quinacrine and tilorone

quinacrine has been researched along with tilorone in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19908 (47.06)18.7374
1990's1 (5.88)18.2507
2000's2 (11.76)29.6817
2010's3 (17.65)24.3611
2020's3 (17.65)2.80

Authors

AuthorsStudies
Chiang, GH; Unger, SH1
Denny, WA; Feigon, J; Kearns, DR; Leupin, W1
Choi, SS; Contrera, JF; Hastings, KL; Kruhlak, NL; Sancilio, LF; Weaver, JL; Willard, JM1
Glen, RC; Lowe, R; Mitchell, JB1
Atzpodien, EA; Csato, M; Doessegger, L; Fischer, H; Lenz, B; Schmitt, G; Singer, T1
Byun, SY; Choi, I; Jeon, S; Kim, S; Ko, M; Lee, J; Park, S; Shum, D1
Ekins, S; Lane, TR1
Mannering, GJ; Renton, KW1
Ciak, J; Hahn, FE1
Bogdanovsky, D; Pierre, M1
Degré, M; Gláz, ET1
Creuzet, C; Loeb, JE1
Gláz, ET; Tálas, M1
Lüllmann-Rauch, R; Pods, R; von Witzendorff, B1
Avrahami, D; Friedman-Levi, Y; Gabizon, R; Mayer-Sonnenfeld, T1
Comer, JE; Ekins, S; Freiberg, AN; Lane, TR; Madrid, PB1
Dyall, J; Ekins, S; Foil, DH; Goodin, C; Holbrook, MR; Lane, TR; Liang, JY; Madrid, PB; Mercer, L; Postnikova, E; Zhou, H1

Other Studies

17 other study(ies) available for quinacrine and tilorone

ArticleYear
Octanol-physiological buffer distribution coefficients of lipophilic amines by reversed-phase high-performance liquid chromatography and their correlation with biological activity.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:3

    Topics: Amines; Animals; Buffers; Chromatography, High Pressure Liquid; Histamine Release; Lipid Metabolism; Octanols; Protein Binding; Rats; Serum Albumin, Bovine; Sodium-Potassium-Exchanging ATPase; Solubility; Structure-Activity Relationship

1981
Interactions of antitumor drugs with natural DNA: 1H NMR study of binding mode and kinetics.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:4

    Topics: Antineoplastic Agents; Base Composition; Chemical Phenomena; Chemistry; DNA; Hydrogen Bonding; Intercalating Agents; Kinetics; Magnetic Resonance Spectroscopy; Structure-Activity Relationship

1984
Development of a phospholipidosis database and predictive quantitative structure-activity relationship (QSAR) models.
    Toxicology mechanisms and methods, 2008, Volume: 18, Issue:2-3

    Topics:

2008
Predicting phospholipidosis using machine learning.
    Molecular pharmaceutics, 2010, Oct-04, Volume: 7, Issue:5

    Topics: Animals; Artificial Intelligence; Databases, Factual; Drug Discovery; Humans; Lipidoses; Models, Biological; Phospholipids; Support Vector Machine

2010
In silico assay for assessing phospholipidosis potential of small druglike molecules: training, validation, and refinement using several data sets.
    Journal of medicinal chemistry, 2012, Jan-12, Volume: 55, Issue:1

    Topics: Animals; Cattle; Cells, Cultured; Computer Simulation; Cornea; Drug-Related Side Effects and Adverse Reactions; Fibroblasts; Lipidoses; Lysosomal Storage Diseases; Models, Molecular; Pharmaceutical Preparations; Phospholipids; Structure-Activity Relationship; Thermodynamics

2012
Identification of Antiviral Drug Candidates against SARS-CoV-2 from FDA-Approved Drugs.
    Antimicrobial agents and chemotherapy, 2020, 06-23, Volume: 64, Issue:7

    Topics: Animals; Anti-Inflammatory Agents; Antiviral Agents; Betacoronavirus; Cell Line; Chlorocebus aethiops; Coronavirus Infections; COVID-19; Drug Evaluation, Preclinical; Drug Repositioning; Humans; Niclosamide; Pandemics; Pneumonia, Viral; Pregnenediones; SARS-CoV-2; Vero Cells

2020
Toward the Target: Tilorone, Quinacrine, and Pyronaridine Bind to Ebola Virus Glycoprotein.
    ACS medicinal chemistry letters, 2020, Aug-13, Volume: 11, Issue:8

    Topics:

2020
Depression of hepatic cytochrome P-450-dependent monooxygenase systems with administered interferon inducing agents.
    Biochemical and biophysical research communications, 1976, Nov-22, Volume: 73, Issue:2

