quinacrine and carbachol

quinacrine has been researched along with carbachol in 29 studies

Research

Studies (29)

TimeframeStudies, this research(%)All Research%
pre-199018 (62.07)18.7374
1990's9 (31.03)18.2507
2000's1 (3.45)29.6817
2010's1 (3.45)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Albuquerque, EX; Eldefrawi, AT; Eldefrawi, ME; Oliveira, AC; Tsai, MC1
Briley, MS; Changeux, JP1
Changeux, JP; Grünhagen, H1
Changeux, J; Grünhagen, HH; Iwatsubo, M1
Changeux, JP; Grünhagen, HH; Iwatsubo, M1
Changeux, JP; Grünhagen, HH2
Dehaye, JP; Gomez, F; Grosfils, K1
Howlett, AC; O'Donnell, KA1
Olianas, MC; Onali, P1
Fernandes, LB; Goldie, RG; Knight, DA; Paterson, JW; Rigby, PJ; Spina, D1
Bowman, A; Gillespie, JS; Soares-da-Silva, P1
Barnes, PJ; Cuss, FM; Grandordy, BM1
Dandona, P; Jeremy, J; Morrow, C; Murphy, S; Pearce, B1
Lindmar, R; Löffelholz, K; Sandmann, J1
Bade, SC; Gardner, RM1
Adams, PR; Feltz, A1
Craven, PA; DeRubertis, FR1
Kaldany, RR; Karlin, A1
Izumi, F; Kobayashi, H; Sakurai, S; Wada, A; Yanagihara, N1
Leusen, I; Van de Voorde, J1
Arias, HR; Johnson, DA1
Carroll, RT; Davis, RE; Doyle, PD; Emmerling, MR; Moore, CJ1
Ayres, S; Johnson, DA1
Arita, Y; Hou, W; Morisset, J2
Artaud, F; Chéramy, A; Glowinski, J; Godeheu, G; L'hirondel, M1

Other Studies

29 other study(ies) available for quinacrine and carbachol

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Mode of action of quinacrine on the acetylcholine receptor ionic channel complex.
    Molecular pharmacology, 1979, Volume: 16, Issue:2

    Topics: Acetylcholine; Animals; Anura; Carbachol; Female; Fishes; In Vitro Techniques; Ion Channels; Membrane Potentials; Muscle Contraction; Quinacrine; Rana pipiens; Rats; Receptors, Cholinergic

1979
Recovery of some functional properties of the detergent-extracted cholinergic receptor protein from Torpedo marmorata after reintegration into a membrane environment.
    European journal of biochemistry, 1978, Mar-15, Volume: 84, Issue:2

    Topics: Animals; Carbachol; Cell Membrane; Cholic Acids; Deoxycholic Acid; Detergents; Fishes; Humans; Phosphatidylcholines; Prilocaine; Quinacrine; Receptors, Cholinergic; Toxins, Biological

1978
[Structural transitions of the Torpedo cholinergic receptor in its membrane state as demonstrated by a fluorescent local anesthetic: quinacrine].
    Comptes rendus hebdomadaires des seances de l'Academie des sciences. Serie D: Sciences naturelles, 1975, Oct-06, Volume: 281, Issue:14

    Topics: Acetylcholine; Animals; Carbachol; Electric Organ; Fishes; Kinetics; Membranes; Parasympatholytics; Quinacrine; Receptors, Cholinergic; Spectrometry, Fluorescence; Structure-Activity Relationship

1975
[Rapid changes in the intensity of fluorescence observed in the presence of cholinergic agonists with Torpedo marmorata membrane fragments rich in cholinergic receptors and labelled with quinacrine].
    Comptes rendus hebdomadaires des seances de l'Academie des sciences. Serie D: Sciences naturelles, 1976, Oct-18, Volume: 283, Issue:9

    Topics: Acetylcholine; Animals; Carbachol; Electric Organ; Fishes; Fluorescence; Hexamethonium Compounds; Kinetics; Parasympathomimetics; Protein Conformation; Quinacrine; Receptors, Cholinergic

