quinacrine and pyrilamine

quinacrine has been researched along with pyrilamine in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19904 (40.00)18.7374
1990's3 (30.00)18.2507
2000's2 (20.00)29.6817
2010's1 (10.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Castro, GA; Russell, DA1
Dveksler, G; Franchi, AM; Gimeno, AL; Gimeno, MF; Viggiano, M1
Nakajima, K1
Enomoto, K; Maeno, T1
Lot, TY1
Horio, S; Ishida, Y; Moritoki, H; Nagare, T1
Al Obaid, AR; Al Rasheed, NM; Al Sayed, MI; Al Zuhair, HH; Fatani, AJ1

Other Studies

10 other study(ies) available for quinacrine and pyrilamine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
    Journal of medicinal chemistry, 2008, Jan-24, Volume: 51, Issue:2

    Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase

2008
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Immunological regulation of colonic ion transport.
    The American journal of physiology, 1989, Volume: 256, Issue:2 Pt 1

    Topics: Animals; Antigens, Helminth; Bradykinin; Colon; Dinoprostone; Electric Conductivity; Evoked Potentials; Furosemide; Guinea Pigs; Histamine Release; Indomethacin; Jejunum; Male; Pyrilamine; Quinacrine; Reference Values; Tetrodotoxin; Trichinella; Trichinellosis

1989
Is there a prostaglandin involvement in the positive inotropic action of histamine in isolated pregnant rat uterus, apparently mediated via H1-receptors activation?
    Prostaglandins, leukotrienes, and medicine, 1987, Volume: 28, Issue:3

    Topics: Alprostadil; Animals; Aspirin; Chlorpheniramine; Cimetidine; Dinoprost; Dinoprostone; Female; Histamine; Pregnancy; Prostaglandins; Prostaglandins E; Prostaglandins F; Pyrilamine; Quinacrine; Rats; Receptors, Histamine; Receptors, Histamine H1; Stimulation, Chemical; Uterine Contraction

1987
A possible mechanism of vasoactive agents on plasminogen activator release in isolated perfused pig ears.
    Thrombosis research, 1983, Jan-15, Volume: 29, Issue:2

    Topics: Acetylcholine; Animals; Atropine; Bradykinin; Dilazep; Dose-Response Relationship, Drug; Drug Synergism; Ear, External; Histamine; In Vitro Techniques; Indomethacin; Papaverine; Perfusion; Plasminogen Activators; Pressure; Pyrilamine; Quinacrine; Swine; Thrombin; Vasoconstrictor Agents; Vasodilator Agents; Vasomotor System

1983
Effects of vesicular acetylcholine uptake blockers on frequency augmentation-potentiation in frog neuromuscular transmission.
    Neuroscience, 1994, Volume: 59, Issue:2

    Topics: Acetylcholine; Animals; Antidepressive Agents; Azepines; Chloroquine; Ethacridine; Evoked Potentials; In Vitro Techniques; Neuromuscular Depolarizing Agents; Neuromuscular Junction; Piperidines; Pyrilamine; Quinacrine; Ranidae; Regression Analysis; Synaptic Transmission

1994
The effects of chronic administration of chloroquine and quinacrine on the response of normal and denervated smooth muscle to agonist drugs.
    Physiology & behavior, 1993, Volume: 54, Issue:2

    Topics: Acetylcholine; Age Factors; Animals; Atropine; Chickens; Chloroquine; Culture Techniques; Dose-Response Relationship, Drug; Histamine; Male; Muscle, Smooth; Neurotransmitter Agents; Norepinephrine; Potassium Chloride; Pyrilamine; Quinacrine; Serotonin; Synaptic Transmission

1993
Interaction of local anaesthetics with histamine H1 receptors in guinea-pig ileum.
    The Journal of pharmacy and pharmacology, 1997, Volume: 49, Issue:7

    Topics: Anesthetics, Local; Animals; Binding, Competitive; Chloroquine; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine H1 Antagonists; Ileum; Isotope Labeling; Male; Muscle Contraction; Muscle, Smooth; Procaine; Pyrilamine; Quinacrine; Receptors, Histamine H1; Structure-Activity Relationship; Tetracaine

1997
Effects of two newly synthesized analogues of lidocaine on rat arterial blood pressure and heart rate.
    Pharmacological research, 2001, Volume: 43, Issue:4

    Topics: Anesthetics, Local; Animals; Anti-Arrhythmia Agents; Antihypertensive Agents; Atropine; Benzoates; Blood Pressure; Calcium Chloride; Cyproheptadine; Enzyme Inhibitors; Heart Rate; Hexamethonium; Histamine Agonists; Indomethacin; Lidocaine; Male; Monitoring, Physiologic; NG-Nitroarginine Methyl Ester; Pyrilamine; Quinacrine; Ranitidine; Rats; Rats, Wistar; Vasodilator Agents

2001