quinacrine and primaquine

quinacrine has been researched along with primaquine in 64 studies

Research

Studies (64)

TimeframeStudies, this research(%)All Research%
pre-199050 (78.13)18.7374
1990's1 (1.56)18.2507
2000's7 (10.94)29.6817
2010's6 (9.38)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Galanakis, D; Ganellin, CR1
Danis, M; Derouin, F; Farhati, K; Franetich, JF; Galvez, J; Garcia-Domenech, R; Hannoun, L; Mahmoudi, N; Mazier, D; Sauerwein, R1
Fitos, I; Mády, G; Visy, J; Zsila, F1
Lombardo, F; Obach, RS; Waters, NJ1
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Bane, CE; Black, C; Butler, K; Caridha, D; Cooper, RA; Dodean, RA; Gaona, H; Gaynor-Ohnstad, L; Huezo, SJ; Kancharla, P; Kelly, JX; Kreishman-Deitrick, M; Leed, SE; Li, Q; Li, Y; Lin, H; Luong, TL; Marcsisin, S; Melendez, V; Nolan, C; Olmeda, R; Potter, B; Pou, S; Rasmussen, SA; Read, L; Riscoe, MK; Roncal, N; Sciotti, RJ; Smilkstein, MJ; Sousa, J; Stephens, MT; Tan, JC; Vesely, B; Vuong, C; Winter, RW; Xie, L; Zeng, Q; Zhang, J; Zhang, P1
Garfinkel, E; Hirschman, SZ1
Mattock, NM; Peters, W1
Holbrook, DJ; Washington, ME; Wichard, LP1
Emerole, GO; Nashiru, TO; Thabrew, MI1
Butler, KW; Deslauriers, R; Smith, IC1
Shao, BR; Xu, YQ1
Bohn, E; Hesse, B; Kunze, H; Löffler, BM1
Chou, SC; Conklin, KA; Pan, HY1
Chou, SC; Levy, MR1
Peters, W2
Cowey, FK; Whitehouse, MW1
Fain, JN; Pointer, RH1
Bacchi, CJ; Goldberg, B; Hutner, SH; Lambros, C1
Miller, A; Natsios, G; Smith, HC1
Olatunde, IA1
Botha, D1
Chou, SC; Conklin, KA2
Moxey, PC; Robles, E; Schimmel, EM; Trier, JS1
Dawkins, AT; Stahler, N; Terzian, LA1
Schmidt, LH1
Fink, E; Kretschmar, W1
Chou, SC; Conklin, KA; Heu, P1
Aviado, DM; Bass, SW; Ramirez, MA1
Bruce-Chwatt, LJ1
Miller, A; Smith, HC2
Ball, EG; Markus, HB1
Cenedella, RJ; Saxe, LH; Van Dyke, K1
Cenedella, R; Saxe, LH; Szustkiewicz, C; Van Dyke, K1
Polet, H1
Gregory, KG; Peters, W1
Bishop, A1
Clancy, CF1
Schneider, MD1
Ott, KJ1
Elslager, EF; Tendick, FH; Werbel, LM1
Purcell, WP; Singer, JA1
Doberstyn, EB1
Ferrante, A; Goh, DH1
Dubin, NH; Ghodgaonkar, RB; King, TM; Parmley, TH1
Ioannides, C; Thabrew, MI1
Bohn, E; Hesse, B; Kunze, H1
Gu, HM; Qu, ZX; Zeng, YL1
Arnold, W; Gahl, GM; Hess, G; Meyer zum Büschenfelde, KH; Möller, B1
Bächinger, HP; Hinrichs, DJ; Ignatushchenko, MV; Riscoe, MK; Winter, RW1
SASLAW, S; SCHAEFER, J1
ARORA, RB; LAL, A1
SULLI, G; VARRONE, F1
NEAL, RA1
Haystead, TA; Kwiek, JJ; Rudolph, J1
Nishikawa, T; Omura, M; Suematsu, S1
Baird, JK1
Barth, H; Benz, R; Kreidler, AM1

