Compounds > quadazocine
Page last updated: 2024-09-03

quadazocine and enkephalin, ala(2)-mephe(4)-gly(5)-

quadazocine has been researched along with enkephalin, ala(2)-mephe(4)-gly(5)- in 5 studies

Compound Research Comparison

Studies
(quadazocine)		Trials
(quadazocine)		Recent Studies (post-2010)
(quadazocine)		Studies
(enkephalin, ala(2)-mephe(4)-gly(5)-)		Trials
(enkephalin, ala(2)-mephe(4)-gly(5)-)		Recent Studies (post-2010) (enkephalin, ala(2)-mephe(4)-gly(5)-)
8100151071
81002,7271374

Protein Interaction Comparison

ProteinTaxonomyquadazocine (IC50)enkephalin, ala(2)-mephe(4)-gly(5)- (IC50)
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)0.003
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)0.003
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)0.003
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)0.003
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)0.003
Delta-type opioid receptorMus musculus (house mouse)1.2415
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0132
Mu-type opioid receptorHomo sapiens (human)0.004
Delta-type opioid receptorHomo sapiens (human)0.0014
Mu-type opioid receptorMus musculus (house mouse)0.0048
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.0283

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (80.00)18.2507
2000's1 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Adapa, ID; Auh, JS; Berzetei-Gurske, IP; Brandt, SR; Craymer, K; Farrington, L; Haggart, D; Kennedy, JM; O'Brien, A; Polgar, WE; Rodriguez, L; Schwartz, RW; Toll, L; White, A1
Gannon, RL; Terrian, DM1
Brusa, L; D'Amore, A; Lorenzini, P; Massotti, M1
Butelman, ER; Ko, MC; Woods, JH1
David Clark, J; Demirci, H; Gharagozlou, P; Lameh, J1

Other Studies

5 other study(ies) available for quadazocine and enkephalin, ala(2)-mephe(4)-gly(5)-

ArticleYear
Standard binding and functional assays related to medications development division testing for potential cocaine and opiate narcotic treatment medications.
    NIDA research monograph, 1998, Volume: 178

    Topics: Animals; Aorta, Thoracic; Cocaine; Cyclic AMP; Electric Stimulation; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Male; Mice; Muscle, Smooth; Opioid-Related Disorders; Rats; Receptors, Dopamine; Receptors, Opioid; Receptors, Serotonin; Substance-Related Disorders

1998
Kappa opioid agonists inhibit transmitter release from guinea pig hippocampal mossy fiber synaptosomes.
    Neurochemical research, 1992, Volume: 17, Issue:8

    Topics: Animals; Azocines; Calcium; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; Glutamates; Glutamic Acid; Guinea Pigs; Hippocampus; Male; Potassium; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Synaptosomes

1992
Area tempestas modulates the behavioural responses to nociceptive stimuli in rats.
    Annali dell'Istituto superiore di sanita, 1993, Volume: 29, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Anticonvulsants; Azocines; Bicuculline; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Escape Reaction; Foot; Hot Temperature; Male; Morphine; Naltrexone; Narcotic Antagonists; Olfactory Pathways; Pain; Phenazocine; Pressure; Pyrrolidines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, Opioid; Seizures; Tail

1993
The role of peripheral mu opioid receptors in the modulation of capsaicin-induced thermal nociception in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 286, Issue:1

    Topics: Animals; Azocines; Capsaicin; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Female; Hot Temperature; Macaca mulatta; Male; Naltrexone; Pain; Receptors, Opioid, mu

1998
Activity of opioid ligands in cells expressing cloned mu opioid receptors.
    BMC pharmacology, 2003, Jan-04, Volume: 3

    Topics: Azocines; beta-Endorphin; Binding, Competitive; Butorphanol; Cell Line; Colforsin; Cyclic AMP; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Etorphine; Fentanyl; Humans; Hydromorphone; Ligands; Morphine; Naltrexone; Phenazocine; Radioligand Assay; Receptors, Opioid, mu; Tritium

2003