1976
Fast kinetic studies on the interaction of cholinergic agonists with the membrane-bound acetylcholine receptor from Torpedo marmorata as revealed by quinacrine fluorescence.
    European journal of biochemistry, 1977, Oct-17, Volume: 80, Issue:1

    Topics: Acetylcholine; Animals; Carbachol; Choline; Electric Organ; Fishes; Fluorescence; In Vitro Techniques; Kinetics; Parasympathomimetics; Quinacrine; Receptors, Cholinergic; Spectrometry, Fluorescence; Temperature

1977
Studies on the electrogenic action of acetylcholine with Torpedo marmorata electric organ. IV. Quinacrine: a fluorescent probe for the conformational transitions of the cholinergic receptor protein in its membrane-bound state.
    Journal of molecular biology, 1976, Sep-25, Volume: 106, Issue:3

    Topics: Acetylcholine; Animals; Binding, Competitive; Carbachol; Cell Membrane; Decamethonium Compounds; Electric Organ; Fishes; Gallamine Triethiodide; Hexamethonium Compounds; Kinetics; Prilocaine; Protein Conformation; Quinacrine; Receptors, Cholinergic; Spectrometry, Fluorescence

1976
Studies on the electrogenic action of acetylcholine with Torpedo marmorata electric organ. V. Qualitative correlation between pharmacological effects and equilibration processes of the cholinergic receptor protein as revealed by the structural probe quina
    Journal of molecular biology, 1976, Sep-25, Volume: 106, Issue:3

    Topics: Acetylcholine; Animals; Binding Sites; Carbachol; Cell Membrane; Electric Organ; Energy Transfer; Fishes; Prilocaine; Quaternary Ammonium Compounds; Quinacrine; Receptors, Cholinergic; Snake Venoms; Spectrometry, Fluorescence

1976
Inhibition by mepacrine and amylase secretion from intact and permeabilized rat pancreatic acini.
    Biochemical and biophysical research communications, 1992, Apr-15, Volume: 184, Issue:1

    Topics: Amylases; Animals; Calcium; Carbachol; Cell Membrane Permeability; Dose-Response Relationship, Drug; Egtazic Acid; In Vitro Techniques; Kinetics; Male; Pancreas; Quinacrine; Rats; Rats, Inbred Strains; Sincalide

1992
Muscarinic receptor binding is inhibited by quinacrine.
    Neuroscience letters, 1991, Jun-10, Volume: 127, Issue:1

    Topics: Binding, Competitive; Calcium; Carbachol; Cyclic AMP; Muscarinic Antagonists; Neuroblastoma; Quinacrine; Quinuclidinyl Benzilate; Receptors, Muscarinic; Secretin; Tumor Cells, Cultured

1991
Ca2(+)-independent stimulation of adenylate cyclase activity by muscarinic receptors in rat olfactory bulb.
    Journal of neurochemistry, 1990, Volume: 55, Issue:3

    Topics: Adenylyl Cyclases; Alkaloids; Animals; Calcium; Calmodulin; Carbachol; Cell Membrane; Egtazic Acid; Male; Olfactory Bulb; Quinacrine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Staurosporine; Tetradecanoylphorbol Acetate

1990
Beta-adrenoceptor desensitization in guinea-pig isolated trachea.
    European journal of pharmacology, 1988, Nov-22, Volume: 157, Issue:2-3

    Topics: Animals; Autoradiography; Carbachol; Female; Fenoterol; Guinea Pigs; Hydrocortisone; In Vitro Techniques; Indomethacin; Isoproterenol; Male; Muscle Relaxation; Norepinephrine; Quinacrine; Receptors, Adrenergic, beta; Theophylline; Trachea

1988
A comparison of the action of the endothelium-derived relaxant factor and the inhibitory factor from the bovine retractor penis on rabbit aortic smooth muscle.
    British journal of pharmacology, 1986, Volume: 87, Issue:1

