quinacrine and 4-bromophenacyl bromide

quinacrine has been researched along with 4-bromophenacyl bromide in 69 studies

Research

Studies (69)

TimeframeStudies, this research(%)All Research%
pre-199034 (49.28)18.7374
1990's30 (43.48)18.2507
2000's4 (5.80)29.6817
2010's0 (0.00)24.3611
2020's1 (1.45)2.80

Authors

AuthorsStudies
Fujii, T; Hashizume, T; Sato, T1
Larsson, C; Mau, S; Saermark, T; Simonsson, P1
Bonnet, P; Bourdeau, A; Herviaux, P; Lieberherr, M; Sachs, C; Souberbielle, JC1
Farkas, T; Kuehn, H; Nemecz, G; Wallukat, G; Wollenberger, A1
Brown, EJ; Lennartz, MR1
Madamba, S; Schweitzer, P; Siggins, GR1
Frithz, G; Jansson, A; Ronquist, G1
Imamura, K; Kufe, DW; Mohri, M; Robbins, G; Rodriguez, C; Sherman, ML; Spriggs, DR1
Kufe, D; Mohri, M; Spriggs, DR1
Abayasekara, DR; Band, AM; Cooke, BA1
Dennis, EA; Glaser, KB; Lister, MD; Ulevitch, RJ1
Anderson, RA; Bielfeld, P; Feathergill, KA; Johnson, SK; Zaneveld, LJ1
Andersson, RG; Toll, JB1
Paul, SM; Schwartz, RD; Skolnick, P1
Choi, SH; Fukutomi, O; Inagaki, N; Koda, A; Matsuura, N; Nagai, H; Sakamoto, T1
McMorris, FA; Shin, ML; Shirazi, Y1
Chappell, JB; Henderson, LM; Jones, OT1
Borowitz, SM; Montgomery, C1
Aeberhard, EE; Barrett, CT; Kaplan, SA; Scott, ML1
Bergstrand, H; Brattsand, R; Dahlbäck, M1
Ofenstein, JP; Rillema, JA1
Mishra, OP; Wagerle, LC1
Nakagawa, Y; Waku, K1
Cei de Job, C; Suburo, A1
Cameron, CM; Etindi, RN; Rillema, JA1
Beckman, JK; Borowitz, SM; Burr, IM1
Kojima, I; Kojima, K; Rasmussen, H1
Fujimoto, Y; Fujita, T; Kagen, C; Ueno, T; Uno, H1
Best, L; Malaisse, WJ; Mathias, PC; Sener, A1
Pelicci, PG; Rochant, H; Testa, U; Thomopoulos, P; Titeux, M1
Kagey-Sobotka, A; Lichtenstein, LM; Marone, G1
Furchgott, RF1
Batenburg, JJ; Post, M; Schuurmans, EA; Van Golde, LM1
Kato, R; Kumakura, K; Sasakawa, N; Yamamoto, S1
Carine, K; Hudig, D1
Kodama, H; Mikasa, H; Miyahara, M; Okimasu, E; Terada, S; Utsumi, K1
Akamatsu, N; Fujimoto, Y; Fujita, T; Hattori, A1
Douglas, WW; Nemeth, EF1
Kuno, M; Yawo, H1
Hofmann, SL; Majerus, PW; Prescott, SM1
Abdel-Latif, AA; Smith, JP1
Izumi, F; Kobayashi, H; Sakurai, S; Wada, A; Yanagihara, N1
Frye, RA; Holz, RW1
Azuri, R; Erman, A; Raz, A1
Cranston, WI; Hellon, RF; Mitchell, D; Townsend, Y1
Haigler, HT; Pastan, I; Willingham, MC1
Nakamura, S1
Villarroel, A1
Johnson, MS; Mitchell, R; Thomson, FJ; Wolbers, B1
Dana, R; Levy, R; Malech, HL1
Burch, RA; Kulp, GV; Leff, AR; Neeley, SP; Spaethe, SM; Strek, ME; White, SR1
Andersson, R; Ar'Rajab, A; Bengmark, S; Fabia, R; Willén, R1
Beraud, M; Bessieres, MH; Frisach, MF; M'Rini, C; Pipy, B; Seguela, JP; Thardin, JF; Vandaele, J1
Berman, JD; Brendle, J; Middleton, W; Ray, P1
Chang, JP; Garofalo, R; Neumann, CM1
Chen, SS; Jiang, MC; Lin, JK1
Haberman, HF; Kumar, JR; Ranadive, NS1
Csaba, G; Kovács, P2
Bashan, N; Kozlovsky, N; Shohami, E1
Matzel, LD; Muzzio, IA; Talk, AC1
Boucrot, P; Bourass, J; Elkihel, L; Letourneux, Y; Petit, JY1
Hemontolor, ME; Sastry, BV1
Hur, GH; Kim, YB; Shin, S1
Bader, BW; Bankhurst, AD; Doshi, RN; Whalen, MM1
Cantoni, O; Fiorani, M; Guidarelli, A1
Llanos, MN; Moraga, PF; Ronco, AM1
Furuyama, S; Kuboyama, N; Moriwaki, K; Nakao, S; Ogata, Y; Sakurai, T; Sugiya, H1
Cui, Y; Li, L; Lu, Y; Qian, Z; Wang, Z; Yang, K; Zhang, Y; Zhu, K; Zong, S1

