pyrroles has been researched along with cp 154526 in 117 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 9 (7.69) | 18.2507 |
2000's | 67 (57.26) | 29.6817 |
2010's | 38 (32.48) | 24.3611 |
2020's | 3 (2.56) | 2.80 |
Authors | Studies |
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Braselton, JP; Chen, YL; Collins, J; Corman, M; Dunaiskis, A; Faraci, S; Heym, J; Mansbach, RS; Schmidt, AW; Schulz, DW; Seeger, T; Seymour, P; Sprouse, J; Tingley, FD; Winston, EN | 1 |
Bartfai, T; Chai, Z; Hasanvan, H; Jenck, F; Lundkvist, J; Moreau, JL; Teheranian, R; Widmer, U | 1 |
Brooks, EN; Chen, YL; Mansbach, RS | 1 |
Brooks, E; Chen, YL; Collins, J; Corman, ML; Dunaiskis, AR; Faraci, WS; Gallaschun, RJ; Mansbach, RS; Schmidt, A; Schulz, DW; Winter, SM | 1 |
Buczek, Y; Erb, S; Leung, S; Shaham, Y; Stewart, J | 1 |
Griebel, G; Perrault, G; Sanger, DJ | 1 |
Grigoriadis, DE; Heinrichs, SC; McCarthy, JR | 1 |
Berridge, CW; Dikkes, P; Dunn, AJ; Majzoub, JA; Miczek, KA; Muglia, LJ; Swiergiel, AH; Weninger, SC | 1 |
Banks, MC; Huhman, KL; Jasnow, AM; Owens, EC | 1 |
Miyata, K; Yamano, M; Yasuda, S; Yuki, H | 1 |
Alvaro, JD; Chen, YL; Duman, RS; Iredale, PA; Lee, Y; Terwilliger, R | 1 |
Kawahara, H; Kawahara, Y; Westerink, BH | 1 |
Bruijnzeel, A; Croiset, G; de Wied, D; Diamant, M; Nijsen, MJ; Stam, R; Wiegant, VM | 1 |
Cassella, JV; Coverdale, S; Hoffman, DC; Kehne, JH; McCloskey, TC | 1 |
Brown, J; Connor, HE; Giles, H; Parsons, SJ; Rees, S; Rhodes, SA | 1 |
Arborelius, L; Owens, MJ; Plotsky, PM; Schulz, DW; Skelton, KH; Thrivikraman, KV | 1 |
Harding, S; Juzytsch, W; Lê, AD; Shaham, Y; Shalev, U; Watchus, J | 1 |
Ceng, X; Huang, M; Lu, L | 1 |
Goeders, NE; Guerin, GF | 1 |
Davidson, A; Finlay, TH; Funai, EF; O'Neill, LM; Roqué, H | 1 |
Akiyoshi, J; Hikichi, T; Isogawa, K; Nagayama, H; Tsutsumi, T; Yamamoto, Y | 1 |
Gauthier, A; Maillot, C; Million, M; Taché, Y; Wei, JY | 1 |
Ceng, X; Liu, D; Lu, L; Ma, L | 1 |
Ceng, X; Liu, D; Lu, L | 1 |
Imaki, J; Imaki, T; Katsumata, H; Minami, S; Miyata, M; Naruse, M | 1 |
Hirata, M; Murakami, Y; Okada, S; Yokotani, K | 1 |
Chaki, S; Kameo, K; Kawashima, N; Nakazato, A; Takamori, K | 1 |
Brocco, M; Casara, P; Dekeyne, A; Dorey, G; Gobert, A; Millan, MJ | 1 |
Bernardini, R; Cantarella, G; Chiarenza, A; Lempereur, L; Lombardo, G; Pafumi, C; Zappalà, G | 1 |
Martínez, V; Rivier, JE; Taché, Y; Wang, L | 1 |
Goeders, NE; Gurkovskaya, O | 1 |
Maillot, C; Million, M; Rivier, J; Saunders, P; Taché, Y; Vale, W | 1 |
Bruelisauer, A; Enz, A; Keller, C; Lemaire, M | 1 |
Maillot, C; Miampamba, M; Million, M; Taché, Y | 1 |
Clampitt, DM; Goeders, NE | 1 |
Blank, T; Nijholt, I; Spiess, J; Vollstaedt, S | 1 |
Schmidt, AW; Schulz, DW; Seymour, PA | 1 |
Blessing, WW; Nalivaiko, E | 2 |
