quinacrine has been researched along with indomethacin in 185 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 91 (49.19) | 18.7374 |
1990's | 71 (38.38) | 18.2507 |
2000's | 19 (10.27) | 29.6817 |
2010's | 4 (2.16) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET | 1 |
Alcaraz, MJ; Ballesteros, JF; Iborra, S; Miranda, MA; Payá, M; Sanz, MJ; Ubeda, A | 1 |
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Lombardo, F; Obach, RS; Waters, NJ | 1 |
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A | 1 |
García-Mera, X; González-Díaz, H; Prado-Prado, FJ | 1 |
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
Folco, GC; Galli, C; Omini, C; Spagnuolo, C | 1 |
Landgraf, R; Landgraf-Leurs, MM | 1 |
Bentley, PJ; Yorio, T | 1 |
Chauvelot, L; Gagnon, D; Heisler, S; Huot, J | 1 |
Burnstock, G; Cocks, T; Crowe, R | 1 |
Blackwell, GJ; Duncombe, WG; Flower, RJ; Parsons, MF; Vane, JR | 1 |
Ally, AI; Horrobin, DF; Karmali, RA; Karmazyn, M; Manku, MS; Morgan, RO | 1 |
Dempster, JA; Kellett, GL | 1 |
Fujita, A; Hata, F; Takeuchi, T; Yagasaki, O | 1 |
Morii, M; Okada, Y; Sakai, H; Takeguchi, N | 1 |
Carganico, G; Ferrer, X; Moreno, JJ; Ortega, E | 1 |
Bonnet, P; Bourdeau, A; Herviaux, P; Lieberherr, M; Sachs, C; Souberbielle, JC | 1 |
Borrell, J; Cambronero, JC; Guaza, C; Rivas, FJ | 1 |
Ball, S; de Belleroche, J; Gardiner, IM; Li, A; Patel, N | 1 |
Capito, K; Gembal, M; Hedeskov, CJ; Malik, T; Thams, P | 1 |
McCann, JD; Smith, JJ; Welsh, MJ | 1 |
Okuda, M; Takeuchi, T; Yagasaki, O | 1 |
Gall, DG; MacNaughton, WK | 1 |
Dettori, C; Magistretti, J; Meldolesi, J | 1 |
al-Bayati, ZA; Stohs, SJ | 1 |
Bond, JA; Calder, PC; Newsholme, EA | 1 |
Fujii, T; Hashizume, T; Kawamoto, A; Sato, T; Tamura, A; Yamaguchi, H | 1 |
Busija, DW; Leffler, CW | 1 |
Diener, M; Rummel, W | 2 |
Aguila, MC; McCann, SM; Milenkovic, L; Snyder, GD | 1 |
Kimura, A; Nakagawa, H; Tu, AT | 1 |
Andres-Trelles, F; Baamonde, A; Cantabrana, B; Fernandez, A; Hidalgo, A | 1 |
Fitzgerald, TP; Granger, GA; Knauer, MF; Longmuir, KJ; Yamamoto, RS | 1 |
Ralph, RK; Wojcik, S | 1 |
Burgoyne, RD; Morgan, A | 1 |
Delbarre, B; Delbarre, G; Ferger, A | 1 |
Bergström, M; Carlsson, J; Csòka, K; Gàti, I; Muhr, C; Westerberg, G | 1 |
Levy, R; Tarsi-Tsuk, D | 1 |
Linssen, MJ; Lipponer, L; Seilnacht, W; Wilhelms, OH | 1 |
Hallbrucker, C; Lang, F; Rehwald, W | 1 |
Fuchimoto, S; Orita, K; Shiiki, S | 1 |
Andres-Trelles, F; Baamonde, A; Cantabrana, B; Hidalgo, A | 1 |
Furukawa, O; Niida, H; Okabe, S; Okada, M; Takeuchi, K | 1 |
Green, K; Recasens, JF | 1 |
de Graeff, PA; de Langen, CD; Scholtens, E; van Gilst, WH; van Wijngaarden, J; Wesseling, H | 1 |
Castro, GA; Russell, DA | 1 |
Bjerregaard, HF | 1 |
Yazaki, K | 2 |
Argenzio, RA; Henrikson, CK; Liacos, JA | 1 |
Evans, J; Shaw, KP; Vernon, LP; Wang, YD | 1 |
Klaas, M; Wadsworth, R | 1 |
Gartner, SL; Shakir, KM; Simpkins, CO; Sobel, DO; Williams, TJ | 1 |
Calixto, JB; Trebien, HA | 1 |
Calixto, JB; Medeiros, YS; Torres, RC | 1 |
Banitt, PF; Guerra, R; Harrison, DG; Myers, PR | 1 |
Fernandes, LB; Goldie, RG; Knight, DA; Paterson, JW; Rigby, PJ; Spina, D | 1 |
Canonico, PL; Cronin, MJ; MacLeod, RM; Scapagnini, U; Sortino, MA; Speciale, C | 1 |
Goldie, RG; Paterson, JW; Spina, D | 1 |
Azuma, H; Nakajima, T; Satoh, A; Sekizaki, S | 1 |
Hardcastle, J; Hardcastle, PT | 1 |
Harakawa, M; Ishitani, K; Mikami, T; Nagase, T; Suzuki, M; Suzuki, S | 1 |
Arita, H; Hanasaki, K; Nakano, T | 1 |
Canonico, PL; Judd, AM; Koike, K; MacLeod, RM; Valdenegro, CA | 1 |
Pasquini, JM; Speziale, EH; Speziale, N | 1 |
Knepel, W; Meyen, G | 1 |
Evans, PM; Lanham, DF | 1 |
Maridonneau-Parini, I; Tauber, AI; Tringale, SM | 1 |
Schaeffer, BE; Zadunaisky, JA | 1 |
Cooper, CL; Malik, KU | 1 |
Azuma, H; Ishikawa, M; Sekizaki, S | 1 |
Beer, CT; Buckley, AR; Gout, PW; Kibler, R; Larson, NA; Montgomery, DW; Putnam, CW; Russell, DH; Zukoski, CF | 1 |
Bevan, JA; Tayo, FM | 1 |
Ohshima, Y; Usui, Y; Yoshida, K | 1 |
Takeuchi, T; Yagasaki, O | 1 |
Mishra, OP; Wagerle, LC | 1 |
Fiera, RA; Matthews, N; Neale, ML | 1 |
Duncan, CJ | 1 |
Harper, MJ; Herlihy, JT; Johns, A | 1 |
Nakahata, N; Nakanishi, H; Ono, T | 1 |
Lang, F; Rehwald, W | 1 |
Furukawa, O; Nishiwaki, H; Okabe, S; Takeuchi, K | 1 |
Furukawa, O; Okabe, S; Takeuchi, K; Tanaka, H | 1 |
Fletcher, JE; Rosenberg, H | 2 |
Chazenbalk, GD; De Tomás, M; Juvenal, GJ; Kleiman de Pisarev, DL; Mercuri, H; Pisarev, MA | 1 |
Rubanyi, GM; Vanhoutte, PM | 1 |
Erlij, D; Gersten, L | 1 |
Karaki, H; Murakami, K; Urakawa, N | 1 |
Cooper, CL; Malik, KU; Shaffer, JE | 1 |
Carlini, CR; Guimarães, JA; Ribeiro, JM | 1 |
Odessey, R | 1 |
Kojima, I; Kojima, K; Rasmussen, H | 1 |
Austen, KF; Schick, B | 1 |
Kimura, T; Satoh, S | 1 |
Clark, JS; Jubb, SN; Maloney, PJ; Young, JM | 1 |
Boström, H; Whitehouse, MW | 1 |
Fenton, JW; McKinney, M; Richelson, E; Snider, RM | 1 |
Binder, SB; Michener, M; Peach, MJ; Sybertz, EJ; Trachte, GJ | 1 |
Kumagai, K; Kurane, I; Sekizawa, T; Tsuchiya, Y | 1 |
Andersson, RG; Norrby, K | 1 |
Axelrod, J; Crews, FT; Hirata, F; McGivney, A; Morita, Y; Siraganian, RP | 1 |
Sinha, BK | 1 |
Bloom, AS; Hillard, CJ | 1 |
Ishii, M; Kato, R; Nakadate, T; Yamamoto, S | 2 |
Foley, KA; Rillema, JA | 1 |
Hosono, M; Satoh, H; Satoh, S | 1 |
Bult, H; Claeys, M; Herman, AG; Rampart, M; Van Hove, C | 1 |
Peach, MJ; Singer, HA | 1 |
Canonico, PL; MacLeod, RM; Schettini, G; Valdenegro, CA | 1 |
Grandison, L | 1 |
Canonico, PL; Judd, AM; MacLeod, RM; Valdenegro, CA | 1 |
Brammer, JP; Maguire, MH | 1 |
Mitchell, HW | 2 |
Ibayashi, H; Umeda, F; Wasada, T; Watanabe, J | 1 |
Nakajima, K | 1 |
Kennedy, I; Langley, M; Whelan, CJ | 1 |
Abdel-Latif, AA; Smith, JP | 1 |
Catt, KJ; Naor, Z | 1 |
Vadas, P | 1 |
Chan, AC; Choy, PC; Gerrard, JM; Man, RY; Pritchard, ET | 1 |
Bennett, T; Lot, TY | 1 |
Ikegami, K; Sakanashi, M; Ueda, S; Yonemura, K | 1 |
Brown, CA; Zusman, RM | 1 |
Hwang, DH | 1 |
Bascands, JL; Bompart, G; Girolami, JP; Pecher, C; Rakotoarivony, J; Tack, JL | 1 |
Benicourt, C; Junien, JL; Lockhart, BP; Privat, A | 1 |
Fujimoto, R; Hata, F; Kubo, T; Nagao, T; Nishio, H; Takeuchi, T | 1 |
Ahn, DS; Choi, EJ; Kang, BS; Kang, SI; Lee, HY; Lee, YH | 1 |
Eguchi, S; Hirata, Y; Imai, T; Marumo, F | 1 |
de Lima, WT; Jancar, S; Kwasniewski, FH; Sirois, P | 1 |
Hodgson, WC; Hopkins, BJ; Sutherland, SK | 1 |
Martin, D; Nadler, JV; Peterson, CL; Thompson, MA | 1 |
Li, ZY; Lian, EC; Yu, TF | 1 |
Bustamante, D; Paeile, C | 1 |
Hollenberg, MD; Laniyonu, A; Saifeddine, M; Yang, SG | 1 |
Beraud, M; Bessieres, MH; Frisach, MF; M'Rini, C; Pipy, B; Seguela, JP; Thardin, JF; Vandaele, J | 1 |
Alexander, RW; Berk, BC; Griendling, KK; Lasségue, B; Rao, GN | 1 |
Arnould, T; Dieu, M; Knott, I; Michiels, C; Remacle, J | 1 |
Berman, JD; Brendle, J; Middleton, W; Ray, P | 1 |
Chang, B; Chang, WC; Jen, CJ; Lin, MT; Shi, GY; Tasi, CF; Wang, SJ; Wing, LY; Wu, HL | 1 |
Dazy, AC; Diogène, G; Marano, F; Venant, A | 1 |
Hata, F; Nishio, H; Takeuchi, T; Yagasaki, O | 1 |
Haberman, HF; Kumar, JR; Ranadive, NS | 1 |
Abdel-Latif, AA; Marathe, GK; Yousufzai, SY | 1 |
Breder, CD; Caggiano, AO; Kraig, RP | 1 |
Imanaga, I; Inoue, M; Sakamoto, Y | 1 |
Castell, A; González, L; Nekrassov, V; Sitges, M | 1 |
Fyfe, GK; Kemp, PJ; Olver, RE | 1 |
Matzel, LD; Muzzio, IA; Talk, AC | 1 |
Araújo, CV; Cordeiro, RS; Estato, V; Lopes-Martins, RA; Moreira, S; Tibiriçá, EV | 1 |
Al Moutaery, AR; Tariq, M | 1 |
Van de Voorde, J; Vanheel, B | 1 |
Hollenberg, MD; Mokashi, S; Zheng, XL | 1 |
Adeagbo, AS | 1 |
Corvaïa, N; Coutant, KD; Ryder, NS | 1 |
Ishiguro, S; Matsuoka, Y; Miyamoto, A; Nakamoto, T; Nishio, A | 1 |
Olianas, MC; Onali, P | 1 |
Erdem, SR; Tuncer, M; Yasar, U | 1 |
Farndale, RW; Maddrell, SH; Riegel, JA | 1 |
Chan, PH; Hirvonen, T; Keinänen, R; Koistinaho, J; Koponen, S; Närhi, M; Roivainen, R | 1 |
Folkerts, G; Hedenstierna, G; Hjoberg, J; Högman, M; Nijkamp, FP; van Gessel, SB | 1 |
Hirata, M; Murakami, Y; Okada, S; Wang, M; Yokotani, K | 1 |
Csaba, G; Kovács, P | 1 |
Herlenius, E; Lindahl, SG; Takita, K; Yamamoto, Y | 1 |
Murphy, HS; Quddus, J; Yu, C | 1 |
Biondi, C; Corradini, FG; Ferretti, ME; Neri, LM; Pavan, B; Vesce, F | 1 |
Al Obaid, AR; Al Rasheed, NM; Al Sayed, MI; Al Zuhair, HH; Fatani, AJ | 1 |
Eriksson, E; Hellstrand, M; Nilsson, CL | 1 |
Balasubramanian, KA; Karnik, S; Thomas, S | 1 |
Barrachina, MD; Calatayud, S; Esplugues, JV; Felipo, V; García-Zaragozá, E; Hernández, C; Quintana, E | 1 |
Kanda, M; Kurahashi, K; Nakamura, S; Shirahase, H; Tarumi, T | 1 |
Davies, JE; Jennings, SC; Ng, LL; Pettit, AI; Quinn, PA; Wong, RK | 1 |
Caruso-Neves, C; Fernandes, MS; Leão-Ferreira, LR; Lopes, AG; Quintana-Gomes, E; Santos, DP; Soares, AC | 1 |
Duret, JF; El Habach, T; Haury, L; Tiritilli, A | 1 |
Coen, N; Faherty, S; Flatharta, CO; Harvey, BJ; Thomas, W | 1 |
Campello-Costa, P; Fosse-Júnior, AM; Oliveira-Silva, P; Serfaty, CA | 1 |
Calvès, P; Nonnotte, G; Nonnotte, L; Ollivier, H; Pichavant-Rafini, K; Puill-Stephan, E | 1 |
Fang, GD; Fonteles, MC; Guerrant, RL; Lima, AA; Nascimento, NR; Toyama, MH; Yotseff, P | 1 |
Bühler, MI; Ortiz, ME; Zelarayán, LI | 1 |
185 other study(ies) available for quinacrine and indomethacin
Article | Year |
---|---|
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium | 1985 |
Synthesis and pharmacological evaluation of 2'-hydroxychalcones and flavones as inhibitors of inflammatory mediators generation.
