Page last updated: 2024-09-03

quinapyramine and suramin

quinapyramine has been researched along with suramin in 19 studies

Compound Research Comparison

Studies
(quinapyramine)
Trials
(quinapyramine)
Recent Studies (post-2010)
(quinapyramine)
Studies
(suramin)
Trials
(suramin)
Recent Studies (post-2010) (suramin)
810103,02392431

Protein Interaction Comparison

ProteinTaxonomyquinapyramine (IC50)suramin (IC50)
ATP-dependent 6-phosphofructokinaseTrypanosoma brucei brucei3
Tyrosine-protein phosphatase non-receptor type 1Homo sapiens (human)9.76
P2X purinoceptor 2Rattus norvegicus (Norway rat)4
DNA-dependent protein kinase catalytic subunitHomo sapiens (human)1.7
DNA primaseMycobacterium tuberculosis CDC15518.2
RmtAAspergillus nidulans5.9
Reverse transcriptase/RNaseH Human immunodeficiency virus 19.4
NAD-dependent protein deacetylase sirtuin-2Homo sapiens (human)1.15
NAD-dependent protein deacetylase sirtuin-1Homo sapiens (human)1.5667
Protein arginine N-methyltransferase 1Homo sapiens (human)5.33
NAD-dependent protein deacylase sirtuin-5, mitochondrialHomo sapiens (human)2.5

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19909 (47.37)18.7374
1990's7 (36.84)18.2507
2000's2 (10.53)29.6817
2010's1 (5.26)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baltz, T; Giroud, C; Zhang, ZQ2
Kaminsky, R; Webster, P; Zweygarth, E1
Ali, BH; Hassan, T; Malik, KH1
Borowy, NK; Hirumi, H; Mkoji, G; Waithaka, HK1
Williamson, J1
Kinabo, LD1
Kaminsky, R; Moloo, SK; Zweygarth, E1
Barns, AM; Ross, CA; Sutherland, DV1
El Malik, KH; El Rayah, IE; Kaminsky, R; Schmid, C1
HAWKING, F; SEN, AB1
BHATTACHARYA, BK; DAS, P; SEN, AB1
GRAY, AR1
STEPHEN, LE1
ORMEROD, WE; SHAW, JJ1
Liao, D; Lin, J; Shen, J; Zhou, J; Zhou, Y1
Konnai, S; Ohashi, K; Onuma, M; Tsuda, A; Witola, WH1
TOWN, BW; WILLS, ED; WORMALL, A1
Arafa, RK; Boykin, DW; Brun, R; Gillingwater, K; Ismail, MA; Kumar, A; Stephens, CE; Tidwell, RR1

Reviews

1 review(s) available for quinapyramine and suramin

ArticleYear
Pharmacology of existing drugs for animal trypanosomiasis.
    Acta tropica, 1993, Volume: 54, Issue:3-4

    Topics: Animals; Arsenicals; Diminazene; Ethidium; Phenanthridines; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosomiasis, African

1993

Other Studies

18 other study(ies) available for quinapyramine and suramin

ArticleYear
In vivo and in vitro sensitivity of Trypanosoma evansi and T. equiperdum to diminazene, suramin, MelCy, quinapyramine and isometamidium.
    Acta tropica, 1991, Volume: 50, Issue:2

    Topics: Animals; Arsenicals; Diminazene; Female; Mice; Phenanthridines; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosoma; Trypanosomiasis

1991
Trypanosoma brucei evansi: dyskinetoplasia and loss of infectivity after long-term in vitro cultivation.
    Acta tropica, 1990, Volume: 48, Issue:2

    Topics: Animals; Diminazene; DNA, Circular; DNA, Kinetoplast; Female; Male; Mice; Microscopy, Electron; Phenanthridines; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

1990
The efficacy of furazolidone against experimental infections with Trypanosoma evansi in camels and mice in Sudan: comparisons with quinapyramine and suramin.
    Revue d'elevage et de medecine veterinaire des pays tropicaux, 1986, Volume: 39, Issue:2

    Topics: Animals; Camelus; Female; Furazolidone; Male; Mice; Quinolinium Compounds; Sudan; Suramin; Trypanocidal Agents; Trypanosomiasis

1986
An assay for screening drugs against animal-infective bloodstream forms of Trypanosoma brucei brucei in vitro.
    Drugs under experimental and clinical research, 1985, Volume: 11, Issue:3

    Topics: Animals; Diminazene; Mice; Parasitology; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosoma brucei brucei

1985
Drug sensitivity of pleomorphic Trypanosoma rhodesiense.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1983, Volume: 77, Issue:2

    Topics: Animals; Arsenicals; Drug Resistance, Microbial; Ethidium; Mice; Pentamidine; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosomiasis, African

1983
Trypanosoma simiae: in vitro studies on drug susceptibility.
    Acta tropica, 1993, Volume: 54, Issue:3-4

    Topics: Animals; Arsenicals; Diminazene; Drug Resistance; Eflornithine; Parasitology; Quinolinium Compounds; Species Specificity; Suramin; Trypanocidal Agents; Trypanosoma

