quinacrine has been researched along with 4-bromophenacyl bromide in 69 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 34 (49.28) | 18.7374 |
1990's | 30 (43.48) | 18.2507 |
2000's | 4 (5.80) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 1 (1.45) | 2.80 |
Authors | Studies |
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Fujii, T; Hashizume, T; Sato, T | 1 |
Larsson, C; Mau, S; Saermark, T; Simonsson, P | 1 |
Bonnet, P; Bourdeau, A; Herviaux, P; Lieberherr, M; Sachs, C; Souberbielle, JC | 1 |
Farkas, T; Kuehn, H; Nemecz, G; Wallukat, G; Wollenberger, A | 1 |
Brown, EJ; Lennartz, MR | 1 |
Madamba, S; Schweitzer, P; Siggins, GR | 1 |
Frithz, G; Jansson, A; Ronquist, G | 1 |
Imamura, K; Kufe, DW; Mohri, M; Robbins, G; Rodriguez, C; Sherman, ML; Spriggs, DR | 1 |
Kufe, D; Mohri, M; Spriggs, DR | 1 |
Abayasekara, DR; Band, AM; Cooke, BA | 1 |
Dennis, EA; Glaser, KB; Lister, MD; Ulevitch, RJ | 1 |
Anderson, RA; Bielfeld, P; Feathergill, KA; Johnson, SK; Zaneveld, LJ | 1 |
Andersson, RG; Toll, JB | 1 |
Paul, SM; Schwartz, RD; Skolnick, P | 1 |
Choi, SH; Fukutomi, O; Inagaki, N; Koda, A; Matsuura, N; Nagai, H; Sakamoto, T | 1 |
McMorris, FA; Shin, ML; Shirazi, Y | 1 |
Chappell, JB; Henderson, LM; Jones, OT | 1 |
Borowitz, SM; Montgomery, C | 1 |
Aeberhard, EE; Barrett, CT; Kaplan, SA; Scott, ML | 1 |
Bergstrand, H; Brattsand, R; Dahlbäck, M | 1 |
Ofenstein, JP; Rillema, JA | 1 |
Mishra, OP; Wagerle, LC | 1 |
Nakagawa, Y; Waku, K | 1 |
Cei de Job, C; Suburo, A | 1 |
Cameron, CM; Etindi, RN; Rillema, JA | 1 |
Beckman, JK; Borowitz, SM; Burr, IM | 1 |
Kojima, I; Kojima, K; Rasmussen, H | 1 |
Fujimoto, Y; Fujita, T; Kagen, C; Ueno, T; Uno, H | 1 |
Best, L; Malaisse, WJ; Mathias, PC; Sener, A | 1 |
Pelicci, PG; Rochant, H; Testa, U; Thomopoulos, P; Titeux, M | 1 |
Kagey-Sobotka, A; Lichtenstein, LM; Marone, G | 1 |
Furchgott, RF | 1 |
Batenburg, JJ; Post, M; Schuurmans, EA; Van Golde, LM | 1 |
Kato, R; Kumakura, K; Sasakawa, N; Yamamoto, S | 1 |
Carine, K; Hudig, D | 1 |
Kodama, H; Mikasa, H; Miyahara, M; Okimasu, E; Terada, S; Utsumi, K | 1 |
Akamatsu, N; Fujimoto, Y; Fujita, T; Hattori, A | 1 |
Douglas, WW; Nemeth, EF | 1 |
Kuno, M; Yawo, H | 1 |
Hofmann, SL; Majerus, PW; Prescott, SM | 1 |
Abdel-Latif, AA; Smith, JP | 1 |
Izumi, F; Kobayashi, H; Sakurai, S; Wada, A; Yanagihara, N | 1 |
Frye, RA; Holz, RW | 1 |
Azuri, R; Erman, A; Raz, A | 1 |
Cranston, WI; Hellon, RF; Mitchell, D; Townsend, Y | 1 |
Haigler, HT; Pastan, I; Willingham, MC | 1 |
Nakamura, S | 1 |
Villarroel, A | 1 |
Johnson, MS; Mitchell, R; Thomson, FJ; Wolbers, B | 1 |
Dana, R; Levy, R; Malech, HL | 1 |
Burch, RA; Kulp, GV; Leff, AR; Neeley, SP; Spaethe, SM; Strek, ME; White, SR | 1 |
Andersson, R; Ar'Rajab, A; Bengmark, S; Fabia, R; Willén, R | 1 |
Beraud, M; Bessieres, MH; Frisach, MF; M'Rini, C; Pipy, B; Seguela, JP; Thardin, JF; Vandaele, J | 1 |
Berman, JD; Brendle, J; Middleton, W; Ray, P | 1 |
Chang, JP; Garofalo, R; Neumann, CM | 1 |
Chen, SS; Jiang, MC; Lin, JK | 1 |
Haberman, HF; Kumar, JR; Ranadive, NS | 1 |
Csaba, G; Kovács, P | 2 |
Bashan, N; Kozlovsky, N; Shohami, E | 1 |
Matzel, LD; Muzzio, IA; Talk, AC | 1 |
Boucrot, P; Bourass, J; Elkihel, L; Letourneux, Y; Petit, JY | 1 |
Hemontolor, ME; Sastry, BV | 1 |
Hur, GH; Kim, YB; Shin, S | 1 |
Bader, BW; Bankhurst, AD; Doshi, RN; Whalen, MM | 1 |
Cantoni, O; Fiorani, M; Guidarelli, A | 1 |
Llanos, MN; Moraga, PF; Ronco, AM | 1 |
Furuyama, S; Kuboyama, N; Moriwaki, K; Nakao, S; Ogata, Y; Sakurai, T; Sugiya, H | 1 |
Cui, Y; Li, L; Lu, Y; Qian, Z; Wang, Z; Yang, K; Zhang, Y; Zhu, K; Zong, S | 1 |
2 review(s) available for quinacrine and 4-bromophenacyl bromide
Article | Year |
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Macrophage phospholipase A2 activity and eicosanoid production: studies with phospholipase A2 inhibitors in P388D1 cells.
