Page last updated: 2024-08-18

pyrroles and cp 154526

pyrroles has been researched along with cp 154526 in 117 studies

Research

Studies (117)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's9 (7.69)18.2507
2000's67 (57.26)29.6817
2010's38 (32.48)24.3611
2020's3 (2.56)2.80

Authors

AuthorsStudies
Braselton, JP; Chen, YL; Collins, J; Corman, M; Dunaiskis, A; Faraci, S; Heym, J; Mansbach, RS; Schmidt, AW; Schulz, DW; Seeger, T; Seymour, P; Sprouse, J; Tingley, FD; Winston, EN1
Bartfai, T; Chai, Z; Hasanvan, H; Jenck, F; Lundkvist, J; Moreau, JL; Teheranian, R; Widmer, U1
Brooks, EN; Chen, YL; Mansbach, RS1
Brooks, E; Chen, YL; Collins, J; Corman, ML; Dunaiskis, AR; Faraci, WS; Gallaschun, RJ; Mansbach, RS; Schmidt, A; Schulz, DW; Winter, SM1
Buczek, Y; Erb, S; Leung, S; Shaham, Y; Stewart, J1
Griebel, G; Perrault, G; Sanger, DJ1
Grigoriadis, DE; Heinrichs, SC; McCarthy, JR1
Berridge, CW; Dikkes, P; Dunn, AJ; Majzoub, JA; Miczek, KA; Muglia, LJ; Swiergiel, AH; Weninger, SC1
Banks, MC; Huhman, KL; Jasnow, AM; Owens, EC1
Miyata, K; Yamano, M; Yasuda, S; Yuki, H1
Alvaro, JD; Chen, YL; Duman, RS; Iredale, PA; Lee, Y; Terwilliger, R1
Kawahara, H; Kawahara, Y; Westerink, BH1
Bruijnzeel, A; Croiset, G; de Wied, D; Diamant, M; Nijsen, MJ; Stam, R; Wiegant, VM1
Cassella, JV; Coverdale, S; Hoffman, DC; Kehne, JH; McCloskey, TC1
Brown, J; Connor, HE; Giles, H; Parsons, SJ; Rees, S; Rhodes, SA1
Arborelius, L; Owens, MJ; Plotsky, PM; Schulz, DW; Skelton, KH; Thrivikraman, KV1
Harding, S; Juzytsch, W; Lê, AD; Shaham, Y; Shalev, U; Watchus, J1
Ceng, X; Huang, M; Lu, L1
Goeders, NE; Guerin, GF1
Davidson, A; Finlay, TH; Funai, EF; O'Neill, LM; Roqué, H1
Akiyoshi, J; Hikichi, T; Isogawa, K; Nagayama, H; Tsutsumi, T; Yamamoto, Y1
Gauthier, A; Maillot, C; Million, M; Taché, Y; Wei, JY1
Ceng, X; Liu, D; Lu, L; Ma, L1
Ceng, X; Liu, D; Lu, L1
Imaki, J; Imaki, T; Katsumata, H; Minami, S; Miyata, M; Naruse, M1
Hirata, M; Murakami, Y; Okada, S; Yokotani, K1
Chaki, S; Kameo, K; Kawashima, N; Nakazato, A; Takamori, K1
Brocco, M; Casara, P; Dekeyne, A; Dorey, G; Gobert, A; Millan, MJ1
Bernardini, R; Cantarella, G; Chiarenza, A; Lempereur, L; Lombardo, G; Pafumi, C; Zappalà, G1
Martínez, V; Rivier, JE; Taché, Y; Wang, L1
Goeders, NE; Gurkovskaya, O1
Maillot, C; Million, M; Rivier, J; Saunders, P; Taché, Y; Vale, W1
Bruelisauer, A; Enz, A; Keller, C; Lemaire, M1
Maillot, C; Miampamba, M; Million, M; Taché, Y1
Clampitt, DM; Goeders, NE1
Blank, T; Nijholt, I; Spiess, J; Vollstaedt, S1
Schmidt, AW; Schulz, DW; Seymour, PA1
Blessing, WW; Nalivaiko, E2
Huang, M; Liu, Z; Lu, L; Zhang, Z1
Okada, S; Shimizu, T; Yokotani, K1
Facci, L; Franceschini, D; Pangallo, M; Skaper, SD; Stevens, DA; Strijbos, PJ1
Bradesi, S; Mayer, EA; McRoberts, JA; Miller, JC; Ohning, G; Sablad, M; Schwetz, I; Zhou, H1
Berggård, C; Damberg, M; Eller, M; Harro, J; Mällo, T; Oreland, L1
Hager, P; Hagman, B; Strömmer, L; Wikström, AC1
Hogg, S; Keeney, A; Overstreet, DH1
Dominguez, G; Kuhar, MJ1
Anisman, H; Khan, S; Merali, Z; Michaud, DS; Shippy, SA1
Houshyar, H; Hsin, LW; Jutkiewicz, EM; Rice, KC; Wood, SK; Woods, JH1
Breese, GR; Knapp, DJ; Navarro, M; Overstreet, DH1
Chen, XQ; Du, JZ; Wang, TY; Xu, JF1
Dettloff, SL; Jones, JE; Seymour, PL; Wade, GN1
Baccei, CS; Bristow, LJ; Correa, LD; Lorrain, DS1
Goeders, NE; Gurkovskaya, OV; Palamarchouk, V; Smagin, G1
Chen, XQ; Du, JZ; Xu, JF1
Filip, M; Frankowska, M; Papla, I; Przegaliński, E; Zaniewska, M1
Khan, S; Plamondon, H1
Bonaz, B; Canini, F; Meregnani, J; Peinnequin, A; Pellissier, S; Porcher, C; Sinniger, V1
Fang, Q; Liu, Z; Lu, L; Wang, J1
Gannon, RL; Millan, MJ1
Blanton, MG; Hicks, MP; Janak, PH; Kinder, JR; Kullberg, EF; Mcgeehan, AJ; Olive, MF; Sahuque, LL1
Keller, PA; McCluskey, A; Morgan, J; O'connor, SM1
Goeders, NE; Moffett, MC1
Ramos, AT; Troncone, LR; Tufik, S1
Chaki, S; Iijima, M1
Guthrie, DH; Guzzi, MF; Higgins, GA; Hodgson, RA; Lu, SX; Mullins, DE; Parker, EM; Pond, AJ; Varty, GB1
Chen, XQ; Dong, J; Du, JZ; Fan, JM; Niu, CY1
Fee, JR; Picker, MJ; Sparta, DR; Thiele, TE1
Fee, JR; Knapp, DJ; Lowery, EG; Sparrow, AM; Sparta, DR; Thiele, TE1
Breese, GR; Knapp, DJ; Lowery, EG; Sparrow, AM; Thiele, TE1
Bradesi, S; Larauche, M; Mayer, EA; McLean, P; McRoberts, JA; Million, M; Taché, Y1
Chen, XQ; Du, JZ; He, JJ; Wang, L; Xu, JF1
Burkhart-Kasch, S; Coste, SC; McKinnon, CS; Pastor, R; Phillips, TJ; Reed, C; Ryabinin, AE; Scibelli, AC; Stenzel-Poore, MP1
Fukudo, S; Hasegawa, R; Ito, H; Nagura, Y; Saito-Nakaya, K1
Breese, GR; Fee, JR; Ferraro, FM; Knapp, DJ; Sparta, DR; Thiele, TE1
Berga, SL; Kaplan, JR; Michopoulos, V; Wilson, ME1
Inagaki, H; Kiyokawa, Y; Mori, Y; Takeuchi, Y1
Hodge, CW; Lowery, EG; Lyons, AM; Navarro, M; Spanos, M; Thiele, TE1
Cummons, T; Harrison, JE; Hummel, M; Kennedy, JD; Lu, P; Mark, L; Whiteside, GT1
Cooper, MA; Huhman, KL1
Baimoukhametova, DV; Bains, JS; Kuzmiski, JB; Marty, V1
Conti, LH; Sutherland, JE1
Contoreggi, C; Eckelman, WC; Jagoda, EM; Kiesewetter, DO; Kim, BM; Lang, L; Ma, Y; McCullough, K; Rice, KC; Szajek, LP1
Boyson, CO; Debold, JF; Miczek, KA; Miguel, TT; Quadros, IM1
Kiyokawa, Y; Kobayashi, T; Mori, Y; Takeuchi, Y1
Brielmaier, J; McDonald, CG; Smith, RF1
Aston-Jones, G; Smith, RJ1
Cook, JM; Groenink, L; Hendriksen, H; Huang, S; Millan, MJ; Olivier, B; Rallipalli, S; van Oorschot, R; Vinkers, CH1
Debold, JF; Hwa, LS; Miczek, KA1
Almela, P; García-Carmona, JA; Hidalgo, J; Laorden, ML; Milanés, MV; Mora, L; Navarro-Zaragoza, J1
Andrés, ME; Araya, KA; Carreño, P; Fuentealba, JA; Gysling, K; Renard, GM; Sotomayor-Zárate, R1
Bifone, A; Gozzi, A; Lepore, S; Merlo-Pich, E; Vicentini, E1
Boulay, D; Douma, TN; Griebel, G; Groenink, L; Millan, MJ; Olivier, B; Verdouw, PM; Westphal, KG1
Homem, KS; Ramos, Ade T; Suchecki, D; Troncone, LR; Tufik, S1
Grachev, P; Hu, MH; Li, SY; Li, XF; Lightman, SL; Millar, RP; O'Byrne, KT1
Fan, Q; Hou, Y; Li, H; Nie, W; Sun, R; Wang, A; Yu, Z1
Carlson, J; DeBold, JF; Hwa, LS; Miczek, KA; Quadros, IM; Shimamoto, A1
DeBold, JF; Hwa, LS; Kayyali, T; Miczek, KA; Norman, KJ; Shimamoto, A; Valentino, RJ1
Chen, J; Chen, XQ; Du, JZ; Evans, AM; Gao, YQ; Hao, K; Kong, FP; Lightman, SL; Tang, JW1
Fukudo, S; Kanazawa, M; Kano, M; Muratsubaki, T; Su, J; Tanaka, Y1
Laorden, ML; Lasheras, MC; Milanés, MV; Núñez, C1
Boerngen-Lacerda, R; Camarini, R; Correia, D; Martynhak, BJ; Pereira, M; Ribeiro, AF; Siba, IP1
Jiang, H; Li, C; Liu, D; Liu, Y; Lu, C; Pan, F; Yin, S1
Baas, JM; Bijlsma, EY; Groenink, L; Hendriksen, H; Millan, MJ1
Almela, P; Camejo, DM; García-Carmona, JA; Jiménez, A; Laorden, ML; Milanés, MV; Sevilla, F1
Aston-Jones, G; Cason, AM; Kohtz, A1
Groenink, L; Millan, MJ; Peeters, BW; van Esterik, JC; Verdouw, PM1
Spierling, SR; Zorrilla, EP1
DiMicco, JA; Rusyniak, DE; Sarkar, S; Zaretskaia, MV; Zaretsky, DV1
Aisenberg, N; Akirav, I; Sabban, EL; Serova, L1
Abbott, B; Baylie, RL; Board, TN; Bruhn-Olszewska, B; Jackson, TR; Jones, RC; Lawrence, KM; Locke, IC; Richardson, SM; Townsend, PA1
Jiang, H; Liu, D; Liu, Y; Pan, F; Xu, J1
Bayerl, DS; Bosch, OJ; Brunton, PJ; Gaßner, BM; Hübner, K; Klampfl, SM; Schramm, MM; Seasholtz, AF1
Almela, P; Laorden, ML; Martínez-Laorden, E; Milanés, MV; Navarro-Zaragoza, J1
Higashi, Y; Nagao, Y; Saito, M; Shimizu, S; Shimizu, T1
Almela, P; Cánovas, A; Gómez-Murcia, V; Laorden, ML; Martínez-Laorden, E; Milanés, MV; Navarro-Zaragoza, J; Teruel-Fernández, FJ1
Agoglia, AE; Bluitt, MN; Douglass, E; Hanback, T; Herman, MA; Hodge, CW; Quadir, SG; Tella, J; Ying, R; Zhu, M1

