quinacrine has been researched along with primaquine in 64 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 50 (78.13) | 18.7374 |
1990's | 1 (1.56) | 18.2507 |
2000's | 7 (10.94) | 29.6817 |
2010's | 6 (9.38) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Galanakis, D; Ganellin, CR | 1 |
Danis, M; Derouin, F; Farhati, K; Franetich, JF; Galvez, J; Garcia-Domenech, R; Hannoun, L; Mahmoudi, N; Mazier, D; Sauerwein, R | 1 |
Fitos, I; Mády, G; Visy, J; Zsila, F | 1 |
Lombardo, F; Obach, RS; Waters, NJ | 1 |
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M | 1 |
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A | 1 |
García-Mera, X; González-Díaz, H; Prado-Prado, FJ | 1 |
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
Bane, CE; Black, C; Butler, K; Caridha, D; Cooper, RA; Dodean, RA; Gaona, H; Gaynor-Ohnstad, L; Huezo, SJ; Kancharla, P; Kelly, JX; Kreishman-Deitrick, M; Leed, SE; Li, Q; Li, Y; Lin, H; Luong, TL; Marcsisin, S; Melendez, V; Nolan, C; Olmeda, R; Potter, B; Pou, S; Rasmussen, SA; Read, L; Riscoe, MK; Roncal, N; Sciotti, RJ; Smilkstein, MJ; Sousa, J; Stephens, MT; Tan, JC; Vesely, B; Vuong, C; Winter, RW; Xie, L; Zeng, Q; Zhang, J; Zhang, P | 1 |
Garfinkel, E; Hirschman, SZ | 1 |
Mattock, NM; Peters, W | 1 |
Holbrook, DJ; Washington, ME; Wichard, LP | 1 |
Emerole, GO; Nashiru, TO; Thabrew, MI | 1 |
Butler, KW; Deslauriers, R; Smith, IC | 1 |
Shao, BR; Xu, YQ | 1 |
Bohn, E; Hesse, B; Kunze, H; Löffler, BM | 1 |
Chou, SC; Conklin, KA; Pan, HY | 1 |
Chou, SC; Levy, MR | 1 |
Peters, W | 2 |
Cowey, FK; Whitehouse, MW | 1 |
Fain, JN; Pointer, RH | 1 |
Bacchi, CJ; Goldberg, B; Hutner, SH; Lambros, C | 1 |
Miller, A; Natsios, G; Smith, HC | 1 |
Olatunde, IA | 1 |
Botha, D | 1 |
Chou, SC; Conklin, KA | 2 |
Moxey, PC; Robles, E; Schimmel, EM; Trier, JS | 1 |
Dawkins, AT; Stahler, N; Terzian, LA | 1 |
Schmidt, LH | 1 |
Fink, E; Kretschmar, W | 1 |
Chou, SC; Conklin, KA; Heu, P | 1 |
Aviado, DM; Bass, SW; Ramirez, MA | 1 |
Bruce-Chwatt, LJ | 1 |
Miller, A; Smith, HC | 2 |
Ball, EG; Markus, HB | 1 |
Cenedella, RJ; Saxe, LH; Van Dyke, K | 1 |
Cenedella, R; Saxe, LH; Szustkiewicz, C; Van Dyke, K | 1 |
Polet, H | 1 |
Gregory, KG; Peters, W | 1 |
Bishop, A | 1 |
Clancy, CF | 1 |
Schneider, MD | 1 |
Ott, KJ | 1 |
Elslager, EF; Tendick, FH; Werbel, LM | 1 |
Purcell, WP; Singer, JA | 1 |
Doberstyn, EB | 1 |
Ferrante, A; Goh, DH | 1 |
Dubin, NH; Ghodgaonkar, RB; King, TM; Parmley, TH | 1 |
Ioannides, C; Thabrew, MI | 1 |
Bohn, E; Hesse, B; Kunze, H | 1 |
Gu, HM; Qu, ZX; Zeng, YL | 1 |
Arnold, W; Gahl, GM; Hess, G; Meyer zum Büschenfelde, KH; Möller, B | 1 |
Bächinger, HP; Hinrichs, DJ; Ignatushchenko, MV; Riscoe, MK; Winter, RW | 1 |
SASLAW, S; SCHAEFER, J | 1 |
ARORA, RB; LAL, A | 1 |
SULLI, G; VARRONE, F | 1 |
NEAL, RA | 1 |
Haystead, TA; Kwiek, JJ; Rudolph, J | 1 |
Nishikawa, T; Omura, M; Suematsu, S | 1 |
Baird, JK | 1 |
Barth, H; Benz, R; Kreidler, AM | 1 |
5 review(s) available for quinacrine and primaquine
Article | Year |
---|---|
Recent advances in antimalarial chemotherapy and drug resistance.