Huang, M; Liu, Z; Lu, L; Zhang, Z | 1 |
Okada, S; Shimizu, T; Yokotani, K | 1 |
Facci, L; Franceschini, D; Pangallo, M; Skaper, SD; Stevens, DA; Strijbos, PJ | 1 |
Bradesi, S; Mayer, EA; McRoberts, JA; Miller, JC; Ohning, G; Sablad, M; Schwetz, I; Zhou, H | 1 |
Berggård, C; Damberg, M; Eller, M; Harro, J; Mällo, T; Oreland, L | 1 |
Hager, P; Hagman, B; Strömmer, L; Wikström, AC | 1 |
Hogg, S; Keeney, A; Overstreet, DH | 1 |
Dominguez, G; Kuhar, MJ | 1 |
Anisman, H; Khan, S; Merali, Z; Michaud, DS; Shippy, SA | 1 |
Houshyar, H; Hsin, LW; Jutkiewicz, EM; Rice, KC; Wood, SK; Woods, JH | 1 |
Breese, GR; Knapp, DJ; Navarro, M; Overstreet, DH | 1 |
Chen, XQ; Du, JZ; Wang, TY; Xu, JF | 1 |
Dettloff, SL; Jones, JE; Seymour, PL; Wade, GN | 1 |
Baccei, CS; Bristow, LJ; Correa, LD; Lorrain, DS | 1 |
Goeders, NE; Gurkovskaya, OV; Palamarchouk, V; Smagin, G | 1 |
Chen, XQ; Du, JZ; Xu, JF | 1 |
Filip, M; Frankowska, M; Papla, I; Przegaliński, E; Zaniewska, M | 1 |
Khan, S; Plamondon, H | 1 |
Bonaz, B; Canini, F; Meregnani, J; Peinnequin, A; Pellissier, S; Porcher, C; Sinniger, V | 1 |
Fang, Q; Liu, Z; Lu, L; Wang, J | 1 |
Gannon, RL; Millan, MJ | 1 |
Blanton, MG; Hicks, MP; Janak, PH; Kinder, JR; Kullberg, EF; Mcgeehan, AJ; Olive, MF; Sahuque, LL | 1 |
Keller, PA; McCluskey, A; Morgan, J; O'connor, SM | 1 |
Goeders, NE; Moffett, MC | 1 |
Ramos, AT; Troncone, LR; Tufik, S | 1 |
Chaki, S; Iijima, M | 1 |
Guthrie, DH; Guzzi, MF; Higgins, GA; Hodgson, RA; Lu, SX; Mullins, DE; Parker, EM; Pond, AJ; Varty, GB | 1 |
Chen, XQ; Dong, J; Du, JZ; Fan, JM; Niu, CY | 1 |
Fee, JR; Picker, MJ; Sparta, DR; Thiele, TE | 1 |
Fee, JR; Knapp, DJ; Lowery, EG; Sparrow, AM; Sparta, DR; Thiele, TE | 1 |
Breese, GR; Knapp, DJ; Lowery, EG; Sparrow, AM; Thiele, TE | 1 |
Bradesi, S; Larauche, M; Mayer, EA; McLean, P; McRoberts, JA; Million, M; Taché, Y | 1 |
Chen, XQ; Du, JZ; He, JJ; Wang, L; Xu, JF | 1 |
Burkhart-Kasch, S; Coste, SC; McKinnon, CS; Pastor, R; Phillips, TJ; Reed, C; Ryabinin, AE; Scibelli, AC; Stenzel-Poore, MP | 1 |
Fukudo, S; Hasegawa, R; Ito, H; Nagura, Y; Saito-Nakaya, K | 1 |
Breese, GR; Fee, JR; Ferraro, FM; Knapp, DJ; Sparta, DR; Thiele, TE | 1 |
Berga, SL; Kaplan, JR; Michopoulos, V; Wilson, ME | 1 |
Inagaki, H; Kiyokawa, Y; Mori, Y; Takeuchi, Y | 1 |
Hodge, CW; Lowery, EG; Lyons, AM; Navarro, M; Spanos, M; Thiele, TE | 1 |
Cummons, T; Harrison, JE; Hummel, M; Kennedy, JD; Lu, P; Mark, L; Whiteside, GT | 1 |
Cooper, MA; Huhman, KL | 1 |
Baimoukhametova, DV; Bains, JS; Kuzmiski, JB; Marty, V | 1 |
Conti, LH; Sutherland, JE | 1 |
Contoreggi, C; Eckelman, WC; Jagoda, EM; Kiesewetter, DO; Kim, BM; Lang, L; Ma, Y; McCullough, K; Rice, KC; Szajek, LP | 1 |
Boyson, CO; Debold, JF; Miczek, KA; Miguel, TT; Quadros, IM | 1 |
Kiyokawa, Y; Kobayashi, T; Mori, Y; Takeuchi, Y | 1 |