Reviews

4 review(s) available for pyrroles and cp 154526

ArticleYear
Recent advances with the CRF1 receptor: design of small molecule inhibitors, receptor subtypes and clinical indications.
    Current pharmaceutical design, 1999, Volume: 5, Issue:5

    Topics: Animals; Anxiety; Depression; Drug Design; Humans; Kinetics; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Seizures; Substance-Related Disorders

1999
The pharmacology of CP-154,526, a non-peptide antagonist of the CRH1 receptor: a review.
    CNS drug reviews, 2003,Spring, Volume: 9, Issue:1

    Topics: Animals; Anxiety; Autonomic Nervous System; Behavior, Animal; Depression; Digestive System; Disease Models, Animal; Drug Evaluation, Preclinical; Genitalia; Haplorhini; Immune System; Mice; Motor Skills; Neurodegenerative Diseases; Neurosecretory Systems; Pyrimidines; Pyrroles; Rats; Receptors, Corticotropin-Releasing Hormone

2003
The role of the HPA axis in psychiatric disorders and CRF antagonists as potential treatments.
    Archiv der Pharmazie, 2006, Volume: 339, Issue:7

    Topics: Amino Acid Sequence; Animals; Corticotropin-Releasing Hormone; Humans; Hypothalamo-Hypophyseal System; Mental Disorders; Molecular Sequence Data; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone

2006
Don't stress about CRF: assessing the translational failures of CRF
    Psychopharmacology, 2017, Volume: 234, Issue:9-10

    Topics: Animals; Behavior, Addictive; Corticotropin-Releasing Hormone; Depression; Humans; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Stress, Psychological; Substance-Related Disorders; Translational Research, Biomedical

2017

Trials

1 trial(s) available for pyrroles and cp 154526

ArticleYear
Inactivation of corticotropin-releasing hormone-induced insulinotropic role by high-altitude hypoxia.
    Diabetes, 2015, Volume: 64, Issue:3

    Topics: Adenosine Triphosphate; Adolescent; Adult; Altitude; Animals; Blood Glucose; Calcium; Corticosterone; Corticotropin-Releasing Hormone; Cyclic AMP; Humans; Hydrocortisone; Hypoxia; Insulin; Male; Pancreas; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Young Adult

2015

Other Studies

112 other study(ies) available for pyrroles and cp 154526

ArticleYear
CP-154,526: a potent and selective nonpeptide antagonist of corticotropin releasing factor receptors.
    Proceedings of the National Academy of Sciences of the United States of America, 1996, Sep-17, Volume: 93, Issue:19

    Topics: Acoustic Stimulation; Adenylyl Cyclases; Adrenocorticotropic Hormone; Animals; Binding, Competitive; Callithrix; Cell Line; Cell Membrane; Cerebral Cortex; Cerebral Ventricles; Corticotropin-Releasing Hormone; Dogs; Guinea Pigs; Humans; Injections, Intraventricular; Kinetics; Locus Coeruleus; Male; Neurons; Pituitary Gland; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Reflex, Startle

1996
A non peptidic corticotropin releasing factor receptor antagonist attenuates fever and exhibits anxiolytic-like activity.
    European journal of pharmacology, 1996, Aug-08, Volume: 309, Issue:2

    Topics: Analgesics, Non-Narcotic; Animals; Anti-Anxiety Agents; Fever; Interleukin-1; Male; Mice; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Recombinant Proteins; Tumor Cells, Cultured

1996
Antidepressant-like effects of CP-154,526, a selective CRF1 receptor antagonist.
    European journal of pharmacology, 1997, Mar-26, Volume: 323, Issue:1

    Topics: Analysis of Variance; Animals; Antidepressive Agents, Tricyclic; Depression; Disease Models, Animal; Helplessness, Learned; Imipramine; Injections, Intraperitoneal; Male; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone

1997
Synthesis and oral efficacy of a 4-(butylethylamino)pyrrolo[2,3-d]pyrimidine: a centrally active corticotropin-releasing factor1 receptor antagonist.
    Journal of medicinal chemistry, 1997, May-23, Volume: 40, Issue:11

    Topics: Animals; Anti-Anxiety Agents; Fear; Male; Molecular Structure; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Reflex, Startle; Structure-Activity Relationship

1997
CP-154,526, a selective, non-peptide antagonist of the corticotropin-releasing factor1 receptor attenuates stress-induced relapse to drug seeking in cocaine- and heroin-trained rats.
    Psychopharmacology, 1998, Volume: 137, Issue:2

    Topics: Animals; Cocaine; Corticotropin-Releasing Hormone; Heroin; Male; Pyrimidines; Pyrroles; Rats; Receptors, Corticotropin-Releasing Hormone; Self Administration; Stress, Psychological; Sucrose

1998
Characterization of the behavioral profile of the non-peptide CRF receptor antagonist CP-154,526 in anxiety models in rodents. Comparison with diazepam and buspirone.
    Psychopharmacology, 1998, Volume: 138, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Anxiety Disorders; Behavior, Animal; Buspirone; Diazepam; Male; Mice; Mice, Inbred BALB C; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone

1998
Stress-induced behaviors require the corticotropin-releasing hormone (CRH) receptor, but not CRH.
    Proceedings of the National Academy of Sciences of the United States of America, 1999, Jul-06, Volume: 96, Issue:14

