quilostigmine has been researched along with donepezil in 3 studies
Studies (quilostigmine) | Trials (quilostigmine) | Recent Studies (post-2010) (quilostigmine) | Studies (donepezil) | Trials (donepezil) | Recent Studies (post-2010) (donepezil) |
---|---|---|---|---|---|
7 | 1 | 1 | 3,193 | 557 | 1,594 |
Protein | Taxonomy | quilostigmine (IC50) | donepezil (IC50) |
---|---|---|---|
Acetylcholinesterase | Electrophorus electricus (electric eel) | 0.4231 | |
Acetylcholinesterase | Tetronarce californica (Pacific electric ray) | 0.0265 | |
Amyloid-beta precursor protein | Homo sapiens (human) | 0.022 | |
Cholinesterase | Homo sapiens (human) | 4.5742 | |
5-hydroxytryptamine receptor 1A | Rattus norvegicus (Norway rat) | 7.42 | |
Amine oxidase [flavin-containing] B | Rattus norvegicus (Norway rat) | 5 | |
Amine oxidase [flavin-containing] A | Rattus norvegicus (Norway rat) | 7.4 | |
Acetylcholinesterase | Mus musculus (house mouse) | 1.5489 | |
Acetylcholinesterase | Homo sapiens (human) | 0.3257 | |
Acetylcholinesterase | Bos taurus (cattle) | 0.1644 | |
Choline O-acetyltransferase | Rattus norvegicus (Norway rat) | 0.0053 | |
Acetylcholinesterase | Rattus norvegicus (Norway rat) | 0.0182 | |
Beta-secretase 1 | Homo sapiens (human) | 0.8666 | |
Cholinesterase | Equus caballus (horse) | 3.7325 | |
Cholinesterase | Mus musculus (house mouse) | 1.992 | |
Acetylcholine receptor subunit epsilon | Homo sapiens (human) | 0.0324 | |
Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | 3.7844 | |
Acyl-CoA:cholesterol acyltransferase | Oryctolagus cuniculus (rabbit) | 0.008 | |
Carboxylic ester hydrolase | Rattus norvegicus (Norway rat) | 4.715 | |
Carboxylic ester hydrolase | Equus caballus (horse) | 4.5551 | |
Histamine H3 receptor | Homo sapiens (human) | 0.35 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (33.33) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 2 (66.67) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Chaudhaery, SS; Nath, C; Nazir, A; Roy, KK; Sammi, SR; Saxena, AK; Saxena, G; Shakya, N | 1 |
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
Cross, AJ; De Souza, RJ; Green, AR; Misra, A; Murray, TK; Snape, MF; Williams, JL | 1 |
3 other study(ies) available for quilostigmine and donepezil
Article | Year |
---|---|
Novel carbamates as orally active acetylcholinesterase inhibitors found to improve scopolamine-induced cognition impairment: pharmacophore-based virtual screening, synthesis, and pharmacology.
Topics: Acetylcholinesterase; Administration, Oral; Animals; Avoidance Learning; Caenorhabditis elegans; Carbamates; Catalytic Domain; Cholinesterase Inhibitors; Databases, Factual; Hydrogen Bonding; Hydrophobic and Hydrophilic Interactions; Male; Mice; Models, Molecular; Nootropic Agents; Quantitative Structure-Activity Relationship; Scopolamine | 2010 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |
A comparative study in rats of the in vitro and in vivo pharmacology of the acetylcholinesterase inhibitors tacrine, donepezil and NXX-066.
Topics: Acetylcholinesterase; Animals; Butyrylcholinesterase; Carbachol; Cholinesterase Inhibitors; Donepezil; Drug Evaluation, Preclinical; Humans; Indans; Indoles; Injections, Intraperitoneal; Isoquinolines; Logistic Models; Male; Physostigmine; Piperidines; Rats; Structure-Activity Relationship; Tacrine; Tumor Cells, Cultured | 1999 |