    Topics: Animals; Carbachol; Catechols; Cattle; Endothelium; Flurbiprofen; Guanylate Cyclase; In Vitro Techniques; Male; Masoprocol; Methylene Blue; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Neural Inhibition; Neurotransmitter Agents; Nitric Oxide; Nitroprusside; Norepinephrine; Penis; Quinacrine; Rabbits; Vasodilator Agents

1986
Breakdown of phosphoinositides in airway smooth muscle: lack of influence of anti-asthmatic drugs.
    Life sciences, 1987, Sep-28, Volume: 41, Issue:13

    Topics: Animals; Carbachol; Cattle; Dexamethasone; Histamine; Hydrolysis; Isoproterenol; Muscle Contraction; Phosphatidylinositols; Phospholipases; Quinacrine; Theophylline; Trachea; Verapamil

1987
Inositol phospholipids are probably not the source of arachidonic acid for eicosanoid synthesis in astrocytes.
    FEBS letters, 1987, Jan-19, Volume: 211, Issue:1

    Topics: Animals; Animals, Newborn; Arachidonic Acid; Arachidonic Acids; Astrocytes; Calcimycin; Carbachol; Cells, Cultured; Cerebral Cortex; Eicosanoic Acids; Inositol; Inositol Phosphates; Kinetics; Norepinephrine; Phosphatidylinositols; Quinacrine; Rats; Sugar Phosphates

1987
On the mechanism of muscarinic hydrolysis of choline phospholipids in the heart.
    Biochemical pharmacology, 1988, Dec-15, Volume: 37, Issue:24

    Topics: Animals; Atropine Derivatives; Carbachol; Chickens; Choline; Inositol Phosphates; Membrane Lipids; Myocardium; Oleic Acid; Oleic Acids; Phosphatidic Acids; Phosphatidylcholines; Phospholipase D; Phospholipases; Quinacrine; Receptors, Muscarinic; Time Factors

1988
Effects of mepacrine on uterine contractile responses.
    Biology of reproduction, 1985, Volume: 32, Issue:5

    Topics: Animals; Barium; Barium Compounds; Carbachol; Chlorides; Dinoprost; Dose-Response Relationship, Drug; Female; Oxytocin; Prostaglandins F; Quinacrine; Rats; Rats, Inbred Strains; Uterine Contraction

1985
End-plate channel opening and the kinetics of quinacrine (mepacrine) block.
    The Journal of physiology, 1980, Volume: 306

    Topics: Acetylcholine; Animals; Carbachol; Dose-Response Relationship, Drug; In Vitro Techniques; Ion Channels; Kinetics; Membrane Potentials; Motor Endplate; Muscles; Neuromuscular Junction; Quinacrine; Rana esculenta

1980
Stimulation of rat colonic mucosal prostaglandin synthesis by calcium and carbamylcholine: relationship to alterations in cyclic nucleotide metabolism.
    Prostaglandins, 1981, Volume: 21, Issue:1

    Topics: Animals; Calcimycin; Calcium; Carbachol; Colon; Cyclic AMP; Cyclic GMP; Drug Synergism; Fatty Acids; Intestinal Mucosa; Nucleotides, Cyclic; Prostaglandins E; Quinacrine; Rats; Tetracaine

1981
Reaction of quinacrine mustard with the acetylcholine receptor from Torpedo californica.
    The Journal of biological chemistry, 1983, May-25, Volume: 258, Issue:10

    Topics: Animals; Carbachol; Cell Membrane Permeability; Cobra Neurotoxin Proteins; Electric Organ; Ion Channels; Proadifen; Quinacrine; Quinacrine Mustard; Radioisotopes; Receptors, Cholinergic; Rubidium; Torpedo; Tritium; Tubocurarine

1983
Suppression by phospholipase A2 inhibitors of secretion of catecholamines from isolated adrenal medullary cells by suppression of cellular calcium uptake.
    Biochemical pharmacology, 1983, Apr-01, Volume: 32, Issue:7