    Topics: Animals; Avoidance Learning; Cerebral Ventricles; Conditioning, Operant; Corticotropin-Releasing Hormone; Crosses, Genetic; Electroshock; Fear; Female; Gene Expression Regulation; Injections, Intraventricular; Learning; Male; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Mice, Knockout; Motor Activity; Pain; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Reinforcement, Psychology; Stress, Psychological; Transcription, Genetic; Urocortins

1999
Differential effects of two corticotropin-releasing factor antagonists on conditioned defeat in male Syrian hamsters (Mesocricetus auratus).
    Brain research, 1999, Oct-30, Volume: 846, Issue:1

    Topics: Adrenocorticotropic Hormone; Aggression; Animals; Behavior, Animal; Corticotropin-Releasing Hormone; Cricetinae; Dominance-Subordination; Dose-Response Relationship, Drug; Male; Mesocricetus; Microinjections; Pyrimidines; Pyrroles; Stress, Psychological

1999
Corticotropin-releasing hormone receptors mediate consensus interferon-alpha YM643-induced depression-like behavior in mice.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 292, Issue:1

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Antidepressive Agents; Behavior, Animal; Depression, Chemical; Dose-Response Relationship, Drug; Drug Interactions; Imipramine; Indomethacin; Interferon-alpha; Male; Mice; Motor Activity; Naloxone; Narcotic Antagonists; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Time Factors

2000
Role of corticotropin-releasing factor receptor-1 in opiate withdrawal.
    Journal of neurochemistry, 2000, Volume: 74, Issue:1

    Topics: Animals; Behavior, Animal; Male; Morphine; Naltrexone; Narcotic Antagonists; Protein Isoforms; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Substance Withdrawal Syndrome

2000
The role of afferents to the locus coeruleus in the handling stress-induced increase in the release of noradrenaline in the medial prefrontal cortex: a dual-probe microdialysis study in the rat brain.
    European journal of pharmacology, 2000, Jan-17, Volume: 387, Issue:3

    Topics: Animals; Benzylamines; Bicuculline; Idazoxan; Locus Coeruleus; Male; Microdialysis; Norepinephrine; Phosphinic Acids; Piperazines; Prefrontal Cortex; Pyrimidines; Pyrroles; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Corticotropin-Releasing Hormone; Receptors, GABA; Receptors, Glutamate; Stress, Physiological

2000
The role of the CRH type 1 receptor in autonomic responses to corticotropin- releasing hormone in the rat.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2000, Volume: 22, Issue:4

    Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Autonomic Nervous System; Corticotropin-Releasing Hormone; Heart Rate; Male; Motor Activity; Neurosecretory Systems; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone

2000
Effects of the CRF(1) receptor antagonist, CP 154,526, in the separation-induced vocalization anxiolytic test in rat pups.
    Neuropharmacology, 2000, Jun-08, Volume: 39, Issue:8

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Antipsychotic Agents; Anxiety; Behavior, Animal; Buspirone; Clozapine; Desipramine; Diazepam; Dose-Response Relationship, Drug; Female; Haloperidol; Injections, Intraperitoneal; Male; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Social Isolation; Stress, Psychological; Vocalization, Animal; Zimeldine

2000
Use of a dual firefly and Renilla luciferase reporter gene assay to simultaneously determine drug selectivity at human corticotrophin releasing hormone 1 and 2 receptors.
    Analytical biochemistry, 2000, Jun-01, Volume: 281, Issue:2

    Topics: Animals; CHO Cells; Coleoptera; Cricetinae; Genes, Reporter; Humans; Luciferases; Protein Isoforms; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone

2000
Chronic administration of the selective corticotropin-releasing factor 1 receptor antagonist CP-154,526: behavioral, endocrine and neurochemical effects in the rat.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 294, Issue:2

    Topics: Adrenal Glands; Adrenocorticotropic Hormone; Animals; Anti-Anxiety Agents; Behavior, Animal; Brain; Corticosterone; Corticotropin-Releasing Hormone; Drug Administration Schedule; Endocrine System; Male; Organ Size; Pyrimidines; Pyrroles; Rats; Receptors, Corticotropin-Releasing Hormone; Reflex, Startle; RNA, Messenger; Stress, Physiological; Urocortins

2000
The role of corticotrophin-releasing factor in stress-induced relapse to alcohol-seeking behavior in rats.
    Psychopharmacology, 2000, Volume: 150, Issue:3

    Topics: Adrenalectomy; Alcoholism; Animals; Corticosterone; Corticotropin-Releasing Hormone; Electroshock; Extinction, Psychological; Injections, Intraventricular; Male; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Recurrence; Self Administration; Stress, Psychological

2000
Corticotropin-releasing factor receptor type I mediates stress-induced relapse to opiate dependence in rats.
    Neuroreport, 2000, Aug-03, Volume: 11, Issue:11

    Topics: Animals; Behavior, Animal; Conditioning, Psychological; Corticotropin-Releasing Hormone; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Male; Morphine; Neuropsychological Tests; Opioid-Related Disorders; Psychomotor Performance; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Secondary Prevention; Stress, Physiological

2000
Effects of the CRH receptor antagonist CP-154,526 on intravenous cocaine self-administration in rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2000, Volume: 23, Issue:5

    Topics: Animals; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Food; Male; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Reinforcement, Psychology; Self Administration

2000
A corticotropin releasing hormone receptor antagonist does not delay parturition in rats.
    Journal of perinatal medicine, 2000, Volume: 28, Issue:4

    Topics: Animals; Female; Gestational Age; Labor, Obstetric; Pregnancy; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone

2000
Suppression of conditioned fear by administration of CRF receptor antagonist CP-154,526.
    Pharmacopsychiatry, 2000, Volume: 33, Issue:5

    Topics: Animals; Conditioning, Psychological; Electroshock; Fear; Male; Motor Activity; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone

2000
Peripheral corticotropin-releasing factor and stress-stimulated colonic motor activity involve type 1 receptor in rats.
    Gastroenterology, 2000, Volume: 119, Issue:6

    Topics: Animals; Avoidance Learning; Colon; Corticotropin-Releasing Hormone; Defecation; Gastrointestinal Motility; Injections, Intraperitoneal; Injections, Intraventricular; Male; Myoelectric Complex, Migrating; Peptide Fragments; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Stress, Physiological; Urocortins; Water

2000
Differential roles of corticotropin-releasing factor receptor subtypes 1 and 2 in opiate withdrawal and in relapse to opiate dependence.
    The European journal of neuroscience, 2000, Volume: 12, Issue:12

    Topics: Animals; Cerebral Ventricles; Choice Behavior; Corticotropin-Releasing Hormone; Hormone Antagonists; Injections, Intraventricular; Male; Morphine; Morphine Dependence; Naloxone; Peptide Fragments; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Substance Withdrawal Syndrome

2000
Corticotropin-releasing factor receptor type 1 mediates stress-induced relapse to cocaine-conditioned place preference in rats.
    European journal of pharmacology, 2001, Volume: 415, Issue:2-3

    Topics: Animals; Cocaine; Cocaine-Related Disorders; Conditioning, Psychological; Corticotropin-Releasing Hormone; Dopamine Uptake Inhibitors; Hormone Antagonists; Male; Peptide Fragments; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Secondary Prevention; Stress, Physiological

2001
Expression of corticotropin-releasing hormone type 1 receptor in paraventricular nucleus after acute stress.
    Neuroendocrinology, 2001, Volume: 73, Issue:5

    Topics: Adrenocorticotropic Hormone; Animals; Corticotropin-Releasing Hormone; Gene Expression; In Situ Hybridization; Male; Oxytocin; Paraventricular Hypothalamic Nucleus; Proto-Oncogene Proteins c-fos; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; RNA, Messenger; Stress, Physiological; Vasopressins

2001
Role of brain arachidonic acid cascade on central CRF1 receptor-mediated activation of sympatho-adrenomedullary outflow in rats.
    European journal of pharmacology, 2001, May-11, Volume: 419, Issue:2-3

    Topics: Analysis of Variance; Animals; Arachidonic Acid; Brain; Corticotropin-Releasing Hormone; Epinephrine; Injections, Intraventricular; Male; Norepinephrine; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Urocortins

2001
Involvement of corticotropin-releasing factor subtype 1 receptor in the acquisition phase of learned helplessness in rats.
    Life sciences, 2001, Aug-03, Volume: 69, Issue:11

    Topics: Animals; Behavior, Animal; Dose-Response Relationship, Drug; Imipramine; Learning; Male; Pyridines; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone

