Page last updated: 2024-09-03

quadazocine and enkephalin, leucine

quadazocine has been researched along with enkephalin, leucine in 14 studies

Compound Research Comparison

Studies
(quadazocine)
Trials
(quadazocine)
Recent Studies (post-2010)
(quadazocine)
Studies
(enkephalin, leucine)
Trials
(enkephalin, leucine)
Recent Studies (post-2010) (enkephalin, leucine)
8100502
810011,52480754

Protein Interaction Comparison

ProteinTaxonomyquadazocine (IC50)enkephalin, leucine (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.0142
Kappa-type opioid receptorMus musculus (house mouse)0.0417
Mu-type opioid receptorHomo sapiens (human)9.5
Mu-type opioid receptorMus musculus (house mouse)0.0308
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.246

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19908 (57.14)18.7374
1990's6 (42.86)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Adapa, ID; Auh, JS; Berzetei-Gurske, IP; Brandt, SR; Craymer, K; Farrington, L; Haggart, D; Kennedy, JM; O'Brien, A; Polgar, WE; Rodriguez, L; Schwartz, RW; Toll, L; White, A1
Gannon, RL; Terrian, DM1
Cagampang, FR; Maeda, K1
Hahn, EF; Howard, DH; Levison, JA; Pasternak, GW; Paul, D; Pick, CG1
Dodson, BA; Miller, KW1
Agura, V; DeWitt, DS; Faden, AI; Hayes, RL; McIntosh, TK1
Adler, MW; Geller, EB; Tiseo, PJ1
Portoghese, PS; Takemori, AE1
Barber, DJ; Barbour-McMullen, J; Cooper, SJ1
Chandra, A; Diliberto, EJ; Dixon, WR; Holaday, JW; Lewis, JW; Long, JB; Tortella, FC; Unsworth, CD; Viveros, OH; Way, EL1
Faden, AI1
Huidobro-Toro, JP; Way, EL; Yoshimura, K1
Brusa, L; D'Amore, A; Lorenzini, P; Massotti, M1
Butelman, ER; Ko, MC; Woods, JH1

Other Studies

14 other study(ies) available for quadazocine and enkephalin, leucine

ArticleYear
Standard binding and functional assays related to medications development division testing for potential cocaine and opiate narcotic treatment medications.
    NIDA research monograph, 1998, Volume: 178

    Topics: Animals; Aorta, Thoracic; Cocaine; Cyclic AMP; Electric Stimulation; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Male; Mice; Muscle, Smooth; Opioid-Related Disorders; Rats; Receptors, Dopamine; Receptors, Opioid; Receptors, Serotonin; Substance-Related Disorders

1998
Kappa opioid agonists inhibit transmitter release from guinea pig hippocampal mossy fiber synaptosomes.
    Neurochemical research, 1992, Volume: 17, Issue:8

    Topics: Animals; Azocines; Calcium; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; Glutamates; Glutamic Acid; Guinea Pigs; Hippocampus; Male; Potassium; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Synaptosomes

1992
Effects of intracerebroventricular administration of opiate receptor antagonists on the suppressed pulsatile LH release during acute fasting in ovariectomized estradiol-treated rats.
    Life sciences, 1991, Volume: 49, Issue:24

    Topics: Animals; Azocines; Enkephalin, Leucine; Estradiol; Fasting; Female; Injections, Intraventricular; Luteinizing Hormone; Naloxone; Narcotic Antagonists; Ovariectomy; Periodicity; Rats; Rats, Inbred Strains; Receptors, Opioid

1991
Naloxone benzoylhydrazone (NalBzoH) analgesia.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 255, Issue:2

    Topics: Analgesia; Analgesics; Animals; Azocines; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Male; Mice; Naloxone; Narcotic Antagonists; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

1990
Evidence for a dual mechanism in the anesthetic action of an opioid peptide.
    Anesthesiology, 1985, Volume: 62, Issue:5

