Page last updated: 2024-09-03

quadazocine and dynorphins

quadazocine has been researched along with dynorphins in 10 studies

Compound Research Comparison

Studies
(quadazocine)
Trials
(quadazocine)
Recent Studies (post-2010)
(quadazocine)
Studies
(dynorphins)
Trials
(dynorphins)
Recent Studies (post-2010) (dynorphins)
81003,09624514
8100368415

Protein Interaction Comparison

ProteinTaxonomyquadazocine (IC50)dynorphins (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.0077
Kappa-type opioid receptorHomo sapiens (human)0.0001

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19905 (50.00)18.7374
1990's5 (50.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gannon, RL; Terrian, DM1
Agura, V; DeWitt, DS; Faden, AI; Hayes, RL; McIntosh, TK1
Faden, AI; Fernyak, S; McIntosh, TK1
Adler, MW; Geller, EB; Tiseo, PJ1
Huidobro-Toro, JP; Way, EL; Yoshimura, K1
Billington, CJ; Gosnell, BA; Levine, AS; Morley, JE1
Butelman, ER; Ko, MC; Woods, JH1
Butelman, ER; Harris, TJ; Kreek, MJ; Perez, A1
Butelman, ER; Harris, TJ; Kreek, MJ1
Adapa, ID; Auh, JS; Berzetei-Gurske, IP; Brandt, SR; Craymer, K; Farrington, L; Haggart, D; Kennedy, JM; O'Brien, A; Polgar, WE; Rodriguez, L; Schwartz, RW; Toll, L; White, A1

Other Studies

10 other study(ies) available for quadazocine and dynorphins

ArticleYear
Kappa opioid agonists inhibit transmitter release from guinea pig hippocampal mossy fiber synaptosomes.
    Neurochemical research, 1992, Volume: 17, Issue:8

    Topics: Animals; Azocines; Calcium; Dynorphins; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; Glutamates; Glutamic Acid; Guinea Pigs; Hippocampus; Male; Potassium; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Synaptosomes

1992
Endogenous opioids may mediate secondary damage after experimental brain injury.
    The American journal of physiology, 1987, Volume: 253, Issue:5 Pt 1

    Topics: Animals; Azocines; Blood Flow Velocity; Blood Pressure; Brain; Brain Injuries; Cats; Cerebrovascular Circulation; Dopamine; Dynorphins; Electroencephalography; Endorphins; Enkephalin, Leucine; Female; Intracranial Pressure; Isomerism; Male; Narcotic Antagonists

1987
Endogenous opioids, opiate receptors and traumatic brain injury.
    NIDA research monograph, 1986, Volume: 75

    Topics: Animals; Azocines; beta-Endorphin; Brain Chemistry; Brain Injuries; Cats; Cerebrovascular Circulation; Dynorphins; Female; Male; Narcotic Antagonists; Receptors, Opioid

1986
Antinociceptive action of intracerebroventricularly administered dynorphin and other opioid peptides in the rat.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Azocines; Cold Temperature; Drug Interactions; Dynorphins; Enkephalins; Injections, Intraventricular; Male; Naloxone; Pyrrolidines; Rats; Rats, Inbred Strains; Reaction Time; Receptors, Opioid

1988
Potency of three opiate antagonists to reverse the inhibitory activity of dynorphin, enkephalins and opioid-like alkaloids on the guinea pig ileum.
    European journal of pharmacology, 1982, Oct-15, Volume: 84, Issue:1-2

    Topics: Animals; Azocines; Benzomorphans; Cyclazocine; Dynorphins; Endorphins; Enkephalins; Ethylketocyclazocine; Guinea Pigs; Ileum; In Vitro Techniques; Male; Morphine Derivatives; Muscle, Smooth; Naloxone; Narcotic Antagonists

1982
Which opioid receptor mechanism modulates feeding?
    Appetite, 1984, Volume: 5, Issue:1

    Topics: Animals; Azocines; Diprenorphine; Dynorphins; Endorphins; Feeding Behavior; Humans; Mice; Naloxone; Naltrexone; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, sigma

1984
Activation of peripheral kappa opioid receptors inhibits capsaicin-induced thermal nociception in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Azocines; Benzomorphans; Capsaicin; Dynorphins; Female; Hot Temperature; Ligands; Macaca mulatta; Male; Naltrexone; Narcotic Antagonists; Pain Measurement; Peptide Fragments; Receptors, Opioid, kappa

1999
Effects of systemically administered dynorphin A(1-17) in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:2

    Topics: Analgesics, Opioid; Animals; Azocines; Behavior, Animal; Conditioning, Operant; Cytokines; Dose-Response Relationship, Drug; Dynorphins; Female; Inflammation; Injections, Intravenous; Macaca mulatta; Male; Narcotic Antagonists; Pain Measurement; Prolactin; Reinforcement Schedule

1999
Effects of E-2078, a stable dynorphin A(1-8) analog, on sedation and serum prolactin levels in rhesus monkeys.
    Psychopharmacology, 1999, Volume: 147, Issue:1

    Topics: Animals; Azocines; Dose-Response Relationship, Drug; Dynorphins; Female; Hypnotics and Sedatives; Injections, Subcutaneous; Macaca mulatta; Male; Motor Activity; Muscle Relaxation; Naltrexone; Narcotic Antagonists; Peptide Fragments; Prolactin; Pyrrolidines; Receptors, Opioid, kappa; Time Factors

1999
Standard binding and functional assays related to medications development division testing for potential cocaine and opiate narcotic treatment medications.
    NIDA research monograph, 1998, Volume: 178

    Topics: Animals; Aorta, Thoracic; Cocaine; Cyclic AMP; Electric Stimulation; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Male; Mice; Muscle, Smooth; Opioid-Related Disorders; Rats; Receptors, Dopamine; Receptors, Opioid; Receptors, Serotonin; Substance-Related Disorders

1998