Topics: Acetophenones; Animals; Cell Line; Eicosanoids; Fatty Acids; Macrophages; Mice; Phospholipases A; Phospholipases A2; Quinacrine; Substrate Specificity; Terpenes | 1990 |
The role of endothelium in the responses of vascular smooth muscle to drugs.
Topics: 5,8,11,14-Eicosatetraynoic Acid; Acetophenones; Acetylcholine; Adenosine Diphosphate; Adenosine Triphosphate; Animals; Arachidonic Acid; Arachidonic Acids; Bradykinin; Calcimycin; Catechols; Endothelium; Histamine; Hydroquinones; Hypoxia; Masoprocol; Methylene Blue; Muscle Relaxation; Muscle, Smooth, Vascular; Prostaglandins; Quinacrine; Serotonin; Substance P; Thrombin | 1984 |
67 other study(ies) available for quinacrine and 4-bromophenacyl bromide
Article | Year |
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Preferential activation of phospholipase A2 by low concentrations of phosphatidic acid with long-chain fatty acids in rabbit platelets.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Acetophenones; Animals; Blood Platelets; Cytosol; Enzyme Activation; Kinetics; Phosphatidic Acids; Phospholipases A; Phospholipases A2; Platelet Aggregation; Quinacrine; Rabbits | 1992 |
Activation of protein kinase C in permeabilized human neuroblastoma SH-SY5Y cells.
Topics: Acetophenones; Amino Acid Sequence; Arachidonic Acids; Calcium; Cell Membrane; Cell Membrane Permeability; Digitonin; Diglycerides; Dose-Response Relationship, Drug; Enzyme Activation; Humans; Molecular Sequence Data; Myelin Basic Protein; Neuroblastoma; Phospholipases A; Phospholipases A2; Phosphorus; Phosphorus Radioisotopes; Phosphorylation; Protein Kinase C; Quinacrine; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 1992 |
Phospholipase-A2 action and arachidonic acid metabolism in calcium-mediated parathyroid hormone secretion.
Topics: Acetophenones; Animals; Arachidonic Acid; Calcium; Cells, Cultured; Dose-Response Relationship, Drug; Flavanones; Flavonoids; Ibuprofen; Indomethacin; Lipoxygenase Inhibitors; Masoprocol; Parathyroid Glands; Parathyroid Hormone; Phospholipases A; Phospholipases A2; Pyrazoles; Quinacrine; Swine; Time Factors; Tritium | 1992 |
Modulation of the beta-adrenergic response in cultured rat heart cells. I. Beta-adrenergic supersensitivity is induced by lactate via a phospholipase A2 and 15-lipoxygenase involving pathway.
Topics: Acetophenones; Animals; Arachidonic Acid; Arachidonic Acids; Cells, Cultured; Chronobiology Phenomena; Dose-Response Relationship, Drug; Enzyme Activation; Heart; Hydroxyeicosatetraenoic Acids; Isoproterenol; Lactates; Leukotrienes; Melitten; Phospholipases A; Phospholipases A2; Prostaglandins D; Quinacrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1991 |
Arachidonic acid is essential for IgG Fc receptor-mediated phagocytosis by human monocytes.
Topics: Acetophenones; Antigen-Antibody Complex; Antigens, Differentiation; Arachidonic Acid; Arachidonic Acids; Complement C3b; Eicosanoids; Humans; Immunoglobulin G; In Vitro Techniques; Monocytes; Phagocytosis; Phospholipases; Quinacrine; Receptors, Fc; Receptors, IgG; Signal Transduction; Structure-Activity Relationship; Terpenes; Yeasts | 1991 |
Arachidonic acid metabolites as mediators of somatostatin-induced increase of neuronal M-current.
