quinacrine and lidocaine

quinacrine has been researched along with lidocaine in 23 studies

Research

Studies (23)

TimeframeStudies, this research(%)All Research%
pre-199010 (43.48)18.7374
1990's1 (4.35)18.2507
2000's8 (34.78)29.6817
2010's4 (17.39)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Chiang, GH; Unger, SH1
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY2
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J1
Lombardo, F; Obach, RS; Waters, NJ1
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Choi, SS; Contrera, JF; Hastings, KL; Kruhlak, NL; Sancilio, LF; Weaver, JL; Willard, JM1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Glen, RC; Lowe, R; Mitchell, JB1
Benveniste, J; Cazenave, JP; Mustard, JF1
Medel, M; Stacchetti, E; Zipper, J1
Björkman, S; Elisson, LO; Gabrielsson, J1
Gartner, SL; Shakir, KM; Simpkins, CO; Sobel, DO; Williams, TJ1
Garcia-Martin, E; Gutiérrez-Merino, C1
Joseph, AA; Kincl, FA1
Bartos, J1
Andersson, A; Olsson, S; Tjälve, H1
Imanishi, S; Miyamae, S1
Al Obaid, AR; Al Rasheed, NM; Al Sayed, MI; Al Zuhair, HH; Fatani, AJ1
Barrantes, GE; Ortells, MO1
Marceau, F; Parks, A1

Other Studies

23 other study(ies) available for quinacrine and lidocaine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Octanol-physiological buffer distribution coefficients of lipophilic amines by reversed-phase high-performance liquid chromatography and their correlation with biological activity.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:3

    Topics: Amines; Animals; Buffers; Chromatography, High Pressure Liquid; Histamine Release; Lipid Metabolism; Octanols; Protein Binding; Rats; Serum Albumin, Bovine; Sodium-Potassium-Exchanging ATPase; Solubility; Structure-Activity Relationship

1981
Prediction of volume of distribution values in humans for neutral and basic drugs using physicochemical measurements and plasma protein binding data.
    Journal of medicinal chemistry, 2002, Jun-20, Volume: 45, Issue:13

    Topics: Blood Proteins; Chemical Phenomena; Chemistry, Physical; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding

2002
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
    Journal of medicinal chemistry, 2008, Jan-24, Volume: 51, Issue:2

    Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase

2008
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship

2008
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Development of a phospholipidosis database and predictive quantitative structure-activity relationship (QSAR) models.
    Toxicology mechanisms and methods, 2008, Volume: 18, Issue:2-3

    Topics:

2008
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Predicting phospholipidosis using machine learning.
    Molecular pharmaceutics, 2010, Oct-04, Volume: 7, Issue:5

    Topics: Animals; Artificial Intelligence; Databases, Factual; Drug Discovery; Humans; Lipidoses; Models, Biological; Phospholipids; Support Vector Machine

2010
Aggregation of rabbit platelets by platelet-activating factor is independent of the release reaction and the arachidonate pathway and inhibited by membrane-active drugs.
    Laboratory investigation; a journal of technical methods and pathology, 1979, Volume: 41, Issue:3

    Topics: Animals; Arachidonic Acids; Blood Platelets; Cell Membrane; Chlorpromazine; Edetic Acid; Egtazic Acid; Fibrinogen; Humans; Imipramine; Lidocaine; Methylprednisolone; Platelet Aggregation; Prostaglandins; Quinacrine; Rabbits; Reserpine; Serotonin

1979
Transvaginal chemical sterilization: clinical use of quinacrine plus potentiating adjuvants.
    Contraception, 1975, Volume: 12, Issue:1

    Topics: Cortisone; Drug Combinations; Epinephrine; Evaluation Studies as Topic; Female; Fertility; Humans; Injections; Lidocaine; Menstruation; Pregnancy; Quinacrine; Sterilization, Tubal; Tetracycline; Vagina

1975
Pharmacokinetics of quinacrine after intrapleural instillation in rabbits and man.
    The Journal of pharmacy and pharmacology, 1989, Volume: 41, Issue:3

    Topics: Animals; Female; Injections; Injections, Intravenous; Lidocaine; Male; Pleura; Quinacrine; Rabbits

1989
Phospholipase C activity in human polymorphonuclear leukocytes: partial characterization and effect of indomethacin.
    Enzyme, 1989, Volume: 42, Issue:4

    Topics: Calcium; Deoxycholic Acid; Fatty Acids, Nonesterified; Humans; Indomethacin; Kinetics; Lidocaine; Naloxone; Neutrophils; Quinacrine; Type C Phospholipases