2001
Anxiolytic properties of the selective, non-peptidergic CRF(1) antagonists, CP154,526 and DMP695: a comparison to other classes of anxiolytic agent.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2001, Volume: 25, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Dopamine; Dose-Response Relationship, Drug; Extracellular Space; Interpersonal Relations; Male; Norepinephrine; Postural Balance; Pyridines; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Serotonin; Vocalization, Animal

2001
Divergent effects of corticotropin releasing hormone on endothelial cell nitric oxide synthase are associated with different expression of CRH type 1 and 2 receptors.
    British journal of pharmacology, 2001, Volume: 134, Issue:4

    Topics: Animals; Blotting, Western; Cell Line; Cell Line, Transformed; Corticotropin-Releasing Hormone; Endothelium, Vascular; Gene Expression Regulation; Humans; Interleukin-1; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Nitrites; Peptide Fragments; Protein Isoforms; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Time Factors; Tumor Necrosis Factor-alpha

2001
Peripheral urocortin inhibits gastric emptying and food intake in mice: differential role of CRF receptor 2.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2001, Volume: 281, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Capsaicin; Corticotropin-Releasing Hormone; Eating; Fasting; Gastric Emptying; Humans; Male; Mice; Mice, Inbred C57BL; Peptide Fragments; Pyrazoles; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Urocortins

2001
Effects of CP-154,526 on responding during extinction from cocaine self-administration in rats.
    European journal of pharmacology, 2001, Nov-30, Volume: 432, Issue:1

    Topics: Animals; Behavior, Animal; Cocaine; Extinction, Psychological; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Reinforcement Schedule; Self Administration

2001
Human urocortin II, a new CRF-related peptide, displays selective CRF(2)-mediated action on gastric transit in rats.
    American journal of physiology. Gastrointestinal and liver physiology, 2002, Volume: 282, Issue:1

    Topics: Animals; Colon; Corticotropin-Releasing Hormone; Gastric Emptying; Humans; Male; Mammals; Peptide Fragments; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Restraint, Physical; Stress, Physiological; Urocortins

2002
Brain pharmacokinetics of a nonpeptidic corticotropin-releasing factor receptor antagonist.
    Drug metabolism and disposition: the biological fate of chemicals, 2002, Volume: 30, Issue:2

    Topics: Animals; Blood-Brain Barrier; Brain; Male; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone

2002
Peripheral CRF activates myenteric neurons in the proximal colon through CRF(1) receptor in conscious rats.
    American journal of physiology. Gastrointestinal and liver physiology, 2002, Volume: 282, Issue:5

    Topics: Acetylcholine; Animals; Colon; Consciousness; Corticotropin-Releasing Hormone; Injections, Intraperitoneal; Male; Myenteric Plexus; NADPH Dehydrogenase; Neurons; Proto-Oncogene Proteins c-fos; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone

2002
Potential role for the hypothalamo-pituitary-adrenal axis in the conditioned reinforcer-induced reinstatement of extinguished cocaine seeking in rats.
    Psychopharmacology, 2002, Volume: 161, Issue:3

    Topics: Analysis of Variance; Animals; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Corticosterone; Extinction, Psychological; Hypothalamo-Hypophyseal System; Ketoconazole; Male; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Reinforcement Schedule; Reinforcement, Psychology; Self Administration; Stress, Psychological

2002
The corticotropin-releasing factor receptor 1 antagonist CP-154,526 reverses stress-induced learning deficits in mice.
    Behavioural brain research, 2003, Jan-22, Volume: 138, Issue:2

    Topics: Animals; Arousal; Calcium-Calmodulin-Dependent Protein Kinases; Conditioning, Classical; Culture Techniques; Fear; Hippocampus; Hypothalamo-Hypophyseal System; Injections, Intraperitoneal; Long-Term Potentiation; Male; Mice; Mice, Inbred BALB C; Neuronal Plasticity; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Stress, Psychological

2003
CRF1-receptor antagonist CP-154526 reduces alerting-related cutaneous vasoconstriction in conscious rabbits.
    Neuroscience, 2003, Volume: 117, Issue:1

    Topics: Animals; Arousal; Blood Flow Velocity; Ear; Laser-Doppler Flowmetry; Male; Pain Measurement; Physical Stimulation; Pyrimidines; Pyrroles; Rabbits; Receptors, Corticotropin-Releasing Hormone; Vasoconstriction

2003
Dopamine-dependent responses to cocaine depend on corticotropin-releasing factor receptor subtypes.
    Journal of neurochemistry, 2003, Volume: 84, Issue:6

    Topics: Animals; Behavior, Animal; Cocaine; Corticotropin-Releasing Hormone; Dopamine; Extracellular Space; Hormone Antagonists; Male; Microdialysis; Motor Activity; Nucleus Accumbens; Peptide Fragments; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Spatial Behavior; Ventral Tegmental Area

2003
Extrahypothalamic corticotropin-releasing hormone mediates (-)-nicotine-induced elevation of plasma corticosterone in rats.
    European journal of pharmacology, 2003, Jul-25, Volume: 473, Issue:2-3

    Topics: Animals; Corticosterone; Corticotropin-Releasing Hormone; Cyclooxygenase Inhibitors; Indomethacin; Male; Microdialysis; Nicotine; Norepinephrine; Paraventricular Hypothalamic Nucleus; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Time Factors

2003
Corticotropin-releasing factor (CRF) and related peptides confer neuroprotection via type 1 CRF receptors.
    Neuropharmacology, 2003, Volume: 45, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; Amphibian Proteins; Amyloid beta-Peptides; Animals; Animals, Newborn; Apoptosis; Blotting, Western; Cell Survival; Cells, Cultured; Cerebellum; Cerebral Cortex; Chromatin; Chromones; Colforsin; Corticotropin-Releasing Hormone; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Glycogen Synthase Kinase 3; Hippocampus; In Situ Nick-End Labeling; Inhibitory Concentration 50; L-Lactate Dehydrogenase; Mitogen-Activated Protein Kinase Kinases; Morpholines; Neurons; Neuroprotective Agents; Peptide Fragments; Peptide Hormones; Peptides; Phosphorylation; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Thionucleotides; Time Factors; Urocortins; Urotensins; Vasodilator Agents

2003
Delayed stress-induced colonic hypersensitivity in male Wistar rats: role of neurokinin-1 and corticotropin-releasing factor-1 receptors.
    American journal of physiology. Gastrointestinal and liver physiology, 2004, Volume: 286, Issue:4

    Topics: Animals; Colon; Electromyography; Fear; Hypersensitivity, Delayed; Immunohistochemistry; Indoles; Isoindoles; Male; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Nociceptors; Physical Stimulation; Piperidines; Pyrimidines; Pyrroles; Quinuclidines; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Receptors, Neurokinin-1; Stress, Psychological; Sympathectomy, Chemical; Sympathetic Nervous System

2004
Effect of long-term blockade of CRF(1) receptors on exploratory behaviour, monoamines and transcription factor AP-2.
    Pharmacology, biochemistry, and behavior, 2004, Volume: 77, Issue:4

    Topics: Animals; Biogenic Monoamines; Brain; DNA-Binding Proteins; Exploratory Behavior; Male; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Transcription Factor AP-2; Transcription Factors

2004
CRF-receptor 1 blockade attenuates acute posttraumatic hyperglycemia in rats.
    The Journal of surgical research, 2004, Jun-01, Volume: 119, Issue:1

    Topics: Acute Disease; Adrenocorticotropic Hormone; Animals; Biological Transport; Blood Glucose; Corticosterone; Dexamethasone; Glucocorticoids; Glucose; Hyperglycemia; Insulin; Male; Muscle, Skeletal; Phosphatidylinositol 3-Kinases; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Wounds and Injuries

2004
Antidepressant effects of citalopram and CRF receptor antagonist CP-154,526 in a rat model of depression.
    European journal of pharmacology, 2004, May-25, Volume: 492, Issue:2-3

    Topics: Animals; Antidepressive Agents; Behavior, Animal; Citalopram; Depression; Disease Models, Animal; Dose-Response Relationship, Drug; Pyrimidines; Pyrroles; Rats; Rats, Inbred Strains; Receptors, Corticotropin-Releasing Hormone; Social Behavior; Swimming

2004
Transcriptional regulation of the CART promoter in CATH.a cells.
    Brain research. Molecular brain research, 2004, Jul-05, Volume: 126, Issue:1

    Topics: Animals; Cell Line; Colforsin; Corticotropin-Releasing Hormone; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Gene Expression Regulation; Locus Coeruleus; Mice; Mutagenesis, Site-Directed; Nerve Tissue Proteins; Neurotransmitter Agents; Promoter Regions, Genetic; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; RNA, Messenger; Transcription, Genetic

2004
Does amygdaloid corticotropin-releasing hormone (CRH) mediate anxiety-like behaviors? Dissociation of anxiogenic effects and CRH release.
    The European journal of neuroscience, 2004, Volume: 20, Issue:1