Brielmaier, J; McDonald, CG; Smith, RF | 1 |
Aston-Jones, G; Smith, RJ | 1 |
Cook, JM; Groenink, L; Hendriksen, H; Huang, S; Millan, MJ; Olivier, B; Rallipalli, S; van Oorschot, R; Vinkers, CH | 1 |
Debold, JF; Hwa, LS; Miczek, KA | 1 |
Almela, P; García-Carmona, JA; Hidalgo, J; Laorden, ML; Milanés, MV; Mora, L; Navarro-Zaragoza, J | 1 |
Andrés, ME; Araya, KA; Carreño, P; Fuentealba, JA; Gysling, K; Renard, GM; Sotomayor-Zárate, R | 1 |
Bifone, A; Gozzi, A; Lepore, S; Merlo-Pich, E; Vicentini, E | 1 |
Boulay, D; Douma, TN; Griebel, G; Groenink, L; Millan, MJ; Olivier, B; Verdouw, PM; Westphal, KG | 1 |
Homem, KS; Ramos, Ade T; Suchecki, D; Troncone, LR; Tufik, S | 1 |
Grachev, P; Hu, MH; Li, SY; Li, XF; Lightman, SL; Millar, RP; O'Byrne, KT | 1 |
Fan, Q; Hou, Y; Li, H; Nie, W; Sun, R; Wang, A; Yu, Z | 1 |
Carlson, J; DeBold, JF; Hwa, LS; Miczek, KA; Quadros, IM; Shimamoto, A | 1 |
DeBold, JF; Hwa, LS; Kayyali, T; Miczek, KA; Norman, KJ; Shimamoto, A; Valentino, RJ | 1 |
Chen, J; Chen, XQ; Du, JZ; Evans, AM; Gao, YQ; Hao, K; Kong, FP; Lightman, SL; Tang, JW | 1 |
Fukudo, S; Kanazawa, M; Kano, M; Muratsubaki, T; Su, J; Tanaka, Y | 1 |
Laorden, ML; Lasheras, MC; Milanés, MV; Núñez, C | 1 |
Boerngen-Lacerda, R; Camarini, R; Correia, D; Martynhak, BJ; Pereira, M; Ribeiro, AF; Siba, IP | 1 |
Jiang, H; Li, C; Liu, D; Liu, Y; Lu, C; Pan, F; Yin, S | 1 |
Baas, JM; Bijlsma, EY; Groenink, L; Hendriksen, H; Millan, MJ | 1 |
Almela, P; Camejo, DM; García-Carmona, JA; Jiménez, A; Laorden, ML; Milanés, MV; Sevilla, F | 1 |
Aston-Jones, G; Cason, AM; Kohtz, A | 1 |
Groenink, L; Millan, MJ; Peeters, BW; van Esterik, JC; Verdouw, PM | 1 |
Spierling, SR; Zorrilla, EP | 1 |
DiMicco, JA; Rusyniak, DE; Sarkar, S; Zaretskaia, MV; Zaretsky, DV | 1 |
Aisenberg, N; Akirav, I; Sabban, EL; Serova, L | 1 |
Abbott, B; Baylie, RL; Board, TN; Bruhn-Olszewska, B; Jackson, TR; Jones, RC; Lawrence, KM; Locke, IC; Richardson, SM; Townsend, PA | 1 |
Jiang, H; Liu, D; Liu, Y; Pan, F; Xu, J | 1 |
Bayerl, DS; Bosch, OJ; Brunton, PJ; Gaßner, BM; Hübner, K; Klampfl, SM; Schramm, MM; Seasholtz, AF | 1 |
Almela, P; Laorden, ML; Martínez-Laorden, E; Milanés, MV; Navarro-Zaragoza, J | 1 |
Higashi, Y; Nagao, Y; Saito, M; Shimizu, S; Shimizu, T | 1 |
Almela, P; Cánovas, A; Gómez-Murcia, V; Laorden, ML; Martínez-Laorden, E; Milanés, MV; Navarro-Zaragoza, J; Teruel-Fernández, FJ | 1 |
Agoglia, AE; Bluitt, MN; Douglass, E; Hanback, T; Herman, MA; Hodge, CW; Quadir, SG; Tella, J; Ying, R; Zhu, M | 1 |
4 review(s) available for pyrroles and cp 154526
Article | Year |
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Recent advances with the CRF1 receptor: design of small molecule inhibitors, receptor subtypes and clinical indications.
