quinacrine and colforsin

quinacrine has been researched along with colforsin in 19 studies

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19903 (15.79)18.7374
1990's13 (68.42)18.2507
2000's2 (10.53)29.6817
2010's1 (5.26)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Nicholson, GC; Papadimitriou, JM; Wood, DJ; Zheng, MH1
Wagner, PD; Wu, YN; Yang, YC1
Bylund, DB; Halenda, SP; Jones, SB1
Diener, M; Rummel, W1
Abayasekara, DR; Band, AM; Cooke, BA1
Fuchimoto, S; Orita, K; Shiiki, S1
Lindmar, R; Löffelholz, K; Sandmann, J1
Goldie, RG; Paterson, JW; Spina, D1
Bascands, JL; Girolami, JP; Pecher, C1
Ciaranello, RD; Harrington, MA; Shaw, K; Zhong, P1
Hata, Y; Hiraishi, H; Kawabe, T; Mutoh, H; Ota, S; Shiina, S; Sugimoto, T; Terano, A; Yoshiura, K1
Bast, A; Kramer, K; Smink, CG1
Olianas, MC; Onali, P1
Carranza, ML; Cheval, L; Doucet, A; Favre, H; Féraille, E; Kiroytcheva, M; Martin, PY1
Satake, N; Shibata, S1
Herlenius, E; Lindahl, SG; Takita, K; Yamamoto, Y1
Anderson, LA; Boothe, JR; Danielewicz, MA; Franz, AK; Wong, DM1

Other Studies

19 other study(ies) available for quinacrine and colforsin

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Evidence that protein kinase-A, calcium-calmodulin kinase and cytoskeletal proteins are involved in osteoclast retraction induced by calcitonin.
    Experimental and molecular pathology, 1992, Volume: 57, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Bone Resorption; Calcitonin; Cells, Cultured; Colchicine; Colforsin; Cytoskeletal Proteins; In Vitro Techniques; Isoquinolines; Neomycin; Osteoclasts; Phospholipases A; Piperazines; Protein Kinase C; Protein Kinase Inhibitors; Protein Kinases; Quinacrine; Rats; Rats, Sprague-Dawley; Type C Phospholipases; Verapamil

1992
Modification of chromaffin cells with pertussis toxin or N-ethylmaleimide lowers cytoskeletal F-actin and enhances Ca(2+)-dependent secretion.
    The Journal of biological chemistry, 1992, Apr-25, Volume: 267, Issue:12

    Topics: Actins; Adenosine Diphosphate Ribose; Adrenal Glands; Animals; Calcium; Cations, Divalent; Cattle; Chromaffin Granules; Colforsin; Cytoskeleton; Down-Regulation; Ethylmaleimide; Microscopy, Fluorescence; Norepinephrine; Pertussis Toxin; Protein Kinase C; Quinacrine; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella

1992
Alpha 2-adrenergic receptor stimulation of phospholipase A2 and of adenylate cyclase in transfected Chinese hamster ovary cells is mediated by different mechanisms.
    Molecular pharmacology, 1991, Volume: 39, Issue:2

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Enzyme Activation; Female; Kinetics; Membranes; Ovary; Pertussis Toxin; Phospholipases A; Phospholipases A2; Prazosin; Quinacrine; Receptors, Adrenergic, alpha; Signal Transduction; Stimulation, Chemical; Time Factors; Transfection; Tritium; Virulence Factors, Bordetella; Yohimbine

1991
Phospholipase A2 and mediation of the activation of short-circuit current in the rat colonic mucosa.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 343, Issue:6

    Topics: Animals; Arachidonic Acid; Atropine; Bradykinin; Colforsin; Colon; Dose-Response Relationship, Drug; Drug Interactions; Female; Indomethacin; Intestinal Mucosa; Masoprocol; Melitten; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Inbred Strains; Tetrodotoxin

1991
Evidence for the involvement of phospholipase A2 in the regulation of luteinizing hormone-stimulated steroidogenesis in rat testis Leydig cells.
    Molecular and cellular endocrinology, 1990, Apr-17, Volume: 70, Issue:2

    Topics: Acetophenones; Animals; Arachidonic Acids; Bucladesine; Colforsin; Cyclic AMP; Dexamethasone; Hydroxycholesterols; Leydig Cells; Luteinizing Hormone; Male; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Inbred Strains; Testosterone

1990
A comparison of the antitumor effects of natural human tumor necrosis factors alpha and beta: the roles of arachidonic acid metabolism and intracellular cAMP.
    Japanese journal of clinical oncology, 1990, Volume: 20, Issue:3

    Topics: Arachidonic Acid; Arachidonic Acids; Breast Neoplasms; Colforsin; Colonic Neoplasms; Cyclic AMP; Dexamethasone; Female; Humans; Indomethacin; Lymphotoxin-alpha; Metyrapone; Phospholipases A; Phospholipases A2; Quinacrine; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha

1990
The release of choline from phospholipids mediated by beta-adrenoceptor activation in isolated hearts.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 334, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Calcium; Chickens; Choline; Colforsin; Cyclic AMP; Guinea Pigs; In Vitro Techniques; Myocardial Contraction; Myocardium; Phospholipids; Quinacrine; Receptors, Adrenergic, beta; Receptors, Muscarinic

