quinacrine and dibucaine

quinacrine has been researched along with dibucaine in 19 studies

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19909 (47.37)18.7374
1990's7 (36.84)18.2507
2000's2 (10.53)29.6817
2010's1 (5.26)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Chiang, GH; Unger, SH1
Galanakis, D; Ganellin, CR1
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Frithz, G; Jansson, A; Ronquist, G1
Garcia-Martin, E; Gutiérrez-Merino, C1
Dorman, RV; Schwartz, MA; Terrian, DM1
Andrenyak, DM; Epstein, PM; Feinstein, MB; Sha'afi, RI; Volpi, M1
Chang, HH; Galton, N; Lampe, RA; Magruder, CD; Michaelis, EK; Michaelis, ML1
Harris, EJ; Jackson, MJ; Jones, DA1
Feinstein, MB; Opas, EE; Walenga, RW1
Homma, Y; Nagai, Y; Takenawa, T1
Almeida, AR; Bunnachak, D; Burke, TJ; Gengaro, P; Nemenoff, RA; Schrier, RW; Wetzels, JF1
Capparelli, AW; Jo, OD; Li, L; Wang, YP; Yanagawa, N1
Ardelt, B; Borowitz, JL; Isom, GE; Kanthasamy, AG; Malave, A; Mills, EM; Powley, TL1
Camarasa, J; Camins, A; Escubedo, E; Gabriel, C; Pallàs, M; Sureda, FX1
Creer, MH; McHowat, J1
Honeyman, TW; Kennington, L; Kohjimoto, Y; Scheid, CR1

Other Studies

19 other study(ies) available for quinacrine and dibucaine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Octanol-physiological buffer distribution coefficients of lipophilic amines by reversed-phase high-performance liquid chromatography and their correlation with biological activity.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:3

    Topics: Amines; Animals; Buffers; Chromatography, High Pressure Liquid; Histamine Release; Lipid Metabolism; Octanols; Protein Binding; Rats; Serum Albumin, Bovine; Sodium-Potassium-Exchanging ATPase; Solubility; Structure-Activity Relationship

1981
Defining determinant molecular properties for the blockade of the apamin-sensitive SKCa channel in guinea-pig hepatocytes: the influence of polarizability and molecular geometry.
    Bioorganic & medicinal chemistry letters, 2004, Aug-02, Volume: 14, Issue:15

    Topics: Animals; Apamin; Guinea Pigs; Hepatocytes; Kinetics; Molecular Conformation; Potassium Channels, Calcium-Activated

2004
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
    Journal of medicinal chemistry, 2008, Jan-24, Volume: 51, Issue:2

    Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase

2008
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Phospholipase A activity in seminal plasma of men attending an infertility clinic.
    Urologia internationalis, 1991, Volume: 46, Issue:2

    Topics: Acetophenones; Dibucaine; Humans; Infertility, Male; Male; Oligospermia; Phospholipases A; Quinacrine; Semen; Sperm Count; Triglycerides; Zinc

1991
Local anesthetics inhibit the Ca2+, Mg2+-ATPase activity of rat brain synaptosomes.
    Journal of neurochemistry, 1986, Volume: 47, Issue:3

    Topics: Anesthetics, Local; Animals; Brain; Ca(2+) Mg(2+)-ATPase; Calcium-Transporting ATPases; Dibucaine; Kinetics; Lidocaine; Procaine; Quinacrine; Rats; Rats, Inbred Strains; Synaptosomes; Tetracaine

1986
Depolarization-induced [3H]arachidonic acid accumulation: effects of external Ca2+ and phospholipase inhibitors.
    Brain research bulletin, 1988, Volume: 21, Issue:3

    Topics: Animals; Arachidonic Acid; Arachidonic Acids; Calcium Channel Blockers; Cerebellum; Dibucaine; Enzyme Inhibitors; Phospholipases; Quinacrine; Rats; Verapamil

1988
Local anesthetics, mepacrine, and propranolol are antagonists of calmodulin.
    Proceedings of the National Academy of Sciences of the United States of America, 1981, Volume: 78, Issue:2

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; 3',5'-Cyclic-GMP Phosphodiesterases; Anesthetics, Local; Animals; Brain; Calcium-Binding Proteins; Calcium-Transporting ATPases; Calmodulin; Cyclic Nucleotide Phosphodiesterases, Type 1; Dibucaine; Drug Antagonism; Enzyme Activation; Erythrocyte Membrane; Erythrocytes; Humans; Kinetics; Propranolol; Quinacrine; Rats

1981
Effects of amphipathic drugs on L'[3H]glutamate binding to synaptic membranes and the purified binding protein.
    Neurochemical research, 1984, Volume: 9, Issue:1

    Topics: Anesthetics, Local; Animals; Chlorpromazine; Dibucaine; Glutamates; Kinetics; Male; Quinacrine; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Glutamate; Synaptic Membranes; Tetracaine