Reviews

2 review(s) available for quinacrine and 4-bromophenacyl bromide

ArticleYear
Macrophage phospholipase A2 activity and eicosanoid production: studies with phospholipase A2 inhibitors in P388D1 cells.
    Advances in experimental medicine and biology, 1990, Volume: 275

    Topics: Acetophenones; Animals; Cell Line; Eicosanoids; Fatty Acids; Macrophages; Mice; Phospholipases A; Phospholipases A2; Quinacrine; Substrate Specificity; Terpenes

1990
The role of endothelium in the responses of vascular smooth muscle to drugs.
    Annual review of pharmacology and toxicology, 1984, Volume: 24

    Topics: 5,8,11,14-Eicosatetraynoic Acid; Acetophenones; Acetylcholine; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Arachidonic Acid; Arachidonic Acids; Bradykinin; Calcimycin; Catechols; Endothelium; Histamine; Hydroquinones; Hypoxia; Masoprocol; Methylene Blue; Muscle Relaxation; Muscle, Smooth, Vascular; Prostaglandins; Quinacrine; Serotonin; Substance P; Thrombin

1984

Other Studies

67 other study(ies) available for quinacrine and 4-bromophenacyl bromide

ArticleYear
Preferential activation of phospholipase A2 by low concentrations of phosphatidic acid with long-chain fatty acids in rabbit platelets.
    Journal of biochemistry, 1992, Volume: 112, Issue:6

    Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Acetophenones; Animals; Blood Platelets; Cytosol; Enzyme Activation; Kinetics; Phosphatidic Acids; Phospholipases A; Phospholipases A2; Platelet Aggregation; Quinacrine; Rabbits

1992
Activation of protein kinase C in permeabilized human neuroblastoma SH-SY5Y cells.
    Journal of neurochemistry, 1992, Volume: 59, Issue:2

    Topics: Acetophenones; Amino Acid Sequence; Arachidonic Acids; Calcium; Cell Membrane; Cell Membrane Permeability; Digitonin; Diglycerides; Dose-Response Relationship, Drug; Enzyme Activation; Humans; Molecular Sequence Data; Myelin Basic Protein; Neuroblastoma; Phospholipases A; Phospholipases A2; Phosphorus; Phosphorus Radioisotopes; Phosphorylation; Protein Kinase C; Quinacrine; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured

1992
Phospholipase-A2 action and arachidonic acid metabolism in calcium-mediated parathyroid hormone secretion.
    Endocrinology, 1992, Volume: 130, Issue:3

    Topics: Acetophenones; Animals; Arachidonic Acid; Calcium; Cells, Cultured; Dose-Response Relationship, Drug; Flavanones; Flavonoids; Ibuprofen; Indomethacin; Lipoxygenase Inhibitors; Masoprocol; Parathyroid Glands; Parathyroid Hormone; Phospholipases A; Phospholipases A2; Pyrazoles; Quinacrine; Swine; Time Factors; Tritium

1992
Modulation of the beta-adrenergic response in cultured rat heart cells. I. Beta-adrenergic supersensitivity is induced by lactate via a phospholipase A2 and 15-lipoxygenase involving pathway.
    Molecular and cellular biochemistry, 1991, Mar-27, Volume: 102, Issue:1

    Topics: Acetophenones; Animals; Arachidonic Acid; Arachidonic Acids; Cells, Cultured; Chronobiology Phenomena; Dose-Response Relationship, Drug; Enzyme Activation; Heart; Hydroxyeicosatetraenoic Acids; Isoproterenol; Lactates; Leukotrienes; Melitten; Phospholipases A; Phospholipases A2; Prostaglandins D; Quinacrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1991
Arachidonic acid is essential for IgG Fc receptor-mediated phagocytosis by human monocytes.
    Journal of immunology (Baltimore, Md. : 1950), 1991, Jul-15, Volume: 147, Issue:2

    Topics: Acetophenones; Antigen-Antibody Complex; Antigens, Differentiation; Arachidonic Acid; Arachidonic Acids; Complement C3b; Eicosanoids; Humans; Immunoglobulin G; In Vitro Techniques; Monocytes; Phagocytosis; Phospholipases; Quinacrine; Receptors, Fc; Receptors, IgG; Signal Transduction; Structure-Activity Relationship; Terpenes; Yeasts

1991
Arachidonic acid metabolites as mediators of somatostatin-induced increase of neuronal M-current.
    Nature, 1990, Aug-02, Volume: 346, Issue:6283

    Topics: Acetophenones; Action Potentials; Animals; Arachidonic Acid; Arachidonic Acids; Cyclooxygenase Inhibitors; Electric Conductivity; Hippocampus; Lipoxygenase; Lipoxygenase Inhibitors; Masoprocol; Membrane Potentials; Neurons; Phospholipases A; Phospholipases A2; Potassium; Quinacrine; Rats; Second Messenger Systems; Somatostatin; SRS-A

1990
Phospholipase A activity in seminal plasma of men attending an infertility clinic.
    Urologia internationalis, 1991, Volume: 46, Issue:2

    Topics: Acetophenones; Dibucaine; Humans; Infertility, Male; Male; Oligospermia; Phospholipases A; Quinacrine; Semen; Sperm Count; Triglycerides; Zinc

1991
Phospholipase A2 activation and autoinduction of tumor necrosis factor gene expression by tumor necrosis factor.
    Cancer research, 1990, Nov-15, Volume: 50, Issue:22