Reviews

5 review(s) available for quinacrine and primaquine

ArticleYear
Recent advances in antimalarial chemotherapy and drug resistance.
    Advances in parasitology, 1974, Volume: 12

    Topics: Agglutination; Amodiaquine; Animals; Anti-Bacterial Agents; Antimalarials; Chloroquine; Cross Reactions; Drug Combinations; Drug Evaluation, Preclinical; Drug Resistance; Folic Acid Antagonists; Haplorhini; Humans; Lincomycin; Malaria; Pigments, Biological; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Plasmodium vivax; Primaquine; Pyrimethamine; Quinacrine; Quinine; Quinolines; Structure-Activity Relationship; Sulfonamides; Sulfones

1974
The present status of chloroquine in the drug treatment of malaria.
    The African journal of medical sciences, 1972, Volume: 3, Issue:1

    Topics: Chloroquine; Drug Resistance, Microbial; Humans; Malaria; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfonamides; Sulfones; Triazines

1972
Chemotherapy of the drug-resistant malarias.
    Annual review of microbiology, 1969, Volume: 23

    Topics: Chloroquine; Cinchona; Drug Resistance, Microbial; Malaria; Mutation; Phytotherapy; Plants, Medicinal; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Quinolines; Sulfonamides; Sulfones

1969
Resistance of Plasmodium falciparum.
    Experientia, 1984, Dec-15, Volume: 40, Issue:12

    Topics: Africa; Animals; Antimalarials; Asia; Chloroquine; DNA; Drug Resistance; Drug Synergism; Hemin; Malaria; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Quinolines; Research; RNA; South America

1984
[EXTRAMALARIAL THERAPUETIC APPLICATIONS OF ANTIMALARIAL DRUGS. 1. CLINICAL UTILIZATIONS].
    La Clinica terapeutica, 1963, Oct-31, Volume: 27

    Topics: Amodiaquine; Antimalarials; Chloroquine; Collagen Diseases; Dermatology; Drug Utilization; Epilepsy; Female; Heart Diseases; Hematology; Humans; Hydroxychloroquine; Hypersensitivity; Multiple Sclerosis; Muscular Diseases; Neurology; Parasitic Diseases; Pharmacology; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Toxicology; Uterus

1963

Other Studies

59 other study(ies) available for quinacrine and primaquine

ArticleYear
Defining determinant molecular properties for the blockade of the apamin-sensitive SKCa channel in guinea-pig hepatocytes: the influence of polarizability and molecular geometry.
    Bioorganic & medicinal chemistry letters, 2004, Aug-02, Volume: 14, Issue:15

    Topics: Animals; Apamin; Guinea Pigs; Hepatocytes; Kinetics; Molecular Conformation; Potassium Channels, Calcium-Activated

2004
New active drugs against liver stages of Plasmodium predicted by molecular topology.
    Antimicrobial agents and chemotherapy, 2008, Volume: 52, Issue:4

    Topics: Animals; Antimalarials; Hepatocytes; Humans; Liver; Mice; Models, Biological; Parasitic Sensitivity Tests; Plasmodium yoelii; Structure-Activity Relationship

2008
Selective plasma protein binding of antimalarial drugs to alpha1-acid glycoprotein.
    Bioorganic & medicinal chemistry, 2008, Apr-01, Volume: 16, Issue:7

    Topics: Antimalarials; Binding Sites; Chromatography, Affinity; Circular Dichroism; Humans; Molecular Structure; Orosomucoid; Protein Binding; Serum Albumin; Spectrophotometry; Stereoisomerism; Structure-Activity Relationship

2008
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Discovery and Structural Optimization of Acridones as Broad-Spectrum Antimalarials.
    Journal of medicinal chemistry, 2019, 04-11, Volume: 62, Issue:7

    Topics: Acridones; Animals; Antimalarials; Disease Models, Animal; Drug Discovery; Hep G2 Cells; Humans; Malaria; Mice; Plasmodium; Species Specificity; Structure-Activity Relationship