Topics: Animals; Anxiety; Depression; Drug Design; Humans; Kinetics; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Seizures; Substance-Related Disorders | 1999 |
The pharmacology of CP-154,526, a non-peptide antagonist of the CRH1 receptor: a review.
Topics: Animals; Anxiety; Autonomic Nervous System; Behavior, Animal; Depression; Digestive System; Disease Models, Animal; Drug Evaluation, Preclinical; Genitalia; Haplorhini; Immune System; Mice; Motor Skills; Neurodegenerative Diseases; Neurosecretory Systems; Pyrimidines; Pyrroles; Rats; Receptors, Corticotropin-Releasing Hormone | 2003 |
The role of the HPA axis in psychiatric disorders and CRF antagonists as potential treatments.
Topics: Amino Acid Sequence; Animals; Corticotropin-Releasing Hormone; Humans; Hypothalamo-Hypophyseal System; Mental Disorders; Molecular Sequence Data; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone | 2006 |
Don't stress about CRF: assessing the translational failures of CRF
Topics: Animals; Behavior, Addictive; Corticotropin-Releasing Hormone; Depression; Humans; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Stress, Psychological; Substance-Related Disorders; Translational Research, Biomedical | 2017 |
1 trial(s) available for pyrroles and cp 154526
Article | Year |
---|---|
Inactivation of corticotropin-releasing hormone-induced insulinotropic role by high-altitude hypoxia.
Topics: Adenosine Triphosphate; Adolescent; Adult; Altitude; Animals; Blood Glucose; Calcium; Corticosterone; Corticotropin-Releasing Hormone; Cyclic AMP; Humans; Hydrocortisone; Hypoxia; Insulin; Male; Pancreas; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Young Adult | 2015 |
112 other study(ies) available for pyrroles and cp 154526
Article | Year |
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CP-154,526: a potent and selective nonpeptide antagonist of corticotropin releasing factor receptors.
Topics: Acoustic Stimulation; Adenylyl Cyclases; Adrenocorticotropic Hormone; Animals; Binding, Competitive; Callithrix; Cell Line; Cell Membrane; Cerebral Cortex; Cerebral Ventricles; Corticotropin-Releasing Hormone; Dogs; Guinea Pigs; Humans; Injections, Intraventricular; Kinetics; Locus Coeruleus; Male; Neurons; Pituitary Gland; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Reflex, Startle | 1996 |
A non peptidic corticotropin releasing factor receptor antagonist attenuates fever and exhibits anxiolytic-like activity.
Topics: Analgesics, Non-Narcotic; Animals; Anti-Anxiety Agents; Fever; Interleukin-1; Male; Mice; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Recombinant Proteins; Tumor Cells, Cultured | 1996 |
Antidepressant-like effects of CP-154,526, a selective CRF1 receptor antagonist.
