Page last updated: 2024-08-21

quinazolines and az-628

quinazolines has been researched along with az-628 in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (50.00)24.3611
2020's2 (50.00)2.80

Authors

AuthorsStudies
Dinkel, V; Gloor, SL; Grina, J; Hansen, JD; Hastings, G; Laird, ER; Mathieu, S; Moreno, D; Rana, S; Rasor, K; Ren, L; Rudolph, J; Sturgis, HL; Vigers, G; Voegtli, WC; Wenglowsky, S; Willis, B1
Chu, P; Lou, M; Wang, Z; Yin, M1
Li, H; Ma, C; Su, H; Xiong, J1
Chen, L; Gong, Y; Hong, Z; Jiang, T; Mi, S; Qiu, J; Wang, Z; Ye, J; Zhang, W; Zheng, X; Zhu, Z1

Other Studies

4 other study(ies) available for quinazolines and az-628

ArticleYear
Highly potent and selective 3-N-methylquinazoline-4(3H)-one based inhibitors of B-Raf(V600E) kinase.
    Bioorganic & medicinal chemistry letters, 2014, Apr-15, Volume: 24, Issue:8

    Topics: Animals; Antineoplastic Agents; Crystallography, X-Ray; Drug Design; Enzyme Activation; Humans; Inhibitory Concentration 50; Molecular Structure; Protein Kinase Inhibitors; Proto-Oncogene Proteins B-raf; Quinazolines; Tumor Burden; Xenograft Model Antitumor Assays

2014
STAT3 inhibitor sensitized KRAS-mutant lung cancers to RAF inhibitor by activating MEK/ERK signaling pathway.
    Aging, 2019, 09-04, Volume: 11, Issue:17

    Topics: Aminosalicylic Acids; Animals; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Cell Line, Tumor; Drug Screening Assays, Antitumor; Humans; Lung Neoplasms; MAP Kinase Signaling System; Mice, Inbred BALB C; Mice, Nude; Proto-Oncogene Proteins p21(ras); Quinazolines; raf Kinases; STAT3 Transcription Factor; Sulfonamides

2019
The underlying molecular mechanism and drugs for treatment in adrenal cortical carcinoma.
    International journal of medical sciences, 2021, Volume: 18, Issue:13

    Topics: Adrenal Cortex; Adrenal Cortex Neoplasms; Adrenalectomy; Adrenocortical Carcinoma; Adult; Biomarkers, Tumor; Chemotherapy, Adjuvant; Computational Biology; Databases, Genetic; Female; Follow-Up Studies; Gene Expression Regulation, Neoplastic; Gene Regulatory Networks; Humans; Isoquinolines; Kaplan-Meier Estimate; Male; MicroRNAs; Middle Aged; Prognosis; Protein Kinase Inhibitors; Quinazolines; RNA-Seq; RNA, Messenger; Succinimides; Sulfonamides

2021
AZ-628 delays osteoarthritis progression via inhibiting the TNF-α-induced chondrocyte necroptosis and regulating osteoclast formation.
    International immunopharmacology, 2022, Volume: 111

    Topics: Animals; Chondrocytes; Mice; Necroptosis; NF-kappa B; Osteoarthritis; Osteoclasts; Quinazolines; Tumor Necrosis Factor-alpha

2022