quilostigmine has been researched along with scopolamine hydrobromide in 2 studies
Studies (quilostigmine) | Trials (quilostigmine) | Recent Studies (post-2010) (quilostigmine) | Studies (scopolamine hydrobromide) | Trials (scopolamine hydrobromide) | Recent Studies (post-2010) (scopolamine hydrobromide) |
---|---|---|---|---|---|
7 | 1 | 1 | 7,548 | 563 | 1,401 |
Protein | Taxonomy | quilostigmine (IC50) | scopolamine hydrobromide (IC50) |
---|---|---|---|
Muscarinic acetylcholine receptor M4 | Homo sapiens (human) | 0.003 | |
Muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | 0.006 | |
Muscarinic acetylcholine receptor M3 | Rattus norvegicus (Norway rat) | 0.006 | |
Muscarinic acetylcholine receptor M4 | Rattus norvegicus (Norway rat) | 0.006 | |
Cytochrome P450 3A4 | Homo sapiens (human) | 0.0006 | |
Muscarinic acetylcholine receptor M5 | Rattus norvegicus (Norway rat) | 0.006 | |
Muscarinic acetylcholine receptor M2 | Rattus norvegicus (Norway rat) | 0.006 | |
Muscarinic acetylcholine receptor M1 | Homo sapiens (human) | 0.0026 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 2 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Chaudhaery, SS; Nath, C; Nazir, A; Roy, KK; Sammi, SR; Saxena, AK; Saxena, G; Shakya, N | 1 |
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
2 other study(ies) available for quilostigmine and scopolamine hydrobromide
Article | Year |
---|---|
Novel carbamates as orally active acetylcholinesterase inhibitors found to improve scopolamine-induced cognition impairment: pharmacophore-based virtual screening, synthesis, and pharmacology.
Topics: Acetylcholinesterase; Administration, Oral; Animals; Avoidance Learning; Caenorhabditis elegans; Carbamates; Catalytic Domain; Cholinesterase Inhibitors; Databases, Factual; Hydrogen Bonding; Hydrophobic and Hydrophilic Interactions; Male; Mice; Models, Molecular; Nootropic Agents; Quantitative Structure-Activity Relationship; Scopolamine | 2010 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |