quinacrine and pyrimethamine

quinacrine has been researched along with pyrimethamine in 39 studies

Research

Studies (39)

TimeframeStudies, this research(%)All Research%
pre-199033 (84.62)18.7374
1990's0 (0.00)18.2507
2000's2 (5.13)29.6817
2010's4 (10.26)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Adrián, F; Anderson, P; Brinker, A; Caldwell, JS; Chatterjee, A; Gray, NS; Henson, K; Janes, J; Kato, N; Kuhen, K; Matzen, JT; McNamara, C; Nagle, A; Nam, TG; Plouffe, D; Schultz, PG; Trager, R; Winzeler, EA; Yan, SF; Zhou, Y1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Barnes, SW; Bonamy, GM; Bopp, SE; Borboa, R; Bright, AT; Chatterjee, A; Che, J; Cohen, S; Dharia, NV; Diagana, TT; Fidock, DA; Froissard, P; Gagaring, K; Gettayacamin, M; Glynne, RJ; Gordon, P; Groessl, T; Kato, N; Kuhen, KL; Lee, MC; Mazier, D; McNamara, CW; Meister, S; Nagle, A; Nam, TG; Plouffe, DM; Richmond, W; Roland, J; Rottmann, M; Sattabongkot, J; Schultz, PG; Tuntland, T; Walker, JR; Winzeler, EA; Wu, T; Zhou, B; Zhou, Y1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Hüther, AM; Parnham, MJ; Sauer, A; Zhang, Y1
Peters, W3
Olatunde, IA1
Briesch, PE; Contacos, PG; Glew, RH; Krotoski, WA; Neva, FA1
Botha, D1
Moxey, PC; Robles, E; Schimmel, EM; Trier, JS1
Dawkins, AT; Stahler, N; Terzian, LA1
Ilan, J1
Hunsicker, LG1
Schmidt, LH1
Pinder, RM1
Fink, E; Kretschmar, W1
Bruce-Chwatt, LJ1
Chin, W; Coatney, GR; Contacos, PG; Lunn, JS1
Cenedella, RJ; Saxe, LH; Van Dyke, K1
Cenedella, R; Saxe, LH; Szustkiewicz, C; Van Dyke, K1
Gregory, KG; Peters, W1
Schneider, MD1
Reba, RC; Sheehy, TW1
Trager, W1
Purcell, WP; Singer, JA1
Doberstyn, EB1
Ferrante, A; Goh, DH1
AMMA, MK; GUJRAL, ML; MISRA, N; SAREEN, K; VARMA, DR; VIJAYAMMA, N1
CONTACOS, PG; MILLAR, JW; STITCHER, JE; YOUNG, MD1
COATNEY, GR; CONTACOS, PG; LUNN, JS1
SULLI, G; VARRONE, F1
ALVING, AS; BREWER, GJ; MILLAR, JW; POWELL, RD1
CROSBY, WH; KAUFMAN, RM1
EYLES, DE; MONTGOMERY, R; SANDOSHAM, AA1
NEAL, RA1

Reviews

7 review(s) available for quinacrine and pyrimethamine

ArticleYear
Recent advances in antimalarial chemotherapy and drug resistance.
    Advances in parasitology, 1974, Volume: 12

    Topics: Agglutination; Amodiaquine; Animals; Anti-Bacterial Agents; Antimalarials; Chloroquine; Cross Reactions; Drug Combinations; Drug Evaluation, Preclinical; Drug Resistance; Folic Acid Antagonists; Haplorhini; Humans; Lincomycin; Malaria; Pigments, Biological; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Plasmodium vivax; Primaquine; Pyrimethamine; Quinacrine; Quinine; Quinolines; Structure-Activity Relationship; Sulfonamides; Sulfones

1974
The present status of chloroquine in the drug treatment of malaria.
    The African journal of medical sciences, 1972, Volume: 3, Issue:1

    Topics: Chloroquine; Drug Resistance, Microbial; Humans; Malaria; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfonamides; Sulfones; Triazines

1972
The pharmacology of the antimalarials. A rational approach to the therapy of resistant falciparum malaria.
    Archives of internal medicine, 1969, Volume: 123, Issue:6

    Topics: Amodiaquine; Antimalarials; Chemical Phenomena; Chemistry; Chloroquine; Dapsone; Drug Resistance, Microbial; Humans; Malaria; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Sulfadimethoxine; Sulfisoxazole

1969
Chemotherapy of the drug-resistant malarias.
    Annual review of microbiology, 1969, Volume: 23

    Topics: Chloroquine; Cinchona; Drug Resistance, Microbial; Malaria; Mutation; Phytotherapy; Plants, Medicinal; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Quinolines; Sulfonamides; Sulfones