Topics: Agglutination; Amodiaquine; Animals; Anti-Bacterial Agents; Antimalarials; Chloroquine; Cross Reactions; Drug Combinations; Drug Evaluation, Preclinical; Drug Resistance; Folic Acid Antagonists; Haplorhini; Humans; Lincomycin; Malaria; Pigments, Biological; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Plasmodium vivax; Primaquine; Pyrimethamine; Quinacrine; Quinine; Quinolines; Structure-Activity Relationship; Sulfonamides; Sulfones | 1974 |
The present status of chloroquine in the drug treatment of malaria.
Topics: Chloroquine; Drug Resistance, Microbial; Humans; Malaria; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfonamides; Sulfones; Triazines | 1972 |
Chemotherapy of the drug-resistant malarias.
Topics: Chloroquine; Cinchona; Drug Resistance, Microbial; Malaria; Mutation; Phytotherapy; Plants, Medicinal; Plasmodium falciparum; Plasmodium malariae; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Quinolines; Sulfonamides; Sulfones | 1969 |
Resistance of Plasmodium falciparum.
Topics: Africa; Animals; Antimalarials; Asia; Chloroquine; DNA; Drug Resistance; Drug Synergism; Hemin; Malaria; Plasmodium falciparum; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Quinolines; Research; RNA; South America | 1984 |
[EXTRAMALARIAL THERAPUETIC APPLICATIONS OF ANTIMALARIAL DRUGS. 1. CLINICAL UTILIZATIONS].
Topics: Amodiaquine; Antimalarials; Chloroquine; Collagen Diseases; Dermatology; Drug Utilization; Epilepsy; Female; Heart Diseases; Hematology; Humans; Hydroxychloroquine; Hypersensitivity; Multiple Sclerosis; Muscular Diseases; Neurology; Parasitic Diseases; Pharmacology; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Toxicology; Uterus | 1963 |
59 other study(ies) available for quinacrine and primaquine
Article | Year |
---|---|
Defining determinant molecular properties for the blockade of the apamin-sensitive SKCa channel in guinea-pig hepatocytes: the influence of polarizability and molecular geometry.
Topics: Animals; Apamin; Guinea Pigs; Hepatocytes; Kinetics; Molecular Conformation; Potassium Channels, Calcium-Activated | 2004 |
New active drugs against liver stages of Plasmodium predicted by molecular topology.
Topics: Animals; Antimalarials; Hepatocytes; Humans; Liver; Mice; Models, Biological; Parasitic Sensitivity Tests; Plasmodium yoelii; Structure-Activity Relationship | 2008 |
Selective plasma protein binding of antimalarial drugs to alpha1-acid glycoprotein.
Topics: Antimalarials; Binding Sites; Chromatography, Affinity; Circular Dichroism; Humans; Molecular Structure; Orosomucoid; Protein Binding; Serum Albumin; Spectrophotometry; Stereoisomerism; Structure-Activity Relationship | 2008 |
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding | 2008 |
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship | 2008 |
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship | 2010 |
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics | 2010 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |
Discovery and Structural Optimization of Acridones as Broad-Spectrum Antimalarials.
Topics: Acridones; Animals; Antimalarials; Disease Models, Animal; Drug Discovery; Hep G2 Cells; Humans; Malaria; Mice; Plasmodium; Species Specificity; Structure-Activity Relationship | 2019 |
Inhibition of hepatitis B DNA polymerase by intercalating agents.
Topics: Chloroquine; Chlorpromazine; Drug Synergism; Ethidium; Hepatitis B; Hepatitis B virus; Humans; Indicators and Reagents; Methylene Blue; Nucleic Acid Synthesis Inhibitors; Primaquine; Quinacrine | 1978 |
The experimental chemotherapy of leishmaniasis. II. The activity in tissue culture of some antiparasitic and antimicrobial compounds in clinical use.