Topics: Animals; Cell Degranulation; Chalcone; Chalcones; Eicosanoids; Flavonoids; Free Radical Scavengers; Humans; Inflammation Mediators; Lipid Peroxidation; Mice; Neutrophils; Pancreatic Elastase; Phospholipases A; Phospholipases A2; Synovial Fluid | 1995 |
Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding | 2008 |
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship | 2010 |
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics | 2010 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |
Antipyretic action of mepacrine without blockade of prostaglandin (PG) synthesis in the C.N.S.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Brain; Indomethacin; Male; Pentylenetetrazole; Prostaglandins; Prostaglandins F; Quinacrine; Rats | 1978 |
The prostaglandins system and insulin release. Studies with the isolated perfused rat pancreas.
Topics: Animals; Aspirin; Furosemide; Glucose; Indomethacin; Insulin; Insulin Secretion; Islets of Langerhans; Male; Prostaglandins; Prostaglandins E; Prostaglandins F; Quinacrine; Rats | 1979 |
Phospholipase A and the mechanism of action of aldosterone.
Topics: Aldosterone; Animals; Anura; Biological Transport; Bufo marinus; Cyclooxygenase Inhibitors; Epithelium; In Vitro Techniques; Indomethacin; Mineralocorticoid Receptor Antagonists; Phospholipases; Quinacrine; Skin; Sodium; Urinary Bladder | 1978 |
Prostaglandins and enzyme secretion from dispersed rat pancreatic acinar cells.
Topics: Amylases; Animals; Arachidonic Acids; Female; Imidazoles; Indomethacin; Pancreas; Phospholipids; Prostaglandins; Quinacrine; Rats; Time Factors | 1979 |
Evidence for purinergic innervation of the anococcygeus muscle.
Topics: Adenosine Triphosphate; Animals; Biogenic Amines; Female; Histocytochemistry; In Vitro Techniques; Indomethacin; Male; Microscopy, Fluorescence; Muscle, Smooth; Purine Nucleotides; Quinacrine; Rabbits; Rats; Rectum | 1978 |
The distribution and metabolism of arachidonic acid in rabbit platelets during aggregation and its modification by drugs.
Topics: Animals; Arachidonic Acids; Blood Platelets; Carbon Radioisotopes; Chemical Phenomena; Chemistry; Chromatography, Gas; Collagen; Fatty Acids; Hydrolysis; In Vitro Techniques; Indomethacin; Lipids; Male; Phosphatidylcholines; Phospholipases; Phospholipids; Phosphorus; Platelet Aggregation; Quinacrine; Rabbits; Thrombin | 1977 |
Quinacrine is a prostaglandin antagonist.
Topics: Animals; Indomethacin; Kinetics; Male; Mesenteric Arteries; Muscle, Smooth; Norepinephrine; Perfusion; Prostaglandin Antagonists; Prostaglandins E; Prostaglandins F; Quinacrine; Rats; Stomach | 1977 |
Metabolism of absorbed glucose in mouse jejunum: influence of arachidonic acid, non-steroidal anti-inflammatory drugs and eicosanoids.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Arachidonic Acids; Cyclooxygenase Inhibitors; Eicosanoids; Glucose; Indomethacin; Intestinal Absorption; Jejunum; Lipoxygenase Inhibitors; Male; Masoprocol; Mice; Mice, Inbred BALB C; Phospholipases; Quinacrine | 1992 |
Role of PGE2 in neurotransmission from pre- to post-ganglionic hypogastric nerves of guinea pigs.
Topics: Animals; Arachidonic Acid; Dinoprostone; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Indomethacin; Male; Quinacrine; Synaptic Transmission; Vas Deferens | 1992 |
Arachidonic acid and prostaglandin E2 activate small-conductance Cl- channels in the basolateral membrane of rabbit parietal cells.
Topics: Animals; Arachidonic Acid; Chlorine; Dinoprostone; Dose-Response Relationship, Drug; Indomethacin; Ion Channels; Male; Membrane Potentials; Nitrobenzoates; Parietal Cells, Gastric; Quinacrine; Rabbits; Umbelliferones | 1992 |
PLA2-induced oedema in rat skin and histamine release in rat mast cells. Evidence for involvement of lysophospholipids in the mechanism of action.
Topics: Animals; Aristolochic Acids; Cytoplasmic Granules; Dexamethasone; Edema; Histamine Release; In Vitro Techniques; Indomethacin; Lysophospholipids; Male; Mast Cells; Phenanthrenes; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Inbred Strains; Skin | 1992 |
Phospholipase-A2 action and arachidonic acid metabolism in calcium-mediated parathyroid hormone secretion.
Topics: Acetophenones; Animals; Arachidonic Acid; Calcium; Cells, Cultured; Dose-Response Relationship, Drug; Flavanones; Flavonoids; Ibuprofen; Indomethacin; Lipoxygenase Inhibitors; Masoprocol; Parathyroid Glands; Parathyroid Hormone; Phospholipases A; Phospholipases A2; Pyrazoles; Quinacrine; Swine; Time Factors; Tritium | 1992 |
Role of arachidonic acid metabolism on corticotropin-releasing factor (CRF)-release induced by interleukin-1 from superfused rat hypothalami.
Topics: Animals; Arachidonic Acid; Corticotropin-Releasing Hormone; Dinoprost; Hypothalamus; Indomethacin; Interleukin-1; Male; Perfusion; Quinacrine; Rats; Rats, Inbred Strains | 1992 |
Excitotoxin induction of ornithine decarboxylase in cerebral cortex is reduced by phospholipase A2 inhibition.
Topics: Animals; Cerebral Cortex; Dexamethasone; Enzyme Induction; Indomethacin; Kainic Acid; Male; Masoprocol; Neurotoxins; Ornithine Decarboxylase; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Inbred Strains | 1992 |
Characteristics of phosphoinositide-specific phospholipase C activity from mouse pancreatic islets.
Topics: Animals; Arachidonic Acid; Calcium; Chlorpromazine; Cyclic AMP; Glucose; Glyceraldehyde 3-Phosphate; Indomethacin; Islets of Langerhans; Male; Mice; Phosphatidylinositols; Putrescine; Quinacrine; Spermine; Substrate Specificity; Tetracaine; Type C Phospholipases | 1991 |
Bradykinin stimulates airway epithelial Cl- secretion via two second messenger pathways.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Bradykinin; Calcimycin; Cells, Cultured; Charybdotoxin; Chlorides; Cyclic AMP; Dogs; Epithelium; Indomethacin; Inositol 1,4,5-Trisphosphate; Isoproterenol; Kinetics; Mucous Membrane; Muscle, Smooth; Prostaglandin Antagonists; Quinacrine; Scorpion Venoms; Second Messenger Systems; Thionucleotides; Trachea; Xanthenes; Xanthones | 1990 |
The differential contribution of endogenous prostaglandins to the release of acetylcholine from the myenteric plexus of the guinea-pig ileum.
Topics: Acetylcholine; Animals; Arachidonic Acid; Arachidonic Acids; Dimethylphenylpiperazinium Iodide; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Indomethacin; Male; Myenteric Plexus; Prostaglandins; Quinacrine; Serotonin; Substance P | 1991 |
Mechanisms of platelet-activating factor-induced electrolyte transport in the rat jejunum.
Topics: Animals; Arachidonic Acids; Azepines; Biological Transport, Active; Chlorides; Dinoprostone; Eicosanoic Acids; Electrophysiology; Female; Indomethacin; Jejunum; Platelet Activating Factor; Quinacrine; Rats; Triazoles | 1991 |
Glucose transport stimulation by bradykinin in Swiss 3T3 fibroblasts: a pertussis toxin-sensitive mechanism operates without involvement of arachidonic acid and cyclic AMP.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Arachidonic Acid; Arachidonic Acids; Biological Transport; Bradykinin; Calcium; Cells, Cultured; Cyclic AMP; Deoxyglucose; Fibroblasts; Glucose; Indomethacin; Insulin; Mice; Pertussis Toxin; Phorbol Esters; Quinacrine; Receptors, Bradykinin; Receptors, Neurotransmitter; Tritium; Virulence Factors, Bordetella | 1991 |
The possible role of phospholipase A2 in hepatic microsomal lipid peroxidation induced by 2,3,7,8-tetrachlorodibenzo-p-dioxin in rats.
Topics: Aminopyrine; Animals; Benzphetamine; beta Carotene; Carotenoids; Female; Indomethacin; Lipid Peroxidation; Microsomes, Liver; Phospholipases A; Phospholipases A2; Phosphorylases; Polychlorinated Dibenzodioxins; Quercetin; Quinacrine; Rats; Rats, Inbred Strains | 1991 |
Effect of inhibitors of eicosanoid synthesis upon lymphocyte proliferation.
Topics: Animals; Aspirin; Caffeic Acids; Cells, Cultured; DNA Replication; Eicosanoids; Indomethacin; Lymph Nodes; Lymphocyte Activation; Male; Masoprocol; Quinacrine; Rats; T-Lymphocytes; Thymidine | 1991 |
Lipid peroxide makes rabbit platelet hyperaggregable to agonists through phospholipase A2 activation.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Blood Platelets; Calcium; Cyclooxygenase Inhibitors; Enzyme Activation; Ferrous Compounds; Indomethacin; Lipid Peroxidation; Lysophosphatidylcholines; Peroxides; Phospholipases A; Phospholipases A2; Platelet Aggregation; Prostaglandin-Endoperoxide Synthases; Quinacrine; Rabbits; tert-Butylhydroperoxide; Vitamin E | 1991 |
Effects of phorbol esters on pial arteriolar diameter and brain production of prostanoids in piglets.