1969
Recent advances in the chemotherapy of malaria.
    Progress in medicinal chemistry, 1971, Volume: 8, Issue:2

    Topics: Acridines; Animals; Anti-Bacterial Agents; Antimalarials; Antineoplastic Agents; Cinchona; Culture Media; Humans; Malaria; Microbial Sensitivity Tests; Naphthoquinones; Phytotherapy; Plants, Medicinal; Plasmodium; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Proguanil; Pyrimethamine; Quinacrine; Quinolines; Sulfonamides; Sulfones

1971
Resistance of Plasmodium falciparum.
    Experientia, 1984, Dec-15, Volume: 40, Issue:12

    Topics: Africa; Animals; Antimalarials; Asia; Chloroquine; DNA; Drug Resistance; Drug Synergism; Hemin; Malaria; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Quinolines; Research; RNA; South America

1984
[EXTRAMALARIAL THERAPUETIC APPLICATIONS OF ANTIMALARIAL DRUGS. 1. CLINICAL UTILIZATIONS].
    La Clinica terapeutica, 1963, Oct-31, Volume: 27

    Topics: Amodiaquine; Antimalarials; Chloroquine; Collagen Diseases; Dermatology; Drug Utilization; Epilepsy; Female; Heart Diseases; Hematology; Humans; Hydroxychloroquine; Hypersensitivity; Multiple Sclerosis; Muscular Diseases; Neurology; Parasitic Diseases; Pharmacology; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Toxicology; Uterus

1963

Other Studies

32 other study(ies) available for quinacrine and pyrimethamine

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
In silico activity profiling reveals the mechanism of action of antimalarials discovered in a high-throughput screen.
    Proceedings of the National Academy of Sciences of the United States of America, 2008, Jul-01, Volume: 105, Issue:26

    Topics: Animals; Antimalarials; Cluster Analysis; Computational Biology; Drug Evaluation, Preclinical; Drug Resistance; Folic Acid Antagonists; Malaria; Models, Molecular; Parasites; Plasmodium falciparum; Reproducibility of Results; Structure-Activity Relationship; Tetrahydrofolate Dehydrogenase

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Imaging of Plasmodium liver stages to drive next-generation antimalarial drug discovery.
    Science (New York, N.Y.), 2011, Dec-09, Volume: 334, Issue:6061

    Topics: Animals; Antimalarials; Cell Line, Tumor; Drug Discovery; Drug Evaluation, Preclinical; Drug Resistance; Erythrocytes; Humans; Imidazoles; Liver; Malaria; Mice; Mice, Inbred BALB C; Molecular Structure; Piperazines; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Plasmodium yoelii; Polymorphism, Single Nucleotide; Protozoan Proteins; Random Allocation; Small Molecule Libraries; Sporozoites

2011
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Antimalarial properties of ebselen.
    Parasitology research, 1989, Volume: 75, Issue:5

    Topics: Animals; Antimalarials; Antioxidants; Azoles; Cell Line; Humans; Isoindoles; Macrophages; Malaria; Male; Mice; Molecular Structure; Organoselenium Compounds; Plasmodium berghei; Plasmodium falciparum; Pyrimethamine; Quinacrine; Selenium

1989
Multidrug-resistant strain of Plasmodium falciparum from eastern Colombia.
    The Journal of infectious diseases, 1974, Volume: 129, Issue:4

    Topics: Adolescent; Adult; Antimalarials; Chloroquine; Colombia; Drug Combinations; Drug Resistance, Microbial; Female; Humans; Malaria; Male; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine

1974
Some pharmacological aspects of antimalarial drugs.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 1974, Jun-15, Volume: 48, Issue:29

    Topics: Antimalarials; Chloroquine; Dapsone; Drug Resistance, Microbial; Humans; Malaria; Plasmodium falciparum; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfonamides; Trimethoprim

1974
Chronic intestinal coccidiosis in man: intestinal morphology and response to treatment.
    Gastroenterology, 1974, Volume: 66, Issue:5

    Topics: Antiprotozoal Agents; Biopsy; Chloroquine; Chronic Disease; Coccidiosis; Diagnosis, Differential; Diarrhea; Diet Therapy; Drug Therapy, Combination; Duodenum; Follow-Up Studies; Humans; Intestinal Diseases, Parasitic; Intestine, Small; Isospora; Jejunum; Malabsorption Syndromes; Male; Metronidazole; Microscopy, Electron; Middle Aged; Nitrofurantoin; Primaquine; Pyrimethamine; Quinacrine; Sulfadiazine; Tetracycline; Time Factors

1974
The sporogonous of Plasmodium vivax in Anopheles mosquitoes as a system for evaluating the prophylactic and curative capabilities of potential antimalarial compounds.
    Experimental parasitology, 1968, Volume: 23, Issue:1