Topics: Acetophenones; Action Potentials; Animals; Arachidonic Acid; Arachidonic Acids; Cyclooxygenase Inhibitors; Electric Conductivity; Hippocampus; Lipoxygenase; Lipoxygenase Inhibitors; Masoprocol; Membrane Potentials; Neurons; Phospholipases A; Phospholipases A2; Potassium; Quinacrine; Rats; Second Messenger Systems; Somatostatin; SRS-A | 1990 |
Phospholipase A activity in seminal plasma of men attending an infertility clinic.
Topics: Acetophenones; Dibucaine; Humans; Infertility, Male; Male; Oligospermia; Phospholipases A; Quinacrine; Semen; Sperm Count; Triglycerides; Zinc | 1991 |
Phospholipase A2 activation and autoinduction of tumor necrosis factor gene expression by tumor necrosis factor.
Topics: Acetophenones; Arachidonic Acid; Arachidonic Acids; Blotting, Northern; Choline; Enzyme Activation; Gene Expression Regulation, Neoplastic; Humans; In Vitro Techniques; Inositol Phosphates; Leukemia, Myeloid; Lipoxygenase Inhibitors; Lysophosphatidylcholines; Phospholipases A; Phospholipases A2; Precipitin Tests; Quinacrine; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha; Type C Phospholipases | 1990 |
Effects of lipopolysaccharide on phospholipase A2 activity and tumor necrosis factor expression in HL-60 cells.
Topics: Acetophenones; Bucladesine; Dinoprostone; Enzyme Activation; Gene Expression; Ketoconazole; Leukocytes, Mononuclear; Lipopolysaccharides; Masoprocol; Melitten; Phospholipases; Phospholipases A; Phospholipases A2; Protein Kinase C; Quinacrine; RNA, Messenger; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha | 1990 |
Evidence for the involvement of phospholipase A2 in the regulation of luteinizing hormone-stimulated steroidogenesis in rat testis Leydig cells.
Topics: Acetophenones; Animals; Arachidonic Acids; Bucladesine; Colforsin; Cyclic AMP; Dexamethasone; Hydroxycholesterols; Leydig Cells; Luteinizing Hormone; Male; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Inbred Strains; Testosterone | 1990 |
Characterization and inhibitor sensitivity of human sperm phospholipase A2: evidence against pivotal involvement of phospholipase A2 in the acrosome reaction.
Topics: 1,2-Dipalmitoylphosphatidylcholine; Acetophenones; Acrosome; Adult; Calcium; Deoxycholic Acid; Dimethyl Sulfoxide; Humans; Hydrogen-Ion Concentration; Kinetics; Lysophosphatidylcholines; Male; Phospholipases A; Phospholipases A2; Quinacrine; Spermatozoa; Temperature; Trifluoperazine | 1990 |
Effects of mepacrine and p-bromophenacyl bromide on anti-IgE and phospholipase A2-induced histamine release from human basophils.
Topics: Acetophenones; Antibodies, Anti-Idiotypic; Basophils; Calcium; Histamine Release; Humans; Immunoglobulin E; Kinetics; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine | 1986 |
Regulation of gamma-aminobutyric acid/barbiturate receptor-gated chloride ion flux in brain vesicles by phospholipase A2: possible role of oxygen radicals.
Topics: Acetophenones; Animals; Brain; Chlorides; Fatty Acids; Free Radicals; Ion Channels; Male; Oxygen; Pentobarbital; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Neurotransmitter; Serum Albumin, Bovine; Superoxide Dismutase; Synaptosomes; Xanthine; Xanthine Oxidase; Xanthines | 1988 |
Pharmacological study of phospholipase A2-induced histamine release from rat peritoneal mast cells.
Topics: Acetophenones; Animals; Cinnarizine; Cromolyn Sodium; Glucocorticoids; Histamine H1 Antagonists; Histamine Release; In Vitro Techniques; Male; Mast Cells; Nifedipine; ortho-Aminobenzoates; Phospholipases; Phospholipases A; Phospholipases A2; Piperazines; Pyridines; Quinacrine; Rats; Rats, Inbred Strains | 1989 |
Arachidonic acid mobilization and phosphoinositide turnover by the terminal complement complex, C5b-9, in rat oligodendrocyte x C6 glioma cell hybrids.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Animals; Arachidonic Acid; Arachidonic Acids; Calcimycin; Calcium; Clone Cells; Complement Membrane Attack Complex; Complement System Proteins; Glioma; Humans; Hybrid Cells; Isoquinolines; Neuroglia; Oligodendroglia; Phosphatidylinositols; Piperazines; Protein Kinase C; Quinacrine; Rats | 1989 |
Superoxide generation is inhibited by phospholipase A2 inhibitors. Role for phospholipase A2 in the activation of the NADPH oxidase.