Topics: Aminoquinolines; Animals; Anti-Bacterial Agents; Antimalarials; Antimony; Antiprotozoal Agents; Ascitic Fluid; Cell Line; Chloroquine; Cricetinae; Culture Techniques; Dogs; Drug Evaluation, Preclinical; Folic Acid Antagonists; Leishmania; Niridazole; Pentamidine; Primaquine; Quinacrine; Quinine; Sarcoma; Sulfonamides; Sulfones; Suramin | 1975 |
Effect of nucleic-acid-binding compounds on the hydrolytic activity of various ribonucleases.
Topics: Acridines; Aminoquinolines; Animals; Binding Sites; Cattle; Chloroquine; Ethidium; Kinetics; Pancreas; Primaquine; Proflavine; Protein Binding; Quinacrine; Ribonucleases; Spermidine; Spermine; Structure-Activity Relationship | 1975 |
Drug induced alterations in some rat hepatic microsomal components: a comparative study of four structurally different antimalarials.
Topics: Aminopyrine N-Demethylase; Aniline Hydroxylase; Animals; Antimalarials; Aryl Hydrocarbon Hydroxylases; Chloroquine; Cholesterol; Cytosol; Glutathione Transferase; Liver; Male; Microsomes, Liver; Phospholipids; Primaquine; Quinacrine; Quinine; Rats; Rats, Inbred Strains | 1985 |
Effects of antimalarial drugs on oxygen consumption by erythrocytes infected with Plasmodium berghei: an ESR study.
Topics: Animals; Antimalarials; Depression, Chemical; Electron Spin Resonance Spectroscopy; Erythrocytes; Malaria; Male; Mice; Oxygen Consumption; Plasmodium berghei; Primaquine; Quinacrine; Quinine | 1986 |
[The mouse micronucleus test for mutagenicity of pyronaridine, chloroquine, quinacrine, primaquine, furapyrimidone and phenthiourezine].
Topics: Animals; Anthelmintics; Antimalarials; Chloroquine; Filaricides; Male; Mice; Micronucleus Tests; Mutagenicity Tests; Naphthyridines; Nitrofurans; Piperazines; Primaquine; Quinacrine | 1988 |
Effects of antimalarial drugs on phospholipase A and lysophospholipase activities in plasma membrane, mitochondrial, microsomal and cytosolic subcellular fractions of rat liver.
Topics: Animals; Antimalarials; Cell Membrane; Chloroquine; Cytosol; Endoplasmic Reticulum; Liver; Lysophospholipase; Male; Microsomes, Liver; Mitochondria, Liver; Phospholipases; Phospholipases A; Phospholipases A1; Phospholipases A2; Primaquine; Quinacrine; Rats; Rats, Inbred Strains | 1985 |
Effects of antimalarial drugs and clofibrate on in vitro lipid synthesis in Tetrahymena pyriformis GL.
Topics: Acetates; Adenosine Triphosphate; Carbon Radioisotopes; Cell Division; Cell-Free System; Chloroquine; Chromatography, Thin Layer; Clofibrate; Depression, Chemical; Fatty Acids, Nonesterified; Lipids; NADH, NADPH Oxidoreductases; Phospholipids; Primaquine; Quinacrine; Quinine; Stimulation, Chemical; Tetrahymena pyriformis; Triglycerides | 1974 |
Activity and some properties of an acid proteinase from normal and Plasmodium berghei-infected red cells.
Topics: Acid Phosphatase; Animals; Cell-Free System; Chloroquine; Dithiothreitol; Edetic Acid; Erythrocytes; Female; Hemoglobins; Hemolysis; Hydrogen-Ion Concentration; Malaria; Mice; Mice, Inbred BALB C; Peptide Hydrolases; Plasmodium berghei; Primaquine; Quinacrine; Rats; Solubility; Surface-Active Agents; Ultracentrifugation | 1973 |
Biochemical properties of anti-inflammatory drugs. VII. Inhibition of proteolytic enzymes in connective tissue by chloroquine (resochin) and related antimalarial antirheumatic drugs.