    Topics: Animals; Anopheles; Antimalarials; Chloroquine; Malaria; Naphthoquinones; Oxytetracycline; Penicillin G; Plasmodium vivax; Primaquine; Proguanil; Pyridines; Pyrimethamine; Quinacrine; Quinine; Quinolines; Sulfadiazine; Thiosemicarbazones

1968
Aminoacyl transfer ribonucleic acid synthetases from cell-free extract of Plasmodium berghei.
    Science (New York, N.Y.), 1969, May-02, Volume: 164, Issue:3879

    Topics: Acridines; Amino Acids; Carbon Isotopes; Cell-Free System; Escherichia coli; Genetic Code; Histidine; Leucine; Ligases; Liver; Lysine; Plasmodium; Proline; Pyrimethamine; Quinacrine; RNA, Transfer; Species Specificity; Stilbamidines; Threonine; Tyrosine; Valine

1969
[Chemotherapeutic activity of standard antimalarials in a simplified test for Plasmodium vinckey infection in the NMPI mouse].
    Zeitschrift fur Tropenmedizin und Parasitologie, 1970, Volume: 21, Issue:2

    Topics: Animals; Antimalarials; Chloroquine; Long-Term Care; Malaria; Mice; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Sulfonamides; Time Factors

1970
The role of drugs in a malaria program.
    The American journal of tropical medicine and hygiene, 1972, Volume: 21, Issue:5

    Topics: Amodiaquine; Antimalarials; Chloroquine; Dose-Response Relationship, Drug; Humans; Malaria; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Recurrence; Sulfonamides; Sulfones; Trimethoprim

1972
Resistance to cycloguanil pamoate (CI-501) by falciparum malaria in West Pakistan.
    The American journal of tropical medicine and hygiene, 1965, Volume: 14, Issue:6

    Topics: Adolescent; Antimalarials; Child; Child, Preschool; Female; Humans; Infant; Malaria; Male; Pakistan; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Quinine

1965
An automated method of mass drug testing applied to screening for antimalarial activity.
    Chemotherapy, 1970, Volume: 15, Issue:3

    Topics: Animals; Antimalarials; Automation; Chloroquine; Erythrocytes; Glucose; Glycolysis; Lactates; Male; Methods; Neoplasms, Experimental; Pharmacology; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rats; Sulfadiazine; Sulfones

1970
A unique antinucleic acid approach to the mass screening of antimalarial drugs.
    Chemotherapy, 1970, Volume: 15, Issue:3

    Topics: Animals; Antimalarials; Cell Membrane; Chemical Phenomena; Chemistry; Chloroquine; Computers; DNA, Bacterial; Erythrocytes; Hydrogen-Ion Concentration; Nucleosides; Pharmacology; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rats; RNA, Bacterial; Sulfones; Temperature; Tritium

1970
The chemotherapy of rodent malaria. IX. Causal prophylaxis. I. A method for demonstrating drug action on exo-erythrocytic stages.
    Annals of tropical medicine and parasitology, 1970, Volume: 64, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Dapsone; Malaria; Male; Mice; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Triazines

1970
The chemotherapy of rodent malaria. XII. Substituted tetrahydrofurans, a new chemical family of antimalarials. The action of 2-(p-chlorophenyl)-2-(4-piperidyl)-tetrahydrofuran against Plasmodium berghei and Plasmodium chabaudi.
    Annals of tropical medicine and parasitology, 1970, Volume: 64, Issue:2

    Topics: Aminobenzoates; Animals; Antimalarials; Chloroquine; Diet; Drug Resistance, Microbial; Drug Synergism; Folic Acid; Furans; Mice; Piperidines; Plasmodium; Pyrimethamine; Quinacrine; Sulfadiazine; Triazines

1970
Characteristics and cross-resistance patterns of chloroquine-resistant Plasmodium berghei infections in mice.
    Experimental parasitology, 1968, Volume: 23, Issue:1

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Dapsone; Drug Resistance, Microbial; Female; Hematocrit; Isoenzymes; L-Lactate Dehydrogenase; Malaria; Mice; Organ Size; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rodent Diseases; Serum Albumin; Serum Globulins; Spleen; Splenomegaly; Sulfadiazine

1968
Drug resistance in Plasmodium berghei Vincke and Lips, 1948. I. Chloroquine resistance.
    Experimental parasitology, 1965, Volume: 17, Issue:1

    Topics: Amodiaquine; Animals; Chloroquine; Dapsone; Malaria; Mice; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Sulfadiazine; Triazines

1965
Treatment of chloroquine-resistant Plasmodium falciparum infections in Vietnam.
    Annals of internal medicine, 1967, Volume: 66, Issue:3