    Topics: Amygdala; Animals; Anti-Anxiety Agents; Anxiety; Avoidance Learning; Behavior, Animal; Bombesin; Brain Chemistry; Corticotropin-Releasing Hormone; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Eating; Electroshock; Environment; Glutamic Acid; Hormone Antagonists; Male; Microdialysis; Peptide Fragments; Pyrimidines; Pyrroles; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone

2004
CRF1 receptor antagonist CP-154,526 reduces cardiovascular responses during acute psychological stress in rabbits.
    Brain research, 2004, Aug-13, Volume: 1017, Issue:1-2

    Topics: Adrenergic beta-Antagonists; Animals; Blood Pressure; Electroencephalography; Heart Rate; Propranolol; Pyrimidines; Pyrroles; Rabbits; Receptors, Corticotropin-Releasing Hormone; Stress, Psychological

2004
The effects of CRF antagonists, antalarmin, CP154,526, LWH234, and R121919, in the forced swim test and on swim-induced increases in adrenocorticotropin in rats.
    Psychopharmacology, 2005, Volume: 180, Issue:2

    Topics: Adrenocorticotropic Hormone; Animals; Antidepressive Agents; Corticotropin-Releasing Hormone; Hypothalamo-Hypophyseal System; Male; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Restraint, Physical; Stress, Psychological; Swimming; Triazoles

2005
Prior multiple ethanol withdrawals enhance stress-induced anxiety-like behavior: inhibition by CRF1- and benzodiazepine-receptor antagonists and a 5-HT1a-receptor agonist.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2005, Volume: 30, Issue:9

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Buspirone; Central Nervous System Depressants; Drug Interactions; Ethanol; Flumazenil; Food, Formulated; GABA Modulators; Interpersonal Relations; Male; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Restraint, Physical; Serotonin Receptor Agonists; Stress, Psychological; Substance Withdrawal Syndrome; Time Factors

2005
CRF receptor type 1 mediates continual hypoxia-induced CRF peptide and CRF mRNA expression increase in hypothalamic PVN of rats.
    Peptides, 2005, Volume: 26, Issue:4

    Topics: Adrenocorticotropic Hormone; Animals; Cell Hypoxia; Corticosterone; Gene Expression Regulation; Immunohistochemistry; In Situ Hybridization; Male; Paraventricular Hypothalamic Nucleus; Pituitary Gland; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger

2005
Corticotropin-releasing factor receptor subtypes mediating nutritional suppression of estrous behavior in Syrian hamsters.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2005, Volume: 289, Issue:2

    Topics: Animal Nutritional Physiological Phenomena; Animals; Corticotropin-Releasing Hormone; Cricetinae; Estrus; Female; Food Deprivation; Mesocricetus; Neuropeptide Y; Peptide Fragments; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Sexual Behavior, Animal; Urocortins

2005
Comparison of the effects of diazepam, the CRF1 antagonist CP-154,526 and the group II mGlu receptor agonist LY379268 on stress-evoked extracellular norepinephrine levels.
    Neuropharmacology, 2005, Volume: 48, Issue:7

    Topics: Amino Acids; Animals; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; Extracellular Fluid; Male; Norepinephrine; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Receptors, Metabotropic Glutamate; Stress, Physiological

2005
Effects of corticotropin-releasing hormone receptor antagonists on cocaine-induced dopamine overflow in the medial prefrontal cortex and nucleus accumbens of rats.
    Synapse (New York, N.Y.), 2005, Sep-15, Volume: 57, Issue:4

    Topics: Animals; Chromatography, High Pressure Liquid; Cocaine; Corticotropin-Releasing Hormone; Dopamine; Dopamine Uptake Inhibitors; Male; Microdialysis; Nucleus Accumbens; Prefrontal Cortex; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone

2005
CRH receptor type 1 mediates continual hypoxia-induced changes of immunoreactive prolactin and prolactin mRNA expression in rat pituitary.
    Hormones and behavior, 2006, Volume: 49, Issue:2

    Topics: Adrenalectomy; Adrenocorticotropic Hormone; Animals; Cold Temperature; Corticotropin-Releasing Hormone; Hypoxia; Immunohistochemistry; Male; Paraventricular Hypothalamic Nucleus; Peptide Fragments; Pituitary Gland; Prolactin; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Restraint, Physical; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Stress, Psychological

2006
Effects of CP 154,526, a CRF1 receptor antagonist, on behavioral responses to cocaine in rats.
    Neuropeptides, 2005, Volume: 39, Issue:5

    Topics: Animals; Behavior, Animal; Cocaine; Discrimination, Psychological; Dose-Response Relationship, Drug; Male; Motor Activity; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Reinforcement, Psychology; Self Administration

2005
The CRH1 antagonist CP154,526 failed to alter ischemia-induced neurodegeneration and spatial memory deficits in rats but inhibited behavioral activity in the novel open field.
    Behavioural brain research, 2006, Jan-06, Volume: 166, Issue:1

    Topics: Animals; Behavior, Animal; Cell Count; Dose-Response Relationship, Drug; Exploratory Behavior; Hippocampus; Ischemia; Male; Memory Disorders; Nerve Degeneration; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Spatial Behavior; Time Factors

2006
Endogenous expression and in vitro study of CRF-related peptides and CRF receptors in the rat gastric antrum.
    Peptides, 2006, Volume: 27, Issue:6

    Topics: Animals; Corticotropin-Releasing Hormone; DNA Primers; Gastric Emptying; Gene Expression Regulation; Immunohistochemistry; Male; Neurons; Pyloric Antrum; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Urocortins

2006
Region-specific effects of brain corticotropin-releasing factor receptor type 1 blockade on footshock-stress- or drug-priming-induced reinstatement of morphine conditioned place preference in rats.
    Psychopharmacology, 2006, Volume: 185, Issue:1

    Topics: Amygdala; Animals; Behavior, Animal; Brain; Central Nervous System Agents; Cocaine; Conditioning, Operant; Extinction, Psychological; Heroin; Injections, Intraventricular; Learning; Male; Morphine; Nucleus Accumbens; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Reinforcement, Psychology; Septal Nuclei; Stress, Psychological

2006
The corticotropin-releasing factor (CRF)(1) receptor antagonists CP154,526 and DMP695 inhibit light-induced phase advances of hamster circadian activity rhythms.
    Brain research, 2006, Apr-14, Volume: 1083, Issue:1

    Topics: Animals; Circadian Rhythm; Corticotropin-Releasing Hormone; Cricetinae; Depressive Disorder; Dose-Response Relationship, Drug; Hypothalamo-Hypophyseal System; Jet Lag Syndrome; Light; Male; Mesocricetus; Pituitary-Adrenal System; Pyridines; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Stress, Psychological; Suprachiasmatic Nucleus

2006
Anxiogenic and aversive effects of corticotropin-releasing factor (CRF) in the bed nucleus of the stria terminalis in the rat: role of CRF receptor subtypes.
    Psychopharmacology, 2006, Volume: 186, Issue:1

    Topics: Animals; Anxiety; Avoidance Learning; Behavior, Animal; Conditioning, Psychological; Corticotropin-Releasing Hormone; Male; Peptide Fragments; Pyrimidines; Pyrroles; Rats; Rats, Long-Evans; Receptors, Corticotropin-Releasing Hormone; Septal Nuclei

2006
CP-154,526, a CRF type-1 receptor antagonist, attenuates the cue-and methamphetamine-induced reinstatement of extinguished methamphetamine-seeking behavior in rats.
    Psychopharmacology, 2007, Volume: 190, Issue:2

    Topics: Amphetamine-Related Disorders; Animals; Corticotropin-Releasing Hormone; Cues; Dose-Response Relationship, Drug; Extinction, Psychological; Hypothalamo-Hypophyseal System; Infusions, Intravenous; Injections, Intraperitoneal; Injections, Intraventricular; Ketoconazole; Male; Methamphetamine; Motivation; Pituitary-Adrenal System; Premedication; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Self Administration

2007
Suppression of adrenocorticotrophic hormone secretion by simultaneous antagonism of vasopressin 1b and CRH-1 receptors on three different stress models.
    Neuroendocrinology, 2006, Volume: 84, Issue:5

    Topics: Adrenocorticotropic Hormone; Animals; Antidiuretic Hormone Receptor Antagonists; Drug Administration Routes; Drug Administration Schedule; Drug Combinations; Drug Evaluation, Preclinical; Ether; Indoles; Male; Pyrimidines; Pyrroles; Pyrrolidines; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Restraint, Physical; Stress, Psychological; Swimming

2006
An arginine vasopressin V1b antagonist, SSR149415 elicits antidepressant-like effects in an olfactory bulbectomy model.
    Progress in neuro-psychopharmacology & biological psychiatry, 2007, Apr-13, Volume: 31, Issue:3