    Topics: Acetophenones; Arachidonic Acid; Arachidonic Acids; Blotting, Northern; Choline; Enzyme Activation; Gene Expression Regulation, Neoplastic; Humans; In Vitro Techniques; Inositol Phosphates; Leukemia, Myeloid; Lipoxygenase Inhibitors; Lysophosphatidylcholines; Phospholipases A; Phospholipases A2; Precipitin Tests; Quinacrine; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha; Type C Phospholipases

1990
Effects of lipopolysaccharide on phospholipase A2 activity and tumor necrosis factor expression in HL-60 cells.
    Journal of immunology (Baltimore, Md. : 1950), 1990, Apr-01, Volume: 144, Issue:7

    Topics: Acetophenones; Bucladesine; Dinoprostone; Enzyme Activation; Gene Expression; Ketoconazole; Leukocytes, Mononuclear; Lipopolysaccharides; Masoprocol; Melitten; Phospholipases; Phospholipases A; Phospholipases A2; Protein Kinase C; Quinacrine; RNA, Messenger; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha

1990
Evidence for the involvement of phospholipase A2 in the regulation of luteinizing hormone-stimulated steroidogenesis in rat testis Leydig cells.
    Molecular and cellular endocrinology, 1990, Apr-17, Volume: 70, Issue:2

    Topics: Acetophenones; Animals; Arachidonic Acids; Bucladesine; Colforsin; Cyclic AMP; Dexamethasone; Hydroxycholesterols; Leydig Cells; Luteinizing Hormone; Male; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Inbred Strains; Testosterone

1990
Characterization and inhibitor sensitivity of human sperm phospholipase A2: evidence against pivotal involvement of phospholipase A2 in the acrosome reaction.
    Molecular reproduction and development, 1990, Volume: 27, Issue:4

    Topics: 1,2-Dipalmitoylphosphatidylcholine; Acetophenones; Acrosome; Adult; Calcium; Deoxycholic Acid; Dimethyl Sulfoxide; Humans; Hydrogen-Ion Concentration; Kinetics; Lysophosphatidylcholines; Male; Phospholipases A; Phospholipases A2; Quinacrine; Spermatozoa; Temperature; Trifluoperazine

1990
Effects of mepacrine and p-bromophenacyl bromide on anti-IgE and phospholipase A2-induced histamine release from human basophils.
    Agents and actions, 1986, Volume: 18, Issue:5-6

    Topics: Acetophenones; Antibodies, Anti-Idiotypic; Basophils; Calcium; Histamine Release; Humans; Immunoglobulin E; Kinetics; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine

1986
Regulation of gamma-aminobutyric acid/barbiturate receptor-gated chloride ion flux in brain vesicles by phospholipase A2: possible role of oxygen radicals.
    Journal of neurochemistry, 1988, Volume: 50, Issue:2

    Topics: Acetophenones; Animals; Brain; Chlorides; Fatty Acids; Free Radicals; Ion Channels; Male; Oxygen; Pentobarbital; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Neurotransmitter; Serum Albumin, Bovine; Superoxide Dismutase; Synaptosomes; Xanthine; Xanthine Oxidase; Xanthines

1988
Pharmacological study of phospholipase A2-induced histamine release from rat peritoneal mast cells.
    Journal of pharmacobio-dynamics, 1989, Volume: 12, Issue:9

    Topics: Acetophenones; Animals; Cinnarizine; Cromolyn Sodium; Glucocorticoids; Histamine H1 Antagonists; Histamine Release; In Vitro Techniques; Male; Mast Cells; Nifedipine; ortho-Aminobenzoates; Phospholipases; Phospholipases A; Phospholipases A2; Piperazines; Pyridines; Quinacrine; Rats; Rats, Inbred Strains

1989
Arachidonic acid mobilization and phosphoinositide turnover by the terminal complement complex, C5b-9, in rat oligodendrocyte x C6 glioma cell hybrids.
    Journal of immunology (Baltimore, Md. : 1950), 1989, Jun-15, Volume: 142, Issue:12

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Animals; Arachidonic Acid; Arachidonic Acids; Calcimycin; Calcium; Clone Cells; Complement Membrane Attack Complex; Complement System Proteins; Glioma; Humans; Hybrid Cells; Isoquinolines; Neuroglia; Oligodendroglia; Phosphatidylinositols; Piperazines; Protein Kinase C; Quinacrine; Rats

1989
Superoxide generation is inhibited by phospholipase A2 inhibitors. Role for phospholipase A2 in the activation of the NADPH oxidase.
    The Biochemical journal, 1989, Nov-15, Volume: 264, Issue:1

    Topics: Acetophenones; Amino Alcohols; Arachidonic Acid; Arachidonic Acids; Cell-Free System; Enzyme Activation; Humans; In Vitro Techniques; N-Formylmethionine Leucyl-Phenylalanine; NADH, NADPH Oxidoreductases; NADPH Oxidases; Neutrophils; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Sodium Dodecyl Sulfate; Superoxides; Tetradecanoylphorbol Acetate

1989
The role of phospholipase A2 in microsomal lipid peroxidation induced with t-butyl hydroperoxide.
    Biochemical and biophysical research communications, 1989, Feb-15, Volume: 158, Issue:3