Topics: Animals; Arterioles; Brain; Indomethacin; Phorbol 12,13-Dibutyrate; Pia Mater; Prostaglandin Antagonists; Prostaglandins; Quinacrine; Swine; Vasoconstriction | 1991 |
Phospholipase A2 and mediation of the activation of short-circuit current in the rat colonic mucosa.
Topics: Animals; Arachidonic Acid; Atropine; Bradykinin; Colforsin; Colon; Dose-Response Relationship, Drug; Drug Interactions; Female; Indomethacin; Intestinal Mucosa; Masoprocol; Melitten; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Inbred Strains; Tetrodotoxin | 1991 |
Role of arachidonic acid or its metabolites in growth-hormone-releasing factor-induced release of somatostatin from the median eminence.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Cyclooxygenase Inhibitors; Cytochrome P-450 Enzyme Inhibitors; Growth Hormone-Releasing Hormone; Indomethacin; Kinetics; Lipoxygenase Inhibitors; Male; Masoprocol; Median Eminence; Metyrapone; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Inbred Strains; Somatostatin | 1990 |
Purification and characterization of Contractin A from the pedicellarial venom of sea urchin, Toxopneustes pileolus.
Topics: Amino Acid Sequence; Animals; Guinea Pigs; Indomethacin; Male; Marine Toxins; Molecular Sequence Data; Muscle Contraction; Muscle Proteins; Muscle, Smooth; Quinacrine; Sea Urchins; Trachea; Venoms | 1991 |
Effects of some inhibitors of arachidonic acid metabolism in rat uterus in vitro.
Topics: Animals; Arachidonic Acids; Eicosanoids; Female; Imidazoles; Indomethacin; Masoprocol; Ovariectomy; Quinacrine; Rats; Rats, Inbred Strains; Uterine Contraction; Uterus | 1991 |
Mechanism of human lymphotoxin and tumor necrosis factor induced destruction of cells in vitro: phospholipase activation and deacylation of specific-membrane phospholipids.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Cell Survival; Dexamethasone; Enzyme Activation; Humans; Hydrocortisone; Indomethacin; Lymphotoxin-alpha; Membrane Lipids; Mice; Phospholipases; Phospholipids; Quinacrine; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha | 1990 |
Inhibitors of lipoxygenase have antiproliferative effects on P815 murine mastocytoma cells.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Cell Division; Indomethacin; Leukotrienes; Lipoxygenase; Lipoxygenase Inhibitors; Masoprocol; Mast-Cell Sarcoma; Mice; Phospholipases A; Quinacrine; Tumor Cells, Cultured | 1990 |
Distension-induced secretion in the rat colon: mediation by prostaglandins and submucosal neurons.
Topics: Animals; Anthracenes; Arachidonic Acid; Arachidonic Acids; Atropine; Bufanolides; Capsaicin; Colon; Electrophysiology; Female; Half-Life; Indomethacin; Intestinal Mucosa; Neurons; Phospholipases A; Phospholipases A2; Prostaglandins; Quinacrine; Rats; Rats, Inbred Strains; Tetrodotoxin | 1990 |
Relationship between arachidonic acid release and Ca2(+)-dependent exocytosis in digitonin-permeabilized bovine adrenal chromaffin cells.
Topics: Adrenal Glands; Alkaloids; Animals; Arachidonic Acid; Arachidonic Acids; Calcium; Cattle; Cell Membrane Permeability; Chromaffin Granules; Cyclohexanones; Digitonin; Ethylmaleimide; Exocytosis; Indomethacin; Phospholipases A; Phospholipases A2; Protein Kinase C; Quinacrine; Staurosporine | 1990 |
[Role of prostaglandins in the mechanism of action of indapamide].
Topics: Animals; Blood Pressure; Endothelium, Vascular; Epoprostenol; Female; Indapamide; Indomethacin; Male; Nephrectomy; Quinacrine; Rats; Rats, Brattleboro; Rats, Inbred SHR; Tranylcypromine | 1990 |
Effects of prostaglandin and leukotriene inhibitors on the growth of human glioma spheroids.
Topics: Arachidonic Acids; Dexamethasone; Glioma; Humans; Indomethacin; Ketoprofen; Leukotriene Antagonists; Lipoxygenase Inhibitors; Masoprocol; Mitosis; Prostaglandin Antagonists; Quinacrine; Tumor Cells, Cultured | 1990 |
Stimulation of the respiratory burst in peripheral blood monocytes by lipoteichoic acid. The involvement of calcium ions and phospholipase A2.
Topics: Antigens, Bacterial; Calcium; Cytochrome c Group; Egtazic Acid; Enterococcus faecalis; Humans; In Vitro Techniques; Indomethacin; Ionomycin; Lipopolysaccharides; Monocytes; Oxygen Consumption; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Signal Transduction; Teichoic Acids; Tetradecanoylphorbol Acetate; Zymosan | 1990 |
Nimesulide, indomethacin, BW 755 C, phenidon, mepacrin and nedocromil inhibit the activation of human and rat leucocytes.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Humans; In Vitro Techniques; Indomethacin; Leukocytes; Lipoxygenase Inhibitors; Luminescent Measurements; Nedocromil; Phospholipases A; Pyrazoles; Quinacrine; Quinolones; Rats; Sulfonamides | 1990 |
Influence of mepacrine, indomethacin, and nordihydroguaiaretic acid on the electrical properties of frog renal proximal tubules.
Topics: Animals; Carrier Proteins; Cell Membrane; Electric Conductivity; Indomethacin; Kidney Tubules, Proximal; Masoprocol; Membrane Potentials; Perfusion; Phenylalanine; Quinacrine; Rana esculenta; Sodium-Hydrogen Exchangers | 1990 |
A comparison of the antitumor effects of natural human tumor necrosis factors alpha and beta: the roles of arachidonic acid metabolism and intracellular cAMP.
Topics: Arachidonic Acid; Arachidonic Acids; Breast Neoplasms; Colforsin; Colonic Neoplasms; Cyclic AMP; Dexamethasone; Female; Humans; Indomethacin; Lymphotoxin-alpha; Metyrapone; Phospholipases A; Phospholipases A2; Quinacrine; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha | 1990 |
Effects of inhibitors of eicosanoid synthesis in the uterus of ovariectomized rats and rats in natural oestrus: relation with calcium.
Topics: Animals; Calcium; Dinoprost; Eicosanoids; Estrus; Female; Imidazoles; In Vitro Techniques; Indomethacin; Masoprocol; Methacholine Compounds; Ovariectomy; Oxytocin; Quinacrine; Rats; Uterine Contraction; Uterus | 1990 |
Influences of stress on gastric alkaline secretion in rats.
Topics: Animals; Gastric Acidity Determination; Gastric Mucosa; Immersion; Indomethacin; Male; Omeprazole; Quinacrine; Rats; Rats, Inbred Strains; Stress, Physiological; Vasopressins | 1990 |
Effects of endotoxin and anti-inflammatory agents on superoxide dismutase in the rabbit iris.
Topics: Animals; Anti-Inflammatory Agents; Cycloheximide; Dexamethasone; Endotoxins; Enzyme Induction; Indomethacin; Iris; Masoprocol; Pregnenediones; Quinacrine; Rabbits; Superoxide Dismutase | 1990 |
Captopril-induced increase in coronary flow: an SH-dependent effect on arachidonic acid metabolism?
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Bridged Bicyclo Compounds; Captopril; Chromones; Coronary Circulation; Glutathione; In Vitro Techniques; Indomethacin; Male; Quinacrine; Ramipril; Rats; Rats, Inbred Strains; Sulfhydryl Compounds | 1987 |
Immunological regulation of colonic ion transport.
Topics: Animals; Antigens, Helminth; Bradykinin; Colon; Dinoprostone; Electric Conductivity; Evoked Potentials; Furosemide; Guinea Pigs; Histamine Release; Indomethacin; Jejunum; Male; Pyrilamine; Quinacrine; Reference Values; Tetrodotoxin; Trichinella; Trichinellosis | 1989 |
Mechanism of calcium ionophore stimulated Cl secretion from frog skin glands.
Topics: Amiloride; Animals; Calcimycin; Chlorides; Female; Indomethacin; Ion Channels; Male; Nervous System Physiological Phenomena; Potassium; Quinacrine; Rana esculenta; Skin; Sodium; Stimulation, Chemical; Tetrodotoxin; Trifluoperazine | 1989 |
[Study of behavioral pharmacology on rats. Tranquilizing effects induced by endogenous or exogenous bradykinin].
Topics: Angiotensin II; Animals; Behavior, Animal; Bradykinin; Eugenol; Hypnotics and Sedatives; Indomethacin; Kallikreins; Prostaglandins; Quinacrine; Rats | 1989 |
Effect of prostaglandin inhibitors on bile salt-induced mucosal damage of porcine colon.
Topics: Animals; Body Water; Colon; Deoxycholic Acid; Dinoprostone; Female; Indomethacin; Intestinal Mucosa; Mannitol; Masoprocol; Permeability; Prostaglandin Antagonists; Quinacrine; Swine | 1989 |
Cellular responses to Pyrularia thionin are mediated by Ca2+ influx and phospholipase A2 activation and are inhibited by thionin tyrosine iodination.
Topics: Animals; Antimicrobial Cationic Peptides; Arachidonic Acid; Arachidonic Acids; Calcium; Cell Line; Cell Survival; Cells, Cultured; Dexamethasone; Enzyme Activation; Hemolysis; Humans; Indomethacin; Iodides; Membrane Potentials; Mice; Muscles; Phospholipases; Phospholipases A; Phospholipases A2; Plant Proteins; Quinacrine; Seeds; Tyrosine | 1989 |
Contraction followed by relaxation in response to hypoxia in the sheep isolated middle cerebral artery.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Cerebral Arteries; Endothelium; Hypoxia; Indomethacin; Methylene Blue; Muscle Contraction; Muscle Relaxation; Quinacrine; Serotonin; Sheep | 1989 |
Studies on the mechanism of the sedational state; "tranquilization" evoked by bradykinin or kallikrein in rats.
Topics: Animals; Bradykinin; Brain; Cerebral Ventricles; Dopamine; Epinephrine; Indomethacin; Injections, Intraventricular; Kallikreins; Male; Motor Activity; Prostaglandins; Prostaglandins E; Quinacrine; Rats; Rats, Inbred Strains; Reference Values; Serotonin; Tranquilizing Agents | 1989 |
Phospholipase C activity in human polymorphonuclear leukocytes: partial characterization and effect of indomethacin.
Topics: Calcium; Deoxycholic Acid; Fatty Acids, Nonesterified; Humans; Indomethacin; Kinetics; Lidocaine; Naloxone; Neutrophils; Quinacrine; Type C Phospholipases | 1989 |
Pharmacological evaluation of rat paw oedema induced by Bothrops jararaca venom.
Topics: Animals; Captopril; Crotalid Venoms; Dexamethasone; Edema; Hot Temperature; Indomethacin; Male; Masoprocol; Platelet Activating Factor; Prazosin; Quinacrine; Rats; Rats, Inbred Strains; Reference Values; Yohimbine | 1989 |
Tracheal responsiveness to histamine, PAF-acether and acetylcholine in normal and actively ovalbumin-sensitized guinea pigs.
Topics: Acetylcholine; Animals; Female; Guinea Pigs; Histamine; Immunization; Indomethacin; Isometric Contraction; Male; Ovalbumin; Platelet Activating Factor; Quinacrine; Trachea | 1989 |
Characteristics of canine coronary resistance arteries: importance of endothelium.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetylcholine; Animals; Atropine; Biological Factors; Blood Pressure; Coronary Vessels; Dogs; Endothelium, Vascular; Female; In Vitro Techniques; Indomethacin; Male; Microscopy, Electron; Muscle, Smooth, Vascular; Nitric Oxide; Potassium; Prostaglandin Endoperoxides, Synthetic; Quinacrine; Thrombin; Vascular Resistance; Vasoconstriction; Vasodilation; Vasopressins | 1989 |
Beta-adrenoceptor desensitization in guinea-pig isolated trachea.