    Topics: Animals; Cytochrome P-450 Enzyme System; Interferons; Male; Mengovirus; Microsomes, Liver; Oxygenases; Pertussis Vaccine; Poly I-C; Quinacrine; Rats; RNA; Tilorone

1976
Bactericidal effects of combinations of ampicillin with anti-R-plasmid compounds on Salmonella typhimurium R1+.
    Antimicrobial agents and chemotherapy, 1977, Volume: 11, Issue:1

    Topics: Acridines; Ampicillin; Drug Combinations; Ethidium; Quinacrine; R Factors; Salmonella typhimurium; Tilorone

1977
Effect of tilorone and quinacrine on translation in reticulocyte lysates.
    Biochemical pharmacology, 1979, Dec-15, Volume: 28, Issue:24

    Topics: Animals; Fluorenes; Hemin; Leucine; Phenylhydrazines; Protein Biosynthesis; Quinacrine; Rabbits; Reticulocytes; Tilorone

1979
Interferon induction in human cell cultures by small molecular inducers (tilorone and acridines).
    Acta pathologica et microbiologica Scandinavica. Section B, Microbiology, 1977, Volume: 85, Issue:3

    Topics: Acridines; Cells, Cultured; Fibroblasts; Fluorenes; Humans; Interferon Inducers; Interferons; Leukocytes; Molecular Weight; Quinacrine; Tilorone

1977
Action of hemin on chromatin protein kinases of rat liver.
    FEBS letters, 1977, Sep-15, Volume: 81, Issue:2

    Topics: Animals; Caseins; Chromatin; Heme; Hemin; In Vitro Techniques; Liver; Male; Phosvitin; Protein Kinase Inhibitors; Protein Kinases; Quinacrine; Rats; Tilorone

1977
Comparison of the ability of small molecular interferon inducers: tilorone and acridine drugs.
    Archives of virology, 1975, Volume: 48, Issue:4

    Topics: Acridines; Aminacrine; Animals; Body Temperature; Chick Embryo; Chickens; Culture Techniques; Cycloheximide; Dactinomycin; Female; Fluorenes; Interferon Inducers; Interferons; Male; Mice; Propanolamines; Quinacrine; Rabbits; Tilorone; Vaccinia virus

1975
The antimalarials quinacrine and chloroquine induce weak lysosomal storage of sulphated glycosaminoglycans in cell culture and in vivo.
    Toxicology, 1996, Jun-17, Volume: 110, Issue:1-3

    Topics: Animals; Anti-Inflammatory Agents; Antimalarials; beta-N-Acetylhexosaminidases; Cattle; Cells, Cultured; Chloroquine; Dose-Response Relationship, Drug; Female; Fibroblasts; Glycosaminoglycans; Histocytochemistry; Lipidoses; Liver; Lysosomes; Microscopy, Electron; Microscopy, Fluorescence; Mucopolysaccharidoses; Quinacrine; Rats; Rats, Wistar; Structure-Activity Relationship; Sulfates; Tilorone

1996
Chemically induced accumulation of GAGs delays PrP(Sc) clearance but prolongs prion disease incubation time.
    Cellular and molecular neurobiology, 2008, Volume: 28, Issue:7

    Topics: Animals; Antiviral Agents; Central Nervous System; CHO Cells; Cricetinae; Cricetulus; Enzyme Inhibitors; Glycosaminoglycans; Infectious Disease Incubation Period; Lysosomes; Metabolic Clearance Rate; Mice; Mice, Inbred C57BL; Neurons; Prion Diseases; Protein Conformation; PrPSc Proteins; Quinacrine; Subcellular Fractions; Tilorone; Time Factors

2008
Repurposing Quinacrine against Ebola Virus Infection
    Antimicrobial agents and chemotherapy, 2019, Volume: 63, Issue:9

    Topics: Animals; Antimalarials; Antiviral Agents; Caco-2 Cells; Chlorocebus aethiops; Disease Models, Animal; Drug Repositioning; Ebolavirus; HeLa Cells; Hemorrhagic Fever, Ebola; Humans; Mice; Mice, Inbred BALB C; Microbial Sensitivity Tests; Quinacrine; Survival Analysis; Tilorone; Vero Cells; Viral Load

2019
Repurposing Pyramax®, quinacrine and tilorone as treatments for Ebola virus disease.
    Antiviral research, 2020, Volume: 182

    Topics: Antiviral Agents; Artesunate; Drug Combinations; Drug Repositioning; Drug Synergism; Ebolavirus; HeLa Cells; Hemorrhagic Fever, Ebola; Humans; Lysosomes; Machine Learning; MCF-7 Cells; Naphthyridines; Quinacrine; Tilorone; Virus Internalization

2020