    Topics: Acetophenones; Adrenal Medulla; Animals; Calcium; Carbachol; Catecholamines; Cattle; Chloroquine; Dose-Response Relationship, Drug; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Quinine

1983
Influence of prostaglandin-synthesis inhibitors on carbachol- and histamine-induced vasodilatation in perfused rat hindquarters.
    Pflugers Archiv : European journal of physiology, 1983, Jun-01, Volume: 397, Issue:4

    Topics: Animals; Arachidonic Acids; Carbachol; Hindlimb; Histamine; Histamine Antagonists; Male; Perfusion; Prostaglandin Antagonists; Quinacrine; Rats; Receptors, Histamine; Vasodilation

1983
Differential agonist-induced displacement of quinacrine and ethidium from their respective histrionicotoxin-sensitive binding sites on the Torpedo acetylcholine receptor.
    Biochemistry, 1995, Feb-07, Volume: 34, Issue:5

    Topics: Acetylcholine; Amphibian Venoms; Animals; Binding Sites; Binding, Competitive; Carbachol; Choline; Cholinergic Agonists; Cholinergic Antagonists; Ethidium; Quinacrine; Receptors, Cholinergic; Torpedo

1995
Phospholipase A2 activation influences the processing and secretion of the amyloid precursor protein.
    Biochemical and biophysical research communications, 1993, Nov-30, Volume: 197, Issue:1

    Topics: Amyloid beta-Protein Precursor; Animals; Carbachol; CHO Cells; Cricetinae; Enzyme Activation; Homosteroids; Melitten; Phospholipases A; Phospholipases A2; Protein Processing, Post-Translational; Quinacrine; Receptors, Muscarinic; Sesterterpenes; Terpenes

1993
Quinacrine noncompetitive inhibitor binding site localized on the Torpedo acetylcholine receptor in the open state.
    Biochemistry, 1996, May-21, Volume: 35, Issue:20

    Topics: Animals; Binding Sites; Carbachol; Cyclic N-Oxides; Dansyl Compounds; Electric Organ; Fluorescent Dyes; In Vitro Techniques; Kinetics; Lipid Bilayers; Nicotinic Antagonists; Protein Conformation; Quaternary Ammonium Compounds; Quinacrine; Receptors, Nicotinic; Spin Labels; Torpedo

1996
Caerulein-stimulated arachidonic acid release in rat pancreatic acini: a diacylglycerol lipase affair.
    The American journal of physiology, 1996, Volume: 271, Issue:5 Pt 1

    Topics: Androstadienes; Animals; Arachidonic Acid; Aristolochic Acids; Carbachol; Cells, Cultured; Ceruletide; Cyclohexanones; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Estrenes; Kinetics; Lipoprotein Lipase; Lipoxygenase Inhibitors; Male; Pancreas; Phenanthrenes; Phospholipase D; Phospholipases A; Phospholipases A2; Pyrrolidinones; Quinacrine; Rats; Rats, Sprague-Dawley; Wortmannin

1996
Endogenous arachidonic acid release and pancreatic amylase secretion.
    Pancreas, 1997, Volume: 14, Issue:3

    Topics: Amylases; Animals; Arachidonic Acid; Aristolochic Acids; Carbachol; Cyclohexanones; Enzyme Inhibitors; In Vitro Techniques; Lipoprotein Lipase; Male; Melitten; Pancreas; Phenanthrenes; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Sprague-Dawley

1997
Contribution of endogenously formed arachidonic acid in the presynaptic facilitatory effects of NMDA and carbachol on dopamine release in the mouse striatum.
    The European journal of neuroscience, 1999, Volume: 11, Issue:4

    Topics: Animals; Arachidonic Acid; Carbachol; Corpus Striatum; Dopamine; Drug Resistance; Drug Synergism; Enzyme Inhibitors; Magnesium; Male; Mice; N-Methylaspartate; Phospholipases A; Phospholipases A2; Presynaptic Terminals; Quinacrine; Synapses; Tetrodotoxin

1999