Topics: Animals; Autoradiography; Carbachol; Female; Fenoterol; Guinea Pigs; Hydrocortisone; In Vitro Techniques; Indomethacin; Isoproterenol; Male; Muscle Relaxation; Norepinephrine; Quinacrine; Receptors, Adrenergic, beta; Theophylline; Trachea | 1988 |
Growth hormone releasing factor (GRF) increases free arachidonate levels in the pituitary: a role for lipoxygenase products.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Arachidonic Acid; Arachidonic Acids; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Growth Hormone-Releasing Hormone; Indomethacin; Lipoxygenase; Lipoxygenase Inhibitors; Male; Peptide Fragments; Pituitary Gland; Pyrazoles; Quinacrine; Rats; Rats, Inbred Strains; Somatostatin | 1986 |
Beta agonist-induced desensitization in pig bronchus.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Airway Resistance; Animals; Bronchi; Colforsin; Fenoterol; Hydrocortisone; In Vitro Techniques; Indomethacin; Isoproterenol; Muscle Contraction; Muscle Relaxation; Norepinephrine; Phenylephrine; Quinacrine; Receptors, Adrenergic, beta; Stereoisomerism; Swine; Theophylline | 1986 |
Platelet aggregation caused by Carybdea rastonii toxins (CrTX-I, II and III) obtained from a jellyfish, Carybdea rastonii.
Topics: Animals; Blood Platelets; Calcium; Cell Membrane; Chromatography, Gel; Cnidarian Venoms; Dose-Response Relationship, Drug; Indomethacin; Membrane Potentials; Platelet Aggregation; Quinacrine; Rabbits; Scyphozoa; Sodium; Verapamil | 1986 |
Involvement of prostaglandins in histamine-induced fluid and electrolyte secretion by rat colon.
Topics: Animals; Body Fluids; Colon; Electrolytes; Electrophysiology; Histamine; In Vitro Techniques; Indomethacin; Male; Prostaglandins; Quinacrine; Rats | 1988 |
Production of leukotrienes from mouse peritoneal macrophages by treatment with a neutral subfraction of bakers' yeast mannan.
Topics: Animals; Autacoids; Chromatography, High Pressure Liquid; Dexamethasone; Guinea Pigs; Indomethacin; Leukotrienes; Macrophages; Male; Mannans; Mice; Mice, Inbred C3H; Muscle Contraction; Muscle, Smooth; Quinacrine; Saccharomyces cerevisiae | 1988 |
Two phasic generation of thromboxane A2 by the action of collagen on rat platelets.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Blood Platelets; Collagen; Dose-Response Relationship, Drug; Indomethacin; Kinetics; Phospholipases; Platelet Aggregation; Prostaglandin Endoperoxides, Synthetic; Prostaglandins, Synthetic; Quinacrine; Rats; Receptors, Prostaglandin; Receptors, Thromboxane; Sulfonamides; Thromboxane A2 | 1987 |
Arachidonate stimulates prolactin release in vitro: a role for the fatty acid and its metabolites as intracellular regulator(s) in mammotrophs.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Arachidonic Acid; Arachidonic Acids; Bucladesine; Catechols; Cells, Cultured; Female; In Vitro Techniques; Indomethacin; Lipoxygenase Inhibitors; Masoprocol; Oleic Acid; Oleic Acids; Phospholipases A; Phospholipases A2; Pituitary Gland; Pituitary Gland, Anterior; Prolactin; Pyrazoles; Quinacrine; Rats; Rats, Inbred Strains; Stearic Acids; Tetradecanoylphorbol Acetate | 1985 |
Bradykinin stimulates phospholipase C in rat renal medullary slices.
Topics: Animals; Bradykinin; Bucladesine; Diglycerides; Enzyme Activation; Indomethacin; Kidney Medulla; Male; Phosphatidylinositols; Phospholipases; Phospholipids; Quinacrine; Rats; Rats, Inbred Strains; Type C Phospholipases | 1985 |
Effect of various blockers of arachidonic acid metabolism on release of beta-endorphin- and adrenocorticotropin-like immunoreactivity induced by phospholipase A2 from rat adenohypophysis in vitro.
Topics: Acetophenones; Adrenocorticotropic Hormone; Animals; Arachidonic Acid; Arachidonic Acids; beta-Endorphin; Cobalt; Endorphins; In Vitro Techniques; Indomethacin; Male; Phospholipases; Phospholipases A; Phospholipases A2; Pituitary Gland, Anterior; Quinacrine; Radioimmunoassay; Rats; Rats, Inbred Strains | 1986 |
Effects of inhibitors of arachidonic acid metabolism on intercellular adhesion of SV40-3T3 cells.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Aspirin; Catechols; Cell Aggregation; Cell Transformation, Viral; Cells, Cultured; Cyclooxygenase Inhibitors; Indomethacin; Masoprocol; Mice; Quinacrine; Simian virus 40 | 1986 |
Identification of distinct activation pathways of the human neutrophil NADPH-oxidase.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Arachidonic Acid; Arachidonic Acids; Aspirin; Calcium; Enzyme Activation; Humans; Indomethacin; Isoquinolines; NADH, NADPH Oxidoreductases; NADPH Oxidases; Neutrophils; Phospholipases A; Phospholipases A2; Phospholipids; Piperazines; Pyrazoles; Quinacrine; Superoxides; Tetradecanoylphorbol Acetate; Zymosan | 1986 |
Mechanism for leukotriene C4 stimulation of chloride transport in cornea.
Topics: Animals; Biological Transport, Active; Chlorides; Cornea; Cyclic AMP; Dinoprostone; Endothelium; Epithelium; Indomethacin; Kinetics; Prostaglandins E; Quinacrine; Ranidae; SRS-A; Trifluoperazine | 1986 |
Contribution of Ca++ and calmodulin to the action of norepinephrine on renal prostaglandin synthesis and vascular tone.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Blood Pressure; Calcium; Calcium Channel Blockers; Calmodulin; Indomethacin; Kidney; Male; Norepinephrine; Perfusion; Prazosin; Prostaglandins; Quinacrine; Rats; Rats, Inbred Strains; Trifluoperazine; Vasoconstriction | 1986 |
Endothelium-dependent inhibition of platelet aggregation.
Topics: Acetylcholine; Animals; Aorta, Thoracic; Arachidonic Acid; Arachidonic Acids; Catechols; Endothelium; In Vitro Techniques; Indomethacin; Male; Masoprocol; Perfusion; Platelet Aggregation; Quinacrine; Rabbits; Vasodilation | 1986 |
Prolactin-dependent mitogenesis in Nb 2 node lymphoma cells: effects of immunosuppressive cyclopeptides.
Topics: Animals; Calcimycin; Cell Division; Cyclosporins; Depsipeptides; DNA; Enzyme Induction; Estradiol; Gossypol; Indomethacin; Lymphoma; Male; Masoprocol; Ornithine Decarboxylase; Peptides, Cyclic; Prolactin; Quercetin; Quinacrine; Rats; Receptors, Prolactin; Tetradecanoylphorbol Acetate | 1987 |
Extracellular calcium dependence of contraction and endothelium-dependent relaxation varies along the length of the aorta and its branches.
Topics: Acetylcholine; Animals; Aorta; Calcimycin; Calcium; Diltiazem; Endothelium; Extracellular Space; Gallopamil; In Vitro Techniques; Indomethacin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Quinacrine; Rabbits; Vasoconstriction | 1987 |
Platelet aggregation by group B streptococci.
Topics: Aspirin; Blood Platelets; Edetic Acid; Humans; Indomethacin; L-Lactate Dehydrogenase; Platelet Aggregation; Platelet Count; Quinacrine; Serotonin; Streptococcus agalactiae | 1987 |
Modulation of acetylcholine release from guinea-pig Ileum myenteric plexus by arachidonic acid cascade inhibitors.
Topics: Acetylcholine; Animals; Arachidonic Acid; Arachidonic Acids; Dinoprostone; Guinea Pigs; Ileum; In Vitro Techniques; Indomethacin; Male; Myenteric Plexus; Nicotine; Phospholipases A; Prostaglandins E; Quinacrine | 1987 |
Mechanism of CO2 response in cerebral arteries of the newborn pig: role of phospholipase, cyclooxygenase, and lipoxygenase pathways.
Topics: Acetophenones; Animals; Animals, Newborn; Arterioles; Carbon Dioxide; Cerebrovascular Circulation; Indomethacin; Lipoxygenase; Masoprocol; Phospholipases A; Pia Mater; Prostaglandin-Endoperoxide Synthases; Quinacrine; Swine | 1988 |
Involvement of phospholipase A2 activation in tumour cell killing by tumour necrosis factor.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Arachidonic Acids; Cell Survival; Dexamethasone; Humans; Indomethacin; Phospholipases; Phospholipases A; Phospholipases A2; Proadifen; Pyrazoles; Quinacrine; Time Factors; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha | 1988 |
The role of phospholipase A2 in calcium-induced damage in cardiac and skeletal muscle.
Topics: Animals; Calcium; Chlorpromazine; Enzyme Inhibitors; In Vitro Techniques; Indomethacin; Lipoxygenase; Mice; Mice, Inbred BALB C; Microscopy, Electron; Mitochondria; Muscles; Myocardium; Phospholipases; Phospholipases A; Phospholipases A2; Prostaglandin-Endoperoxide Synthases; Quinacrine; Rana temporaria; Sarcoplasmic Reticulum | 1988 |
Modulation of vascular smooth muscle sensitivity by preload and eicosanoid synthesis inhibition.
Topics: 5,8,11,14-Eicosatetraynoic Acid; Animals; Dose-Response Relationship, Drug; Eicosanoic Acids; Female; Indomethacin; Masoprocol; Meclofenamic Acid; Methacrylates; Muscle, Smooth, Vascular; Phenylephrine; Potassium Chloride; Quinacrine; Rabbits; Serotonin | 1987 |
Contribution of prostaglandin E2 to bradykinin-induced contraction in rabbit urinary detrusor.
Topics: Acetylcholine; Adenosine Triphosphate; Animals; Arachidonic Acids; Bradykinin; Caffeic Acids; Dinoprostone; Female; In Vitro Techniques; Indomethacin; Male; Muscle Contraction; Muscle, Smooth; Prostaglandins E; Quinacrine; Rabbits; Urinary Bladder | 1987 |
On the nature of delayed repolarization during sustained sodium coupled transport in frog proximal tubules.
Topics: Animals; In Vitro Techniques; Indomethacin; Kidney Tubules, Proximal; Membrane Potentials; Microelectrodes; Perfusion; Phenylalanine; Quinacrine; Rana esculenta; Sodium; Trifluoperazine | 1987 |
Effects of prostaglandin biosynthesis inhibitors and ouabain on duodenal mucosa and HCO3- secretion in rats.
Topics: Animals; Aspirin; Bicarbonates; Drug Interactions; Duodenum; Gastric Mucosa; Histamine; Indomethacin; Intestinal Mucosa; Male; Ouabain; Prostaglandin Antagonists; Quinacrine; Rats | 1987 |
Determination of acid-neutralizing capacity in rat duodenum. Influences of 16,16-dimethyl prostaglandin E2 and nonsteroidal antiinflammatory drugs.
Topics: 16,16-Dimethylprostaglandin E2; Animals; Anti-Inflammatory Agents; Aspirin; Bicarbonates; Duodenum; Gastric Acid; Gastric Acidity Determination; Hydrogen-Ion Concentration; Indomethacin; Male; Prostaglandins E, Synthetic; Quinacrine; Rats; Rats, Inbred Strains | 1986 |
In vitro muscle contractures induced by halothane and suxamethonium. I: The rat diaphragm.
Topics: Animals; Dantrolene; Diaphragm; Drug Synergism; Halothane; In Vitro Techniques; Indomethacin; Male; Muscle Contraction; Quinacrine; Rats; Rats, Inbred Strains; Spermine; Succinylcholine; Tubocurarine | 1986 |
In vitro muscle contractures induced by halothane and suxamethonium. II: Human skeletal muscle from normal and malignant hyperthermia susceptible patients.
Topics: Disease Susceptibility; Fatty Acids, Nonesterified; Halothane; Humans; In Vitro Techniques; Indomethacin; Malignant Hyperthermia; Muscle Contraction; Muscles; Phospholipases A; Phospholipases A2; Quinacrine; Spermine; Succinylcholine | 1986 |
Biosynthesis and regulation of iodolipids in calf thyroid.
Topics: Animals; Cattle; Imidazoles; Indomethacin; Iodine; Lipid Metabolism; Pancreatin; Propylthiouracil; Quinacrine; Subcellular Fractions; Thyroid Gland; Thyroid Hormones; Thyrotropin; Thyroxine; Triiodothyronine | 1985 |
Hypoxia releases a vasoconstrictor substance from the canine vascular endothelium.