2019
Inhibition of hepatitis B DNA polymerase by intercalating agents.
    Nature, 1978, Feb-16, Volume: 271, Issue:5646

    Topics: Chloroquine; Chlorpromazine; Drug Synergism; Ethidium; Hepatitis B; Hepatitis B virus; Humans; Indicators and Reagents; Methylene Blue; Nucleic Acid Synthesis Inhibitors; Primaquine; Quinacrine

1978
The experimental chemotherapy of leishmaniasis. II. The activity in tissue culture of some antiparasitic and antimicrobial compounds in clinical use.
    Annals of tropical medicine and parasitology, 1975, Volume: 69, Issue:3

    Topics: Aminoquinolines; Animals; Anti-Bacterial Agents; Antimalarials; Antimony; Antiprotozoal Agents; Ascitic Fluid; Cell Line; Chloroquine; Cricetinae; Culture Techniques; Dogs; Drug Evaluation, Preclinical; Folic Acid Antagonists; Leishmania; Niridazole; Pentamidine; Primaquine; Quinacrine; Quinine; Sarcoma; Sulfonamides; Sulfones; Suramin

1975
Effect of nucleic-acid-binding compounds on the hydrolytic activity of various ribonucleases.
    European journal of biochemistry, 1975, Dec-15, Volume: 60, Issue:2

    Topics: Acridines; Aminoquinolines; Animals; Binding Sites; Cattle; Chloroquine; Ethidium; Kinetics; Pancreas; Primaquine; Proflavine; Protein Binding; Quinacrine; Ribonucleases; Spermidine; Spermine; Structure-Activity Relationship

1975
Drug induced alterations in some rat hepatic microsomal components: a comparative study of four structurally different antimalarials.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1985, Volume: 81, Issue:1

    Topics: Aminopyrine N-Demethylase; Aniline Hydroxylase; Animals; Antimalarials; Aryl Hydrocarbon Hydroxylases; Chloroquine; Cholesterol; Cytosol; Glutathione Transferase; Liver; Male; Microsomes, Liver; Phospholipids; Primaquine; Quinacrine; Quinine; Rats; Rats, Inbred Strains

1985
Effects of antimalarial drugs on oxygen consumption by erythrocytes infected with Plasmodium berghei: an ESR study.
    Magnetic resonance in medicine, 1986, Volume: 3, Issue:2

    Topics: Animals; Antimalarials; Depression, Chemical; Electron Spin Resonance Spectroscopy; Erythrocytes; Malaria; Male; Mice; Oxygen Consumption; Plasmodium berghei; Primaquine; Quinacrine; Quinine

1986
[The mouse micronucleus test for mutagenicity of pyronaridine, chloroquine, quinacrine, primaquine, furapyrimidone and phenthiourezine].
    Zhongguo ji sheng chong xue yu ji sheng chong bing za zhi = Chinese journal of parasitology & parasitic diseases, 1988, Volume: 6, Issue:4

    Topics: Animals; Anthelmintics; Antimalarials; Chloroquine; Filaricides; Male; Mice; Micronucleus Tests; Mutagenicity Tests; Naphthyridines; Nitrofurans; Piperazines; Primaquine; Quinacrine

1988
Effects of antimalarial drugs on phospholipase A and lysophospholipase activities in plasma membrane, mitochondrial, microsomal and cytosolic subcellular fractions of rat liver.
    Biochimica et biophysica acta, 1985, Jul-31, Volume: 835, Issue:3

    Topics: Animals; Antimalarials; Cell Membrane; Chloroquine; Cytosol; Endoplasmic Reticulum; Liver; Lysophospholipase; Male; Microsomes, Liver; Mitochondria, Liver; Phospholipases; Phospholipases A; Phospholipases A1; Phospholipases A2; Primaquine; Quinacrine; Rats; Rats, Inbred Strains

1985
Effects of antimalarial drugs and clofibrate on in vitro lipid synthesis in Tetrahymena pyriformis GL.
    Pharmacology, 1974, Volume: 12, Issue:1

    Topics: Acetates; Adenosine Triphosphate; Carbon Radioisotopes; Cell Division; Cell-Free System; Chloroquine; Chromatography, Thin Layer; Clofibrate; Depression, Chemical; Fatty Acids, Nonesterified; Lipids; NADH, NADPH Oxidoreductases; Phospholipids; Primaquine; Quinacrine; Quinine; Stimulation, Chemical; Tetrahymena pyriformis; Triglycerides