Topics: Acetophenones; Amino Alcohols; Arachidonic Acid; Arachidonic Acids; Cell-Free System; Enzyme Activation; Humans; In Vitro Techniques; N-Formylmethionine Leucyl-Phenylalanine; NADH, NADPH Oxidoreductases; NADPH Oxidases; Neutrophils; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Sodium Dodecyl Sulfate; Superoxides; Tetradecanoylphorbol Acetate | 1989 |
The role of phospholipase A2 in microsomal lipid peroxidation induced with t-butyl hydroperoxide.
Topics: Acetophenones; Animals; Chlorpromazine; Enzyme Activation; Fatty Acids; Lipid Peroxidation; Melitten; Microsomes, Liver; Peroxides; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Rats; tert-Butylhydroperoxide; Thiobarbiturates | 1989 |
Regulation of phospholipid synthesis by intracellular phospholipases in fetal rabbit type II pneumocytes.
Topics: Acetophenones; Animals; Choline; Choline-Phosphate Cytidylyltransferase; Female; Lung; Nucleotidyltransferases; Palmitic Acid; Palmitic Acids; Phospholipases; Phospholipases A; Phospholipases A2; Phospholipids; Pregnancy; Quinacrine; Rabbits; Time Factors; Type C Phospholipases | 1985 |
Antigen-induced bronchial anaphylaxis in actively sensitized SD rats. Effects of glucocorticoid treatment.
Topics: Acetophenones; Administration, Topical; Alum Compounds; Aluminum; Anaphylaxis; Animals; Antigens; Bronchial Diseases; Budesonide; Cromolyn Sodium; Dexamethasone; Dose-Response Relationship, Drug; Drug Interactions; Glucocorticoids; Immunization; Injections, Intraperitoneal; Injections, Intravenous; Male; Ovalbumin; Pregnenediones; Quinacrine; Rats; Rats, Inbred Strains; Respiration; Sulfates; Time Factors | 1986 |
Possible involvement of the phospholipases in the mitogenic actions of prolactin (PRL) on Nb2 node lymphoma cells.
Topics: Acetophenones; Animals; Arachidonic Acid; Arachidonic Acids; Cell Division; Cell Line; Lymphoma; Phospholipases; Phospholipases A; Phospholipases A2; Prolactin; Quinacrine; Rats; Stimulation, Chemical; Type C Phospholipases | 1987 |
Mechanism of CO2 response in cerebral arteries of the newborn pig: role of phospholipase, cyclooxygenase, and lipoxygenase pathways.
Topics: Acetophenones; Animals; Animals, Newborn; Arterioles; Carbon Dioxide; Cerebrovascular Circulation; Indomethacin; Lipoxygenase; Masoprocol; Phospholipases A; Pia Mater; Prostaglandin-Endoperoxide Synthases; Quinacrine; Swine | 1988 |
Selective inhibition of free arachidonic acid production in activated alveolar macrophages by calmodulin antagonists.
Topics: Acetophenones; Animals; Arachidonic Acid; Arachidonic Acids; Calmodulin; Chlorpromazine; Chromatography, High Pressure Liquid; Cytochalasin B; Linoleic Acid; Linoleic Acids; Macrophage Activation; Macrophages; Oleic Acid; Oleic Acids; Opsonin Proteins; Phosphatidylcholines; Phosphatidylinositols; Phospholipases A; Pulmonary Alveoli; Quinacrine; Rabbits; Sulfonamides; Trifluoperazine; Zymosan | 1988 |
The biphasic effect of phospholipase A2 inhibitors on axon elongation.
Topics: Acetophenones; Animals; Axons; Cells, Cultured; Enzyme Inhibitors; Ganglia, Spinal; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Inbred Strains; Strontium | 1986 |
Prolactin actions on casein and lipid biosynthesis in mouse and rabbit mammary gland explants are abolished by p-bromphenacyl bromide and quinacrine, phospholipase A2 inhibitors.
Topics: Acetophenones; Animals; Caseins; Lipids; Mammary Glands, Animal; Mice; Phospholipases A; Phospholipases A2; Prolactin; Quinacrine; Rabbits | 1986 |
The role of phospholipase A activity in rat liver microsomal lipid peroxidation.
Topics: Acetophenones; Adenosine Diphosphate; Alloxan; Animals; Chlorpromazine; Copper; Ferrous Compounds; Glutathione; Hydrogen-Ion Concentration; Lipid Peroxides; Male; Microsomes, Liver; Phospholipases; Phospholipases A; Phospholipases A1; Phospholipases A2; Quinacrine; Rats; Rats, Inbred Strains | 1987 |
Possible role of phospholipase A2 action and arachidonic acid metabolism in angiotensin II-mediated aldosterone secretion.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; 5,8,11,14-Eicosatetraynoic Acid; Acetophenones; Aldosterone; Angiotensin II; Animals; Arachidonic Acid; Arachidonic Acids; Caffeic Acids; Calcium; Cattle; Cyclooxygenase Inhibitors; Dantrolene; Dose-Response Relationship, Drug; Indomethacin; Lipoxygenase Inhibitors; Phospholipases; Phospholipases A; Phospholipases A2; Pyrazoles; Quinacrine | 1985 |
Effect of diarachidonin on prostaglandin E2 synthesis in rabbit kidney medulla slices.