Topics: Acetylcholine; Adenosine Diphosphate; Animals; Coronary Vessels; Dinoprost; Dogs; Endothelium; Female; In Vitro Techniques; Indomethacin; Isometric Contraction; Male; Methylene Blue; Muscle, Smooth, Vascular; Oxygen; Prostaglandins F; Pyrazoles; Quinacrine; Vasoconstriction | 1985 |
Prostaglandin release mediates drug-induced stimulation of sodium transport in frog skin: the effects of quinacrine.
Topics: Amiloride; Animals; Biological Transport, Active; Dinoprostone; Ethers; Indomethacin; Ionomycin; Prostaglandins; Prostaglandins E; Quinacrine; Rana catesbeiana; Skin; Sodium | 1985 |
Role of endothelium in the contractions induced by norepinephrine and clonidine in rat aorta.
Topics: Angiotensin II; Animals; Aorta, Thoracic; Clonidine; Endothelium; In Vitro Techniques; Indomethacin; Male; Methylene Blue; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide; Norepinephrine; Potassium; Prazosin; Quinacrine; Rats; Rats, Inbred Strains; Tetraethylammonium Compounds; Vasodilator Agents; Yohimbine | 1985 |
Mechanism of action of angiotensin II and bradykinin on prostaglandin synthesis and vascular tone in the isolated rat kidney. Effect of Ca++ antagonists and calmodulin inhibitors.
Topics: 6-Ketoprostaglandin F1 alpha; Angiotensin II; Animals; Bradykinin; Calcimycin; Calcium; Calcium Channel Blockers; Calmodulin; Dantrolene; Diltiazem; Dinoprostone; Gallic Acid; Imidazoles; Indomethacin; Kidney; Male; Nicotinic Acids; Nimodipine; Prostaglandins E; Quinacrine; Rats; Rats, Inbred Strains; Ryanodine; Stimulation, Chemical; Sulfonamides; Trifluoperazine; Vasoconstriction | 1985 |
Platelet release reaction and aggregation induced by canatoxin, a convulsant protein: evidence for the involvement of the platelet lipoxygenase pathway.
Topics: 5,8,11,14-Eicosatetraynoic Acid; Adenosine Monophosphate; Animals; Arachidonate Lipoxygenases; Blood Platelets; Caffeine; Creatine Kinase; Drug Interactions; Edetic Acid; Epoprostenol; Guinea Pigs; Humans; In Vitro Techniques; Indicators and Reagents; Indomethacin; Lectins; Lipoxygenase; Phosphocreatine; Plant Proteins; Platelet Aggregation; Quinacrine; Rabbits; Species Specificity; Synaptosomes; Thrombin; Toxins, Biological | 1985 |
Effect of inhibitors of proteolysis and arachidonic acid metabolism on burn-induced protein breakdown.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Aspirin; Burns; Hindlimb; Ibuprofen; In Vitro Techniques; Indomethacin; Leupeptins; Lysosomes; Muscles; Oligopeptides; Peptide Hydrolases; Protease Inhibitors; Proteins; Quinacrine; Rats; Rats, Inbred Strains; Tyrosine | 1985 |
Possible role of phospholipase A2 action and arachidonic acid metabolism in angiotensin II-mediated aldosterone secretion.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; 5,8,11,14-Eicosatetraynoic Acid; Acetophenones; Aldosterone; Angiotensin II; Animals; Arachidonic Acid; Arachidonic Acids; Caffeic Acids; Calcium; Cattle; Cyclooxygenase Inhibitors; Dantrolene; Dose-Response Relationship, Drug; Indomethacin; Lipoxygenase Inhibitors; Phospholipases; Phospholipases A; Phospholipases A2; Pyrazoles; Quinacrine | 1985 |
Pharmacological modulation of activation-secretion of rat serosal mast cells by chymase, an endogenous secretory granule protease.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Arachidonic Acids; Catechols; Chymases; Deoxyadenosines; Dideoxyadenosine; Diethylcarbamazine; Dose-Response Relationship, Drug; Endopeptidases; Exocytosis; Hexosaminidases; Immunoglobulin E; In Vitro Techniques; Indomethacin; Masoprocol; Mast Cells; Prostaglandin D2; Prostaglandins D; Pyrazoles; Quinacrine; Rats; Rats, Inbred Strains; Serine Endopeptidases; Theophylline | 1985 |
Inhibitory effect of quinacrine on myocardial reactive hyperemia in the dog.
Topics: Acetylcholine; Adenosine; Animals; Blood Flow Velocity; Catechols; Coronary Circulation; Dogs; Female; Heart Rate; Hyperemia; Indomethacin; Male; Masoprocol; Pyrazoles; Quinacrine; Regional Blood Flow; Theophylline; Verapamil | 1985 |
Pharmacological investigation of the mechanisms of platelet-activating factor induced mortality in the mouse.
Topics: Anaphylaxis; Animals; Chloroquine; Chlortetracycline; Dexamethasone; Dose-Response Relationship, Drug; Female; Indomethacin; Injections, Intravenous; Male; Mice; Mice, Inbred DBA; Naproxen; Nicardipine; Nifedipine; Platelet Activating Factor; Pyrazoles; Quinacrine; Tetracycline; Verapamil | 1985 |
Biochemical properties of anti-inflammatory drugs. VI. The effects of chloroquine (resochin), mepacrine (quinacrine) and some of their potential metabolites on cartilage metabolism and oxidative phosphorylation.
Topics: Animals; Cartilage; Chloroquine; Glycosaminoglycans; Gold; Hydroxychloroquine; In Vitro Techniques; Indomethacin; Oxidative Phosphorylation; Polysaccharides; Quinacrine; Quinolines; Rats; Sulfates; Sulfur Isotopes; Thiosulfates | 1965 |
Activation of cyclic nucleotide formation in murine neuroblastoma N1E-115 cells by modified human thrombins.
Topics: 5,8,11,14-Eicosatetraynoic Acid; Animals; Antioxidants; Catechols; Cell Line; Cyclic GMP; Humans; Indomethacin; Kinetics; Masoprocol; Mice; Neuroblastoma; Quinacrine; Structure-Activity Relationship; Thrombin | 1984 |
Angiotensin III-induced modulation of neurogenic responses in the rabbit vas deferens and portal vein.
Topics: Angiotensin II; Angiotensin III; Animals; Cyclooxygenase Inhibitors; Dinoprostone; Electric Stimulation; In Vitro Techniques; Indomethacin; Male; Meclofenamic Acid; Muscle, Smooth; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Phospholipases; Portal Vein; Prostaglandins E; Quinacrine; Rabbits; Receptors, Neurotransmitter; Sympathetic Nervous System; Vas Deferens | 1984 |
Inhibition by indomethacin of in vitro reactivation of latent herpes simplex virus type 1 in murine trigeminal ganglia.
Topics: Animals; Female; Indomethacin; Mefenamic Acid; Mice; Mice, Inbred BALB C; Quinacrine; Simplexvirus; Tetracaine; Time Factors; Trigeminal Ganglion; Trigeminal Nerve; Virus Activation | 1984 |
On the role of arachidonic acid metabolites in mast-cell mediated mitogenesis in the rat.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Arachidonic Acid; Arachidonic Acids; Cyclooxygenase Inhibitors; DNA; Histamine; Indomethacin; Lipoxygenase Inhibitors; Male; Mast Cells; Mesentery; Mitosis; p-Methoxy-N-methylphenethylamine; Phospholipases A; Phospholipases A2; Prostaglandins; Pyrazoles; Quinacrine; Rats; Rats, Inbred Strains; SRS-A | 1984 |
Phospholipase activation in the IgE-mediated and Ca2+ ionophore A23187-induced release of histamine from rat basophilic leukemia cells.
Topics: Animals; Anti-Bacterial Agents; Arachidonic Acid; Arachidonic Acids; Basophils; Calcimycin; Calcium; Cell Line; Enzyme Activation; Histamine Release; Immunoglobulin E; Indomethacin; Kinetics; Leukemia, Experimental; Phospholipases; Quinacrine; Rats | 1981 |
Irreversible binding of quinacrine to nucleic acids during horseradish peroxidase- and prostaglandin synthetase-catalyzed oxidation.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; DNA; Horseradish Peroxidase; Indomethacin; Kinetics; Male; Microsomes; Oxidation-Reduction; Peroxidases; Prostaglandin-Endoperoxide Synthases; Quinacrine; RNA; Seminal Vesicles; Sheep | 1983 |
Possible role of prostaglandins in the effects of the cannabinoids on adenylate cyclase activity.
Topics: Adenosine Triphosphate; Adenylyl Cyclases; Animals; Aspirin; Cannabinoids; Dronabinol; Guanosine Triphosphate; Indomethacin; Male; Mice; Mice, Inbred ICR; Phospholipases A; Phospholipases A2; Prostaglandins; Quinacrine | 1983 |
Stimulation of 6-keto-prostaglandin F1 alpha release from isolated pancreatic islets by an insulinotropic concentration of glucose.
Topics: 6-Ketoprostaglandin F1 alpha; Animals; Culture Techniques; Dose-Response Relationship, Drug; Glucose; Indomethacin; Islets of Langerhans; Male; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Secretory Rate | 1983 |
Characteristics of the action of prolactin on [3H]-thymidine incorporation into DNA in mammary gland explants from virgin mice.
Topics: Animals; Culture Techniques; DNA; Female; Hydrocortisone; Indomethacin; Insulin; Kinetics; Mammary Glands, Animal; Mice; Mice, Inbred C3H; Prolactin; Quinacrine; Thymidine | 1983 |
Distinctive effect of angiotensin II on prostaglandin production in dog renal and femoral arteries.
Topics: 6-Ketoprostaglandin F1 alpha; Angiotensin II; Animals; Dinoprostone; Dogs; Epoprostenol; Female; Femoral Artery; Femur; Indomethacin; Kidney; Male; Prostaglandins E; Quinacrine; Regional Blood Flow; Renal Artery; Saralasin | 1984 |
Mechanism of complement-induced stimulation of prostacyclin production by isolated rabbit peritoneum.
Topics: 6-Ketoprostaglandin F1 alpha; Animals; Arachidonic Acid; Arachidonic Acids; Complement C3; Complement C5; Complement System Proteins; Dexamethasone; Epoprostenol; Female; Indomethacin; Male; Molecular Weight; Peptide Fragments; Peritoneum; Prostaglandins; Quinacrine; Rabbits; Trypsin | 1983 |
Endothelium-dependent relaxation of rabbit aorta. II. Inhibition of relaxation stimulated by methacholine and A23187 with antagonists of arachidonic acid metabolism.
Topics: 5,8,11,14-Eicosatetraynoic Acid; Animals; Anti-Bacterial Agents; Aorta, Thoracic; Arachidonic Acid; Arachidonic Acids; Calcimycin; Endothelium; Indomethacin; Isoproterenol; Male; Methacholine Chloride; Methacholine Compounds; Muscle Contraction; Muscle Relaxation; Prostaglandin Antagonists; Quinacrine; Rabbits | 1983 |
Arachidonic acid metabolism and prolactin secretion in vitro: a possible role for the lipoxygenase products.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Catechols; Female; Indomethacin; Lipoxygenase; Masoprocol; Phospholipases A; Phospholipases A2; Pituitary Gland, Anterior; Prolactin; Quinacrine; Rats; Rats, Inbred Strains | 1983 |
Stimulation of anterior pituitary prolactin release by melittin, an activator of phospholipase A2.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Bee Venoms; Biological Transport; Cattle; Cells, Cultured; Indomethacin; Kinetics; Leucine; Melitten; Phospholipases; Phospholipases A; Phospholipases A2; Pituitary Gland, Anterior; Prolactin; Quinacrine; Tritium | 1984 |
Arachidonic acid metabolism and thyrotropin secretion in vitro.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Arachidonic Acid; Arachidonic Acids; Catechols; Female; In Vitro Techniques; Indomethacin; Masoprocol; Phospholipases A; Phospholipases A2; Pituitary Gland; Pyrazoles; Quinacrine; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Thyrotropin; Thyrotropin-Releasing Hormone | 1984 |
Arachidonate metabolism, 5-hydroxytryptamine release and aggregation in human platelets activated by palmitaldehyde acetal phosphatidic acid.