Topics: Analysis of Variance; Animals; Antidepressive Agents, Tricyclic; Depression; Disease Models, Animal; Helplessness, Learned; Imipramine; Injections, Intraperitoneal; Male; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone | 1997 |
Synthesis and oral efficacy of a 4-(butylethylamino)pyrrolo[2,3-d]pyrimidine: a centrally active corticotropin-releasing factor1 receptor antagonist.
Topics: Animals; Anti-Anxiety Agents; Fear; Male; Molecular Structure; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Reflex, Startle; Structure-Activity Relationship | 1997 |
CP-154,526, a selective, non-peptide antagonist of the corticotropin-releasing factor1 receptor attenuates stress-induced relapse to drug seeking in cocaine- and heroin-trained rats.
Topics: Animals; Cocaine; Corticotropin-Releasing Hormone; Heroin; Male; Pyrimidines; Pyrroles; Rats; Receptors, Corticotropin-Releasing Hormone; Self Administration; Stress, Psychological; Sucrose | 1998 |
Characterization of the behavioral profile of the non-peptide CRF receptor antagonist CP-154,526 in anxiety models in rodents. Comparison with diazepam and buspirone.
Topics: Animals; Anti-Anxiety Agents; Anxiety Disorders; Behavior, Animal; Buspirone; Diazepam; Male; Mice; Mice, Inbred BALB C; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone | 1998 |
Stress-induced behaviors require the corticotropin-releasing hormone (CRH) receptor, but not CRH.
Topics: Animals; Avoidance Learning; Cerebral Ventricles; Conditioning, Operant; Corticotropin-Releasing Hormone; Crosses, Genetic; Electroshock; Fear; Female; Gene Expression Regulation; Injections, Intraventricular; Learning; Male; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Mice, Knockout; Motor Activity; Pain; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Reinforcement, Psychology; Stress, Psychological; Transcription, Genetic; Urocortins | 1999 |
Differential effects of two corticotropin-releasing factor antagonists on conditioned defeat in male Syrian hamsters (Mesocricetus auratus).
Topics: Adrenocorticotropic Hormone; Aggression; Animals; Behavior, Animal; Corticotropin-Releasing Hormone; Cricetinae; Dominance-Subordination; Dose-Response Relationship, Drug; Male; Mesocricetus; Microinjections; Pyrimidines; Pyrroles; Stress, Psychological | 1999 |
Corticotropin-releasing hormone receptors mediate consensus interferon-alpha YM643-induced depression-like behavior in mice.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Antidepressive Agents; Behavior, Animal; Depression, Chemical; Dose-Response Relationship, Drug; Drug Interactions; Imipramine; Indomethacin; Interferon-alpha; Male; Mice; Motor Activity; Naloxone; Narcotic Antagonists; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Time Factors | 2000 |
Role of corticotropin-releasing factor receptor-1 in opiate withdrawal.
Topics: Animals; Behavior, Animal; Male; Morphine; Naltrexone; Narcotic Antagonists; Protein Isoforms; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Substance Withdrawal Syndrome | 2000 |
The role of afferents to the locus coeruleus in the handling stress-induced increase in the release of noradrenaline in the medial prefrontal cortex: a dual-probe microdialysis study in the rat brain.
Topics: Animals; Benzylamines; Bicuculline; Idazoxan; Locus Coeruleus; Male; Microdialysis; Norepinephrine; Phosphinic Acids; Piperazines; Prefrontal Cortex; Pyrimidines; Pyrroles; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Corticotropin-Releasing Hormone; Receptors, GABA; Receptors, Glutamate; Stress, Physiological | 2000 |
The role of the CRH type 1 receptor in autonomic responses to corticotropin- releasing hormone in the rat.
Topics: Adrenergic beta-Antagonists; Animals; Atenolol; Autonomic Nervous System; Corticotropin-Releasing Hormone; Heart Rate; Male; Motor Activity; Neurosecretory Systems; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone | 2000 |
Effects of the CRF(1) receptor antagonist, CP 154,526, in the separation-induced vocalization anxiolytic test in rat pups.
Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Antipsychotic Agents; Anxiety; Behavior, Animal; Buspirone; Clozapine; Desipramine; Diazepam; Dose-Response Relationship, Drug; Female; Haloperidol; Injections, Intraperitoneal; Male; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Social Isolation; Stress, Psychological; Vocalization, Animal; Zimeldine | 2000 |
Use of a dual firefly and Renilla luciferase reporter gene assay to simultaneously determine drug selectivity at human corticotrophin releasing hormone 1 and 2 receptors.