1986
Beta agonist-induced desensitization in pig bronchus.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:1

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Airway Resistance; Animals; Bronchi; Colforsin; Fenoterol; Hydrocortisone; In Vitro Techniques; Indomethacin; Isoproterenol; Muscle Contraction; Muscle Relaxation; Norepinephrine; Phenylephrine; Quinacrine; Receptors, Adrenergic, beta; Stereoisomerism; Swine; Theophylline

1986
Indirect inhibition by bradykinin of cyclic AMP generation in isolated rat glomeruli and mesangial cells.
    Molecular pharmacology, 1993, Volume: 44, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Bradykinin; Cells, Cultured; Colforsin; Cyclic AMP; Diglycerides; Dinoprostone; Down-Regulation; Drug Interactions; Enzyme Activation; Glomerular Mesangium; Isoproterenol; Kidney Glomerulus; Male; Pertussis Toxin; Protein Kinase C; Quinacrine; Rats; Rats, Sprague-Dawley; Receptors, Bradykinin; Stimulation, Chemical; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella

1993
Agonist-induced desensitization and loss of high-affinity binding sites of stably expressed human 5-HT1A receptors.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 268, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclase Inhibitors; Arachidonic Acid; Binding Sites; Calcium; Colforsin; Enzyme Activation; HeLa Cells; Humans; Ligands; Phosphatidylinositols; Phospholipases A; Phospholipases A2; Phosphorylation; Protein Kinase C; Quinacrine; Receptors, Serotonin; Serotonin; Tetradecanoylphorbol Acetate

1994
Roles of Ca2+ and protein kinase C in regulation of prostaglandin E2 release by cultured rabbit gastric epithelial cells.
    Digestive diseases and sciences, 1993, Volume: 38, Issue:8

    Topics: 2-Chloroadenosine; Animals; Calcimycin; Calcium; Calcium Channel Blockers; Calmodulin; Cells, Cultured; Colforsin; Cyclic AMP; Dinoprostone; Drug Interactions; Epithelium; Female; Gallic Acid; Gastric Mucosa; Male; Protein Kinase C; Quinacrine; Rabbits; Stomach

1993
Effect of phospholipase A2 activation on the receptor function in the rat left atrium: unmasking of a positive inotropic effect of methacholine.
    General pharmacology, 1997, Volume: 29, Issue:3

    Topics: Adrenergic beta-Agonists; Animals; Cardiotonic Agents; Colforsin; Enzyme Activation; Enzyme Inhibitors; Heart; Heart Atria; In Vitro Techniques; Isoproterenol; Melitten; Methacholine Chloride; Muscarinic Agonists; Myocardial Contraction; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Wistar; Receptors, Neurotransmitter

1997
GABA(B) receptor-mediated stimulation of adenylyl cyclase activity in membranes of rat olfactory bulb.
    British journal of pharmacology, 1999, Volume: 126, Issue:3

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Baclofen; Calcium; Calmodulin; Colforsin; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Vitro Techniques; Indomethacin; Injections, Intraventricular; Male; Membranes; Neuropeptides; Neuroprotective Agents; Olfactory Bulb; Organophosphorus Compounds; Pertussis Toxin; Phosphinic Acids; Phospholipases A; Phospholipids; Pituitary Adenylate Cyclase-Activating Polypeptide; Propanolamines; Propylamines; Quinacrine; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Transducin; Virulence Factors, Bordetella

1999
Effect of cAMP on the activity and the phosphorylation of Na+,K(+)-ATPase in rat thick ascending limb of Henle.
    Kidney international, 1999, Volume: 55, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Adenosine Monophosphate; Adenosine Triphosphate; Animals; Bucladesine; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Kidney Medulla; Loop of Henle; Male; Organ Culture Techniques; Oxygen; Phosphodiesterase Inhibitors; Phosphorylation; Quinacrine; Rats; Rats, Wistar; Rubidium Radioisotopes; Sodium; Sodium-Potassium-Exchanging ATPase

1999
The potentiating effect of genistein on the relaxation induced by isoproterenol in rat aortic rings.
    General pharmacology, 1999, Volume: 33, Issue:3

    Topics: Adrenergic beta-Agonists; Animals; Aorta; Benzoflavones; Bucladesine; Colforsin; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Genistein; In Vitro Techniques; Isoproterenol; Male; Methoxsalen; Muscle Relaxation; Phosphodiesterase Inhibitors; Quinacrine; Rats; Rats, Wistar; Theophylline

1999
Effects of neuroactive substances on the morphine-induced respiratory depression; an in vitro study.
    Brain research, 2000, Nov-24, Volume: 884, Issue:1--2

    Topics: Acetylcholine; Animals; Animals, Newborn; Colforsin; Drug Interactions; Efferent Pathways; Haloperidol; Indomethacin; Morphine; Neurons; Neurotransmitter Agents; Quinacrine; Rats; Rats, Sprague-Dawley; Respiratory Center; Respiratory Insufficiency; Spinal Cord; Substance P; Thyrotropin-Releasing Hormone

2000
Phenotypic screening with oleaginous microalgae reveals modulators of lipid productivity.
    ACS chemical biology, 2013, May-17, Volume: 8, Issue:5

    Topics: Antioxidants; Batch Cell Culture Techniques; Biomass; Butylated Hydroxyanisole; Catechin; Colforsin; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Fluorescent Dyes; Lipid Metabolism; Lipids; Microalgae; Oxazines; Phenotype; Quinacrine; Small Molecule Libraries

2013