    Topics: Acetophenones; Animals; Chlorpromazine; Enzyme Activation; Fatty Acids; Lipid Peroxidation; Melitten; Microsomes, Liver; Peroxides; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Rats; tert-Butylhydroperoxide; Thiobarbiturates

1989
Regulation of phospholipid synthesis by intracellular phospholipases in fetal rabbit type II pneumocytes.
    Biochimica et biophysica acta, 1985, Mar-06, Volume: 833, Issue:3

    Topics: Acetophenones; Animals; Choline; Choline-Phosphate Cytidylyltransferase; Female; Lung; Nucleotidyltransferases; Palmitic Acid; Palmitic Acids; Phospholipases; Phospholipases A; Phospholipases A2; Phospholipids; Pregnancy; Quinacrine; Rabbits; Time Factors; Type C Phospholipases

1985
Antigen-induced bronchial anaphylaxis in actively sensitized SD rats. Effects of glucocorticoid treatment.
    Allergy, 1986, Volume: 41, Issue:3

    Topics: Acetophenones; Administration, Topical; Alum Compounds; Aluminum; Anaphylaxis; Animals; Antigens; Bronchial Diseases; Budesonide; Cromolyn Sodium; Dexamethasone; Dose-Response Relationship, Drug; Drug Interactions; Glucocorticoids; Immunization; Injections, Intraperitoneal; Injections, Intravenous; Male; Ovalbumin; Pregnenediones; Quinacrine; Rats; Rats, Inbred Strains; Respiration; Sulfates; Time Factors

1986
Possible involvement of the phospholipases in the mitogenic actions of prolactin (PRL) on Nb2 node lymphoma cells.
    Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), 1987, Volume: 185, Issue:2

    Topics: Acetophenones; Animals; Arachidonic Acid; Arachidonic Acids; Cell Division; Cell Line; Lymphoma; Phospholipases; Phospholipases A; Phospholipases A2; Prolactin; Quinacrine; Rats; Stimulation, Chemical; Type C Phospholipases

1987
Mechanism of CO2 response in cerebral arteries of the newborn pig: role of phospholipase, cyclooxygenase, and lipoxygenase pathways.
    Circulation research, 1988, Volume: 62, Issue:5

    Topics: Acetophenones; Animals; Animals, Newborn; Arterioles; Carbon Dioxide; Cerebrovascular Circulation; Indomethacin; Lipoxygenase; Masoprocol; Phospholipases A; Pia Mater; Prostaglandin-Endoperoxide Synthases; Quinacrine; Swine

1988
Selective inhibition of free arachidonic acid production in activated alveolar macrophages by calmodulin antagonists.
    Biochemical and biophysical research communications, 1988, Oct-31, Volume: 156, Issue:2

    Topics: Acetophenones; Animals; Arachidonic Acid; Arachidonic Acids; Calmodulin; Chlorpromazine; Chromatography, High Pressure Liquid; Cytochalasin B; Linoleic Acid; Linoleic Acids; Macrophage Activation; Macrophages; Oleic Acid; Oleic Acids; Opsonin Proteins; Phosphatidylcholines; Phosphatidylinositols; Phospholipases A; Pulmonary Alveoli; Quinacrine; Rabbits; Sulfonamides; Trifluoperazine; Zymosan

1988
The biphasic effect of phospholipase A2 inhibitors on axon elongation.
    International journal of developmental neuroscience : the official journal of the International Society for Developmental Neuroscience, 1986, Volume: 4, Issue:4

    Topics: Acetophenones; Animals; Axons; Cells, Cultured; Enzyme Inhibitors; Ganglia, Spinal; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Inbred Strains; Strontium

1986
Prolactin actions on casein and lipid biosynthesis in mouse and rabbit mammary gland explants are abolished by p-bromphenacyl bromide and quinacrine, phospholipase A2 inhibitors.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 1986, Volume: 18, Issue:10

    Topics: Acetophenones; Animals; Caseins; Lipids; Mammary Glands, Animal; Mice; Phospholipases A; Phospholipases A2; Prolactin; Quinacrine; Rabbits

1986
The role of phospholipase A activity in rat liver microsomal lipid peroxidation.
    The Journal of biological chemistry, 1987, Feb-05, Volume: 262, Issue:4

    Topics: Acetophenones; Adenosine Diphosphate; Alloxan; Animals; Chlorpromazine; Copper; Ferrous Compounds; Glutathione; Hydrogen-Ion Concentration; Lipid Peroxides; Male; Microsomes, Liver; Phospholipases; Phospholipases A; Phospholipases A1; Phospholipases A2; Quinacrine; Rats; Rats, Inbred Strains

1987
Possible role of phospholipase A2 action and arachidonic acid metabolism in angiotensin II-mediated aldosterone secretion.
    Endocrinology, 1985, Volume: 117, Issue:3

    Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; 5,8,11,14-Eicosatetraynoic Acid; Acetophenones; Aldosterone; Angiotensin II; Animals; Arachidonic Acid; Arachidonic Acids; Caffeic Acids; Calcium; Cattle; Cyclooxygenase Inhibitors; Dantrolene; Dose-Response Relationship, Drug; Indomethacin; Lipoxygenase Inhibitors; Phospholipases; Phospholipases A; Phospholipases A2; Pyrazoles; Quinacrine

1985
Effect of diarachidonin on prostaglandin E2 synthesis in rabbit kidney medulla slices.
    The Biochemical journal, 1985, Dec-15, Volume: 232, Issue:3