Topics: Acridines; Animals; Cartilage; Cattle; Chloroquine; Chondroitin; Connective Tissue; Hyaluronoglucosaminidase; Hydrogen-Ion Concentration; Hydroxychloroquine; Microbial Collagenase; Mucoproteins; Papain; Primaquine; Quaternary Ammonium Compounds; Quinacrine; Rabbits | 1966 |
Response of isolated white fat cells to anti-malarial drugs.
Topics: Adenylyl Cyclase Inhibitors; Adipose Tissue; Animals; Antimalarials; Bucladesine; Chloroquine; Drug Synergism; Fatty Acids, Nonesterified; Female; Glycerol; Norepinephrine; Primaquine; Proteins; Quinacrine; Quinidine; Rats; Theophylline; Triglycerides | 1973 |
Inhibition by several standard antiprotozoal drugs of growth and O2 uptake of cells and particulate preparations of a Leptomonas.
Topics: Acridines; Alkanesulfonates; Amidines; Arsenicals; Culture Media; Ethidium; Eukaryota; Glycerophosphates; Hydrogen-Ion Concentration; Oxygen Consumption; Phenyl Ethers; Primaquine; Proline; Pyrimidines; Quinacrine; Quinolinium Compounds; Rotenone; Stilbamidines; Succinates; Suramin; Triazines; Trypanocidal Agents | 1974 |
Effect of antimalarial drugs on the efflux of K+ from Streptococcus pyogenes.
Topics: Antimalarials; Biological Transport; Cell Membrane Permeability; Chloroquine; Culture Media; Potassium; Potassium Isotopes; Primaquine; Quinacrine; Quinine; Streptococcus pneumoniae; Streptococcus pyogenes | 1971 |
Some pharmacological aspects of antimalarial drugs.
Topics: Antimalarials; Chloroquine; Dapsone; Drug Resistance, Microbial; Humans; Malaria; Plasmodium falciparum; Plasmodium vivax; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfonamides; Trimethoprim | 1974 |
The effects of antimalarial drugs on uptake and incorporation of macromolecular precursors by Tetrahymena pyriformis.
Topics: Amino Acids; Animals; Antimalarials; Carbon Isotopes; Cell Division; Chloroquine; Cycloheximide; Dactinomycin; DNA; Kinetics; Macromolecular Substances; Nalidixic Acid; Primaquine; Quinacrine; Quinine; RNA; Tetrahymena pyriformis; Thymidine; Uridine | 1972 |
Chronic intestinal coccidiosis in man: intestinal morphology and response to treatment.
Topics: Antiprotozoal Agents; Biopsy; Chloroquine; Chronic Disease; Coccidiosis; Diagnosis, Differential; Diarrhea; Diet Therapy; Drug Therapy, Combination; Duodenum; Follow-Up Studies; Humans; Intestinal Diseases, Parasitic; Intestine, Small; Isospora; Jejunum; Malabsorption Syndromes; Male; Metronidazole; Microscopy, Electron; Middle Aged; Nitrofurantoin; Primaquine; Pyrimethamine; Quinacrine; Sulfadiazine; Tetracycline; Time Factors | 1974 |
The sporogonous of Plasmodium vivax in Anopheles mosquitoes as a system for evaluating the prophylactic and curative capabilities of potential antimalarial compounds.
Topics: Animals; Anopheles; Antimalarials; Chloroquine; Malaria; Naphthoquinones; Oxytetracycline; Penicillin G; Plasmodium vivax; Primaquine; Proguanil; Pyridines; Pyrimethamine; Quinacrine; Quinine; Quinolines; Sulfadiazine; Thiosemicarbazones | 1968 |
[Chemotherapeutic activity of standard antimalarials in a simplified test for Plasmodium vinckey infection in the NMPI mouse].
Topics: Animals; Antimalarials; Chloroquine; Long-Term Care; Malaria; Mice; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Sulfonamides; Time Factors | 1970 |
Quinine: effect of Tetrahymena pyriformis. 3. Energetics of isolated mitochondria in the presence of quinine and other antimalarial drugs.