    Topics: Animals; Antidepressive Agents; Depression; Disease Models, Animal; Drug Administration Schedule; Indoles; Male; Olfactory Bulb; Pyrimidines; Pyrroles; Pyrrolidines; Rats; Rats, Wistar; Statistics, Nonparametric

2007
Comparison of the V1b antagonist, SSR149415, and the CRF1 antagonist, CP-154,526, in rodent models of anxiety and depression.
    Pharmacology, biochemistry, and behavior, 2007, Volume: 86, Issue:3

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Anxiety; Conditioning, Psychological; Depression; Female; Guinea Pigs; Humans; Indoles; Male; Maze Learning; Mice; Pyrimidines; Pyrroles; Pyrrolidines; Rats; Receptors, Corticotropin-Releasing Hormone; Receptors, Vasopressin; Vocalization, Animal

2007
Effects of hypoxia on glucose, insulin, glucagon, and modulation by corticotropin-releasing factor receptor type 1 in the rat.
    Endocrinology, 2007, Volume: 148, Issue:7

    Topics: Altitude; Animals; Blood Glucose; Body Weight; Corticosterone; Eating; Glucagon; Hypoxia; Insulin; Leptin; Liver Glycogen; Male; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone

2007
Corticotropin releasing factor-1 receptor antagonist, CP-154,526, blocks the expression of ethanol-induced behavioral sensitization in DBA/2J mice.
    Neuroscience, 2007, Nov-30, Volume: 150, Issue:1

    Topics: Analysis of Variance; Animals; Behavior, Animal; Central Nervous System Depressants; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; Hormone Antagonists; Male; Mice; Mice, Inbred DBA; Motor Activity; Pyrimidines; Pyrroles; Time Factors

2007
Blockade of the corticotropin releasing factor type 1 receptor attenuates elevated ethanol drinking associated with drinking in the dark procedures.
    Alcoholism, clinical and experimental research, 2008, Volume: 32, Issue:2

    Topics: Alcohol Drinking; Alcoholism; Animals; Association Learning; Circadian Rhythm; Darkness; Dose-Response Relationship, Drug; Ethanol; Hypothalamo-Hypophyseal System; Injections, Intraperitoneal; Male; Mice; Mice, Inbred C57BL; Motor Activity; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone

2008
The CRF-1 receptor antagonist, CP-154,526, attenuates stress-induced increases in ethanol consumption by BALB/cJ mice.
    Alcoholism, clinical and experimental research, 2008, Volume: 32, Issue:2

    Topics: Alcohol Drinking; Alcoholism; Animals; Brain; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Signal Transduction; Species Specificity; Stress, Psychological

2008
Corticotropin-releasing factor type 1 receptors mediate the visceral hyperalgesia induced by repeated psychological stress in rats.
    American journal of physiology. Gastrointestinal and liver physiology, 2008, Volume: 294, Issue:4

    Topics: Animals; Blood-Brain Barrier; Chronic Disease; Colon; Corticotropin-Releasing Hormone; Disease Models, Animal; Hyperalgesia; Infusion Pumps, Implantable; Injections, Subcutaneous; Male; Mechanotransduction, Cellular; Peptide Fragments; Pressure; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Rectum; Stress, Psychological

2008
Corticotropin-releasing hormone receptor 1 coexists with endothelin-1 and modulates its mRNA expression and release in rat paraventricular nucleus during hypoxia.
    Neuroscience, 2008, Apr-09, Volume: 152, Issue:4

    Topics: Animals; Corticosterone; Endothelin-1; Gene Expression Regulation; Hypoxia; Male; Paraventricular Hypothalamic Nucleus; Pyrimidines; Pyrroles; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; RNA, Messenger; Time Factors

2008
Corticotropin-releasing factor-1 receptor involvement in behavioral neuroadaptation to ethanol: a urocortin1-independent mechanism.
    Proceedings of the National Academy of Sciences of the United States of America, 2008, Jul-01, Volume: 105, Issue:26

    Topics: Adaptation, Biological; Adrenocorticotropic Hormone; Animals; Behavior, Animal; Ethanol; Gene Deletion; Mice; Mice, Inbred C57BL; Mice, Knockout; Mifepristone; Nervous System Physiological Phenomena; Psychomotor Performance; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Urocortins

2008
Corticotropin-releasing hormone receptor 1 antagonist blocks colonic hypersensitivity induced by a combination of inflammation and repetitive colorectal distension.
    Neurogastroenterology and motility, 2008, Volume: 20, Issue:10

    Topics: Animals; Colitis; Colon; Dilatation, Pathologic; Electromyography; Humans; Inflammation; Irritable Bowel Syndrome; Male; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Trinitrobenzenesulfonic Acid

2008
The alcohol deprivation effect in C57BL/6J mice is observed using operant self-administration procedures and is modulated by CRF-1 receptor signaling.
    Alcoholism, clinical and experimental research, 2009, Volume: 33, Issue:1

    Topics: Alcoholism; Animals; Conditioning, Operant; Ethanol; Male; Mice; Mice, Inbred C57BL; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Self Administration; Signal Transduction; Substance Withdrawal Syndrome

2009
Social subordination and polymorphisms in the gene encoding the serotonin transporter enhance estradiol inhibition of luteinizing hormone secretion in female rhesus monkeys.
    Biology of reproduction, 2009, Volume: 81, Issue:6

    Topics: Analysis of Variance; Animals; Body Weight; Dominance-Subordination; Estradiol; Female; Hydrocortisone; Hypothalamo-Hypophyseal System; Individuality; Luteinizing Hormone; Macaca mulatta; Pituitary-Adrenal System; Polymorphism, Genetic; Pyrimidines; Pyrroles; Radioimmunoassay; Receptors, Corticotropin-Releasing Hormone; Serotonin Plasma Membrane Transport Proteins; Social Environment; Stress, Psychological

2009
The alarm pheromone in male rats as a unique anxiety model: psychopharmacological evidence using anxiolytics.
    Pharmacology, biochemistry, and behavior, 2010, Volume: 94, Issue:4

    Topics: Administration, Inhalation; Animals; Anti-Anxiety Agents; Anxiety; Buspirone; Clonidine; Disease Models, Animal; Male; Midazolam; Phenelzine; Pheromones; Propranolol; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Reflex, Startle

2010
CRF-1 antagonist and CRF-2 agonist decrease binge-like ethanol drinking in C57BL/6J mice independent of the HPA axis.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2010, Volume: 35, Issue:6

    Topics: Alcohol-Induced Disorders, Nervous System; Animals; Corticotropin-Releasing Hormone; Disease Models, Animal; Hormone Antagonists; Hypothalamo-Hypophyseal System; Injections, Intraperitoneal; Injections, Intraventricular; Male; Mice; Mice, Inbred C57BL; Mifepristone; Peptide Fragments; Pyridines; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Signal Transduction; Urocortins

2010
Pain is a salient "stressor" that is mediated by corticotropin-releasing factor-1 receptors.
    Neuropharmacology, 2010, Volume: 59, Issue:3

    Topics: Aniline Compounds; Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Corticotropin-Releasing Hormone; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Hyperalgesia; Indomethacin; Inflammation; Male; Mice; Pain; Pain Threshold; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Spinal Cord Injuries; Stomach Ulcer; Stress, Psychological

2010
Blocking corticotropin-releasing factor-2 receptors, but not corticotropin-releasing factor-1 receptors or glucocorticoid feedback, disrupts the development of conditioned defeat.
    Physiology & behavior, 2010, Nov-02, Volume: 101, Issue:4

    Topics: Aggression; Analysis of Variance; Animals; Antimetabolites; Association Learning; Conditioning, Classical; Cricetinae; Dominance-Subordination; Feedback, Physiological; Glucocorticoids; Hormone Antagonists; Hypothalamo-Hypophyseal System; Male; Mesocricetus; Metyrapone; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone

2010
Stress-induced priming of glutamate synapses unmasks associative short-term plasticity.
    Nature neuroscience, 2010, Volume: 13, Issue:10

    Topics: Animals; Biophysical Phenomena; Biophysics; Chelating Agents; Corticotropin-Releasing Hormone; Dizocilpine Maleate; Drug Interactions; Egtazic Acid; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Exocytosis; Freezing Reaction, Cataleptic; Glutamic Acid; In Vitro Techniques; Male; Neuronal Plasticity; Neurons; Paraventricular Hypothalamic Nucleus; Patch-Clamp Techniques; Pyrimidines; Pyrroles; Quinoxalines; Rats; Rats, Sprague-Dawley; SNARE Proteins; Stress, Physiological; Synapses; Time Factors

