pyrroles and s 33084
pyrroles has been researched along with s 33084 in 14 studies
Research
Studies (14)
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 11 (78.57) | 29.6817 |
2010's | 3 (21.43) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors
Authors | Studies |
---|---|
Cussac, D; Millan, MJ; Newman-Tancredi, A; Sezgin, L | 2 |
Audinot, V; Cussac, D; Dubuffet, T; Gobert, A; Lavielle, G; Lejeune, F; Millan, MJ; Newman-Tancredi, A; Rivet, JM | 1 |
Brocco, M; Dekeyne, A; Dubuffet, T; Lavielle, G; Millan, MJ; Rivet, JM | 1 |
Biala, G; Duarte, C; Hamon, M; Le Bihan, C; Thiébot, MH | 1 |
Hanger, D; Joyce, JN; Reploge, M; Yarkov, AV | 1 |
Brotchie, JM; Crossman, AR; Millan, MJ; Nicholson, SL; Ravenscroft, P; Silverdale, MA | 1 |
Gyertyán, I; Sághy, K | 1 |
Kolasiewicz, W; Maj, J; Ossowska, K | 1 |
Loiseau, F; Millan, MJ | 1 |
Brotchie, JM; Fox, SH; Johnston, T; Millan, MJ; Reyes, G; Visanji, NP | 1 |
Brocco, M; Mela, F; Millan, MJ; Morari, M | 1 |
Fan, X; Hess, EJ; Xu, M | 1 |
Fone, KC; Ingallinesi, M; Loiseau, F; Marsden, CA; Millan, MJ; Watson, DJ | 1 |
Other Studies
14 other study(ies) available for pyrroles and s 33084
Article | Year |
---|---|
The novel antagonist, S33084, and GR218,231 interact selectively with cloned and native, rat dopamine D(3) receptors as compared with native, rat dopamine D(2) receptors.
Topics: Animals; Benzopyrans; Binding, Competitive; CHO Cells; Cricetinae; Dopamine Antagonists; Olfactory Pathways; Oxazines; Pyrroles; Rats; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombinant Proteins; Spiperone; Sulfones; Tetrahydronaphthalenes | 2000 |
[3H]S33084: a novel, selective and potent radioligand at cloned, human dopamine D3 receptors.
Topics: Animals; Benzopyrans; Binding, Competitive; Cells, Cultured; CHO Cells; Cricetinae; Dopamine Antagonists; Humans; Pyrroles; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombinant Proteins; Spiperone; Transfection; Tritium | 2000 |
S33084, a novel, potent, selective, and competitive antagonist at dopamine D(3)-receptors: I. Receptorial, electrophysiological and neurochemical profile compared with GR218,231 and L741,626.
Topics: Animals; Benzopyrans; Brain; Dopamine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Enzyme Activation; Guanosine 5'-O-(3-Thiotriphosphate); Indoles; Male; Mitogen-Activated Protein Kinases; Norepinephrine; Oxazines; Piperidines; Pyrroles; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Serotonin; Sulfones; Tetrahydronaphthalenes | 2000 |
S33084, a novel, potent, selective, and competitive antagonist at dopamine D(3)-receptors: II. Functional and behavioral profile compared with GR218,231 and L741,626.