1974
Activity and some properties of an acid proteinase from normal and Plasmodium berghei-infected red cells.
    The Journal of parasitology, 1973, Volume: 59, Issue:6

    Topics: Acid Phosphatase; Animals; Cell-Free System; Chloroquine; Dithiothreitol; Edetic Acid; Erythrocytes; Female; Hemoglobins; Hemolysis; Hydrogen-Ion Concentration; Malaria; Mice; Mice, Inbred BALB C; Peptide Hydrolases; Plasmodium berghei; Primaquine; Quinacrine; Rats; Solubility; Surface-Active Agents; Ultracentrifugation

1973
Biochemical properties of anti-inflammatory drugs. VII. Inhibition of proteolytic enzymes in connective tissue by chloroquine (resochin) and related antimalarial antirheumatic drugs.
    Biochemical pharmacology, 1966, Volume: 15, Issue:8

    Topics: Acridines; Animals; Cartilage; Cattle; Chloroquine; Chondroitin; Connective Tissue; Hyaluronoglucosaminidase; Hydrogen-Ion Concentration; Hydroxychloroquine; Microbial Collagenase; Mucoproteins; Papain; Primaquine; Quaternary Ammonium Compounds; Quinacrine; Rabbits

1966
Response of isolated white fat cells to anti-malarial drugs.
    Biochemical pharmacology, 1973, Dec-01, Volume: 22, Issue:23

    Topics: Adenylyl Cyclase Inhibitors; Adipose Tissue; Animals; Antimalarials; Bucladesine; Chloroquine; Drug Synergism; Fatty Acids, Nonesterified; Female; Glycerol; Norepinephrine; Primaquine; Proteins; Quinacrine; Quinidine; Rats; Theophylline; Triglycerides

1973
Inhibition by several standard antiprotozoal drugs of growth and O2 uptake of cells and particulate preparations of a Leptomonas.
    The Journal of protozoology, 1974, Volume: 21, Issue:2

    Topics: Acridines; Alkanesulfonates; Amidines; Arsenicals; Culture Media; Ethidium; Eukaryota; Glycerophosphates; Hydrogen-Ion Concentration; Oxygen Consumption; Phenyl Ethers; Primaquine; Proline; Pyrimidines; Quinacrine; Quinolinium Compounds; Rotenone; Stilbamidines; Succinates; Suramin; Triazines; Trypanocidal Agents

1974
Effect of antimalarial drugs on the efflux of K+ from Streptococcus pyogenes.
    Biochemical pharmacology, 1971, Volume: 20, Issue:11

    Topics: Antimalarials; Biological Transport; Cell Membrane Permeability; Chloroquine; Culture Media; Potassium; Potassium Isotopes; Primaquine; Quinacrine; Quinine; Streptococcus pneumoniae; Streptococcus pyogenes

1971
Some pharmacological aspects of antimalarial drugs.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 1974, Jun-15, Volume: 48, Issue:29

    Topics: Antimalarials; Chloroquine; Dapsone; Drug Resistance, Microbial; Humans; Malaria; Plasmodium falciparum; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfonamides; Trimethoprim

1974
The effects of antimalarial drugs on uptake and incorporation of macromolecular precursors by Tetrahymena pyriformis.
    The Journal of pharmacology and experimental therapeutics, 1972, Volume: 180, Issue:1

    Topics: Amino Acids; Animals; Antimalarials; Carbon Isotopes; Cell Division; Chloroquine; Cycloheximide; Dactinomycin; DNA; Kinetics; Macromolecular Substances; Nalidixic Acid; Primaquine; Quinacrine; Quinine; RNA; Tetrahymena pyriformis; Thymidine; Uridine

1972
Chronic intestinal coccidiosis in man: intestinal morphology and response to treatment.
    Gastroenterology, 1974, Volume: 66, Issue:5