Topics: Acetophenones; Animals; Arachidonic Acid; Arachidonic Acids; Diglycerides; Dinoprostone; Dose-Response Relationship, Drug; Egtazic Acid; Glycerides; In Vitro Techniques; Kidney Medulla; Male; Phosphatidic Acids; Prostaglandins E; Quinacrine; Rabbits | 1985 |
Inhibition by mepacrine and p-bromophenacylbromide of phosphoinositide hydrolysis, glucose oxidation, calcium uptake and insulin release in rat pancreatic islets.
Topics: Acetophenones; Animals; Calcium; Dose-Response Relationship, Drug; Glucose; Hydrolysis; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Oxidation-Reduction; Phosphatidylinositols; Quinacrine; Rats; Rubidium; Type C Phospholipases | 1984 |
The number of the Trf receptors on human hematopoietic cell lines is influenced by membrane phospholipids.
Topics: Acetophenones; Cell Line; Cell Membrane; Humans; Kinetics; Leukemia, Myeloid, Acute; Membrane Lipids; Phospholipases; Phospholipids; Quinacrine; Receptors, Cell Surface; Receptors, Transferrin; Tetracaine; Transferrin | 1983 |
Possible role of phospholipase A2 in triggering histamine secretion from human basophils in vitro.
Topics: Acetophenones; Arachidonic Acids; Basophils; Calcium; Edetic Acid; Histamine Release; Humans; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine | 1981 |
Mechanisms involved in the synthesis of disaturated phosphatidylcholine by alveolar type II cells isolated from adult rat lung.
Topics: Acetophenones; Animals; Cell Membrane; Diacylglycerol Cholinephosphotransferase; Ethanolaminephosphotransferase; Glycerol; Kinetics; Lung; Male; Phosphatidylcholines; Quinacrine; Rats; Rats, Inbred Strains | 1983 |
Prevention of catecholamine release from adrenal chromaffin cells by phospholipase A2- and lipoxygenase-inhibitors.
Topics: 4,5-Dihydro-1-(3-(trifluoromethyl)phenyl)-1H-pyrazol-3-amine; Acetophenones; Adrenal Medulla; Animals; Arachidonic Acids; Aspirin; Catecholamines; Cattle; Chromaffin System; In Vitro Techniques; Lipoxygenase Inhibitors; Phospholipases; Phospholipases A; Phospholipases A2; Pyrazoles; Quinacrine | 1983 |
Assessment of a role for phospholipase A2 and arachidonic acid metabolism in human lymphocyte natural cytotoxicity.
Topics: Acetophenones; Arachidonic Acid; Arachidonic Acids; Binding, Competitive; Cyclooxygenase Inhibitors; Cytotoxicity, Immunologic; Dexamethasone; Humans; Hydrocortisone; Killer Cells, Natural; Kinetics; Lipoxygenase Inhibitors; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine | 1984 |
Improvement of the anoxia-induced mitochondrial dysfunction by membrane modulation.
Topics: Acetophenones; Adenine Nucleotides; Alkaloids; Animals; Benzylisoquinolines; Chlorpromazine; Egtazic Acid; Hypoxia; Kinetics; Male; Mitochondria, Liver; Mitochondrial Swelling; Oxidative Phosphorylation; Oxygen Consumption; Phospholipids; Quinacrine; Rats; Rats, Inbred Strains | 1984 |
Stimulation of prostaglandin E2 synthesis by exogenous phospholipase A2 and C in rabbit kidney medulla slices.
Topics: Acetophenones; Animals; Dinoprostone; Fatty Acids; In Vitro Techniques; Kidney Medulla; Lipolysis; Male; Phospholipases; Phospholipases A; Phospholipases A2; Prostaglandins E; Quinacrine; Rabbits; Stimulation, Chemical; Type C Phospholipases | 1984 |
Calmodulin, phospholipase, and exocytosis. p-Bromophenacyl bromide inhibits but mepacrine stimulates secretion in rat mast cells.
Topics: Acetophenones; Animals; Calcium; Calmodulin; Exocytosis; In Vitro Techniques; Male; Mast Cells; Phenothiazines; Phospholipases; Quinacrine; Rats; Rats, Inbred Strains | 1983 |
How a nerve fiber repairs its cut end: involvement of phospholipase A2.