Topics: Adenosine Diphosphate; Arachidonic Acid; Arachidonic Acids; Blood Platelets; Chlorpromazine; Humans; In Vitro Techniques; Indomethacin; Lipids; Malondialdehyde; Platelet Aggregation; Platelet Count; Quinacrine; Serotonin; Thionucleotides; Thrombin | 1984 |
Pharmacological studies into cyclo-oxygenase, lipoxygenase and phospholipase in smooth muscle contraction in the isolated trachea.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Animals; Arachidonate Lipoxygenases; Cyclooxygenase Inhibitors; Female; Guinea Pigs; Histamine; In Vitro Techniques; Indomethacin; Lipoxygenase Inhibitors; Male; Muscle Contraction; Muscle, Smooth; Phospholipases; Phospholipases A; Pyrazoles; Quinacrine; Swine; Trachea | 1984 |
Effect of prostaglandin synthetase inhibitors on platelet aggregation and thromboxane production in diabetes mellitus.
Topics: Adult; Diabetes Mellitus; Diabetic Retinopathy; Female; Humans; Imidazoles; Indomethacin; Male; Middle Aged; Platelet Aggregation; Quinacrine; Thromboxane B2; Thromboxanes | 1984 |
A possible mechanism of vasoactive agents on plasminogen activator release in isolated perfused pig ears.
Topics: Acetylcholine; Animals; Atropine; Bradykinin; Dilazep; Dose-Response Relationship, Drug; Drug Synergism; Ear, External; Histamine; In Vitro Techniques; Indomethacin; Papaverine; Perfusion; Plasminogen Activators; Pressure; Pyrilamine; Quinacrine; Swine; Thrombin; Vasoconstrictor Agents; Vasodilator Agents; Vasomotor System | 1983 |
The release and metabolism of [3H]arachidonic acid from guinea pig perfused lungs in vitro: a simple method for the study of the action of drugs on the release and metabolism of arachidonic acid.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Bradykinin; Guinea Pigs; In Vitro Techniques; Indomethacin; Lung; Quinacrine | 1981 |
The effect of inhibitors of arachidonic acid metabolism on drug-induced contractions in isolated tracheal smooth muscle of the pig.
Topics: 5,8,11,14-Eicosatetraynoic Acid; Acetylcholine; Animals; Arachidonic Acid; Arachidonic Acids; Dexamethasone; In Vitro Techniques; Indomethacin; Muscle Contraction; Muscle, Smooth; Potassium; Prostaglandins E; Quinacrine; Receptors, Histamine; Sodium Salicylate; Swine; Trachea | 1982 |
Inhibition of 12-O-tetradecanoylphorbol-13-acetate-induced epidermal ornithine decarboxylase activity by phospholipase A2 inhibitors and lipoxygenase inhibitor.
Topics: Animals; Antioxidants; Arachidonic Acid; Arachidonic Acids; Carboxy-Lyases; Catechols; Dinoprostone; Female; Indomethacin; Lipoxygenase Inhibitors; Masoprocol; Mice; Ornithine Decarboxylase; Phorbols; Phospholipases; Phospholipases A; Phospholipases A2; Prostaglandins E; Quinacrine; Skin; Tetracaine; Tetradecanoylphorbol Acetate | 1982 |
Studies on the incorporation of [1-14C]arachidonic acid into glycerolipids and its conversion into prostaglandins by rabbit iris. Effects of anti-inflammatory drugs and phospholipase A2 inhibitors.
Topics: Acetophenones; Animals; Anti-Inflammatory Agents; Arachidonic Acid; Arachidonic Acids; Aspirin; Diglycerides; Female; Indomethacin; Iris; Lipid Metabolism; Male; Microsomes; Muscle, Smooth; Phospholipases; Phospholipases A; Phospholipases A2; Phospholipids; Prostaglandins; Quinacrine; Rabbits; Triglycerides | 1982 |
Mechanism of action of gonadotropin-releasing hormone. Involvement of phospholipid turnover in luteinizing hormone release.
Topics: Animals; Arachidonic Acids; Calcium; Cells, Cultured; Chloroquine; Female; Gonadotropin-Releasing Hormone; Indomethacin; Kinetics; Luteinizing Hormone; Phospholipases A; Phospholipases A2; Pituitary Gland; Quinacrine; Rats | 1981 |
The efficacy of anti-inflammatory agents with respect to extracellular phospholipase A2 activity.
Topics: Animals; Anti-Inflammatory Agents; Cycloheximide; Dexamethasone; Enzyme Activation; Indomethacin; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Rabbits | 1982 |
Biphasic modulation of platelet phospholipase A2 activity and platelet aggregation by mepacrine (quinacrine).
Topics: Animals; Aspirin; Blood Platelets; Dose-Response Relationship, Drug; Indomethacin; Male; Phospholipases; Phospholipases A; Phospholipases A2; Platelet Aggregation; Quinacrine; Rats; Substrate Specificity | 1982 |
Comparison of the effects of chloroquine quinacrine and quinidine on autonomic neuroeffector mechanisms.
Topics: Animals; Autonomic Nervous System; Chickens; Chloroquine; Electric Stimulation; Female; Indomethacin; Male; Mice; Norepinephrine; Quinacrine; Quinidine; Rats; Rats, Inbred Strains; Receptors, Cholinergic; Tetrodotoxin | 1982 |
Further investigations on potassium-induced automaticity of isolated human renal artery.
Topics: Adult; Aged; Aspirin; Bradykinin; Female; Humans; In Vitro Techniques; Indomethacin; Male; Middle Aged; Muscle Contraction; Muscle, Smooth, Vascular; Phospholipases A; Phospholipases A2; Potassium; Prostaglandins; Quinacrine; Renal Artery; Tranylcypromine | 1981 |
Role of phospholipase in the regulation of prostaglandin E2 biosynthesis by rabbit renomedullary interstitial cells in tissue culture: effects of angiotensin II, potassium, hyperosmolality, dexamethasone, and protein synthesis inhibition.
Topics: Angiotensin II; Animals; Cycloheximide; Dexamethasone; Indomethacin; Kidney Medulla; Kinetics; Osmolar Concentration; Phospholipases; Potassium; Prostaglandins E; Quinacrine; Rabbits | 1980 |
Aggregation and inhibition of rat platelets, and the formation of endoperoxide metabolites.
Topics: Animals; Heparin; Indomethacin; Male; Platelet Aggregation; Prostaglandin Endoperoxides; Prostaglandins; Quinacrine; Rats; Thromboxane A2; Thromboxane B2; Vitamin E | 1980 |
Bradykinin-induced in vitro contraction of rat mesangial cells via a B2 receptor type.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic beta-2 Receptor Antagonists; Angiotensin II; Animals; Arginine Vasopressin; Bombesin; Bradykinin; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Cells, Cultured; Dinoprost; Dinoprostone; Dose-Response Relationship, Drug; Endothelins; Fatty Acids, Unsaturated; Glomerular Mesangium; Indomethacin; Kinetics; Naphthalenes; Neomycin; Polycyclic Compounds; Prostaglandin Endoperoxides, Synthetic; Protein Kinase C; Quinacrine; Rats; Receptors, Adrenergic, beta-2; Surface Properties; Tetradecanoylphorbol Acetate; Thromboxane A2; Vasoconstrictor Agents | 1994 |
Inhibitors of free radical formation fail to attenuate direct beta-amyloid25-35 peptide-mediated neurotoxicity in rat hippocampal cultures.
Topics: Allopurinol; Alzheimer Disease; Amino Acid Oxidoreductases; Amyloid beta-Peptides; Animals; Arginine; Catalase; Cell Death; Cells, Cultured; Embryo, Mammalian; Free Radical Scavengers; Free Radicals; Hippocampus; Humans; Indomethacin; Masoprocol; Neurons; Neurotoxins; Nitric Oxide Synthase; Nitroarginine; omega-N-Methylarginine; Oxypurinol; Peptide Fragments; Quinacrine; Rats; Rats, Sprague-Dawley; Superoxide Dismutase; Xanthine Oxidase | 1994 |
Ca(2+)-independent fusion of secretory granules with phospholipase A2-treated plasma membranes in vitro.
Topics: 5,8,11,14-Eicosatetraynoic Acid; Albumins; Amylases; Animals; Arachidonic Acid; Benzoquinones; Calcium; Cell Membrane; Cytoplasmic Granules; Egtazic Acid; Exocytosis; Fatty Acids; Indomethacin; Lipoxygenase Inhibitors; Lysophosphatidylcholines; Male; Membrane Fusion; Microscopy, Electron; Parotid Gland; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Wistar | 1995 |
Effects of mastoparan on a vascular contractility in rabbit aorta.
Topics: Animals; Aorta; Arginine; Calcium; In Vitro Techniques; Indomethacin; Intercellular Signaling Peptides and Proteins; Neomycin; Nitroarginine; Peptides; Quinacrine; Rabbits; Vasoconstriction; Wasp Venoms | 1995 |
Endothelin receptor subtypes are coupled to adenylate cyclase via different guanyl nucleotide-binding proteins in vasculature.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Base Sequence; Blotting, Northern; Cattle; Cells, Cultured; Cyclic AMP; DNA Probes; Dose-Response Relationship, Drug; Endothelin Receptor Antagonists; Endothelins; Endothelium, Vascular; GTP-Binding Proteins; Indomethacin; Isoproterenol; Kinetics; Molecular Sequence Data; Muscle, Smooth, Vascular; Oligodeoxyribonucleotides; Peptides, Cyclic; Pertussis Toxin; Poly A; Quinacrine; Rats; Receptors, Endothelin; RNA; RNA, Messenger; Virulence Factors, Bordetella | 1993 |
Studies on the mechanism of PAF-induced vasopermeability in rat lungs.
Topics: Animals; Blood Proteins; Bronchi; Capillary Permeability; Evans Blue; Extravasation of Diagnostic and Therapeutic Materials; Imidazoles; Indomethacin; Lung; Male; Platelet Activating Factor; Quinacrine; Rats; Rats, Wistar; Trachea | 1995 |
Pharmacological studies of stonefish (Synanceja trachynis) venom.
Topics: Animals; Biphenyl Compounds; Blood Pressure; Captopril; Chromones; Dose-Response Relationship, Drug; Fish Venoms; Fishes; Guinea Pigs; Heptanoic Acids; Histamine; Ileum; Imidazoles; In Vitro Techniques; Indomethacin; Losartan; Male; Mecamylamine; Muscle Contraction; Muscle, Smooth; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Receptors, Thromboxane; Serotonin; SRS-A; Tetrazoles; Vas Deferens | 1994 |
Modulation of glutamate and aspartate release from slices of hippocampal area CA1 by inhibitors of arachidonic acid metabolism.
Topics: Animals; Arachidonate 5-Lipoxygenase; Arachidonic Acid; Arginine; Aspartic Acid; Female; Flavanones; Flavonoids; gamma-Aminobutyric Acid; Glutamates; Hippocampus; In Vitro Techniques; Indoles; Indomethacin; Masoprocol; omega-N-Methylarginine; Platelet Activating Factor; Potassium; Prostaglandin-Endoperoxide Synthases; Quinacrine; Rats; Rats, Sprague-Dawley; Receptors, Glutamate; Taurine | 1995 |
Purification and characterization of L-amino acid oxidase from king cobra (Ophiophagus hannah) venom and its effects on human platelet aggregation.
Topics: Alprostadil; Amino Acid Oxidoreductases; Animals; Antimycin A; Aspirin; Blood Coagulation Tests; Blood Platelets; Catalase; Chromatography, Gel; Chromatography, Ion Exchange; Drug Interactions; Edetic Acid; Elapid Venoms; Electrophoresis, Polyacrylamide Gel; Heparin; Hirudins; Humans; Hydrogen Peroxide; Indomethacin; Isoelectric Point; L-Amino Acid Oxidase; Molecular Weight; Nitroprusside; Platelet Aggregation; Quinacrine; Thromboxane A2; Verapamil | 1994 |
Ketorolac tromethamine: an experimental study of its analgesic effects in the rat.
