pyrroles has been researched along with l 750667 in 11 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (18.18) | 18.2507 |
2000's | 7 (63.64) | 29.6817 |
2010's | 2 (18.18) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Curtis, NR; Emms, F; Freedman, SB; Kulagowski, JJ; Leeson, PD; Marston, D; Marwood, R; Patel, S | 1 |
Chumpradit, S; Kung, HF; Kung, MP; Stevenson, DA; Sun, XM; Vessotskie, JM; Zhuang, ZP | 1 |
Benjamin, PS; Schetz, JA; Sibley, DR | 1 |
Al Tikriti, MS; Baldwin, RM; Eshima, L; Fujita, M; Innis, RB; Lu, L; Roe, D; Seibyl, JP; Staley, JK; Tamagnan, G; Thornback, J | 1 |
Pittman, QJ; Price, CJ | 1 |
Chapman, KL; Hutson, PH; Marston, D; Patel, S; Ragan, CI | 1 |
Chen, S; Floresca, CZ; Kortagere, S; Schetz, JA | 1 |
Anderson, SM; Pierce, RC; Schmidt, HD | 1 |
Hashimoto, K; Higashi, T; Matsushita, S; Nakano, K; Takagi, R; Tanaka, Y | 1 |
Kaneko, A; Kawano, M; Matsushita, S; Takagi, R | 1 |
Chang, SE; Hwang, JS; Jung, JM; Kim, SY; Lee, WJ | 1 |
11 other study(ies) available for pyrroles and l 750667
Article | Year |
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Identification and pharmacological characterization of [125I]L-750,667, a novel radioligand for the dopamine D4 receptor.
Topics: Animals; Cell Line; Dopamine Antagonists; Humans; Iodine Radioisotopes; Kinetics; Pyridines; Pyrroles; Radioligand Assay; Rats; Receptors, Dopamine D2; Receptors, Dopamine D4 | 1996 |
Characterization of a novel iodinated ligand, IPMPP, for human dopamine D4 receptors expressed in CHO cells.
Topics: Animals; Binding, Competitive; CHO Cells; Cricetinae; Dopamine Agonists; Guanine Nucleotides; Humans; Magnesium; Pyridines; Pyrroles; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins | 1997 |
Nonconserved residues in the second transmembrane-spanning domain of the D(4) dopamine receptor are molecular determinants of D(4)-selective pharmacology.
Topics: Animals; Binding Sites; COS Cells; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Ligands; Membrane Proteins; Mutagenesis, Site-Directed; Protein Conformation; Pyridines; Pyrroles; Rats; Receptors, Dopamine D2; Receptors, Dopamine D4; Structure-Activity Relationship; Transfection | 2000 |
SPECT imaging with the D(4) receptor antagonist L-750,667 in nonhuman primate brain.
Topics: Animals; Basal Ganglia; Binding, Competitive; Brain; Brain Stem; Cerebellum; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Frontal Lobe; Gyrus Cinguli; Imidazoles; Iodine Radioisotopes; Occipital Lobe; Organ Specificity; Papio; Parietal Lobe; Pyridines; Pyrimidines; Pyrroles; Receptors, Dopamine D4; Temporal Lobe; Tissue Distribution; Tomography, Emission-Computed, Single-Photon | 2000 |
Dopamine D4 receptor activation inhibits presynaptically glutamatergic neurotransmission in the rat supraoptic nucleus.
Topics: Animals; Benzamides; Benzazepines; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Glutamic Acid; Male; Patch-Clamp Techniques; Piperazines; Presynaptic Terminals; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D4; Sulpiride; Supraoptic Nucleus; Synaptic Transmission | 2001 |
Pharmacological and functional characterisation of dopamine D4 receptors in the rat retina.
Topics: Animals; Binding Sites; Cyclic AMP; Darkness; Dopamine Agonists; Dopamine Antagonists; In Vitro Techniques; Indoles; Male; Piperidines; Pyridines; Pyrroles; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D4; Retina; Spiperone | 2003 |
Reciprocal mutations in TM2/TM3 in a D2 dopamine receptor background confirms the importance of this microdomain as a selective determinant of para-halogenated 1,4-disubstituted aromatic piperazines.
Topics: Animals; Chemistry, Pharmaceutical; Chlorocebus aethiops; COS Cells; Membrane Microdomains; Membrane Transport Proteins; Mutation; Piperazine; Piperazines; Pyrazoles; Pyridines; Pyrroles; Rats; Receptors, Dopamine D2; Spiperone; Tritium | 2005 |
Administration of the D2 dopamine receptor antagonist sulpiride into the shell, but not the core, of the nucleus accumbens attenuates cocaine priming-induced reinstatement of drug seeking.
Topics: Analysis of Variance; Animals; Behavior, Addictive; Behavior, Animal; Cocaine; Conditioning, Operant; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Extinction, Psychological; Indans; Male; Microinjections; Nucleus Accumbens; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Reinforcement Schedule; Self Administration; Sulpiride | 2006 |
Antagonizing dopamine D1-like receptor inhibits Th17 cell differentiation: preventive and therapeutic effects on experimental autoimmune encephalomyelitis.
Topics: Adoptive Transfer; Animals; Benzazepines; Cell Differentiation; Cell Polarity; Dendritic Cells; Disease Models, Animal; Encephalomyelitis, Autoimmune, Experimental; Female; Humans; Interleukin-17; Lymphocyte Activation; Mice; Pyridines; Pyrroles; Receptors, Dopamine D1; T-Lymphocytes, Helper-Inducer | 2008 |
Berberine is a dopamine D1- and D2-like receptor antagonist and ameliorates experimentally induced colitis by suppressing innate and adaptive immune responses.
Topics: Adaptive Immunity; Animals; Benzazepines; Berberine; Bone Marrow; Colitis; Cytokines; Dendritic Cells; Dextran Sulfate; Disease Models, Animal; Dopamine Antagonists; Immunity, Innate; Lipopolysaccharides; Lymph Nodes; Lymphocytes; Macrophages; Mice; Mice, Inbred C57BL; Protein Binding; Pyridines; Pyrroles; Receptors, Dopamine; Receptors, Serotonin; Time Factors | 2015 |
Dopamine D4 receptor antagonist inhibits melanogenesis through transcriptional downregulation of MITF via ERK signalling.
Topics: Cell Survival; Dopamine; Dose-Response Relationship, Drug; Down-Regulation; Extracellular Signal-Regulated MAP Kinases; Humans; Melanins; Melanocytes; Microphthalmia-Associated Transcription Factor; Pyridines; Pyrroles; Receptors, Dopamine D4; RNA, Messenger; Signal Transduction | 2016 |