    Topics: Acetophenones; Animals; Arachidonic Acid; Arachidonic Acids; Diglycerides; Dinoprostone; Dose-Response Relationship, Drug; Egtazic Acid; Glycerides; In Vitro Techniques; Kidney Medulla; Male; Phosphatidic Acids; Prostaglandins E; Quinacrine; Rabbits

1985
Inhibition by mepacrine and p-bromophenacylbromide of phosphoinositide hydrolysis, glucose oxidation, calcium uptake and insulin release in rat pancreatic islets.
    Biochemical pharmacology, 1984, Aug-15, Volume: 33, Issue:16

    Topics: Acetophenones; Animals; Calcium; Dose-Response Relationship, Drug; Glucose; Hydrolysis; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Oxidation-Reduction; Phosphatidylinositols; Quinacrine; Rats; Rubidium; Type C Phospholipases

1984
The number of the Trf receptors on human hematopoietic cell lines is influenced by membrane phospholipids.
    Biochemistry international, 1983, Volume: 7, Issue:2

    Topics: Acetophenones; Cell Line; Cell Membrane; Humans; Kinetics; Leukemia, Myeloid, Acute; Membrane Lipids; Phospholipases; Phospholipids; Quinacrine; Receptors, Cell Surface; Receptors, Transferrin; Tetracaine; Transferrin

1983
Possible role of phospholipase A2 in triggering histamine secretion from human basophils in vitro.
    Clinical immunology and immunopathology, 1981, Volume: 20, Issue:2

    Topics: Acetophenones; Arachidonic Acids; Basophils; Calcium; Edetic Acid; Histamine Release; Humans; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine

1981
Mechanisms involved in the synthesis of disaturated phosphatidylcholine by alveolar type II cells isolated from adult rat lung.
    Biochimica et biophysica acta, 1983, Jan-07, Volume: 750, Issue:1

    Topics: Acetophenones; Animals; Cell Membrane; Diacylglycerol Cholinephosphotransferase; Ethanolaminephosphotransferase; Glycerol; Kinetics; Lung; Male; Phosphatidylcholines; Quinacrine; Rats; Rats, Inbred Strains

1983
Prevention of catecholamine release from adrenal chromaffin cells by phospholipase A2- and lipoxygenase-inhibitors.
    Japanese journal of pharmacology, 1983, Volume: 33, Issue:5

    Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Acetophenones; Adrenal Medulla; Animals; Arachidonic Acids; Aspirin; Catecholamines; Cattle; Chromaffin System; In Vitro Techniques; Lipoxygenase Inhibitors; Phospholipases; Phospholipases A; Phospholipases A2; Pyrazoles; Quinacrine

1983
Assessment of a role for phospholipase A2 and arachidonic acid metabolism in human lymphocyte natural cytotoxicity.
    Cellular immunology, 1984, Volume: 87, Issue:1

    Topics: Acetophenones; Arachidonic Acid; Arachidonic Acids; Binding, Competitive; Cyclooxygenase Inhibitors; Cytotoxicity, Immunologic; Dexamethasone; Humans; Hydrocortisone; Killer Cells, Natural; Kinetics; Lipoxygenase Inhibitors; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine

1984
Improvement of the anoxia-induced mitochondrial dysfunction by membrane modulation.
    Archives of biochemistry and biophysics, 1984, Aug-15, Volume: 233, Issue:1

    Topics: Acetophenones; Adenine Nucleotides; Alkaloids; Animals; Benzylisoquinolines; Chlorpromazine; Egtazic Acid; Hypoxia; Kinetics; Male; Mitochondria, Liver; Mitochondrial Swelling; Oxidative Phosphorylation; Oxygen Consumption; Phospholipids; Quinacrine; Rats; Rats, Inbred Strains

1984
Stimulation of prostaglandin E2 synthesis by exogenous phospholipase A2 and C in rabbit kidney medulla slices.
    The Biochemical journal, 1984, Feb-15, Volume: 218, Issue:1

    Topics: Acetophenones; Animals; Dinoprostone; Fatty Acids; In Vitro Techniques; Kidney Medulla; Lipolysis; Male; Phospholipases; Phospholipases A; Phospholipases A2; Prostaglandins E; Quinacrine; Rabbits; Stimulation, Chemical; Type C Phospholipases

1984
Calmodulin, phospholipase, and exocytosis. p-Bromophenacyl bromide inhibits but mepacrine stimulates secretion in rat mast cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 324, Issue:1

    Topics: Acetophenones; Animals; Calcium; Calmodulin; Exocytosis; In Vitro Techniques; Male; Mast Cells; Phenothiazines; Phospholipases; Quinacrine; Rats; Rats, Inbred Strains

1983
How a nerve fiber repairs its cut end: involvement of phospholipase A2.
    Science (New York, N.Y.), 1983, Dec-23, Volume: 222, Issue:4630

    Topics: Acetophenones; Animals; Axons; Calcium; Cell Membrane; Denervation; Enzyme Activation; Membrane Potentials; Periplaneta; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Temperature

1983
The effects of mepacrine and p-bromophenacyl bromide on arachidonic acid release in human platelets.
    Archives of biochemistry and biophysics, 1982, Apr-15, Volume: 215, Issue:1

    Topics: Acetophenones; Arachidonic Acid; Arachidonic Acids; Blood Platelets; Dose-Response Relationship, Drug; Humans; Quinacrine; Serotonin; Thrombin; Type C Phospholipases