1989
Local anesthetics inhibit the Ca2+, Mg2+-ATPase activity of rat brain synaptosomes.
    Journal of neurochemistry, 1986, Volume: 47, Issue:3

    Topics: Anesthetics, Local; Animals; Brain; Ca(2+) Mg(2+)-ATPase; Calcium-Transporting ATPases; Dibucaine; Kinetics; Lidocaine; Procaine; Quinacrine; Rats; Rats, Inbred Strains; Synaptosomes; Tetracaine

1986
Toxic and antifertility effects of quinacrine hydrochloride in rats.
    American journal of obstetrics and gynecology, 1974, Aug-01, Volume: 119, Issue:7

    Topics: Animals; Atrophy; Autopsy; Colonic Diseases; Dose-Response Relationship, Drug; Drug Synergism; Embryo Implantation; Epinephrine; Female; Fertility; Gastrointestinal Motility; Hydrogen-Ion Concentration; Infertility, Female; Intestinal Obstruction; Kidney; Lidocaine; Metaraminol; Necrosis; Ovary; Pregnancy; Quinacrine; Rats; Sodium Chloride; Uterus

1974
[Bacteriostatic effect of 8 non-antibiotic drugs on E. coli strains obtained from dead piglets and from those suffering from diarrhea].
    Veterinarni medicina, 1971, Volume: 16, Issue:2

    Topics: Animals; Anti-Bacterial Agents; Copper; Culture Media; Diarrhea; Escherichia coli; Furazolidone; Lidocaine; Nalidixic Acid; Procaine; Quinacrine; Serotyping; Sodium Salicylate; Swine; Swine Diseases

1971
The uptake of 14C-chloroquine by mouse pancreatic islets in vitro.
    Acta pharmacologica et toxicologica, 1980, Volume: 47, Issue:1

    Topics: Absorption; Animals; Chloroquine; Chlorpromazine; Desipramine; Glucose; Hydrogen-Ion Concentration; Imipramine; Islets of Langerhans; Lidocaine; Mice; Nicotine; Nitrogen; Ouabain; Quinacrine; Temperature

1980
Hyperpolarization induced by sodium removal in rabbit sinoatrial node cells. Possible role of electrogenic sodium-calcium exchange.
    Journal of electrocardiology, 1995, Volume: 28, Issue:2

    Topics: Animals; Calcium; In Vitro Techniques; Lidocaine; Membrane Potentials; Ouabain; Quinacrine; Quinidine; Rabbits; Sinoatrial Node; Sodium; Sodium-Potassium-Exchanging ATPase; Verapamil

1995
Effects of two newly synthesized analogues of lidocaine on rat arterial blood pressure and heart rate.
    Pharmacological research, 2001, Volume: 43, Issue:4

    Topics: Anesthetics, Local; Animals; Anti-Arrhythmia Agents; Antihypertensive Agents; Atropine; Benzoates; Blood Pressure; Calcium Chloride; Cyproheptadine; Enzyme Inhibitors; Heart Rate; Hexamethonium; Histamine Agonists; Indomethacin; Lidocaine; Male; Monitoring, Physiologic; NG-Nitroarginine Methyl Ester; Pyrilamine; Quinacrine; Ranitidine; Rats; Rats, Wistar; Vasodilator Agents

2001
Understanding channel blocking in the nicotinic acetylcholine receptor.
    Receptors & channels, 2001, Volume: 7, Issue:4

    Topics: Acetylcholine; Animals; Binding Sites; Chlorisondamine; Ethidium; Hexamethonium; Lidocaine; Mice; Nicotinic Antagonists; Onium Compounds; Pempidine; Proadifen; Quinacrine; Receptors, Nicotinic; Trityl Compounds

2001
Lysosomotropic cationic drugs induce cytostatic and cytotoxic effects: Role of liposolubility and autophagic flux and antagonism by cholesterol ablation.
    Toxicology and applied pharmacology, 2016, 08-15, Volume: 305

    Topics: Amiodarone; Anticholesteremic Agents; Autophagy; beta-Cyclodextrins; Cell Line, Tumor; Cell Proliferation; Cells, Cultured; Chloroquine; Cholesterol; Cytostatic Agents; Cytotoxins; Human Umbilical Vein Endothelial Cells; Humans; Hydroxychloroquine; Lidocaine; Lovastatin; Lysosomes; Microtubule-Associated Proteins; Poly (ADP-Ribose) Polymerase-1; Procainamide; Quinacrine

2016