1984
Inhibition of lipid peroxidation in muscle homogenates by phospholipase A2 inhibitors.
    Bioscience reports, 1984, Volume: 4, Issue:7

    Topics: Animals; Chloroquine; Chlorpromazine; Dibucaine; Female; Free Radicals; In Vitro Techniques; Iron; Lipid Peroxides; Mice; Muscles; Phospholipases; Phospholipases A; Phospholipases A2; Procaine; Quinacrine; Tetracaine

1984
Differential effects of calmodulin antagonists on phospholipases A2 and C in thrombin-stimulated platelets.
    The Journal of biological chemistry, 1981, Dec-10, Volume: 256, Issue:23

    Topics: Arachidonic Acid; Arachidonic Acids; Blood Platelets; Calcium-Binding Proteins; Calmodulin; Chlorpromazine; Dibucaine; Fluphenazine; Humans; Kinetics; Phospholipases; Phospholipases A; Phospholipids; Platelet Aggregation; Quinacrine; Thrombin; Trifluoperazine; Type C Phospholipases

1981
Effect of calmodulin antagonists on lysosomal enzyme secretion and phospholipid metabolism in guinea-pig macrophages.
    The Biochemical journal, 1982, Dec-15, Volume: 208, Issue:3

    Topics: Acetylglucosaminidase; Animals; Arachidonic Acid; Arachidonic Acids; Calcium-Binding Proteins; Calmodulin; Dibucaine; Female; Guinea Pigs; Hexosaminidases; In Vitro Techniques; Lysosomes; Macrophages; Phospholipids; Quinacrine; Trifluoperazine; Triglycerides

1982
Ca2+ uptake, fatty acid, and LDH release during proximal tubule hypoxia: effects of mepacrine and dibucaine.
    The American journal of physiology, 1994, Volume: 266, Issue:2 Pt 2

    Topics: Animals; Biological Transport; Calcium; Dibucaine; Dose-Response Relationship, Drug; Fatty Acids, Nonesterified; Hypoxia; In Vitro Techniques; Kidney Tubules, Proximal; Kinetics; L-Lactate Dehydrogenase; Quinacrine; Rats; Time Factors

1994
Effect of luminal angiotensin II on proximal tubule fluid transport: role of apical phospholipase A2.
    The American journal of physiology, 1994, Volume: 266, Issue:2 Pt 2

    Topics: Angiotensin II; Animals; Dibucaine; Dose-Response Relationship, Drug; In Vitro Techniques; Kidney Tubules, Proximal; Kinetics; Male; Perfusion; Phospholipases A; Phospholipases A2; Quinacrine; Rabbits

1994
Reactive oxygen species generated by cyanide mediate toxicity in rat pheochromocytoma cells.
    Toxicology letters, 1997, Sep-19, Volume: 93, Issue:1

    Topics: Amitrole; Animals; Ascorbic Acid; Catalase; Cell Death; Dibucaine; Dose-Response Relationship, Drug; Enzyme Inhibitors; Lipid Peroxidation; Microscopy, Confocal; PC12 Cells; Potassium Cyanide; Quinacrine; Rats; Reactive Oxygen Species; Superoxide Dismutase

1997
Modulation of neuronal mitochondrial membrane potential by the NMDA receptor: role of arachidonic acid.
    Brain research, 1997, Nov-28, Volume: 777, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; Anesthetics, Local; Animals; Arachidonic Acid; Biomarkers; Cells, Cultured; Cerebellum; Dibucaine; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Flow Cytometry; Fluorescent Dyes; Glycine; Intracellular Membranes; Kynurenic Acid; Membrane Potentials; Mitochondria; N-Methylaspartate; Piperidines; Quinacrine; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Rhodamine 123; Rhodamines; Sulfonamides

1997
Thrombin activates a membrane-associated calcium-independent PLA2 in ventricular myocytes.
    The American journal of physiology, 1998, Volume: 274, Issue:2

    Topics: Animals; Arachidonic Acid; Calcium; Cell Membrane; Dibucaine; Enzyme Activation; Enzyme Inhibitors; Female; Heart Ventricles; In Vitro Techniques; Myocardium; Naphthalenes; Peptide Fragments; Phospholipases A; Phospholipases A2; Pyrones; Quinacrine; Rabbits; Receptors, Thrombin; Thrombin

1998
Role of phospholipase A2 in the cytotoxic effects of oxalate in cultured renal epithelial cells.
    Kidney international, 1999, Volume: 56, Issue:4

    Topics: Anesthetics, Local; Animals; Arachidonic Acid; Arachidonic Acids; Biological Transport; Cell Line; Cyclohexanones; Dibucaine; Diglycerides; Dogs; Enzyme Inhibitors; Epithelial Cells; Free Radicals; Kidney Tubules, Distal; Oleic Acid; Oxalates; Phospholipases A; Phospholipases A2; Protease Inhibitors; Quinacrine; Tritium

1999