Topics: Analgesics; Animals; Dose-Response Relationship, Drug; Drug Combinations; Electromyography; Formaldehyde; Indomethacin; Ketorolac Tromethamine; Morphine; Nociceptors; Pain Measurement; Prostaglandin Antagonists; Quinacrine; Rats; Rats, Wistar; Reflex; Tolmetin; Tromethamine | 1993 |
Distinct signal transduction pathways for angiotensin-II in guinea pig gastric smooth muscle: differential blockade by indomethacin and tyrosine kinase inhibitors.
Topics: Angiotensin II; Animals; Biphenyl Compounds; Calcium; Catechols; Cyclohexanones; Dose-Response Relationship, Drug; Epidermal Growth Factor; Genistein; Guinea Pigs; Imidazoles; In Vitro Techniques; Indoles; Indomethacin; Isoflavones; Losartan; Male; Muscle, Smooth; Nitriles; Protein-Tyrosine Kinases; Pyridines; Quinacrine; Signal Transduction; Stomach; Tetrazoles; Tyrphostins | 1993 |
Eicosanoid production by mouse peritoneal macrophages during Toxoplasma gondii penetration: role of parasite and host cell phospholipases.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Animals; Arachidonic Acid; Calcium; Cyclooxygenase Inhibitors; Eicosanoids; Female; Indomethacin; Isoquinolines; Lipoxygenase; Macrophages; Mice; Peritoneal Cavity; Phospholipases; Piperazines; Prostaglandin-Endoperoxide Synthases; Protein Kinase C; Quinacrine; Toxoplasma; Toxoplasmosis, Animal | 1993 |
Hydrogen peroxide-induced c-fos expression is mediated by arachidonic acid release: role of protein kinase C.
Topics: Animals; Arachidonic Acid; Blotting, Northern; Cells, Cultured; Gene Expression; Hydrogen Peroxide; Indomethacin; Male; Masoprocol; Protein Kinase C; Proto-Oncogene Proteins c-fos; Quinacrine; Rats; Rats, Sprague-Dawley; RNA, Messenger | 1993 |
Stimulation of prostaglandin synthesis by human endothelial cells exposed to hypoxia.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Arachidonic Acid; Calcium; Carbon Radioisotopes; Cell Hypoxia; Endothelium, Vascular; Humans; Indomethacin; Kinetics; Oxygen; Phospholipases A; Phospholipases A2; Prostaglandins; Quinacrine; Stearic Acids; Tritium; Umbilical Veins; Verapamil | 1993 |
Botulinum toxin inhibits arachidonic acid release associated with acetylcholine release from PC12 cells.
Topics: Acetophenones; Acetylcholine; Animals; Arachidonic Acid; Botulinum Toxins; Cell Differentiation; Dose-Response Relationship, Drug; Ethacrynic Acid; Indomethacin; Kinetics; Masoprocol; Melitten; Models, Biological; Nerve Growth Factors; PC12 Cells; Phospholipases A; Phospholipases A2; Potassium; Protein Kinase C; Quinacrine; Terpenes | 1993 |
Regulation of plasminogen activator inhibitor activity by plasmin in endothelial cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Aspirin; Cells, Cultured; Cyclooxygenase Inhibitors; Endothelium, Vascular; Enzyme Inhibitors; Fibrinolysin; Fibrinolysis; Gene Expression Regulation; GTP-Binding Proteins; Humans; Indomethacin; Isoquinolines; Lipoxygenase Inhibitors; Masoprocol; Pertussis Toxin; Phospholipases A; Phospholipases A2; Piperazines; Plasminogen Activator Inhibitor 1; Protein Kinase C; Quinacrine; Staurosporine; Tissue Plasminogen Activator; Umbilical Veins; Virulence Factors, Bordetella | 1996 |
Differential effects of maitotoxin on calcium entry and ciliary beating in the rabbit ciliated tracheal epithelium.
Topics: Animals; Arachidonic Acids; Biological Transport, Active; Bradykinin; Calcium; Calcium Channel Blockers; Chelating Agents; Cilia; Cyclic AMP; Cyclooxygenase Inhibitors; Egtazic Acid; Enzyme Inhibitors; Epithelium; Indomethacin; Inositol Phosphates; Ionomycin; Kinetics; Lipoxygenase Inhibitors; Marine Toxins; Masoprocol; Motion; Oxocins; Phospholipases A; Quinacrine; Rabbits; Signal Transduction; Stimulation, Chemical; Terpenes; Thapsigargin; Trachea; Trifluoperazine; Verapamil | 1995 |
Ca(2+)-independent fusion of synaptic vesicles with phospholipase A2-treated presynaptic membranes in vitro.
Topics: 5,8,11,14-Eicosatetraynoic Acid; Acetylcholine; Albumins; Animals; Arachidonic Acid; Benzoquinones; Brain; Calcium; Egtazic Acid; Exocytosis; In Vitro Techniques; Indomethacin; Male; Membrane Fusion; Neurotransmitter Agents; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Wistar; Swine; Synaptic Membranes; Synaptic Vesicles | 1996 |
Modulation of 8-methoxypsoralen-photoinduced cutaneous inflammatory reactions by various chemotherapeutic agents in vivo.
Topics: Acetophenones; Animals; Capillary Permeability; Erythema; Ibuprofen; Indoles; Indomethacin; Masoprocol; Methoxsalen; Neutrophils; PUVA Therapy; Quinacrine; Rabbits; Skin | 1996 |
Mediation by prostaglandins of the stimulatory effect of substance P on cyclic AMP production in dog iris sphincter smooth muscle.
Topics: Adenylyl Cyclases; Animals; Cyclic AMP; Cyclooxygenase Inhibitors; Dinoprostone; Dogs; Dose-Response Relationship, Drug; Enzyme Inhibitors; In Vitro Techniques; Indomethacin; Iris; Kinetics; Muscle Contraction; Muscle, Smooth; Phospholipases A; Phospholipases A2; Prostaglandins; Quinacrine; Receptors, Prostaglandin; Substance P | 1996 |
Long-term elevation of cyclooxygenase-2, but not lipoxygenase, in regions synaptically distant from spreading depression.
Topics: Adrenergic alpha-Agonists; Animals; Antibody Specificity; Cerebral Cortex; Cortical Spreading Depression; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Dexamethasone; Enzyme Inhibitors; Glucocorticoids; Hippocampus; Immunohistochemistry; Indomethacin; Isoenzymes; Lipoxygenase; Lipoxygenase Inhibitors; Male; Masoprocol; Nitroprusside; Phenylephrine; Prostaglandin-Endoperoxide Synthases; Quinacrine; Rats; Rats, Wistar; Synapses; Time Factors; Vasodilator Agents | 1996 |
Mn(2+)-induced transient contraction of the longitudinal muscle of guinea-pig stomach through prostaglandin synthesis.
Topics: Animals; Atropine; Calcium; Calcium Channel Blockers; Cyclooxygenase Inhibitors; Electric Stimulation; Enzyme Inhibitors; Female; Gastric Mucosa; Guinea Pigs; In Vitro Techniques; Indomethacin; Male; Manganese; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Nifedipine; Phospholipases A; Phospholipases A2; Prostaglandins; Quinacrine; Stomach; Tetrodotoxin | 1996 |
Characterization of melittin effects in synaptosomes.
Topics: Animals; Arachidonic Acid; Brain; Calcium; gamma-Aminobutyric Acid; Indomethacin; L-Lactate Dehydrogenase; Male; Masoprocol; Melitten; Mice; Microscopy, Electron; Quinacrine; Synaptosomes; Tritium | 1997 |
Conductive Na+ transport in fetal lung alveolar apical membrane vesicles is regulated by fatty acids and G proteins.
Topics: 5,8,11,14-Eicosatetraynoic Acid; Amiloride; Animals; Arachidonic Acid; Biological Transport; Cell Membrane; Enzyme Inhibitors; Fatty Acids; Fetus; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Guanosine Triphosphate; Guinea Pigs; Indomethacin; Masoprocol; Pulmonary Alveoli; Quinacrine; Sodium; Sodium Channels; Thionucleotides | 1997 |
Phospholipases and arachidonic acid contribute independently to sensory transduction and associative neuronal facilitation in Hermissenda type B photoreceptors.
Topics: Acetophenones; Animals; Arachidonic Acid; Association Learning; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Indomethacin; Lipoxygenase Inhibitors; Masoprocol; Mollusca; Neurons; Phospholipases; Photoreceptor Cells, Invertebrate; Quinacrine; Sensation; Signal Transduction | 1997 |
Platelet-activating factor. A possible role in the modulation of the vasomotor tone and blood pressure.
Topics: Adrenergic alpha-Agonists; Animals; Anti-Inflammatory Agents, Non-Steroidal; Azepines; Blood Pressure; Carotid Arteries; Diterpenes; Enzyme Inhibitors; Ginkgolides; Indomethacin; Lactones; Muscle Tonus; Muscle, Smooth, Vascular; Norepinephrine; Phospholipases A; Platelet Activating Factor; Platelet Aggregation Inhibitors; Quinacrine; Rabbits; Triazoles | 1996 |
Effect of quinacrine, a phospholipase A2 inhibitor on stress and chemically induced gastroduodenal ulcers.
Topics: Animals; Cyclooxygenase Inhibitors; Cysteamine; Duodenal Ulcer; Enzyme Inhibitors; Ethanol; Female; Gastric Acid; Gastric Juice; Gastric Mucosa; Immersion; Indomethacin; Male; Peptic Ulcer; Phospholipases A; Phospholipases A2; Pylorus; Quinacrine; Radiation-Protective Agents; Rats; Stomach Ulcer; Stress, Physiological; Sulfhydryl Compounds | 1997 |
Evidence against the involvement of cytochrome P450 metabolites in endothelium-dependent hyperpolarization of the rat main mesenteric artery.
Topics: Animals; Arachidonic Acid; Biological Factors; Cyclooxygenase Inhibitors; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Electric Stimulation; Electrophysiology; Endothelium, Vascular; Enzyme Inhibitors; In Vitro Techniques; Indomethacin; Kinetics; Membrane Potentials; Mesenteric Arteries; Phospholipases A; Quinacrine; Rats; Rats, Wistar | 1997 |
Contractile action of ethanol in guinea pig gastric smooth muscle: inhibition by tyrosine kinase inhibitors and comparison with the contractile action of epidermal growth factor-urogastrone.
Topics: Animals; Calcium; Cyclohexanones; Dose-Response Relationship, Drug; Enzyme Inhibitors; Epidermal Growth Factor; Ethanol; Guinea Pigs; Indomethacin; Male; Muscle Contraction; Protein Tyrosine Phosphatases; Protein-Tyrosine Kinases; Quinacrine; Stomach; Type C Phospholipases | 1997 |
Endothelium-derived hyperpolarizing factor: characterization as a cytochrome P450 1A-linked metabolite of arachidonic acid in perfused rat mesenteric prearteriolar bed.
Topics: Acetylcholine; Animals; Arachidonic Acid; Biological Factors; Cyclooxygenase Inhibitors; Cytochrome P-450 CYP1A1; Enzyme Inhibitors; Histamine; Indomethacin; Male; Mesenteric Arteries; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Perfusion; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Sprague-Dawley; Vasodilation | 1997 |
Bradykinin induces actin reorganization and enhances cell motility in HaCaT keratinocytes.
Topics: Actins; Bradykinin; Cell Line, Transformed; Cell Movement; Enzyme Inhibitors; Humans; Indomethacin; Keratinocytes; Masoprocol; Phospholipases A; Phospholipases A2; Quinacrine | 1997 |
The role of thromboxane A2 in regulating porcine basilar arterial tone.
Topics: Animals; Basilar Artery; Coronary Vessels; Cyclooxygenase Inhibitors; Endothelium, Vascular; Enzyme Inhibitors; Female; In Vitro Techniques; Indomethacin; Male; Mesenteric Arteries; Methacrylates; Muscle, Smooth, Vascular; Pulmonary Artery; Quinacrine; Swine; Thromboxane A2; Thromboxane B2; Thromboxane-A Synthase; Vasoconstriction | 1998 |
GABA(B) receptor-mediated stimulation of adenylyl cyclase activity in membranes of rat olfactory bulb.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Baclofen; Calcium; Calmodulin; Colforsin; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Vitro Techniques; Indomethacin; Injections, Intraventricular; Male; Membranes; Neuropeptides; Neuroprotective Agents; Olfactory Bulb; Organophosphorus Compounds; Pertussis Toxin; Phosphinic Acids; Phospholipases A; Phospholipids; Pituitary Adenylate Cyclase-Activating Polypeptide; Propanolamines; Propylamines; Quinacrine; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Transducin; Virulence Factors, Bordetella | 1999 |
Cyclosporine A preparations and their vehicles induce contraction of the guinea pig gallbladder in vitro: the role of cyclooxygenase metabolites.
