats; Rats, Wistar

2003
Cell surface receptors activate p21-activated kinase 1 via multiple Ras and PI3-kinase-dependent pathways.
    Cellular signalling, 2003, Volume: 15, Issue:12

    Topics: Androstadienes; Animals; Carbachol; cdc42 GTP-Binding Protein; Cell Line, Tumor; Chlorocebus aethiops; COS Cells; Epidermal Growth Factor; ErbB Receptors; Humans; Indoles; Kinetics; Lysophospholipids; Maleimides; Mice; Models, Biological; Myelin Basic Protein; NIH 3T3 Cells; p21-Activated Kinases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Kinase C; Protein Serine-Threonine Kinases; Quinazolines; rac GTP-Binding Proteins; ras Proteins; Receptor, Muscarinic M2; Receptors, Cell Surface; rho GTP-Binding Proteins; Signal Transduction; Tetradecanoylphorbol Acetate; Transfection; Tyrphostins; Wortmannin

2003
Epidermal growth factor receptor tyrosine kinase-mediated signalling contributes to diabetes-induced vascular dysfunction in the mesenteric bed.
    British journal of pharmacology, 2005, Volume: 145, Issue:6

    Topics: Angiotensin II; Animals; Carbachol; Cell Line; Diabetes Mellitus, Experimental; Endothelin-1; ErbB Receptors; Female; Genistein; Histamine; Humans; In Vitro Techniques; Mesenteric Arteries; Mesenteric Veins; Norepinephrine; Quinazolines; Rats; Rats, Wistar; Signal Transduction; Streptozocin; Tyrphostins; Vasoconstriction; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents

2005
Interleukin 13 increases contractility of murine tracheal smooth muscle by a phosphoinositide 3-kinase p110delta-dependent mechanism.
    Molecular pharmacology, 2008, Volume: 73, Issue:5

    Topics: Adenine; Animals; Bronchial Hyperreactivity; Carbachol; Chromones; Class I Phosphatidylinositol 3-Kinases; In Vitro Techniques; Interleukin-13; Isoenzymes; Lung; Mice; Mice, Mutant Strains; Morpholines; Muscle Contraction; Muscle, Smooth; Mutant Proteins; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Potassium Chloride; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Quinazolines; Tissue Extracts; Trachea

2008
Combination of alfuzosin and tadalafil exerts an additive relaxant effect on human detrusor and prostatic tissues in vitro.
    European urology, 2010, Volume: 57, Issue:4

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Aged; Carbachol; Carbolines; Cholinergic Agonists; Dose-Response Relationship, Drug; Drug Therapy, Combination; Electric Stimulation; Humans; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Phosphodiesterase 5 Inhibitors; Prostate; Quinazolines; Tadalafil; Urinary Bladder

2010
JNK mitogen-activated protein kinase limits calcium-dependent chloride secretion across colonic epithelial cells.
    American journal of physiology. Gastrointestinal and liver physiology, 2010, Volume: 298, Issue:1

    Topics: Amino Acids, Cyclic; Anthracenes; Calcium; Carbachol; Cell Line; Cell Polarity; Chlorides; Cholinergic Agonists; Colon; Enzyme Inhibitors; Epithelial Cells; Flavonoids; Humans; Intestinal Mucosa; JNK Mitogen-Activated Protein Kinases; MAP Kinase Signaling System; Phosphorylation; Potassium; Quinazolines; Thapsigargin; Tyrphostins

2010
Parasympathetic innervation maintains epithelial progenitor cells during salivary organogenesis.
    Science (New York, N.Y.), 2010, Sep-24, Volume: 329, Issue:5999

    Topics: Acetylcholine; Animals; Carbachol; Cell Differentiation; Epithelial Cells; Epithelium; ErbB Receptors; Ganglia, Parasympathetic; Heparin-binding EGF-like Growth Factor; Intercellular Signaling Peptides and Proteins; Keratin-5; Male; Mice; Morphogenesis; Neurons; Organ Culture Techniques; Organogenesis; Prostate; Quinazolines; Receptor, Muscarinic M1; Regeneration; Signal Transduction; Stem Cells; Submandibular Gland

2010
EGFR and PKC are involved in the activation of ERK1/2 and p90 RSK and the subsequent proliferation of SNU-407 colon cancer cells by muscarinic acetylcholine receptors.
    Molecular and cellular biochemistry, 2012, Volume: 370, Issue:1-2

    Topics: Calcium; Carbachol; Cell Line, Tumor; Cell Proliferation; Colonic Neoplasms; Enzyme Activation; ErbB Receptors; Extracellular Signal-Regulated MAP Kinases; Humans; Indoles; Maleimides; Protein Kinase C; Quinazolines; Quinolones; Receptors, Muscarinic; Ribosomal Protein S6 Kinases, 90-kDa; Tyrphostins

2012