2010
Restraint stress-induced reduction in prepulse inhibition in Brown Norway rats: role of the CRF2 receptor.
    Neuropharmacology, 2011, Volume: 60, Issue:4

    Topics: Acoustic Stimulation; Analysis of Variance; Animals; Grooming; Male; Pyrimidines; Pyrroles; Rats; Receptors, Corticotropin-Releasing Hormone; Reflex, Startle; Restraint, Physical; Sensory Gating; Stress, Physiological

2011
[(76) Br]BMK-152, a nonpeptide analogue, with high affinity and low nonspecific binding for the corticotropin-releasing factor type 1 receptor.
    Synapse (New York, N.Y.), 2011, Volume: 65, Issue:9

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Autoradiography; Barium Radioisotopes; Binding Sites; Binding, Competitive; Brain; In Vitro Techniques; Ligands; Macaca mulatta; Male; Mice; Mice, Knockout; Protein Binding; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Triazines

2011
Prevention of social stress-escalated cocaine self-administration by CRF-R1 antagonist in the rat VTA.
    Psychopharmacology, 2011, Volume: 218, Issue:1

    Topics: Animals; Cocaine; Cocaine-Related Disorders; Locomotion; Male; Neurons; Pyrimidines; Pyrroles; Rats; Rats, Long-Evans; Receptors, Corticotropin-Releasing Hormone; Reinforcement Schedule; Self Administration; Stress, Psychological; Ventral Tegmental Area

2011
Pretreatment with CP-154526 blocks the modifying effects of alarm pheromone on components of sexual behavior in male, but not in female, rats.
    Chemical senses, 2011, Volume: 36, Issue:7

    Topics: Animals; Female; Male; Pheromones; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Sex Characteristics; Sexual Behavior, Animal

2011
Effects of acute stress on acquisition of nicotine conditioned place preference in adolescent rats: a role for corticotropin-releasing factor 1 receptors.
    Psychopharmacology, 2012, Volume: 219, Issue:1

    Topics: Acute Disease; Age Factors; Animals; Conditioning, Psychological; Dose-Response Relationship, Drug; Male; Nicotine; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Stress, Psychological

2012
α(2) Adrenergic and imidazoline receptor agonists prevent cue-induced cocaine seeking.
    Biological psychiatry, 2011, Oct-15, Volume: 70, Issue:8

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Cocaine; Cues; Dose-Response Relationship, Drug; Drug Interactions; Drug-Seeking Behavior; Extinction, Psychological; Guanfacine; Imidazoles; Imidazoline Receptors; Isoquinolines; Male; Motor Activity; Naphthyridines; Prazosin; Propranolol; Pyrimidines; Pyrroles; Quinoxalines; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology; Self Administration

2011
Lifelong CRF overproduction is associated with altered gene expression and sensitivity of discrete GABA(A) and mGlu receptor subtypes.
    Psychopharmacology, 2012, Volume: 219, Issue:3

    Topics: Animals; Corticotropin-Releasing Hormone; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Agonists; Gene Expression Regulation; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Pyridines; Pyrimidines; Pyrroles; Rats; Receptors, GABA-A; Receptors, Metabotropic Glutamate

2012
Alcohol in excess: CRF₁ receptors in the rat and mouse VTA and DRN.
    Psychopharmacology, 2013, Volume: 225, Issue:2

    Topics: Alcohol Drinking; Animals; Dose-Response Relationship, Drug; Drinking; Ethanol; Male; Mice; Mice, Inbred C57BL; Pyrimidines; Pyrroles; Raphe Nuclei; Rats; Rats, Long-Evans; Receptors, Corticotropin-Releasing Hormone; Species Specificity; Ventral Tegmental Area

2013
Role of corticotropin-releasing factor (CRF) receptor-1 on the catecholaminergic response to morphine withdrawal in the nucleus accumbens (NAc).
    PloS one, 2012, Volume: 7, Issue:10

    Topics: Animals; Corticosterone; Dopamine; Male; Morphine; Morphine Dependence; Naloxone; Neurons; Norepinephrine; Nucleus Accumbens; Phosphorylation; Proto-Oncogene Proteins c-fos; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Serine; Substance Withdrawal Syndrome; Tyrosine 3-Monooxygenase; Ventral Tegmental Area

2012
Long-term loss of dopamine release mediated by CRF-1 receptors in the rat lateral septum after repeated cocaine administration.
    Behavioural brain research, 2013, Aug-01, Volume: 250

    Topics: Animals; Cocaine; Corticotropin-Releasing Hormone; Dopamine; Dopamine Uptake Inhibitors; Drug Administration Schedule; Drug Interactions; Male; Microdialysis; Peptides, Cyclic; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Septum of Brain; Time Factors

2013
Differential effect of orexin-1 and CRF-1 antagonism on stress circuits: a fMRI study in the rat with the pharmacological stressor Yohimbine.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2013, Volume: 38, Issue:11

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Aminopyridines; Amygdala; Animals; Benzazepines; Corpus Striatum; Corticosterone; Dopamine Antagonists; Functional Neuroimaging; Gyrus Cinguli; Male; Medetomidine; Neural Pathways; Orexin Receptor Antagonists; Piperidines; Pyrimidines; Pyrroles; Rats; Receptors, Corticotropin-Releasing Hormone; Stress, Psychological; Yohimbine

2013
CRF1 receptor antagonists do not reverse pharmacological disruption of prepulse inhibition in rodents.
    Psychopharmacology, 2014, Volume: 231, Issue:7

    Topics: Acoustic Stimulation; Animals; Corticotropin-Releasing Hormone; Dextroamphetamine; Dizocilpine Maleate; Dopamine; Dose-Response Relationship, Drug; Hydrocarbons, Halogenated; Ketamine; Male; Mice; Mice, Transgenic; Nucleus Accumbens; Prefrontal Cortex; Prepulse Inhibition; Pyridines; Pyrimidines; Pyrroles; Rats; Receptors, Corticotropin-Releasing Hormone; Reflex, Startle; Thiazines

2014
Drug-induced suppression of ACTH secretion does not promote anti-depressive or anxiolytic effects.
    Behavioural brain research, 2014, May-15, Volume: 265

    Topics: Adrenocorticotropic Hormone; Analysis of Variance; Animals; Anti-Anxiety Agents; Anxiety; Disease Models, Animal; Dose-Response Relationship, Drug; Indoles; Interpersonal Relations; Male; Maze Learning; Pyrimidines; Pyrroles; Pyrrolidines; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Swimming

2014
Neurokinin B signaling in the female rat: a novel link between stress and reproduction.
    Endocrinology, 2014, Volume: 155, Issue:7

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arcuate Nucleus of Hypothalamus; Corticosterone; Corticotropin-Releasing Hormone; Female; Gonadotropin-Releasing Hormone; Injections, Intraventricular; Lipopolysaccharides; Luteinizing Hormone; Neurokinin B; Neurons; Ovariectomy; Peptide Fragments; Pyrimidines; Pyrroles; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Receptors, Neurokinin-3; Receptors, Vasopressin; Reproduction; Signal Transduction; Stress, Physiological; Substance P

2014
Epigenetic upregulation of corticotrophin-releasing hormone mediates postnatal maternal separation-induced memory deficiency.
    PloS one, 2014, Volume: 9, Issue:4

    Topics: Acetylation; Animals; Animals, Newborn; Corticotropin-Releasing Hormone; Electric Stimulation; Epigenesis, Genetic; Hippocampus; Histones; Long-Term Potentiation; Maternal Deprivation; Maze Learning; Memory Disorders; Methyl-CpG-Binding Protein 2; Neuronal Plasticity; Phosphorylation; Promoter Regions, Genetic; Pyrimidines; Pyrroles; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; RNA, Messenger; Up-Regulation

2014
Prevention of alcohol-heightened aggression by CRF-R1 antagonists in mice: critical role for DRN-PFC serotonin pathway.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2014, Volume: 39, Issue:12

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aggression; Alcohol Drinking; Animals; Central Nervous System Agents; Central Nervous System Depressants; Dorsal Raphe Nucleus; Ethanol; Mice; Neural Pathways; Prefrontal Cortex; Pyridazines; Pyrimidines; Pyrroles; Receptor, Serotonin, 5-HT1A; Receptors, Corticotropin-Releasing Hormone; Self Administration; Serotonin; Serotonin 5-HT1 Receptor Agonists; Thiazoles

2014
Dissociation of μ-opioid receptor and CRF-R1 antagonist effects on escalated ethanol consumption and mPFC serotonin in C57BL/6J mice.
    Addiction biology, 2016, Volume: 21, Issue:1

