quilostigmine has been researched along with physostigmine in 2 studies
Studies (quilostigmine) | Trials (quilostigmine) | Recent Studies (post-2010) (quilostigmine) | Studies (physostigmine) | Trials (physostigmine) | Recent Studies (post-2010) (physostigmine) |
---|---|---|---|---|---|
7 | 1 | 1 | 6,230 | 252 | 331 |
Protein | Taxonomy | quilostigmine (IC50) | physostigmine (IC50) |
---|---|---|---|
Acetylcholinesterase | Electrophorus electricus (electric eel) | 0.1666 | |
Acetylcholinesterase | Tetronarce californica (Pacific electric ray) | 0.3023 | |
Cholinesterase | Homo sapiens (human) | 0.3055 | |
Cytochrome P450 2D6 | Homo sapiens (human) | 0.2 | |
Alpha-1B adrenergic receptor | Rattus norvegicus (Norway rat) | 0.857 | |
Acetylcholinesterase | Mus musculus (house mouse) | 0.0269 | |
Acetylcholinesterase | Homo sapiens (human) | 0.0853 | |
Acetylcholinesterase | Bos taurus (cattle) | 0.7197 | |
Alpha-1D adrenergic receptor | Rattus norvegicus (Norway rat) | 0.857 | |
Delta-type opioid receptor | Mus musculus (house mouse) | 1.1821 | |
Acetylcholinesterase | Gallus gallus (chicken) | 0.02 | |
Acetylcholinesterase | Rattus norvegicus (Norway rat) | 0.0416 | |
Alpha-1A adrenergic receptor | Rattus norvegicus (Norway rat) | 0.857 | |
Cholinesterase | Equus caballus (horse) | 0.4081 | |
Cholinesterase | Mus musculus (house mouse) | 0.28 | |
Acyl-CoA:cholesterol acyltransferase | Oryctolagus cuniculus (rabbit) | 0.0189 | |
Carboxylic ester hydrolase | Rattus norvegicus (Norway rat) | 0.018 | |
Carboxylic ester hydrolase | Equus caballus (horse) | 1.263 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (50.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 1 (50.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Chaudhaery, SS; Nath, C; Nazir, A; Roy, KK; Sammi, SR; Saxena, AK; Saxena, G; Shakya, N | 1 |
Cross, AJ; De Souza, RJ; Green, AR; Misra, A; Murray, TK; Snape, MF; Williams, JL | 1 |
2 other study(ies) available for quilostigmine and physostigmine
Article | Year |
---|---|
Novel carbamates as orally active acetylcholinesterase inhibitors found to improve scopolamine-induced cognition impairment: pharmacophore-based virtual screening, synthesis, and pharmacology.
Topics: Acetylcholinesterase; Administration, Oral; Animals; Avoidance Learning; Caenorhabditis elegans; Carbamates; Catalytic Domain; Cholinesterase Inhibitors; Databases, Factual; Hydrogen Bonding; Hydrophobic and Hydrophilic Interactions; Male; Mice; Models, Molecular; Nootropic Agents; Quantitative Structure-Activity Relationship; Scopolamine | 2010 |
A comparative study in rats of the in vitro and in vivo pharmacology of the acetylcholinesterase inhibitors tacrine, donepezil and NXX-066.
Topics: Acetylcholinesterase; Animals; Butyrylcholinesterase; Carbachol; Cholinesterase Inhibitors; Donepezil; Drug Evaluation, Preclinical; Humans; Indans; Indoles; Injections, Intraperitoneal; Isoquinolines; Logistic Models; Male; Physostigmine; Piperidines; Rats; Structure-Activity Relationship; Tacrine; Tumor Cells, Cultured | 1999 |