Compounds > quinazolines
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quinazolines and benzoxazoles

quinazolines has been researched along with benzoxazoles in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19901 (11.11)18.7374
1990's2 (22.22)18.2507
2000's1 (11.11)29.6817
2010's5 (55.56)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Picciola, G1
Bleasdale, C; Bowman, K; Calvert, AH; Curtin, NJ; Durkacz, BW; Griffin, RJ; Newell, DR; Pemberton, LC; Porteous, JK; Rhodes, D1
Bekhit, AA; Khalil, MA1
Bouregeois, NM; Corbett, TH; Crantz, B; Hazeldine, ST; Horwitz, JP; Kushner, J; Palomino, E; Polin, L; White, K1
Di Paolo, T; Gasparini, F; Gomez-Mancilla, B; Grégoire, L; Hoyer, D; Morissette, M; Ouattara, B1
Aura, C; Baselga, J; Calvo, MT; García-García, C; Grueso, J; Guzmán, M; Ibrahim, YH; Jessen, K; Liu, Y; Pérez, J; Rommel, C; Scaltriti, M; Serra, V; Tabernero, J1
Dinneswara Reddy, G; Mallikarjuna Reddy, L; Padmaja, A; Padmavathi, V1
Lin, J; Xue, L; Yin, S; Zhang, C; Zhou, L1
Borger, D; Chisholm, S; Foster, R; Growdon, WB; Hernandez, SF; Rueda, BR1

Other Studies

9 other study(ies) available for quinazolines and benzoxazoles

ArticleYear
[Synthesis of quinazolinic and benzoxazinonic acids and study of their anti-inflammatory activity].
    Il Farmaco; edizione scientifica, 1976, Volume: 31, Issue:9

    Topics: Anti-Inflammatory Agents; Benzoxazoles; Methods; Quinazolines

1976
Novel potent inhibitors of the DNA repair enzyme poly(ADP-ribose)polymerase (PARP).
    Anti-cancer drug design, 1995, Volume: 10, Issue:6

    Topics: Animals; Benzoxazoles; Binding Sites; Enzyme Inhibitors; Humans; Leukemia L1210; Poly(ADP-ribose) Polymerase Inhibitors; Quinazolines

1995
Non-steroidal anti-inflammatory agents: synthesis of novel benzopyrazolyl, benzoxazolyl and quinazolinyl derivatives of 4(3 H)-quinazolinones.
    Die Pharmazie, 1998, Volume: 53, Issue:8

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzoxazoles; Granuloma; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Quinazolines; Rats; Rats, Sprague-Dawley

1998
II. Synthesis and biological evaluation of some bioisosteres and congeners of the antitumor agent, 2-(4-[(7-chloro-2-quinoxalinyl)oxy]phenoxy)propionic acid (XK469).
    Journal of medicinal chemistry, 2002, Jul-04, Volume: 45, Issue:14

    Topics: Animals; Antineoplastic Agents; Benzoxazoles; Drug Screening Assays, Antitumor; Mice; Neoplasm Transplantation; Propionates; Pyrazines; Pyridines; Quinazolines; Quinolines; Quinoxalines; Stereoisomerism; Structure-Activity Relationship; Thiazoles; Triazines; Tumor Cells, Cultured

2002
Changes of AMPA receptors in MPTP monkeys with levodopa-induced dyskinesias.
    Neuroscience, 2010, Jun-02, Volume: 167, Issue:4

    Topics: Animals; Antiparkinson Agents; Autoradiography; Benzoxazoles; Brain; Cabergoline; Drug Interactions; Dyskinesia, Drug-Induced; Ergolines; Female; Imidazoles; Levodopa; Ligands; Macaca fascicularis; MPTP Poisoning; Piperidines; Quinazolines; Receptors, AMPA; Receptors, Dopamine D2; Receptors, N-Methyl-D-Aspartate

2010
Dual mTORC1/2 and HER2 blockade results in antitumor activity in preclinical models of breast cancer resistant to anti-HER2 therapy.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2012, May-01, Volume: 18, Issue:9

    Topics: Animals; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Apoptosis; Benzoxazoles; Blotting, Western; Breast Neoplasms; Cell Cycle; Drug Resistance, Neoplasm; Drug Synergism; Extracellular Signal-Regulated MAP Kinases; Female; Humans; Lapatinib; Mechanistic Target of Rapamycin Complex 1; Mice; Mice, Nude; Multiprotein Complexes; Phosphatidylinositol 3-Kinases; Phosphorylation; Protein Kinase Inhibitors; Proteins; Proto-Oncogene Proteins c-akt; Pyrimidines; Quinazolines; Receptor, ErbB-2; TOR Serine-Threonine Kinases; Transcription Factors; Trastuzumab; Tumor Cells, Cultured; Xenograft Model Antitumor Assays

2012
Synthesis and antimicrobial activity of amino linked heterocycles.
    Chemical & pharmaceutical bulletin, 2015, Volume: 63, Issue:2

    Topics: Amines; Anti-Infective Agents; Aspergillus niger; Benzimidazoles; Benzothiazoles; Benzoxazoles; Gram-Negative Bacteria; Gram-Positive Bacteria; Microbial Sensitivity Tests; Quinazolines; Staphylococcus aureus

2015
Design, synthesis and biological activities of novel oxazolo[4,5-g]quinazolin-2(1H)-one derivatives as EGFR inhibitors.
    European journal of medicinal chemistry, 2015, Aug-28, Volume: 101

    Topics: Animals; Antineoplastic Agents; Benzoxazoles; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Design; Drug Screening Assays, Antitumor; ErbB Receptors; Humans; Mice; Mice, SCID; Neoplasms, Experimental; Quinazolines; Structure-Activity Relationship

2015
Ridaforolimus improves the anti-tumor activity of dual HER2 blockade in uterine serous carcinoma in vivo models with HER2 gene amplification and PIK3CA mutation.
    Gynecologic oncology, 2016, Volume: 141, Issue:3

    Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Benzoxazoles; Cell Cycle; Cell Proliferation; Class I Phosphatidylinositol 3-Kinases; Cystadenoma, Serous; Drug Synergism; Female; Gene Amplification; Humans; Lapatinib; Mice; Mice, Inbred NOD; Mice, SCID; Phosphatidylinositol 3-Kinases; Pyrimidines; Quinazolines; Receptor, ErbB-2; Sirolimus; TOR Serine-Threonine Kinases; Trastuzumab; Uterine Neoplasms; Xenograft Model Antitumor Assays

2016