Topics: Acetophenones; Animals; Axons; Calcium; Cell Membrane; Denervation; Enzyme Activation; Membrane Potentials; Periplaneta; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Temperature | 1983 |
The effects of mepacrine and p-bromophenacyl bromide on arachidonic acid release in human platelets.
Topics: Acetophenones; Arachidonic Acid; Arachidonic Acids; Blood Platelets; Dose-Response Relationship, Drug; Humans; Quinacrine; Serotonin; Thrombin; Type C Phospholipases | 1982 |
Studies on the incorporation of [1-14C]arachidonic acid into glycerolipids and its conversion into prostaglandins by rabbit iris. Effects of anti-inflammatory drugs and phospholipase A2 inhibitors.
Topics: Acetophenones; Animals; Anti-Inflammatory Agents; Arachidonic Acid; Arachidonic Acids; Aspirin; Diglycerides; Female; Indomethacin; Iris; Lipid Metabolism; Male; Microsomes; Muscle, Smooth; Phospholipases; Phospholipases A; Phospholipases A2; Phospholipids; Prostaglandins; Quinacrine; Rabbits; Triglycerides | 1982 |
Suppression by phospholipase A2 inhibitors of secretion of catecholamines from isolated adrenal medullary cells by suppression of cellular calcium uptake.
Topics: Acetophenones; Adrenal Medulla; Animals; Calcium; Carbachol; Catecholamines; Cattle; Chloroquine; Dose-Response Relationship, Drug; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Quinine | 1983 |
Phospholipase A2 inhibitors block catecholamine secretion and calcium uptake in cultured bovine adrenal medullary cells.
Topics: Acetophenones; Adrenal Medulla; Animals; Biological Transport, Active; Calcium; Catecholamines; Cattle; Cells, Cultured; Exocytosis; Kinetics; Phospholipases; Phospholipases A; Phospholipases A2; Propanolamines; Quinacrine | 1983 |
Phospholipase A2 inhibitors. Differential inhibition of fatty acid acylation into kidney lipids by mepacrine and p-bromophenacyl bromide.
Topics: Acetophenones; Acylation; Animals; Arachidonic Acids; Fatty Acids; In Vitro Techniques; Kidney Medulla; Linoleic Acids; Lipid Metabolism; Male; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Rabbits; Stearic Acids | 1983 |
Intraventricular injections of drugs which inhibit phospholipase A2 suppress fever in rabbits.
Topics: Acetophenones; Animals; Arachidonic Acids; Body Temperature Regulation; Fever; Injections, Intravenous; Injections, Intraventricular; Phospholipases; Phospholipases A; Phospholipases A2; Quinacrine; Rabbits | 1983 |
Inhibitors of 125I-epidermal growth factor internalization.
Topics: Acetophenones; Animals; Azo Compounds; Bacitracin; Cells, Cultured; Chlorpromazine; Endocytosis; Epidermal Growth Factor; Methylamines; Peptides; Phenylglyoxal; Phospholipases; Phospholipases A; Quinacrine; Rats | 1980 |
Effects of phospholipase A2 inhibitors on the antidepressant-induced axonal regeneration of noradrenergic locus coeruleus neurons.
Topics: Acetophenones; Adrenergic Fibers; Animals; Antidepressive Agents; Axons; Fluorescence; Immunohistochemistry; Locus Coeruleus; Microscopy, Electron; Nerve Regeneration; Neurons; Norepinephrine; Oxidopamine; Phospholipases A; Phospholipases A2; Quinacrine; Rats | 1994 |
On the role of arachidonic acid in M-current modulation by muscarine in bullfrog sympathetic neurons.
Topics: Acetophenones; Animals; Arachidonic Acid; Dose-Response Relationship, Drug; Ganglia, Sympathetic; Gonadotropin-Releasing Hormone; In Vitro Techniques; Kinetics; Masoprocol; Membrane Potentials; Muscarine; Neurons; Phospholipases A; Phospholipases A2; Potassium Channels; Quinacrine; Rana catesbeiana | 1994 |
Evidence for a role of phospholipase A2 in the mechanism of LHRH priming in rat anterior pituitary tissue.
Topics: Acetophenones; Aminobenzoates; Animals; Arachidonic Acid; Aristolochic Acids; Calcium; Chlorobenzoates; Cinnamates; Cycloheximide; Female; Gonadotropin-Releasing Hormone; In Vitro Techniques; Luteinizing Hormone; ortho-Aminobenzoates; Phenanthrenes; Phenothiazines; Phospholipases A; Phospholipases A2; Pituitary Gland, Anterior; Proestrus; Quinacrine; Rats; Rats, Wistar | 1994 |
The requirement for phospholipase A2 for activation of the assembled NADPH oxidase in human neutrophils.