1982
Studies on the incorporation of [1-14C]arachidonic acid into glycerolipids and its conversion into prostaglandins by rabbit iris. Effects of anti-inflammatory drugs and phospholipase A2 inhibitors.
    Biochimica et biophysica acta, 1982, Jun-11, Volume: 711, Issue:3

    Topics: Acetophenones; Animals; Anti-Inflammatory Agents; Arachidonic Acid; Arachidonic Acids; Aspirin; Diglycerides; Female; Indomethacin; Iris; Lipid Metabolism; Male; Microsomes; Muscle, Smooth; Phospholipases; Phospholipases A; Phospholipases A2; Phospholipids; Prostaglandins; Quinacrine; Rabbits; Triglycerides

1982
Suppression by phospholipase A2 inhibitors of secretion of catecholamines from isolated adrenal medullary cells by suppression of cellular calcium uptake.
    Biochemical pharmacology, 1983, Apr-01, Volume: 32, Issue:7

    Topics: Acetophenones; Adrenal Medulla; Animals; Calcium; Carbachol; Catecholamines; Cattle; Chloroquine; Dose-Response Relationship, Drug; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Quinine

1983
Phospholipase A2 inhibitors block catecholamine secretion and calcium uptake in cultured bovine adrenal medullary cells.
    Molecular pharmacology, 1983, Volume: 23, Issue:3

    Topics: Acetophenones; Adrenal Medulla; Animals; Biological Transport, Active; Calcium; Catecholamines; Cattle; Cells, Cultured; Exocytosis; Kinetics; Phospholipases; Phospholipases A; Phospholipases A2; Propanolamines; Quinacrine

1983
Phospholipase A2 inhibitors. Differential inhibition of fatty acid acylation into kidney lipids by mepacrine and p-bromophenacyl bromide.
    Biochemical pharmacology, 1983, Jul-01, Volume: 32, Issue:13

    Topics: Acetophenones; Acylation; Animals; Arachidonic Acids; Fatty Acids; In Vitro Techniques; Kidney Medulla; Linoleic Acids; Lipid Metabolism; Male; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Rabbits; Stearic Acids

1983
Intraventricular injections of drugs which inhibit phospholipase A2 suppress fever in rabbits.
    The Journal of physiology, 1983, Volume: 339

    Topics: Acetophenones; Animals; Arachidonic Acids; Body Temperature Regulation; Fever; Injections, Intravenous; Injections, Intraventricular; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Rabbits

1983
Inhibitors of 125I-epidermal growth factor internalization.
    Biochemical and biophysical research communications, 1980, May-30, Volume: 94, Issue:2

    Topics: Acetophenones; Animals; Azo Compounds; Bacitracin; Cells, Cultured; Chlorpromazine; Endocytosis; Epidermal Growth Factor; Methylamines; Peptides; Phenylglyoxal; Phospholipases; Phospholipases A; Quinacrine; Rats

1980
Effects of phospholipase A2 inhibitors on the antidepressant-induced axonal regeneration of noradrenergic locus coeruleus neurons.
    Microscopy research and technique, 1994, Oct-15, Volume: 29, Issue:3

    Topics: Acetophenones; Adrenergic Fibers; Animals; Antidepressive Agents; Axons; Fluorescence; Immunohistochemistry; Locus Coeruleus; Microscopy, Electron; Nerve Regeneration; Neurons; Norepinephrine; Oxidopamine; Phospholipases A; Phospholipases A2; Quinacrine; Rats

1994
On the role of arachidonic acid in M-current modulation by muscarine in bullfrog sympathetic neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1994, Volume: 14, Issue:11 Pt 2

    Topics: Acetophenones; Animals; Arachidonic Acid; Dose-Response Relationship, Drug; Ganglia, Sympathetic; Gonadotropin-Releasing Hormone; In Vitro Techniques; Kinetics; Masoprocol; Membrane Potentials; Muscarine; Neurons; Phospholipases A; Phospholipases A2; Potassium Channels; Quinacrine; Rana catesbeiana

1994
Evidence for a role of phospholipase A2 in the mechanism of LHRH priming in rat anterior pituitary tissue.
    The Journal of endocrinology, 1994, Volume: 141, Issue:1

    Topics: Acetophenones; Aminobenzoates; Animals; Arachidonic Acid; Aristolochic Acids; Calcium; Chlorobenzoates; Cinnamates; Cycloheximide; Female; Gonadotropin-Releasing Hormone; In Vitro Techniques; Luteinizing Hormone; ortho-Aminobenzoates; Phenanthrenes; Phenothiazines; Phospholipases A; Phospholipases A2; Pituitary Gland, Anterior; Proestrus; Quinacrine; Rats; Rats, Wistar

1994
The requirement for phospholipase A2 for activation of the assembled NADPH oxidase in human neutrophils.
    The Biochemical journal, 1994, Jan-01, Volume: 297 ( Pt 1)

    Topics: Acetophenones; Alkaloids; Arachidonic Acid; Biological Transport; Cell Membrane; Enzyme Activation; Humans; NADH, NADPH Oxidoreductases; NADPH Oxidases; Neutrophils; Opsonin Proteins; Phospholipases A; Phospholipases A2; Phosphorylation; Protein Kinase C; Quinacrine; Staurosporine; Superoxides; Tetradecanoylphorbol Acetate; Tritium; Zymosan