Topics: Chloroquine; Citrates; Citric Acid Cycle; Depression, Chemical; Fumarates; Glutamates; Hydroxybutyrates; Isocitrates; Ketoglutaric Acids; Malates; Mitochondria; Oxidative Phosphorylation; Oxygen Consumption; Primaquine; Quinacrine; Quinine; Stimulation, Chemical; Succinates; Tetrahymena pyriformis; Uncoupling Agents | 1971 |
Cardiopulmonary effects of antimalarial drugs. VI. Adenosine, quinacrine and primaquine.
Topics: Adenosine; Animals; Anti-Arrhythmia Agents; Blood Pressure; Cardiac Output; Cats; Coronary Circulation; Dogs; Drug Interactions; Electrocardiography; Female; Heart; Heart Rate; Hemodynamics; Isoproterenol; Male; Mice; Muscle Contraction; Primaquine; Pulmonary Circulation; Quinacrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Vascular Resistance; Ventricular Fibrillation | 1972 |
The role of drugs in a malaria program.
Topics: Amodiaquine; Antimalarials; Chloroquine; Dose-Response Relationship, Drug; Humans; Malaria; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Recurrence; Sulfonamides; Sulfones; Trimethoprim | 1972 |
The influence of glucose and exogenous glutathione on the red cell membrane effect of the antimalarial drugs 1,4-naphthoquinone and beta-naphthol.
Topics: Cell Membrane; Erythrocytes; Glucose; Glutathione; Hemolysis; Humans; In Vitro Techniques; Methemoglobin; Naphthalenes; Naphthoquinones; Osmotic Fragility; Potassium; Primaquine; Quinacrine; Quinine | 1971 |
Inhibition of lipolytic processes in rat adipose tissue by antimalaria drugs.
Topics: Adipose Tissue; Animals; Antimalarials; Chloroquine; Epididymis; Fatty Acids; Heparin; Hydroxychloroquine; Lipid Metabolism; Male; Primaquine; Quinacrine; Quinidine; Quinine; Rats | 1969 |
An automated method of mass drug testing applied to screening for antimalarial activity.
Topics: Animals; Antimalarials; Automation; Chloroquine; Erythrocytes; Glucose; Glycolysis; Lactates; Male; Methods; Neoplasms, Experimental; Pharmacology; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rats; Sulfadiazine; Sulfones | 1970 |
A unique antinucleic acid approach to the mass screening of antimalarial drugs.
Topics: Animals; Antimalarials; Cell Membrane; Chemical Phenomena; Chemistry; Chloroquine; Computers; DNA, Bacterial; Erythrocytes; Hydrogen-Ion Concentration; Nucleosides; Pharmacology; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rats; RNA, Bacterial; Sulfones; Temperature; Tritium | 1970 |
Influence of sucrose on chloroquine-3-H3 content of mammalian cells in vitro: the possible role of lysosomes in chloroquine resistance.
Topics: Animals; Carbon Isotopes; Cell Line; Chloroquine; Cold Temperature; Cricetinae; Culture Techniques; Drug Resistance, Microbial; HeLa Cells; Hexoses; Hydrogen-Ion Concentration; Kidney; Lysosomes; Pinocytosis; Plasmodium; Primaquine; Quinacrine; Quinine; Sucrose; Tritium | 1970 |
The intracellular and membrane effects of oxidant agents on normal red cells.
Topics: Cell Membrane; Erythrocytes; Glutathione; Heinz Bodies; Hemoglobinometry; Hemolysis; Humans; Hydroquinones; Hydroxylamines; Naphthoquinones; Osmotic Fragility; Oxidation-Reduction; Phenols; Phenylhydrazines; Potassium; Primaquine; Quinacrine; Quinine | 1970 |
Antimalarials: effects on in vivo and in vitro protein synthesis.
Topics: Amino Acids; Antimalarials; Carbon Isotopes; Cell-Free System; Chloroquine; Cycloheximide; Primaquine; Protein Biosynthesis; Quinacrine; Quinine; Tetrahymena | 1970 |
The chemotherapy of rodent malaria. IX. Causal prophylaxis. I. A method for demonstrating drug action on exo-erythrocytic stages.
Topics: Animals; Antimalarials; Chloroquine; Dapsone; Malaria; Male; Mice; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Quinine; Sulfadiazine; Triazines | 1970 |
Resistance to primaquine in Plasmodium gallinaceum, and the problem of resistance to quinoline compounds in malaria parasites.