    Topics: 1-Octanol; Analgesics, Opioid; Anesthetics; Animals; Atmospheric Pressure; Azocines; Dose-Response Relationship, Drug; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Lipids; Naloxone; Narcotic Antagonists; Octanols; Postural Balance; Rana pipiens; Receptors, Opioid; Reflex; Solubility; Time Factors

1985
Endogenous opioids may mediate secondary damage after experimental brain injury.
    The American journal of physiology, 1987, Volume: 253, Issue:5 Pt 1

    Topics: Animals; Azocines; Blood Flow Velocity; Blood Pressure; Brain; Brain Injuries; Cats; Cerebrovascular Circulation; Dopamine; Dynorphins; Electroencephalography; Endorphins; Enkephalin, Leucine; Female; Intracranial Pressure; Isomerism; Male; Narcotic Antagonists

1987
Antinociceptive action of intracerebroventricularly administered dynorphin and other opioid peptides in the rat.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Azocines; Cold Temperature; Drug Interactions; Dynorphins; Enkephalins; Injections, Intraventricular; Male; Naloxone; Pyrrolidines; Rats; Rats, Inbred Strains; Reaction Time; Receptors, Opioid

1988
TENA, a selective kappa opioid receptor antagonist.
    Life sciences, 1985, Feb-25, Volume: 36, Issue:8

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Azocines; Benzomorphans; Cyclazocine; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Guinea Pigs; Ileum; Male; Mice; Naloxone; Naltrexone; Narcotic Antagonists; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Vas Deferens

1985
Selective attenuation of sweetened milk consumption by opiate receptor antagonists in male and female rats of the Roman strains.
    Neuropeptides, 1985, Volume: 5, Issue:4-6

    Topics: Animals; Appetite Depressants; Azocines; Benzomorphans; Diprenorphine; Enkephalin, Leucine; Feeding Behavior; Female; Male; Naloxone; Narcotic Antagonists; Rats; Receptors, Opioid; Sex Factors; Species Specificity

1985
Multiple opiate receptors: functional implications.
    Federation proceedings, 1985, Volume: 44, Issue:13

    Topics: Adrenal Medulla; Adrenalectomy; Animals; Azocines; Behavior, Animal; Binding Sites; Blood Pressure; Clonidine; Corticosterone; Enkephalins; Naloxone; Receptors, Opioid; Stress, Physiological; Sympathetic Nervous System

1985
New pharmacologic approaches to spinal cord injury: opiate antagonists and thyrotropin-releasing hormone.
    Central nervous system trauma : journal of the American Paralysis Association, 1985,Spring, Volume: 2, Issue:1

    Topics: Animals; Azocines; Cats; Endorphins; Enkephalin, Leucine; Humans; Naloxone; Narcotic Antagonists; Rabbits; Receptors, Opioid; Spinal Cord Injuries; Thiazolidines; Thyrotropin-Releasing Hormone

1985
Potency of three opiate antagonists to reverse the inhibitory activity of dynorphin, enkephalins and opioid-like alkaloids on the guinea pig ileum.
    European journal of pharmacology, 1982, Oct-15, Volume: 84, Issue:1-2

    Topics: Animals; Azocines; Benzomorphans; Cyclazocine; Dynorphins; Endorphins; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Morphine Derivatives; Muscle, Smooth; Naloxone; Narcotic Antagonists

1982
Area tempestas modulates the behavioural responses to nociceptive stimuli in rats.
    Annali dell'Istituto superiore di sanita, 1993, Volume: 29, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Anticonvulsants; Azocines; Bicuculline; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Escape Reaction; Foot; Hot Temperature; Male; Morphine; Naltrexone; Narcotic Antagonists; Olfactory Pathways; Pain; Phenazocine; Pressure; Pyrrolidines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, Opioid; Seizures; Tail

1993
The role of peripheral mu opioid receptors in the modulation of capsaicin-induced thermal nociception in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 286, Issue:1

    Topics: Animals; Azocines; Capsaicin; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Female; Hot Temperature; Macaca mulatta; Male; Naltrexone; Pain; Receptors, Opioid, mu

1998