    Topics: Antiprotozoal Agents; Biopsy; Chloroquine; Chronic Disease; Coccidiosis; Diagnosis, Differential; Diarrhea; Diet Therapy; Drug Therapy, Combination; Duodenum; Follow-Up Studies; Humans; Intestinal Diseases, Parasitic; Intestine, Small; Isospora; Jejunum; Malabsorption Syndromes; Male; Metronidazole; Microscopy, Electron; Middle Aged; Nitrofurantoin; Primaquine; Pyrimethamine; Quinacrine; Sulfadiazine; Tetracycline; Time Factors

1974
The sporogonous of Plasmodium vivax in Anopheles mosquitoes as a system for evaluating the prophylactic and curative capabilities of potential antimalarial compounds.
    Experimental parasitology, 1968, Volume: 23, Issue:1

    Topics: Animals; Anopheles; Antimalarials; Chloroquine; Malaria; Naphthoquinones; Oxytetracycline; Penicillin G; Plasmodium vivax; Primaquine; Proguanil; Pyridines; Pyrimethamine; Quinacrine; Quinine; Quinolines; Sulfadiazine; Thiosemicarbazones

1968
[Chemotherapeutic activity of standard antimalarials in a simplified test for Plasmodium vinckey infection in the NMPI mouse].
    Zeitschrift fur Tropenmedizin und Parasitologie, 1970, Volume: 21, Issue:2

    Topics: Animals; Antimalarials; Chloroquine; Long-Term Care; Malaria; Mice; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Sulfonamides; Time Factors

1970
Quinine: effect of Tetrahymena pyriformis. 3. Energetics of isolated mitochondria in the presence of quinine and other antimalarial drugs.
    Biochemical pharmacology, 1971, Volume: 20, Issue:8

    Topics: Chloroquine; Citrates; Citric Acid Cycle; Depression, Chemical; Fumarates; Glutamates; Hydroxybutyrates; Isocitrates; Ketoglutaric Acids; Malates; Mitochondria; Oxidative Phosphorylation; Oxygen Consumption; Primaquine; Quinacrine; Quinine; Stimulation, Chemical; Succinates; Tetrahymena pyriformis; Uncoupling Agents

1971
Cardiopulmonary effects of antimalarial drugs. VI. Adenosine, quinacrine and primaquine.
    Toxicology and applied pharmacology, 1972, Volume: 21, Issue:4

    Topics: Adenosine; Animals; Anti-Arrhythmia Agents; Blood Pressure; Cardiac Output; Cats; Coronary Circulation; Dogs; Drug Interactions; Electrocardiography; Female; Heart; Heart Rate; Hemodynamics; Isoproterenol; Male; Mice; Muscle Contraction; Primaquine; Pulmonary Circulation; Quinacrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Vascular Resistance; Ventricular Fibrillation

1972
The role of drugs in a malaria program.
    The American journal of tropical medicine and hygiene, 1972, Volume: 21, Issue:5

    Topics: Amodiaquine; Antimalarials; Chloroquine; Dose-Response Relationship, Drug; Humans; Malaria; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Recurrence; Sulfonamides; Sulfones; Trimethoprim

1972
The influence of glucose and exogenous glutathione on the red cell membrane effect of the antimalarial drugs 1,4-naphthoquinone and beta-naphthol.
    British journal of haematology, 1971, Volume: 20, Issue:6

    Topics: Cell Membrane; Erythrocytes; Glucose; Glutathione; Hemolysis; Humans; In Vitro Techniques; Methemoglobin; Naphthalenes; Naphthoquinones; Osmotic Fragility; Potassium; Primaquine; Quinacrine; Quinine

1971
Inhibition of lipolytic processes in rat adipose tissue by antimalaria drugs.
    Biochimica et biophysica acta, 1969, Dec-17, Volume: 187, Issue:4

    Topics: Adipose Tissue; Animals; Antimalarials; Chloroquine; Epididymis; Fatty Acids; Heparin; Hydroxychloroquine; Lipid Metabolism; Male; Primaquine; Quinacrine; Quinidine; Quinine; Rats

1969
An automated method of mass drug testing applied to screening for antimalarial activity.
    Chemotherapy, 1970, Volume: 15, Issue:3