Topics: Acetophenones; Alkaloids; Arachidonic Acid; Biological Transport; Cell Membrane; Enzyme Activation; Humans; NADH, NADPH Oxidoreductases; NADPH Oxidases; Neutrophils; Opsonin Proteins; Phospholipases A; Phospholipases A2; Phosphorylation; Protein Kinase C; Quinacrine; Staurosporine; Superoxides; Tetradecanoylphorbol Acetate; Tritium; Zymosan | 1994 |
Regulation of human eosinophil degranulation and activation by endogenous phospholipase A2.
Topics: Acetophenones; Arachidonic Acid; Cell Separation; Centrifugation, Density Gradient; Cytochalasin B; Dose-Response Relationship, Drug; Eosinophil Peroxidase; Eosinophils; Homeostasis; In Vitro Techniques; Kinetics; N-Formylmethionine Leucyl-Phenylalanine; Peroxidases; Phospholipases A; Phospholipases A2; Quinacrine; SRS-A; Superoxides | 1993 |
Effect of putative phospholipase A2 inhibitors on acetic acid-induced acute colitis in the rat.
Topics: Acetates; Acetic Acid; Acetophenones; Animals; Colitis; Colon; Enzyme Activation; Female; Intestinal Mucosa; Peroxidase; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Sprague-Dawley; Verapamil | 1993 |
Eicosanoid production by mouse peritoneal macrophages during Toxoplasma gondii penetration: role of parasite and host cell phospholipases.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Animals; Arachidonic Acid; Calcium; Cyclooxygenase Inhibitors; Eicosanoids; Female; Indomethacin; Isoquinolines; Lipoxygenase; Macrophages; Mice; Peritoneal Cavity; Phospholipases; Piperazines; Prostaglandin-Endoperoxide Synthases; Protein Kinase C; Quinacrine; Toxoplasma; Toxoplasmosis, Animal | 1993 |
Botulinum toxin inhibits arachidonic acid release associated with acetylcholine release from PC12 cells.
Topics: Acetophenones; Acetylcholine; Animals; Arachidonic Acid; Botulinum Toxins; Cell Differentiation; Dose-Response Relationship, Drug; Ethacrynic Acid; Indomethacin; Kinetics; Masoprocol; Melitten; Models, Biological; Nerve Growth Factors; PC12 Cells; Phospholipases A; Phospholipases A2; Potassium; Protein Kinase C; Quinacrine; Terpenes | 1993 |
Differences in the acute actions of sGnRH and cGnRH-II on gonadotropin release in goldfish pituitary cells.
Topics: Acetophenones; Analysis of Variance; Animals; Calcium Channel Blockers; Cells, Cultured; Enzyme Inhibitors; Female; Goldfish; Gonadotropin-Releasing Hormone; Gonadotropins; Male; Masoprocol; Pituitary Gland; Quinacrine; Verapamil | 1995 |
Inhibition of HIV-1 Tat-mediated transactivation by quinacrine and chloroquine.
Topics: Acetophenones; Alkaloids; Antimalarials; Benzoquinones; Cell Line; Cell Survival; Chloroquine; Curcumin; Gene Expression Regulation, Viral; Gene Products, tat; HIV Long Terminal Repeat; HIV-1; Humans; Lactams, Macrocyclic; Quinacrine; Quinones; Rifabutin; Staurosporine; tat Gene Products, Human Immunodeficiency Virus; Transcriptional Activation; Tumor Cells, Cultured; Virus Replication | 1996 |
Modulation of 8-methoxypsoralen-photoinduced cutaneous inflammatory reactions by various chemotherapeutic agents in vivo.
Topics: Acetophenones; Animals; Capillary Permeability; Erythema; Ibuprofen; Indoles; Indomethacin; Masoprocol; Methoxsalen; Neutrophils; PUVA Therapy; Quinacrine; Rabbits; Skin | 1996 |
PLA2 activity in Tetrahymena pyriformis. Effects of inhibitors and stimulators.
Topics: Acetophenones; Aluminum Compounds; Animals; Arachidonic Acid; Calcium; Enzyme Activation; Enzyme Inhibitors; Fluorides; Hydrogen Peroxide; Inositol; Lithium Chloride; Melitten; Phorbol 12,13-Dibutyrate; Phosphatidylinositols; Phospholipases A; Phospholipases A2; Phospholipids; Protein-Tyrosine Kinases; Quinacrine; Signal Transduction; Sodium Fluoride; Tetrahymena pyriformis; Vanadates | 1997 |
Increased PLA2 activity is not related to increase GLUT1 expression in L6 myotubes under hypoxic conditions.
Topics: Acetophenones; Animals; Arachidonic Acid; Biological Transport; Cell Hypoxia; Cell Line; Cyclooxygenase Inhibitors; Deoxyglucose; Glucose; Glucose Transporter Type 1; Glucose Transporter Type 4; Insulin; Membrane Proteins; Monosaccharide Transport Proteins; Muscle Proteins; Muscle, Skeletal; Phospholipases A; Phospholipases A2; Prostaglandins; Quinacrine; Rats; Signal Transduction | 1997 |
Phospholipases and arachidonic acid contribute independently to sensory transduction and associative neuronal facilitation in Hermissenda type B photoreceptors.