1993
Trypanosoma evansi: in vivo and in vitro determination of trypanocide resistance profiles.
    Experimental parasitology, 1993, Volume: 77, Issue:4

    Topics: Animals; Arsenicals; Diminazene; Drug Resistance; Phenanthridines; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosoma

1993
Trypanosoma evansi: measurement of pyruvate production as an indicator of the drug sensitivity of isolates in vitro.
    Tropical medicine and parasitology : official organ of Deutsche Tropenmedizinische Gesellschaft and of Deutsche Gesellschaft fur Technische Zusammenarbeit (GTZ), 1995, Volume: 46, Issue:2

    Topics: Animals; Arsenic Poisoning; Arsenicals; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Pyruvates; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosoma

1995
Drug resistance in Sudanese Trypanosoma evansi.
    Veterinary parasitology, 1999, Jan-28, Volume: 80, Issue:4

    Topics: Animals; Camelus; Chromatography, Ion Exchange; Drug Resistance; Female; Hypoxanthine; Inhibitory Concentration 50; Mice; Mice, Inbred ICR; Phenanthridines; Quinolinium Compounds; Scintillation Counting; Sudan; Suramin; Trypanocidal Agents; Trypanosoma; Trypanosomiasis, African

1999
The trypanocidal action of homidium, quinapyramine and suramin.
    British journal of pharmacology and chemotherapy, 1960, Volume: 15

    Topics: Animals; Arsenicals; Ethidium; Mice; Pentamidine; Quinolines; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosomiasis

1960
Changes observed in Trypanosoma evansi from Antrycide and Suramin treated rats.
    Archives internationales de pharmacodynamie et de therapie, 1962, Feb-01, Volume: 135

    Topics: Animals; Quinolines; Quinolinium Compounds; Rats; Suramin; Trypanosoma

1962
Suramin complexes. VIII. A further trial of the prophylactic activity of Antrycide-suramin complex and Antrycide chloride against Trypanosoma simiae in pigs.
    Annals of tropical medicine and parasitology, 1961, Volume: 55

    Topics: Animals; Humans; Quinolines; Quinolinium Compounds; Suramin; Swine; Swine Diseases; Trypanosoma

1961
Suramin complexes, IX. An experiment to test the therapeutic activity of antrycide-suramin complex against Trypanosoma simiae in large white pigs.
    Annals of tropical medicine and parasitology, 1962, Volume: 56

    Topics: Humans; Quinolinium Compounds; Suramin; Trypanosoma

1962
A STUDY OF GRANULES AND OTHER CHANGES IN PHASE-CONTRAST APPEARANCE PRODUCED BY CHEMOTHERAPEUTIC AGENTS IN TRYPANOSOMES.
    British journal of pharmacology and chemotherapy, 1963, Volume: 21

    Topics: Animals; Antineoplastic Agents; Antiprotozoal Agents; Fluorescence; Histology; Mice; Microscopy; Microscopy, Fluorescence; Microscopy, Phase-Contrast; Pharmacology; Quinolines; Quinolinium Compounds; Rats; Research; Stilbamidines; Suramin; Trypan Blue; Trypanocidal Agents; Trypanosoma; Trypanosomiasis

1963
Resistance to drug by different isolates Trypanosoma evansi in China.
    Acta tropica, 2004, Volume: 90, Issue:3

    Topics: Animals; China; Disease Models, Animal; Drug Resistance; Female; Humans; Male; Mice; Parasitic Sensitivity Tests; Quinolinium Compounds; Suramin; Trypanocidal Agents; Trypanosoma; Trypanosomiasis

2004
The effect of TAO expression on PCD-like phenomenon development and drug resistance in Trypanosoma brucei.
    Parasitology international, 2006, Volume: 55, Issue:2

    Topics: Animals; Apoptosis; Dose-Response Relationship, Drug; Drug Resistance; Gene Expression Regulation, Enzymologic; Humans; In Situ Nick-End Labeling; Mitochondrial Proteins; Oxidoreductases; Parasitic Sensitivity Tests; Plant Proteins; Quinolinium Compounds; Reactive Oxygen Species; Suramin; Time Factors; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

2006
Action of suramin and antrycide on enzymes.
    Nature, 1949, Aug-06, Volume: 164, Issue:4162

    Topics: Enzymes; Humans; Quinolinium Compounds; Suramin

1949
In vitro activity and preliminary toxicity of various diamidine compounds against Trypanosoma evansi.
    Veterinary parasitology, 2010, May-11, Volume: 169, Issue:3-4

    Topics: Amidines; Animals; Arsenicals; Cells, Cultured; Diminazene; Drug Resistance; Female; Inhibitory Concentration 50; Mice; Pentamidine; Quinolinium Compounds; Rats; Suramin; Trypanocidal Agents; Trypanosoma; Trypanosomiasis

2010