    Topics: Alcohol Drinking; Aminopyridines; Animals; Behavior, Animal; Central Nervous System Depressants; Dorsal Raphe Nucleus; Ethanol; Immunohistochemistry; Infusions, Intraventricular; Male; Mice; Mice, Inbred C57BL; Microdialysis; Naltrexone; Narcotic Antagonists; Prefrontal Cortex; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Receptors, Opioid, mu; Self Administration; Serotonin; Tryptophan Hydroxylase

2016
Injection of corticotropin-releasing hormone into the amygdala aggravates visceral nociception and induces noradrenaline release in rats.
    Neurogastroenterology and motility, 2015, Volume: 27, Issue:1

    Topics: Amygdala; Animals; Colon; Corticotropin-Releasing Hormone; Dilatation, Pathologic; Dopamine; Male; Nociception; Norepinephrine; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Rectum; Serotonin

2015
Corticotropin-releasing factor 1 receptor mediates the activity of the reward system evoked by morphine-induced conditioned place preference.
    Neuropharmacology, 2015, Volume: 95

    Topics: Animals; Conditioning, Operant; Hormone Antagonists; Locus Coeruleus; Male; Mice; Morphine; Morphine Dependence; Narcotics; Neurons; Nucleus Accumbens; Pyrimidines; Pyrroles; Random Allocation; Receptors, Corticotropin-Releasing Hormone; Reward; Spatial Behavior; Ventral Tegmental Area

2015
Reduction of ethanol intake by corticotropin-releasing factor receptor-1 antagonist in "heavy-drinking" mice in a free-choice paradigm.
    Psychopharmacology, 2015, Volume: 232, Issue:15

    Topics: Alcohol Drinking; Amygdala; Animals; Choice Behavior; Drinking; Ethanol; Male; Mice; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone

2015
Long-term effects of early adolescent stress: dysregulation of hypothalamic-pituitary-adrenal axis and central corticotropin releasing factor receptor 1 expression in adult male rats.
    Behavioural brain research, 2015, Jul-15, Volume: 288

    Topics: Animals; Anxiety; Corticosterone; Depression; Disease Models, Animal; Electroshock; Exercise Therapy; Foot; Hypothalamo-Hypophyseal System; Male; Maze Learning; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Random Allocation; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Running; Stress Disorders, Post-Traumatic; Stress, Psychological

2015
Lifelong disturbance of serotonin transporter functioning results in fear learning deficits: Reversal by blockade of CRF1 receptors.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2015, Volume: 25, Issue:10

    Topics: Animals; Basolateral Nuclear Complex; Disease Models, Animal; Dorsal Raphe Nucleus; Fear; Gene Knockout Techniques; Learning; Learning Disabilities; Male; Neurotransmitter Agents; Paroxetine; Prepulse Inhibition; Pyrimidines; Pyrroles; Rats, Transgenic; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Reflex, Startle; RNA-Binding Proteins; RNA, Messenger

2015
CP-154,526 Modifies CREB Phosphorylation and Thioredoxin-1 Expression in the Dentate Gyrus following Morphine-Induced Conditioned Place Preference.
    PloS one, 2015, Volume: 10, Issue:8

    Topics: Animals; Blotting, Western; Cells, Cultured; Conditioning, Psychological; Cyclic AMP Response Element-Binding Protein; Dentate Gyrus; Fluorescent Antibody Technique; Immunoenzyme Techniques; Male; Mice; Morphine; Morphine Dependence; Narcotics; Neurons; Phosphorylation; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Thioredoxins

2015
Role of Corticotropin Releasing Factor 1 Signaling in Cocaine Seeking during Early Extinction in Female and Male Rats.
    PloS one, 2016, Volume: 11, Issue:6

    Topics: Animals; Cocaine; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Extinction, Psychological; Female; Male; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Self Administration; Signal Transduction

2016
CRF
    Pharmacology, biochemistry, and behavior, 2017, Volume: 154

    Topics: Animals; Anti-Anxiety Agents; Benzodioxoles; Corticotropin-Releasing Hormone; Dose-Response Relationship, Drug; Drug Interactions; Guinea Pigs; Maternal Deprivation; Mice; Mice, Transgenic; Mifepristone; Paroxetine; Pyridines; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Receptors, Glucocorticoid; Steroids; Vocalization, Animal

2017
The non-peptide CRH1-antagonist CP-154,526 elicits a paradoxical route-dependent activation of the HPA axis.
    Neuroscience letters, 2017, Jul-13, Volume: 653

    Topics: Adrenocorticotropic Hormone; Animals; Arterial Pressure; Heart Rate; Hypothalamo-Hypophyseal System; Injections, Intra-Arterial; Injections, Intraperitoneal; Male; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone

2017
The effects of enhancing endocannabinoid signaling and blocking corticotrophin releasing factor receptor in the amygdala and hippocampus on the consolidation of a stressful event.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2017, Volume: 27, Issue:9

    Topics: Amidohydrolases; Animals; Anxiety; Basolateral Nuclear Complex; Benzamides; CA1 Region, Hippocampal; Carbamates; Disease Models, Animal; Endocannabinoids; Male; Memory Consolidation; Nootropic Agents; Pyrimidines; Pyrroles; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Corticotropin-Releasing Hormone; Reflex, Startle; RNA, Messenger; Stress Disorders, Post-Traumatic; Stress, Psychological

2017
Chondroprotection by urocortin involves blockade of the mechanosensitive ion channel Piezo1.
    Scientific reports, 2017, 07-11, Volume: 7, Issue:1

    Topics: Autocrine Communication; Calcium; Cartilage, Articular; Cell Survival; Cells, Cultured; Chondrocytes; Cyclic AMP; Humans; Ion Channels; Paracrine Communication; Peptide Fragments; Peptides, Cyclic; Protein Conformation; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Signal Transduction; Urocortins

2017
Early adolescent stress-induced changes in prefrontal cortex miRNA-135a and hippocampal miRNA-16 in male rats.
    Developmental psychobiology, 2017, Volume: 59, Issue:8

    Topics: Age Factors; Animals; Anxiety; Disease Models, Animal; Hippocampus; Male; MicroRNAs; Paroxetine; Prefrontal Cortex; Pyrimidines; Pyrroles; Rats; Receptor, Serotonin, 5-HT1A; Receptors, Corticotropin-Releasing Hormone; Selective Serotonin Reuptake Inhibitors; Spatial Memory; Stress, Psychological

2017
Maternal stress and the MPOA: Activation of CRF receptor 1 impairs maternal behavior and triggers local oxytocin release in lactating rats.
    Neuropharmacology, 2018, 05-01, Volume: 133

    Topics: Analysis of Variance; Animals; Animals, Newborn; Carrier Proteins; Corticotropin-Releasing Hormone; Female; Gene Expression Regulation; Hormone Antagonists; Lactation; Male; Maternal Behavior; Maze Learning; Microdialysis; Oxytocin; Preoptic Area; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; RNA, Messenger

2018
Conditioned aversive memory associated with morphine withdrawal increases brain-derived neurotrophic factor in dentate gyrus and basolateral amygdala.
    Addiction biology, 2020, Volume: 25, Issue:4

    Topics: Affect; Analgesics, Opioid; Animals; Basolateral Nuclear Complex; Brain-Derived Neurotrophic Factor; Conditioning, Classical; Corticosterone; Corticotropin-Releasing Hormone; Cyclic AMP Response Element-Binding Protein; Dentate Gyrus; Extinction, Psychological; Male; Memory; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Morphine; Naloxone; Narcotic Antagonists; Protein Precursors; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Substance Withdrawal Syndrome

2020
Central angiotensin II type 1 receptor as a therapeutic target against frequent urination.
    Neurourology and urodynamics, 2019, Volume: 38, Issue:8

    Topics: Amphibian Proteins; Angiotensin II; Angiotensin II Type 1 Receptor Blockers; Animals; Male; Peptide Hormones; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Telmisartan; Urination

2019
Naloxone-induced conditioned place aversion score and extinction period are higher in C57BL/6J morphine-dependent mice than in Swiss: Role of HPA axis.
    Pharmacology, biochemistry, and behavior, 2021, Volume: 201

    Topics: Animals; Avoidance Learning; Conditioning, Operant; Extinction, Psychological; Hypothalamo-Hypophyseal System; Male; Memory; Mice; Mice, Inbred C57BL; Morphine; Morphine Dependence; Naloxone; Narcotic Antagonists; Narcotics; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Substance Withdrawal Syndrome

2021
Sex-specific plasticity in CRF regulation of inhibitory control in central amygdala CRF1 neurons after chronic voluntary alcohol drinking.
    Addiction biology, 2022, Volume: 27, Issue:1

    Topics: Alcohol Drinking; Animals; Central Amygdaloid Nucleus; Corticotropin-Releasing Hormone; Ethanol; Female; gamma-Aminobutyric Acid; Male; Mice; Neurons; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Receptors, GABA-A; Sex Characteristics; Synaptic Transmission

2022