Topics: Acetylcholine; Administration, Oral; Animals; Cyclooxygenase Inhibitors; Cyclosporine; Enzyme Inhibitors; Female; Gallbladder; Guinea Pigs; Immunosuppressive Agents; In Vitro Techniques; Indomethacin; Male; Muscle Contraction; Pentanoic Acids; Pharmaceutical Vehicles; Pyridines; Quinacrine; Sphincter of Oddi; Vasodilator Agents | 1999 |
Fluid secretion by isolated Malpighian tubules of Drosophila melanogaster Meig.: effects of organic anions, quinacrine and a diuretic factor found in the secreted fluid.
Topics: Adenylyl Cyclases; Animals; Anions; Body Fluids; Diuresis; Drosophila melanogaster; Female; In Vitro Techniques; Indomethacin; Male; Malpighian Tubules; Nucleotides, Cyclic; Ouabain; Quinacrine | 1999 |
Spreading depression induces expression of calcium-independent protein kinase C subspecies in ischaemia-sensitive cortical layers: regulation by N-methyl-D-aspartate receptors and glucocorticoids.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Brain Ischemia; Cortical Spreading Depression; Cyclooxygenase Inhibitors; Dexamethasone; Diclofenac; Disease Susceptibility; Dizocilpine Maleate; Enzyme Induction; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Gene Expression Regulation, Enzymologic; Indomethacin; Isoenzymes; Male; Nerve Tissue Proteins; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Parietal Lobe; Phospholipases A; Phospholipases A2; Promoter Regions, Genetic; Protein Kinase C; Protein Kinase C-delta; Quinacrine; Quinoxalines; Rats; Rats, Wistar; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Signal Transduction; Transcriptional Activation | 1999 |
Hyperosmolarity-induced relaxation and prostaglandin release in guinea pig trachea in vitro.
Topics: Animals; Dinoprostone; Dose-Response Relationship, Drug; Enzyme Inhibitors; Guinea Pigs; In Vitro Techniques; Indomethacin; Male; Muscle Relaxation; Nitric Oxide Synthase; omega-N-Methylarginine; Osmolar Concentration; Prostaglandins; Quinacrine; Sodium Chloride; Trachea | 2000 |
Brain phospholipase A(2)-arachidonic acid cascade is involved in the activation of central sympatho-adrenomedullary outflow in rats.
Topics: Animals; Arachidonic Acid; Brain; Enzyme Inhibitors; Epinephrine; Indomethacin; Male; Melitten; Norepinephrine; Phospholipases A; Quinacrine; Rats; Rats, Wistar; Signal Transduction | 2000 |
Fluorimetric analysis of phospholipase activity in Tetrahymena pyriformis GL.
Topics: Acetophenones; Aluminum Compounds; Animals; Beryllium; Enzyme Inhibitors; Fluorides; Fluorometry; GTP-Binding Proteins; Indomethacin; Neomycin; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Sodium Fluoride; Tetrahymena pyriformis; Type C Phospholipases | 1999 |
Effects of neuroactive substances on the morphine-induced respiratory depression; an in vitro study.
Topics: Acetylcholine; Animals; Animals, Newborn; Colforsin; Drug Interactions; Efferent Pathways; Haloperidol; Indomethacin; Morphine; Neurons; Neurotransmitter Agents; Quinacrine; Rats; Rats, Sprague-Dawley; Respiratory Center; Respiratory Insufficiency; Spinal Cord; Substance P; Thyrotropin-Releasing Hormone | 2000 |
Functional expression of NAD(P)H oxidase p47 in lung microvascular endothelial cells.
Topics: Allopurinol; Animal Population Groups; Animals; Cells, Cultured; Endothelium, Vascular; Enzyme Inhibitors; HL-60 Cells; Humans; Indomethacin; Mice; Mice, Inbred AKR; Microcirculation; NADH, NADPH Oxidoreductases; NADPH Oxidases; Onium Compounds; Phosphoproteins; Pulmonary Circulation; Quinacrine; Rotenone; Signal Transduction; Superoxides; Tetradecanoylphorbol Acetate | 2000 |
Formyl-methionyl-leucyl-phenylalanine induces prostaglandin E2 release from human amnion-derived WISH cells by phospholipase C-mediated [Ca+]i rise.
Topics: Amnion; Binding Sites; Calcium; Cell Line; Cyclooxygenase Inhibitors; Dinoprostone; Enzyme Inhibitors; Estrenes; Humans; Indomethacin; Microscopy, Confocal; N-Formylmethionine Leucyl-Phenylalanine; Oligopeptides; Pyrrolidinones; Quinacrine; Radioimmunoassay; Signal Transduction; Type C Phospholipases | 2001 |
Effects of two newly synthesized analogues of lidocaine on rat arterial blood pressure and heart rate.
Topics: Anesthetics, Local; Animals; Anti-Arrhythmia Agents; Antihypertensive Agents; Atropine; Benzoates; Blood Pressure; Calcium Chloride; Cyproheptadine; Enzyme Inhibitors; Heart Rate; Hexamethonium; Histamine Agonists; Indomethacin; Lidocaine; Male; Monitoring, Physiologic; NG-Nitroarginine Methyl Ester; Pyrilamine; Quinacrine; Ranitidine; Rats; Rats, Wistar; Vasodilator Agents | 2001 |
Dopamine D(2) receptor-induced COX-2-mediated production of prostaglandin E(2) in D(2)-transfected Chinese hamster ovary cells without simultaneous administration of a Ca(2+)-mobilizing agent.
Topics: Animals; Arachidonic Acids; Calcium; Calcium Channel Blockers; CHO Cells; Cricetinae; Cyclooxygenase 2; Dinoprostone; Dopamine; Dopamine Antagonists; Drug Interactions; Enzyme Inhibitors; Gallic Acid; Indomethacin; Isoenzymes; Naphthalenes; Nitrobenzenes; Phosphatidylcholines; Prostaglandin-Endoperoxide Synthases; Pyrones; Quinacrine; Receptors, Dopamine D2; Salicylamides; Salicylates; Sulfonamides; Tetradecanoylphorbol Acetate; Transfection | 2002 |
Surgical manipulation of the small intestine and its effect on the lung.
Topics: Allopurinol; alpha-Tocopherol; Animals; Arginine; Catalase; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Fatty Acids, Unsaturated; Female; Indomethacin; Intestine, Small; Lung; Male; Neutrophil Activation; Oxidative Stress; Peroxidase; Quinacrine; Rats; Rats, Wistar; Reactive Oxygen Species; Superoxide Dismutase | 2002 |
Downregulation of nNOS and synthesis of PGs associated with endotoxin-induced delay in gastric emptying.
Topics: Animals; Arachidonic Acid; Cyclooxygenase Inhibitors; Endotoxins; Enzyme Inhibitors; Food; Gastric Emptying; Indazoles; Indomethacin; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Nitric Oxide Synthase Type II; Nitrobenzenes; Phospholipases A; Prostaglandins; Pyloric Antrum; Quinacrine; Rats; Rats, Sprague-Dawley; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sulfonamides | 2002 |
Role of intracellular Ca2+ in endothelium-dependent contraction and relaxation of rabbit intrapulmonary arteries.
Topics: Animals; Aspirin; Calcimycin; Calcium; Endothelium, Vascular; Enzyme Inhibitors; Indomethacin; Ionomycin; Ionophores; Male; Methacrylates; Methylene Blue; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Pulmonary Artery; Quinacrine; Rabbits; Terpenes; Thapsigargin | 2003 |
Advanced glycation end products stimulate an enhanced neutrophil respiratory burst mediated through the activation of cytosolic phospholipase A2 and generation of arachidonic Acid.
Topics: Acetylcysteine; Adult; Arachidonic Acid; Arachidonic Acids; Cells, Cultured; Enzyme Inhibitors; Glycation End Products, Advanced; Group IV Phospholipases A2; Humans; Indomethacin; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Organophosphonates; Oxidation-Reduction; Phospholipases A; Phospholipases A2; Quinacrine; Reactive Oxygen Species; Respiratory Burst; Vascular Diseases | 2003 |
PLA2/PGE2 are involved in the inhibitory effect of bradykinin on the angiotensin-(1-7)-stimulated Na(+)-ATPase activity of the proximal tubule.
Topics: Angiotensin I; Animals; Bradykinin; Bradykinin B2 Receptor Antagonists; Cell Membrane; Cyclooxygenase Inhibitors; Diclofenac; Dinoprostone; Dose-Response Relationship, Drug; Indomethacin; Kidney Tubules, Proximal; Peptide Fragments; Phospholipases A; Phospholipases A2; Quinacrine; Receptor, Bradykinin B2; Sodium-Potassium-Exchanging ATPase; Swine | 2004 |
BK2 but not BK1 receptors mediating contractile response in human umbilical arteries: role of thromboxane A2.
Topics: Bradykinin; Bradykinin B1 Receptor Antagonists; Bradykinin B2 Receptor Antagonists; Dose-Response Relationship, Drug; Endothelium; Humans; Imidazoles; Indomethacin; Masoprocol; Muscle Contraction; Muscle, Smooth, Vascular; Quinacrine; Receptor, Bradykinin B1; Receptor, Bradykinin B2; Thromboxane A2; Umbilical Arteries | 2004 |
Estrogen induces phospholipase A2 activation through ERK1/2 to mobilize intracellular calcium in MCF-7 cells.
Topics: Animals; Antineoplastic Agents; Breast Neoplasms; Calcium; Cattle; Cyclooxygenase Inhibitors; Enzyme Activation; Estradiol; Group IV Phospholipases A2; Humans; Indomethacin; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Phospholipases A; Phospholipases A2; Phosphorylation; Protein Transport; Quinacrine; Receptors, Estrogen; Serum Albumin, Bovine; Signal Transduction | 2006 |
Blockade of arachidonic acid pathway induces sprouting in the adult but not in the neonatal uncrossed retinotectal projection.
Topics: Animals; Animals, Newborn; Arachidonic Acid; Enzyme Inhibitors; Immunohistochemistry; Indomethacin; Lipoxygenase Inhibitors; Masoprocol; Neuronal Plasticity; Phospholipases A; Phospholipases A2; Prostaglandin-Endoperoxide Synthases; Quinacrine; Rats; Retina; Signal Transduction; Synapses; Synaptic Transmission; Visual Pathways | 2006 |
Effects of hyposmotic stress on exocytosis in isolated turbot, Scophthalmus maximus, hepatocytes.
Topics: 1-Butanol; Alkaloids; Androstadienes; Animals; Benzophenanthridines; Cell Membrane; Colchicine; Cytochalasin B; Cytoskeleton; Estrenes; Exocytosis; Flatfishes; Fluorescent Dyes; Hepatocytes; Indomethacin; Ionomycin; Isoquinolines; Masoprocol; Osmotic Pressure; Phenanthridines; Pyridinium Compounds; Pyrrolidinones; Quaternary Ammonium Compounds; Quinacrine; Signal Transduction; Sulfonamides; Thapsigargin; Wortmannin | 2006 |
Role of phospholipase A2 and tyrosine kinase in Clostridium difficile toxin A-induced disruption of epithelial integrity, histologic inflammatory damage and intestinal secretion.
Topics: Animals; Bacterial Toxins; Cell Line, Tumor; Disease Models, Animal; Drug Combinations; Enterotoxins; Enzyme Inhibitors; Ileum; Indomethacin; Intestinal Mucosa; Male; Phospholipase A2 Inhibitors; Phospholipases A2; Protein-Tyrosine Kinases; Quinacrine; Rabbits | 2008 |
Involvement of PLA2, COX and LOX in Rhinella arenarum oocyte maturation.
Topics: Animals; Arachidonic Acid; Bufo arenarum; Cells, Cultured; Cyclooxygenase 2 Inhibitors; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Indomethacin; Lactones; Lipoxygenase; Masoprocol; Melitten; Oocytes; Oogenesis; Phospholipases A2; Progesterone; Prostaglandin-Endoperoxide Synthases; Quinacrine; Sulfones | 2014 |