    Topics: Animals; Antimalarials; Automation; Chloroquine; Erythrocytes; Glucose; Glycolysis; Lactates; Male; Methods; Neoplasms, Experimental; Pharmacology; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rats; Sulfadiazine; Sulfones

1970
A unique antinucleic acid approach to the mass screening of antimalarial drugs.
    Chemotherapy, 1970, Volume: 15, Issue:3

    Topics: Animals; Antimalarials; Cell Membrane; Chemical Phenomena; Chemistry; Chloroquine; Computers; DNA, Bacterial; Erythrocytes; Hydrogen-Ion Concentration; Nucleosides; Pharmacology; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rats; RNA, Bacterial; Sulfones; Temperature; Tritium

1970
Influence of sucrose on chloroquine-3-H3 content of mammalian cells in vitro: the possible role of lysosomes in chloroquine resistance.
    The Journal of pharmacology and experimental therapeutics, 1970, Volume: 173, Issue:1

    Topics: Animals; Carbon Isotopes; Cell Line; Chloroquine; Cold Temperature; Cricetinae; Culture Techniques; Drug Resistance, Microbial; HeLa Cells; Hexoses; Hydrogen-Ion Concentration; Kidney; Lysosomes; Pinocytosis; Plasmodium; Primaquine; Quinacrine; Quinine; Sucrose; Tritium

1970
The intracellular and membrane effects of oxidant agents on normal red cells.
    British journal of haematology, 1970, Volume: 19, Issue:3

    Topics: Cell Membrane; Erythrocytes; Glutathione; Heinz Bodies; Hemoglobinometry; Hemolysis; Humans; Hydroquinones; Hydroxylamines; Naphthoquinones; Osmotic Fragility; Oxidation-Reduction; Phenols; Phenylhydrazines; Potassium; Primaquine; Quinacrine; Quinine

1970
Antimalarials: effects on in vivo and in vitro protein synthesis.
    Science (New York, N.Y.), 1970, Dec-11, Volume: 170, Issue:3963

    Topics: Amino Acids; Antimalarials; Carbon Isotopes; Cell-Free System; Chloroquine; Cycloheximide; Primaquine; Protein Biosynthesis; Quinacrine; Quinine; Tetrahymena

1970
The chemotherapy of rodent malaria. IX. Causal prophylaxis. I. A method for demonstrating drug action on exo-erythrocytic stages.
    Annals of tropical medicine and parasitology, 1970, Volume: 64, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Dapsone; Malaria; Male; Mice; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Triazines

1970
Resistance to primaquine in Plasmodium gallinaceum, and the problem of resistance to quinoline compounds in malaria parasites.
    Parasitology, 1967, Volume: 57, Issue:4

    Topics: Aedes; Animals; Chickens; Chloroquine; Drug Resistance, Microbial; Malaria, Avian; Primaquine; Quinacrine; Quinine; Quinolines

1967
The lethal effect of certain antimalarial drugs on Tetrahymena pyriformis.
    The American journal of tropical medicine and hygiene, 1968, Volume: 17, Issue:3

    Topics: Animals; Antimalarials; Antiprotozoal Agents; Chloroquine; Chlortetracycline; Metronidazole; Nitrofurantoin; Penicillins; Primaquine; Proguanil; Quinacrine; Quinine; Streptomycin; Sulfadiazine; Sulfisoxazole; Tetrahymena

1968
Characteristics and cross-resistance patterns of chloroquine-resistant Plasmodium berghei infections in mice.
    Experimental parasitology, 1968, Volume: 23, Issue:1

    Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Dapsone; Drug Resistance, Microbial; Female; Hematocrit; Isoenzymes; L-Lactate Dehydrogenase; Malaria; Mice; Organ Size; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rodent Diseases; Serum Albumin; Serum Globulins; Spleen; Splenomegaly; Sulfadiazine

1968
The Plasmodium chabaudi-mouse system in chemotherapy studies.
    Experimental parasitology, 1969, Volume: 24, Issue:2

    Topics: Animals; Antimalarials; Chloroquine; Injections, Intravenous; Malaria; Male; Mice; Plasmodium; Primaquine; Quinacrine