1994
Regulation of human eosinophil degranulation and activation by endogenous phospholipase A2.
    The Journal of clinical investigation, 1993, Volume: 91, Issue:5

    Topics: Acetophenones; Arachidonic Acid; Cell Separation; Centrifugation, Density Gradient; Cytochalasin B; Dose-Response Relationship, Drug; Eosinophil Peroxidase; Eosinophils; Homeostasis; In Vitro Techniques; Kinetics; N-Formylmethionine Leucyl-Phenylalanine; Peroxidases; Phospholipases A; Phospholipases A2; Quinacrine; SRS-A; Superoxides

1993
Effect of putative phospholipase A2 inhibitors on acetic acid-induced acute colitis in the rat.
    The British journal of surgery, 1993, Volume: 80, Issue:9

    Topics: Acetates; Acetic Acid; Acetophenones; Animals; Colitis; Colon; Enzyme Activation; Female; Intestinal Mucosa; Peroxidase; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Sprague-Dawley; Verapamil

1993
Eicosanoid production by mouse peritoneal macrophages during Toxoplasma gondii penetration: role of parasite and host cell phospholipases.
    Infection and immunity, 1993, Volume: 61, Issue:4

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Animals; Arachidonic Acid; Calcium; Cyclooxygenase Inhibitors; Eicosanoids; Female; Indomethacin; Isoquinolines; Lipoxygenase; Macrophages; Mice; Peritoneal Cavity; Phospholipases; Piperazines; Prostaglandin-Endoperoxide Synthases; Protein Kinase C; Quinacrine; Toxoplasma; Toxoplasmosis, Animal

1993
Botulinum toxin inhibits arachidonic acid release associated with acetylcholine release from PC12 cells.
    The Journal of biological chemistry, 1993, May-25, Volume: 268, Issue:15

    Topics: Acetophenones; Acetylcholine; Animals; Arachidonic Acid; Botulinum Toxins; Cell Differentiation; Dose-Response Relationship, Drug; Ethacrynic Acid; Indomethacin; Kinetics; Masoprocol; Melitten; Models, Biological; Nerve Growth Factors; PC12 Cells; Phospholipases A; Phospholipases A2; Potassium; Protein Kinase C; Quinacrine; Terpenes

1993
Differences in the acute actions of sGnRH and cGnRH-II on gonadotropin release in goldfish pituitary cells.
    General and comparative endocrinology, 1995, Volume: 100, Issue:3

    Topics: Acetophenones; Analysis of Variance; Animals; Calcium Channel Blockers; Cells, Cultured; Enzyme Inhibitors; Female; Goldfish; Gonadotropin-Releasing Hormone; Gonadotropins; Male; Masoprocol; Pituitary Gland; Quinacrine; Verapamil

1995
Inhibition of HIV-1 Tat-mediated transactivation by quinacrine and chloroquine.
    Biochemical and biophysical research communications, 1996, Sep-04, Volume: 226, Issue:1

    Topics: Acetophenones; Alkaloids; Antimalarials; Benzoquinones; Cell Line; Cell Survival; Chloroquine; Curcumin; Gene Expression Regulation, Viral; Gene Products, tat; HIV Long Terminal Repeat; HIV-1; Humans; Lactams, Macrocyclic; Quinacrine; Quinones; Rifabutin; Staurosporine; tat Gene Products, Human Immunodeficiency Virus; Transcriptional Activation; Tumor Cells, Cultured; Virus Replication

1996
Modulation of 8-methoxypsoralen-photoinduced cutaneous inflammatory reactions by various chemotherapeutic agents in vivo.
    Photochemistry and photobiology, 1996, Volume: 63, Issue:4

    Topics: Acetophenones; Animals; Capillary Permeability; Erythema; Ibuprofen; Indoles; Indomethacin; Masoprocol; Methoxsalen; Neutrophils; PUVA Therapy; Quinacrine; Rabbits; Skin

1996
PLA2 activity in Tetrahymena pyriformis. Effects of inhibitors and stimulators.
    Journal of lipid mediators and cell signalling, 1997, Volume: 15, Issue:3

    Topics: Acetophenones; Aluminum Compounds; Animals; Arachidonic Acid; Calcium; Enzyme Activation; Enzyme Inhibitors; Fluorides; Hydrogen Peroxide; Inositol; Lithium Chloride; Melitten; Phorbol 12,13-Dibutyrate; Phosphatidylinositols; Phospholipases A; Phospholipases A2; Phospholipids; Protein-Tyrosine Kinases; Quinacrine; Signal Transduction; Sodium Fluoride; Tetrahymena pyriformis; Vanadates

1997
Increased PLA2 activity is not related to increase GLUT1 expression in L6 myotubes under hypoxic conditions.
    Prostaglandins, leukotrienes, and essential fatty acids, 1997, Volume: 56, Issue:1

    Topics: Acetophenones; Animals; Arachidonic Acid; Biological Transport; Cell Hypoxia; Cell Line; Cyclooxygenase Inhibitors; Deoxyglucose; Glucose; Glucose Transporter Type 1; Glucose Transporter Type 4; Insulin; Membrane Proteins; Monosaccharide Transport Proteins; Muscle Proteins; Muscle, Skeletal; Phospholipases A; Phospholipases A2; Prostaglandins; Quinacrine; Rats; Signal Transduction