Topics: Aedes; Animals; Chickens; Chloroquine; Drug Resistance, Microbial; Malaria, Avian; Primaquine; Quinacrine; Quinine; Quinolines | 1967 |
The lethal effect of certain antimalarial drugs on Tetrahymena pyriformis.
Topics: Animals; Antimalarials; Antiprotozoal Agents; Chloroquine; Chlortetracycline; Metronidazole; Nitrofurantoin; Penicillins; Primaquine; Proguanil; Quinacrine; Quinine; Streptomycin; Sulfadiazine; Sulfisoxazole; Tetrahymena | 1968 |
Characteristics and cross-resistance patterns of chloroquine-resistant Plasmodium berghei infections in mice.
Topics: Amodiaquine; Animals; Antimalarials; Chloroquine; Dapsone; Drug Resistance, Microbial; Female; Hematocrit; Isoenzymes; L-Lactate Dehydrogenase; Malaria; Mice; Organ Size; Plasmodium; Primaquine; Pyrimethamine; Quinacrine; Quinine; Rodent Diseases; Serum Albumin; Serum Globulins; Spleen; Splenomegaly; Sulfadiazine | 1968 |
The Plasmodium chabaudi-mouse system in chemotherapy studies.
Topics: Animals; Antimalarials; Chloroquine; Injections, Intravenous; Malaria; Male; Mice; Plasmodium; Primaquine; Quinacrine | 1969 |
Repository drugs. 8. Ester and amide congeners of amodiaquine, hydroxychloroquine, oxychloroquine, primaquine, quinacrine, and related substances as potential long-acting antimalarial agents.
Topics: Amodiaquine; Animals; Antimalarials; Chemical Phenomena; Chemistry; Delayed-Action Preparations; Esters; Hydroxychloroquine; Malaria; Mice; Primaquine; Quinacrine | 1969 |
Drug resistance in Plasmodium berghei Vincke and Lips, 1948. I. Chloroquine resistance.
Topics: Amodiaquine; Animals; Chloroquine; Dapsone; Malaria; Mice; Plasmodium; Primaquine; Proguanil; Pyrimethamine; Quinacrine; Sulfadiazine; Triazines | 1965 |
Hückel molecular orbital calculations for some antimalarial drugs and related molecules.
Topics: Antimalarials; Chemical Phenomena; Chemistry, Physical; Chloroquine; DNA; Primaquine; Pyrimethamine; Quinacrine; Quinine; RNA | 1967 |
The effect of anti-malarial drugs on human natural killer cells in vitro.
Topics: Antimalarials; Cell Line; Chloroquine; Cytotoxicity, Immunologic; Humans; Killer Cells, Natural; Leukemia, Myeloid, Acute; Mefloquine; Primaquine; Pyrimethamine; Quinacrine; Quinine; Quinolines | 1984 |
Comparative effects of intrauterine instillation of analogues of quinacrine and tetracycline on uterine morphology in the rat.
Topics: Animals; Chloroquine; Demeclocycline; Doxycycline; Female; Primaquine; Quinacrine; Rats; Rats, Inbred Strains; Sodium Chloride; Tetracycline; Tetracyclines; Trimethoprim; Uterus | 1984 |
Inhibition of rat hepatic mixed function oxidases by antimalarial drugs: selectivity for cytochromes P-450 and P-448.
Topics: Animals; Antimalarials; Chloroquine; Cytochrome P-450 CYP1A1; Cytochrome P-450 CYP1A2; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Cytochromes; Male; Microsomes, Liver; Mixed Function Oxygenases; Oxidoreductases; Oxidoreductases, N-Demethylating; Primaquine; Quinacrine; Rats; Rats, Inbred Strains | 1984 |
Effects of antimalarial drugs on several rat-liver lysosomal enzymes involved in phosphatidylethanolamine catabolism.
Topics: Animals; Antimalarials; Carboxylic Ester Hydrolases; Chloroquine; Dose-Response Relationship, Drug; Liver; Lysophospholipase; Lysosomes; Male; Monoacylglycerol Lipases; Phosphatidylethanolamines; Phospholipases; Phospholipases A; Phospholipases A1; Primaquine; Quinacrine; Rats; Rats, Inbred Strains | 1982 |
[The effect of pyracrini phosphas on plasma primaquine level following combined administration to rats (author's transl)].