1969
Repository drugs. 8. Ester and amide congeners of amodiaquine, hydroxychloroquine, oxychloroquine, primaquine, quinacrine, and related substances as potential long-acting antimalarial agents.
    Journal of medicinal chemistry, 1969, Volume: 12, Issue:4

    Topics: Amodiaquine; Animals; Antimalarials; Chemical Phenomena; Chemistry; Delayed-Action Preparations; Esters; Hydroxychloroquine; Malaria; Mice; Primaquine; Quinacrine

1969
Drug resistance in Plasmodium berghei Vincke and Lips, 1948. I. Chloroquine resistance.
    Experimental parasitology, 1965, Volume: 17, Issue:1

    Topics: Amodiaquine; Animals; Chloroquine; Dapsone; Malaria; Mice; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Sulfadiazine; Triazines

1965
Hückel molecular orbital calculations for some antimalarial drugs and related molecules.
    Journal of medicinal chemistry, 1967, Volume: 10, Issue:5

    Topics: Antimalarials; Chemical Phenomena; Chemistry, Physical; Chloroquine; DNA; Primaquine; Pyrimethamine; Quinacrine; Quinine; RNA

1967
The effect of anti-malarial drugs on human natural killer cells in vitro.
    Parasite immunology, 1984, Volume: 6, Issue:6

    Topics: Antimalarials; Cell Line; Chloroquine; Cytotoxicity, Immunologic; Humans; Killer Cells, Natural; Leukemia, Myeloid, Acute; Mefloquine; Primaquine; Pyrimethamine; Quinacrine; Quinine; Quinolines

1984
Comparative effects of intrauterine instillation of analogues of quinacrine and tetracycline on uterine morphology in the rat.
    Contraception, 1984, Volume: 29, Issue:6

    Topics: Animals; Chloroquine; Demeclocycline; Doxycycline; Female; Primaquine; Quinacrine; Rats; Rats, Inbred Strains; Sodium Chloride; Tetracycline; Tetracyclines; Trimethoprim; Uterus

1984
Inhibition of rat hepatic mixed function oxidases by antimalarial drugs: selectivity for cytochromes P-450 and P-448.
    Chemico-biological interactions, 1984, Volume: 51, Issue:3

    Topics: Animals; Antimalarials; Chloroquine; Cytochrome P-450 CYP1A1; Cytochrome P-450 CYP1A2; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Cytochromes; Male; Microsomes, Liver; Mixed Function Oxygenases; Oxidoreductases; Oxidoreductases, N-Demethylating; Primaquine; Quinacrine; Rats; Rats, Inbred Strains

1984
Effects of antimalarial drugs on several rat-liver lysosomal enzymes involved in phosphatidylethanolamine catabolism.
    Biochimica et biophysica acta, 1982, Oct-14, Volume: 713, Issue:1

    Topics: Animals; Antimalarials; Carboxylic Ester Hydrolases; Chloroquine; Dose-Response Relationship, Drug; Liver; Lysophospholipase; Lysosomes; Male; Monoacylglycerol Lipases; Phosphatidylethanolamines; Phospholipases; Phospholipases A; Phospholipases A1; Primaquine; Quinacrine; Rats; Rats, Inbred Strains

1982
[The effect of pyracrini phosphas on plasma primaquine level following combined administration to rats (author's transl)].
    Yao xue xue bao = Acta pharmaceutica Sinica, 1980, Volume: 15, Issue:10

    Topics: Aminoacridines; Animals; Antimalarials; Drug Interactions; Drug Therapy, Combination; Primaquine; Quinacrine; Rats

1980
Inhibition of hepatitis B virus specific DNA polymerase by intercalating agents.
    Medical microbiology and immunology, 1980, Volume: 168, Issue:1

    Topics: Carrier State; Chloroquine; DNA-Directed DNA Polymerase; Ethidium; Hepatitis B; Hepatitis B Antigens; Hepatitis B virus; Humans; Intercalating Agents; Magnesium; Methylene Blue; Nucleic Acid Synthesis Inhibitors; Primaquine; Quinacrine; Quinine