1997
Phospholipases and arachidonic acid contribute independently to sensory transduction and associative neuronal facilitation in Hermissenda type B photoreceptors.
    Brain research, 1997, Mar-21, Volume: 751, Issue:2

    Topics: Acetophenones; Animals; Arachidonic Acid; Association Learning; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Indomethacin; Lipoxygenase Inhibitors; Masoprocol; Mollusca; Neurons; Phospholipases; Photoreceptor Cells, Invertebrate; Quinacrine; Sensation; Signal Transduction

1997
Structure-activity of three phospholipid analogues towards inhibition of phospholipase A2 in macrophages.
    Pharmacological research, 1997, Volume: 35, Issue:1

    Topics: Acetophenones; Animals; Anti-Inflammatory Agents; Cells, Cultured; Culture Media; Dexamethasone; Eicosanoids; Enzyme Inhibitors; Macrophages, Peritoneal; Male; Phospholipases A; Phospholipases A2; Phospholipids; Quinacrine; Rats; Structure-Activity Relationship; Tritium

1997
Influence of nicotine and cotinine on retinal phospholipase A2 and its significance to macular function.
    Journal of ocular pharmacology and therapeutics : the official journal of the Association for Ocular Pharmacology and Therapeutics, 1998, Volume: 14, Issue:5

    Topics: Acetophenones; Acetylcholine; Animals; Cotinine; Enzyme Inhibitors; Macular Degeneration; Nicotine; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Inbred F344; Retina

1998
Involvement of phospholipase A2 activation in anthrax lethal toxin-induced cytotoxicity.
    Cell biology and toxicology, 1999, Volume: 15, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 4-Aminobenzoic Acid; Acetophenones; Aminobenzoates; Animals; Anthrax; Antigens, Bacterial; Antioxidants; Apoptosis; Bacterial Toxins; Cells, Cultured; Dehydroepiandrosterone; DNA Fragmentation; Enzyme Activation; Enzyme Inhibitors; Macrophages, Peritoneal; Melatonin; Mice; Mice, Inbred ICR; Nitric Oxide; para-Aminobenzoates; Phosphodiesterase Inhibitors; Phospholipases A; Phospholipases A2; Protein Kinase Inhibitors; Quinacrine; Reactive Oxygen Species; Staurosporine; Terpenes

1999
Lysophosphatidylcholine and arachidonic acid are required in the cytotoxic response of human natural killer cells to tumor target cells.
    Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology, 1999, Volume: 9, Issue:6

    Topics: Acetophenones; Arachidonic Acid; Cytotoxicity, Immunologic; Enzyme Inhibitors; Humans; K562 Cells; Killer Cells, Natural; Leukotrienes; Linoleic Acid; Lipid Peroxides; Lysophosphatidylcholines; Phospholipases A; Quinacrine

1999
Calcium-dependent mitochondrial formation of species promoting strand scission of genomic DNA in U937 cells exposed to tert-butylhydroperoxide: the role of arachidonic acid.
    Free radical research, 2000, Volume: 33, Issue:5

    Topics: 5,8,11,14-Eicosatetraynoic Acid; Acetophenones; Antimycin A; Arachidonic Acid; Calcium; DNA Damage; Electron Transport; Enzyme Inhibitors; Humans; Melitten; Mitochondria; Phospholipases A; Phospholipases A2; Quinacrine; tert-Butylhydroperoxide; U937 Cells

2000
Effect of quinacrine treatment on the activity of acid hydrolases (phosphatase, N-acetyl-beta-glucosaminidase, glucosidase, galactosidase and esterase) in Tetrahymena.
    Cell biochemistry and function, 2001, Volume: 19, Issue:4

    Topics: Acetophenones; Acetylglucosaminidase; Acid Phosphatase; Animals; Antimalarials; Cell Fractionation; Enzyme Inhibitors; Esterases; Galactosidases; Glucosidases; Hydrolases; Quinacrine; Tetrahymena pyriformis

2001
Arachidonic acid release from rat Leydig cells: the involvement of G protein, phospholipase A2 and regulation of cAMP production.
    The Journal of endocrinology, 2002, Volume: 172, Issue:1

    Topics: Acetophenones; Animals; Arachidonic Acid; Chorionic Gonadotropin; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Leydig Cells; Male; Melitten; Pertussis Toxin; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Inbred Strains; Stimulation, Chemical; Virulence Factors, Bordetella

2002
4-Bromophenacyl bromide induces Ca2+ influx in human gingival fibroblasts.
    Comparative biochemistry and physiology. Toxicology & pharmacology : CBP, 2002, Volume: 131, Issue:3

    Topics: Acetophenones; Aniline Compounds; Arachidonic Acids; Bradykinin; Calcium; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fibroblasts; Fluorescent Dyes; Gingiva; Histamine; Humans; Kinetics; Phospholipases A; Phospholipases A2; Quinacrine; Spectrometry, Fluorescence; Structure-Activity Relationship; Terpenes; Xanthenes

2002
Quaternary-Ammonium-Modulated Surface-Enhanced Raman Spectroscopy Effect: Discovery, Mechanism, and Application for Highly Sensitive
    Analytical chemistry, 2020, 07-21, Volume: 92, Issue:14

    Topics: Acetophenones; Acetylcholine; Animals; Microfluidic Analytical Techniques; PC12 Cells; Quaternary Ammonium Compounds; Quinacrine; Rats; Spectrum Analysis, Raman

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