Topics: Animals; Behavior, Animal; Benzopyrans; Body Temperature; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Extrapyramidal Tracts; Indoles; Male; Mice; Motor Activity; Oxazines; Piperidines; Psychotropic Drugs; Pyrroles; Rats; Rats, Wistar; Receptors, Dopamine D3; Sulfones; Tetrahydronaphthalenes | 2000 |
Respective roles of dopamine D2 and D3 receptors in food-seeking behaviour in rats.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amisulpride; Analysis of Variance; Animals; Apomorphine; Benzazepines; Benzopyrans; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Synergism; Feeding Behavior; Haloperidol; Male; Naphthalenes; Pyrroles; Pyrrolidines; Quinolines; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Reinforcement, Psychology; Sulpiride; Tetrahydronaphthalenes | 2003 |
Behavioral effects of dopamine agonists and antagonists in MPTP-lesioned D3 receptor knockout mice.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Apomorphine; Autoradiography; Behavior, Animal; Benzopyrans; Carbidopa; Cocaine; Dopamine Agents; Dopamine Agonists; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Female; Grooming; Levodopa; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Inbred C57BL; Mice, Knockout; Motor Activity; Nerve Tissue Proteins; Oxazines; Pyrroles; Radiopharmaceuticals; Receptors, Dopamine D2; Receptors, Dopamine D3; Stereotyped Behavior | 2003 |
Selective blockade of D(3) dopamine receptors enhances the anti-parkinsonian properties of ropinirole and levodopa in the MPTP-lesioned primate.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Benzopyrans; Brain; Callithrix; Disease Models, Animal; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Synergism; Drug Therapy, Combination; Indoles; Levodopa; Parkinsonian Disorders; Pyrroles; Receptors, Dopamine D2; Receptors, Dopamine D3 | 2004 |
The selective dopamine D3 receptor antagonists, SB 277011-A and S 33084 block haloperidol-induced catalepsy in rats.
Topics: Animals; Benzopyrans; Catalepsy; Haloperidol; Male; Nitriles; Pyrroles; Rats; Rats, Wistar; Receptors, Dopamine D3; Tetrahydroisoquinolines | 2007 |
The involvement of cerebellar dopamine D3 receptors in locomotor activity of rats.
Topics: Animals; Behavior, Animal; Benzopyrans; Cerebellum; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Administration Routes; Drug Interactions; Male; Motor Activity; Pyrroles; Rats; Rats, Wistar; Receptors, Dopamine D3; Tetrahydronaphthalenes | 2008 |
Blockade of dopamine D(3) receptors in frontal cortex, but not in sub-cortical structures, enhances social recognition in rats: similar actions of D(1) receptor agonists, but not of D(2) antagonists.
Topics: Animals; Benzazepines; Benzopyrans; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Indoles; Male; Microinjections; Nitriles; Piperidines; Prefrontal Cortex; Pyrroles; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D3; Recognition, Psychology; Social Behavior; Tetrahydroisoquinolines | 2009 |
Dopamine D3 receptor stimulation underlies the development of L-DOPA-induced dyskinesia in animal models of Parkinson's disease.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Antiparkinson Agents; Benzopyrans; Callithrix; Corpus Striatum; Disease Models, Animal; Dopamine and cAMP-Regulated Phosphoprotein 32; Dopamine Antagonists; Dyskinesia, Drug-Induced; Enkephalins; Female; Levodopa; Male; Oxidopamine; Parkinsonian Disorders; Protein Precursors; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger | 2009 |
The selective D(3) receptor antagonist, S33084, improves parkinsonian-like motor dysfunction but does not affect L-DOPA-induced dyskinesia in 6-hydroxydopamine hemi-lesioned rats.
Topics: Animals; Antiparkinson Agents; Benzopyrans; Disability Evaluation; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Dyskinesia, Drug-Induced; Hypokinesia; Levodopa; Male; Oxidopamine; Parkinsonian Disorders; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D3; Time Factors; Treatment Outcome | 2010 |
D2 dopamine receptor subtype-mediated hyperactivity and amphetamine responses in a model of ADHD.
Topics: Amphetamine; Animals; Attention Deficit Disorder with Hyperactivity; Benzopyrans; Corpus Striatum; Dihydroxyphenylalanine; Disease Models, Animal; Dopamine; Dopamine Agents; Dopamine D2 Receptor Antagonists; Extracellular Space; Indoles; Locomotion; Mice; Mice, Knockout; Mice, Mutant Strains; Piperidines; Pyridines; Pyrroles; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Dopamine D4 | 2010 |
Selective blockade of dopamine D3 receptors enhances while D2 receptor antagonism impairs social novelty discrimination and novel object recognition in rats: a key role for the prefrontal cortex.
Topics: Animals; Benzopyrans; Discrimination, Psychological; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Indoles; Male; Mice; Mice, Knockout; Microinjections; Piperidines; Prefrontal Cortex; Pyrroles; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Recognition, Psychology | 2012 |