1980
Xanthones as antimalarial agents; studies of a possible mode of action.
    FEBS letters, 1997, Jun-02, Volume: 409, Issue:1

    Topics: Animals; Antimalarials; Chloroquine; Heme; Humans; Plasmodium falciparum; Polymers; Primaquine; Quinacrine; Structure-Activity Relationship; Xanthenes; Xanthones

1997
In vivo and in vitro effects of antimalarials on Histoplasma capsulatum.
    Antibiotics & chemotherapy (Northfield, Ill.), 1962, Volume: 12

    Topics: Amodiaquine; Antimalarials; Chloroquine; Histoplasma; Humans; In Vitro Techniques; Primaquine; Quinacrine

1962
ANTIMALARIAL DRUGS ON THE AUTOMATICITY OF SINO-AURICULAR AND ATRIO-VENTRICULAR NODES.
    The Indian journal of medical research, 1963, Volume: 51

    Topics: Administration, Intravenous; Amodiaquine; Animals; Anti-Arrhythmia Agents; Antimalarials; Atrioventricular Node; Atropine; Chloroquine; Dogs; Heart Conduction System; Humans; Hydroxychloroquine; Hypotension; Injections, Intravenous; Primaquine; Quinacrine; Quinidine; Research; Statistics as Topic

1963
CHEMOTHERAPY OF CUTANEOUS LEISHMANIASIS: LEISHMANIA TROPICA INFECTIONS IN MICE.
    Annals of tropical medicine and parasitology, 1964, Volume: 58

    Topics: Amidines; Animals; Antimony; Antiprotozoal Agents; Chloroquine; Chlortetracycline; Dapsone; Deoxyribonuclease I; Emetine; Hyaluronoglucosaminidase; Hydrastis; Leishmania tropica; Leishmaniasis; Leishmaniasis, Cutaneous; Leishmaniasis, Mucocutaneous; Mice; Pathology; Pharmacology; Primaquine; Pyrimethamine; Quinacrine; Research; Streptodornase and Streptokinase; Streptokinase; Sulfonamides; Surface-Active Agents; Toxicology

1964
Kinetic mechanism of quinone oxidoreductase 2 and its inhibition by the antimalarial quinolines.
    Biochemistry, 2004, Apr-20, Volume: 43, Issue:15

    Topics: Antimalarials; Binding, Competitive; Chloroquine; Copper; Humans; Kinetics; Niacinamide; Oxidation-Reduction; Primaquine; Quinacrine; Quinolines; Quinone Reductases; Recombinant Proteins; Spectrophotometry; Substrate Specificity; Zinc

2004
Role of calcium messenger systems in ACTH-induced cortisol production in bovine adrenal fasciculo-reticularis cells.
    Endocrine journal, 2007, Volume: 54, Issue:4

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adrenocorticotropic Hormone; Animals; Bucladesine; Calcium; Calcium Signaling; Cattle; Cells, Cultured; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Hydrocortisone; Isoquinolines; Naphthalenes; Phospholipase A2 Inhibitors; Phospholipases A2; Primaquine; Protein Kinase C; Protein Kinase Inhibitors; Quinacrine; Second Messenger Systems; Sulfonamides; Zona Fasciculata

2007
Resistance to chloroquine unhinges vivax malaria therapeutics.
    Antimicrobial agents and chemotherapy, 2011, Volume: 55, Issue:5

    Topics: Aminoquinolines; Antimalarials; Chloroquine; Drug Interactions; Drug Resistance; Humans; Malaria, Vivax; Plasmodium vivax; Primaquine; Quinacrine

2011
Chloroquine derivatives block the translocation pores and inhibit cellular entry of Clostridium botulinum C2 toxin and Bacillus anthracis lethal toxin.
    Archives of toxicology, 2017, Volume: 91, Issue:3

    Topics: Antigens, Bacterial; Bacterial Toxins; Biological Transport; Botulinum Toxins; Cell Membrane; Chloroquine; Fluphenazine; HeLa Cells; Humans; Lipid Bilayers; Primaquine; Quinacrine

2017