quinazolines has been researched along with benzimidazole in 13 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (7.69) | 29.6817 |
2010's | 10 (76.92) | 24.3611 |
2020's | 2 (15.38) | 2.80 |
Authors | Studies |
---|---|
Arienzo, R; Cramp, S; Dyke, HJ; Lockey, PM; Norman, D; Roach, AG; Smith, P; Wong, M; Wren, SP | 1 |
Annis, DA; Basso, AD; Chuang, CC; Gray, K; Herbst, R; Lahue, B; Le, HV; Ma, Y; Nickbarg, E; Sanden, D; Seghezzi, W; Sheth, PR; Shipps, GW; Smith, CK; Vilenchik, L | 1 |
Fu, H; Lu, J; Xu, S | 1 |
Kamran Azim, M; Khan, KM; Khan, R; Rashid, Y; Saify, ZS | 1 |
Luxami, V; Paul, K; Sharma, A | 2 |
Shi, L; Wang, Z; Wu, TT; Xu, YG; Xue, JY | 1 |
Anbu, S; Guedes da Silva, MF; Koch, B; Kuznetsov, ML; Paul, A; Pombeiro, AJ; Sharma, G | 1 |
Cimarelli, C; Di Nicola, M; Diomedi, S; Giovannini, R; Hamprecht, D; Marcantoni, E; Properzi, R; Sorana, F | 1 |
Boerneke, MA; Charrette, BP; Hermann, T | 1 |
Banerjee, S; Kumar, A; Roy, P; Sharma, A; Sondhi, SM | 1 |
Chakraborti, AK; Dhameliya, TM; Jadhavar, PS; Krishna, VS; Patel, KI; Saha, N; Sriram, D; Vaja, MD | 1 |
Ahmad, MN; Akunuri, R; Chopra, S; Dasgupta, A; Kaul, G; Madhavi, YV; Malasala, S; Nanduri, S; Shukla, M | 1 |
13 other study(ies) available for quinazolines and benzimidazole
Article | Year |
---|---|
Quinazoline and benzimidazole MCH-1R antagonists.
Topics: Benzimidazoles; Humans; Inhibitory Concentration 50; Protein Binding; Quinazolines; Receptors, Somatostatin; Structure-Activity Relationship | 2007 |
Novel benzimidazole inhibitors bind to a unique site in the kinesin spindle protein motor domain.
Topics: Adenosine Triphosphatases; Antineoplastic Agents; Benzamides; Benzimidazoles; Binding Sites; Circular Dichroism; Humans; Kinesins; Mass Spectrometry; Nucleotides; Protein Structure, Tertiary; Quinazolines | 2010 |
Copper-catalyzed cascade synthesis of benzimidazoquinazoline derivatives under mild condition.
Topics: Benzimidazoles; Catalysis; Copper; Quinazolines | 2011 |
Small molecule activators of proteasome-related HslV peptidase.
Topics: Benzimidazoles; Calorimetry; Chromones; Dose-Response Relationship, Drug; Endopeptidase Clp; Enzyme Activation; Escherichia coli Proteins; High-Throughput Screening Assays; Hydrolysis; Ligands; Models, Molecular; Molecular Structure; Molecular Weight; Proteasome Endopeptidase Complex; Proteolysis; Quinazolines; Small Molecule Libraries; Structure-Activity Relationship | 2012 |
Synthesis, single crystal and antitumor activities of benzimidazole-quinazoline hybrids.
Topics: Antineoplastic Agents; Benzimidazoles; Binding Sites; Catalytic Domain; Cell Line, Tumor; Cell Proliferation; Crystallography, X-Ray; Drug Screening Assays, Antitumor; Humans; Magnetic Resonance Spectroscopy; Mass Spectrometry; Molecular Conformation; Molecular Docking Simulation; Orphan Nuclear Receptors; Quinazolines; Structure-Activity Relationship | 2013 |
Synthesis and in vitro antitumor evaluation of primary amine substituted quinazoline linked benzimidazole.
Topics: Antineoplastic Agents; Benzimidazoles; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; Quinazolines; Structure-Activity Relationship | 2014 |
Discovery of quinazolin-4-amines bearing benzimidazole fragments as dual inhibitors of c-Met and VEGFR-2.
Topics: Antineoplastic Agents; Benzimidazoles; Cell Proliferation; Dose-Response Relationship, Drug; Drug Discovery; Drug Screening Assays, Antitumor; Hep G2 Cells; Humans; MCF-7 Cells; Molecular Docking Simulation; Molecular Structure; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-met; Quinazolines; Structure-Activity Relationship; Vascular Endothelial Growth Factor Receptor-2 | 2014 |
Intracellular detection of Cu(2+) and S(2-) ions through a quinazoline functionalized benzimidazole-based new fluorogenic differential chemosensor.
Topics: Benzimidazoles; Biosensing Techniques; Coordination Complexes; Copper; Crystallography, X-Ray; Fluorescent Dyes; Humans; Lymphoma; Quinazolines; Spectrometry, Fluorescence; Sulfur; Tumor Cells, Cultured | 2015 |
An efficient one-pot two catalyst system in the construction of 2-substituted benzimidazoles: synthesis of benzimidazo[1,2-c]quinazolines.
Topics: Aniline Compounds; Benzimidazoles; Catalysis; Chemistry Techniques, Analytical; Molecular Structure; Quinazolines; Schiff Bases | 2015 |
Ligand Optimization by Improving Shape Complementarity at a Hepatitis C Virus RNA Target.
Topics: Antiviral Agents; Benzimidazoles; Drug Design; Hepacivirus; Hepatitis C; Humans; Internal Ribosome Entry Sites; Ligands; Models, Molecular; Nucleic Acid Conformation; Quinazolines; RNA, Viral | 2016 |
Solvent-free synthesis and anticancer activity evaluation of benzimidazole and perimidine derivatives.
Topics: Antineoplastic Agents; Benzimidazoles; Cell Line, Tumor; Cell Proliferation; Chemistry Techniques, Synthetic; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; Inhibitory Concentration 50; Molecular Structure; Quinazolines; Solvents; Structure-Activity Relationship | 2018 |
Benzimidazoquinazolines as new potent anti-TB chemotypes: Design, synthesis, and biological evaluation.
Topics: Animals; Antitubercular Agents; Benzimidazoles; Cell Survival; Dose-Response Relationship, Drug; Drug Design; Mice; Microbial Sensitivity Tests; Molecular Structure; Mycobacterium tuberculosis; Quinazolines; RAW 264.7 Cells; Structure-Activity Relationship; Tuberculosis | 2020 |
Synthesis and evaluation of new quinazoline-benzimidazole hybrids as potent anti-microbial agents against multidrug resistant Staphylococcus aureus and Mycobacterium tuberculosis.
Topics: Anti-Bacterial Agents; Benzimidazoles; Dose-Response Relationship, Drug; Microbial Sensitivity Tests; Molecular Structure; Mycobacterium tuberculosis; Quinazolines; Staphylococcus aureus; Structure-Activity Relationship | 2021 |