    Topics: Chloroquine; Dapsone; Humans; Malaria; Military Medicine; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Sulfonamides; Vietnam

1967
The different effects of antimalarial drugs on Plasmodium lophurae developing intracellularly and extracellularly in vitro.
    The American journal of tropical medicine and hygiene, 1967, Volume: 16, Issue:1

    Topics: Animals; Chloroquine; In Vitro Techniques; Malaria, Avian; Plasmodium; Pyrimethamine; Quinacrine; Sulfadiazine

1967
Hückel molecular orbital calculations for some antimalarial drugs and related molecules.
    Journal of medicinal chemistry, 1967, Volume: 10, Issue:5

    Topics: Antimalarials; Chemical Phenomena; Chemistry, Physical; Chloroquine; DNA; Primaquine; Pyrimethamine; Quinacrine; Quinine; RNA

1967
The effect of anti-malarial drugs on human natural killer cells in vitro.
    Parasite immunology, 1984, Volume: 6, Issue:6

    Topics: Antimalarials; Cell Line; Chloroquine; Cytotoxicity, Immunologic; Humans; Killer Cells, Natural; Leukemia, Myeloid, Acute; Mefloquine; Primaquine; Pyrimethamine; Quinacrine; Quinine; Quinolines

1984
Oral contraceptives. VII. Antimalarials as antifertility agents.
    Indian journal of physiology and pharmacology, 1962, Volume: 6

    Topics: Amodiaquine; Antimalarials; Chloroquine; Contraceptive Agents; Contraceptives, Oral; Female; Humans; Proguanil; Pyrimethamine; Quinacrine

1962
DRUG RESISTANCE IN PLASMODIUM FALCIPARUM FROM THAILAND.
    The American journal of tropical medicine and hygiene, 1963, Volume: 12

    Topics: Amodiaquine; Antimalarials; Chloroquine; Drug Resistance; Drug Resistance, Microbial; Humans; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Quinine; Thailand

1963
DRUG-RESISTANT FALCIPARUM MALARIA FROM CAMBODIA AND MALAYA.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1963, Volume: 57

    Topics: Animals; Cambodia; Chloroquine; Culicidae; Drug Resistance; Drug Resistance, Microbial; Humans; Malaria; Malaria, Falciparum; Malaysia; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Quinine

1963
STUDIES ON A STRAIN OF CHLOROQUINE-RESISTANT PLASMODIUM FALCIPARUM FROM THAILAND.
    Bulletin of the World Health Organization, 1964, Volume: 30

    Topics: Amodiaquine; Antimalarials; Asia, Southeastern; Biomedical Research; Chloroquine; Drug Resistance; Drug Resistance, Microbial; Humans; Hydroxychloroquine; Malaria; Malaria, Falciparum; Pharmacology; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Quinine; Thailand

1964
DRUG-INDUCED THROMBOCYTOPENIA.
    The Medical annals of the District of Columbia, 1964, Volume: 33

    Topics: Acetazolamide; Anticonvulsants; Arsphenamine; Chloramphenicol; Chlorothiazide; Colchicine; Gold; Hydantoins; Hypoglycemic Agents; Meprobamate; Perchlorates; Phenothiazines; Phenylbutazone; Pyrimethamine; Quinacrine; Quinidine; Quinine; Ristocetin; Streptomycin; Sulfonamides; Thrombocytopenia; Toxicology

1964
DRUG-RESISTANCE IN FALCIPARUM MALARIA IN SOUTH-EAST ASIA.
    The Medical journal of Malaya, 1964, Volume: 18

    Topics: Adolescent; Asia, Southeastern; Child; Chloroquine; Drug Resistance; Drug Resistance, Microbial; Drug Therapy; Humans; Malaria; Plasmodium falciparum; Proguanil; Pyrimethamine; Quinacrine; Quinine; Statistics as Topic; Toxicology

1964
CHEMOTHERAPY OF CUTANEOUS LEISHMANIASIS: LEISHMANIA TROPICA INFECTIONS IN MICE.
    Annals of tropical medicine and parasitology, 1964, Volume: 58

    Topics: Amidines; Animals; Antimony; Antiprotozoal Agents; Chloroquine; Chlortetracycline; Dapsone; Deoxyribonuclease I; Emetine; Hyaluronoglucosaminidase; Hydrastis; Leishmania tropica; Leishmaniasis; Leishmaniasis, Cutaneous; Leishmaniasis, Mucocutaneous; Mice; Pathology; Pharmacology; Primaquine; Pyrimethamine; Quinacrine; Research; Streptodornase and Streptokinase; Streptokinase; Sulfonamides; Surface-Active Agents; Toxicology

1964