Topics: Acetophenones; Animals; Arachidonic Acid; Association Learning; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Indomethacin; Lipoxygenase Inhibitors; Masoprocol; Mollusca; Neurons; Phospholipases; Photoreceptor Cells, Invertebrate; Quinacrine; Sensation; Signal Transduction | 1997 |
Structure-activity of three phospholipid analogues towards inhibition of phospholipase A2 in macrophages.
Topics: Acetophenones; Animals; Anti-Inflammatory Agents; Cells, Cultured; Culture Media; Dexamethasone; Eicosanoids; Enzyme Inhibitors; Macrophages, Peritoneal; Male; Phospholipases A; Phospholipases A2; Phospholipids; Quinacrine; Rats; Structure-Activity Relationship; Tritium | 1997 |
Influence of nicotine and cotinine on retinal phospholipase A2 and its significance to macular function.
Topics: Acetophenones; Acetylcholine; Animals; Cotinine; Enzyme Inhibitors; Macular Degeneration; Nicotine; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Inbred F344; Retina | 1998 |
Involvement of phospholipase A2 activation in anthrax lethal toxin-induced cytotoxicity.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 4-Aminobenzoic Acid; Acetophenones; Aminobenzoates; Animals; Anthrax; Antigens, Bacterial; Antioxidants; Apoptosis; Bacterial Toxins; Cells, Cultured; Dehydroepiandrosterone; DNA Fragmentation; Enzyme Activation; Enzyme Inhibitors; Macrophages, Peritoneal; Melatonin; Mice; Mice, Inbred ICR; Nitric Oxide; para-Aminobenzoates; Phosphodiesterase Inhibitors; Phospholipases A; Phospholipases A2; Protein Kinase Inhibitors; Quinacrine; Reactive Oxygen Species; Staurosporine; Terpenes | 1999 |
Lysophosphatidylcholine and arachidonic acid are required in the cytotoxic response of human natural killer cells to tumor target cells.
Topics: Acetophenones; Arachidonic Acid; Cytotoxicity, Immunologic; Enzyme Inhibitors; Humans; K562 Cells; Killer Cells, Natural; Leukotrienes; Linoleic Acid; Lipid Peroxides; Lysophosphatidylcholines; Phospholipases A; Quinacrine | 1999 |
Calcium-dependent mitochondrial formation of species promoting strand scission of genomic DNA in U937 cells exposed to tert-butylhydroperoxide: the role of arachidonic acid.
Topics: 5,8,11,14-Eicosatetraynoic Acid; Acetophenones; Antimycin A; Arachidonic Acid; Calcium; DNA Damage; Electron Transport; Enzyme Inhibitors; Humans; Melitten; Mitochondria; Phospholipases A; Phospholipases A2; Quinacrine; tert-Butylhydroperoxide; U937 Cells | 2000 |
Effect of quinacrine treatment on the activity of acid hydrolases (phosphatase, N-acetyl-beta-glucosaminidase, glucosidase, galactosidase and esterase) in Tetrahymena.
Topics: Acetophenones; Acetylglucosaminidase; Acid Phosphatase; Animals; Antimalarials; Cell Fractionation; Enzyme Inhibitors; Esterases; Galactosidases; Glucosidases; Hydrolases; Quinacrine; Tetrahymena pyriformis | 2001 |
Arachidonic acid release from rat Leydig cells: the involvement of G protein, phospholipase A2 and regulation of cAMP production.
Topics: Acetophenones; Animals; Arachidonic Acid; Chorionic Gonadotropin; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Leydig Cells; Male; Melitten; Pertussis Toxin; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Inbred Strains; Stimulation, Chemical; Virulence Factors, Bordetella | 2002 |
4-Bromophenacyl bromide induces Ca2+ influx in human gingival fibroblasts.
Topics: Acetophenones; Aniline Compounds; Arachidonic Acids; Bradykinin; Calcium; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fibroblasts; Fluorescent Dyes; Gingiva; Histamine; Humans; Kinetics; Phospholipases A; Phospholipases A2; Quinacrine; Spectrometry, Fluorescence; Structure-Activity Relationship; Terpenes; Xanthenes | 2002 |
Quaternary-Ammonium-Modulated Surface-Enhanced Raman Spectroscopy Effect: Discovery, Mechanism, and Application for Highly Sensitive
Topics: Acetophenones; Acetylcholine; Animals; Microfluidic Analytical Techniques; PC12 Cells; Quaternary Ammonium Compounds; Quinacrine; Rats; Spectrum Analysis, Raman | 2020 |