Topics: Aminoacridines; Animals; Antimalarials; Drug Interactions; Drug Therapy, Combination; Primaquine; Quinacrine; Rats | 1980 |
Inhibition of hepatitis B virus specific DNA polymerase by intercalating agents.
Topics: Carrier State; Chloroquine; DNA-Directed DNA Polymerase; Ethidium; Hepatitis B; Hepatitis B Antigens; Hepatitis B virus; Humans; Intercalating Agents; Magnesium; Methylene Blue; Nucleic Acid Synthesis Inhibitors; Primaquine; Quinacrine; Quinine | 1980 |
Xanthones as antimalarial agents; studies of a possible mode of action.
Topics: Animals; Antimalarials; Chloroquine; Heme; Humans; Plasmodium falciparum; Polymers; Primaquine; Quinacrine; Structure-Activity Relationship; Xanthenes; Xanthones | 1997 |
In vivo and in vitro effects of antimalarials on Histoplasma capsulatum.
Topics: Amodiaquine; Antimalarials; Chloroquine; Histoplasma; Humans; In Vitro Techniques; Primaquine; Quinacrine | 1962 |
ANTIMALARIAL DRUGS ON THE AUTOMATICITY OF SINO-AURICULAR AND ATRIO-VENTRICULAR NODES.
Topics: Administration, Intravenous; Amodiaquine; Animals; Anti-Arrhythmia Agents; Antimalarials; Atrioventricular Node; Atropine; Chloroquine; Dogs; Heart Conduction System; Humans; Hydroxychloroquine; Hypotension; Injections, Intravenous; Primaquine; Quinacrine; Quinidine; Research; Statistics as Topic | 1963 |
CHEMOTHERAPY OF CUTANEOUS LEISHMANIASIS: LEISHMANIA TROPICA INFECTIONS IN MICE.
Topics: Amidines; Animals; Antimony; Antiprotozoal Agents; Chloroquine; Chlortetracycline; Dapsone; Deoxyribonuclease I; Emetine; Hyaluronoglucosaminidase; Hydrastis; Leishmania tropica; Leishmaniasis; Leishmaniasis, Cutaneous; Leishmaniasis, Mucocutaneous; Mice; Pathology; Pharmacology; Primaquine; Pyrimethamine; Quinacrine; Research; Streptodornase and Streptokinase; Streptokinase; Sulfonamides; Surface-Active Agents; Toxicology | 1964 |
Kinetic mechanism of quinone oxidoreductase 2 and its inhibition by the antimalarial quinolines.
Topics: Antimalarials; Binding, Competitive; Chloroquine; Copper; Humans; Kinetics; Niacinamide; Oxidation-Reduction; Primaquine; Quinacrine; Quinolines; Quinone Reductases; Recombinant Proteins; Spectrophotometry; Substrate Specificity; Zinc | 2004 |
Role of calcium messenger systems in ACTH-induced cortisol production in bovine adrenal fasciculo-reticularis cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adrenocorticotropic Hormone; Animals; Bucladesine; Calcium; Calcium Signaling; Cattle; Cells, Cultured; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Hydrocortisone; Isoquinolines; Naphthalenes; Phospholipase A2 Inhibitors; Phospholipases A2; Primaquine; Protein Kinase C; Protein Kinase Inhibitors; Quinacrine; Second Messenger Systems; Sulfonamides; Zona Fasciculata | 2007 |
Resistance to chloroquine unhinges vivax malaria therapeutics.
Topics: Aminoquinolines; Antimalarials; Chloroquine; Drug Interactions; Drug Resistance; Humans; Malaria, Vivax; Plasmodium vivax; Primaquine; Quinacrine | 2011 |
Chloroquine derivatives block the translocation pores and inhibit cellular entry of Clostridium botulinum C2 toxin and Bacillus anthracis lethal toxin.
Topics: Antigens, Bacterial; Bacterial Toxins; Biological Transport; Botulinum Toxins; Cell Membrane; Chloroquine; Fluphenazine; HeLa Cells; Humans; Lipid Bilayers; Primaquine; Quinacrine | 2017 |