Topics: Animals; CHO Cells; Coleoptera; Cricetinae; Genes, Reporter; Humans; Luciferases; Protein Isoforms; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone | 2000 |
Chronic administration of the selective corticotropin-releasing factor 1 receptor antagonist CP-154,526: behavioral, endocrine and neurochemical effects in the rat.
Topics: Adrenal Glands; Adrenocorticotropic Hormone; Animals; Anti-Anxiety Agents; Behavior, Animal; Brain; Corticosterone; Corticotropin-Releasing Hormone; Drug Administration Schedule; Endocrine System; Male; Organ Size; Pyrimidines; Pyrroles; Rats; Receptors, Corticotropin-Releasing Hormone; Reflex, Startle; RNA, Messenger; Stress, Physiological; Urocortins | 2000 |
The role of corticotrophin-releasing factor in stress-induced relapse to alcohol-seeking behavior in rats.
Topics: Adrenalectomy; Alcoholism; Animals; Corticosterone; Corticotropin-Releasing Hormone; Electroshock; Extinction, Psychological; Injections, Intraventricular; Male; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Recurrence; Self Administration; Stress, Psychological | 2000 |
Corticotropin-releasing factor receptor type I mediates stress-induced relapse to opiate dependence in rats.
Topics: Animals; Behavior, Animal; Conditioning, Psychological; Corticotropin-Releasing Hormone; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Male; Morphine; Neuropsychological Tests; Opioid-Related Disorders; Psychomotor Performance; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Secondary Prevention; Stress, Physiological | 2000 |
Effects of the CRH receptor antagonist CP-154,526 on intravenous cocaine self-administration in rats.
Topics: Animals; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Food; Male; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Reinforcement, Psychology; Self Administration | 2000 |
A corticotropin releasing hormone receptor antagonist does not delay parturition in rats.
Topics: Animals; Female; Gestational Age; Labor, Obstetric; Pregnancy; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone | 2000 |
Suppression of conditioned fear by administration of CRF receptor antagonist CP-154,526.
Topics: Animals; Conditioning, Psychological; Electroshock; Fear; Male; Motor Activity; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone | 2000 |
Peripheral corticotropin-releasing factor and stress-stimulated colonic motor activity involve type 1 receptor in rats.
Topics: Animals; Avoidance Learning; Colon; Corticotropin-Releasing Hormone; Defecation; Gastrointestinal Motility; Injections, Intraperitoneal; Injections, Intraventricular; Male; Myoelectric Complex, Migrating; Peptide Fragments; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Stress, Physiological; Urocortins; Water | 2000 |
Differential roles of corticotropin-releasing factor receptor subtypes 1 and 2 in opiate withdrawal and in relapse to opiate dependence.
Topics: Animals; Cerebral Ventricles; Choice Behavior; Corticotropin-Releasing Hormone; Hormone Antagonists; Injections, Intraventricular; Male; Morphine; Morphine Dependence; Naloxone; Peptide Fragments; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Substance Withdrawal Syndrome | 2000 |
Corticotropin-releasing factor receptor type 1 mediates stress-induced relapse to cocaine-conditioned place preference in rats.
Topics: Animals; Cocaine; Cocaine-Related Disorders; Conditioning, Psychological; Corticotropin-Releasing Hormone; Dopamine Uptake Inhibitors; Hormone Antagonists; Male; Peptide Fragments; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Secondary Prevention; Stress, Physiological | 2001 |
Expression of corticotropin-releasing hormone type 1 receptor in paraventricular nucleus after acute stress.
Topics: Adrenocorticotropic Hormone; Animals; Corticotropin-Releasing Hormone; Gene Expression; In Situ Hybridization; Male; Oxytocin; Paraventricular Hypothalamic Nucleus; Proto-Oncogene Proteins c-fos; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; RNA, Messenger; Stress, Physiological; Vasopressins | 2001 |
Role of brain arachidonic acid cascade on central CRF1 receptor-mediated activation of sympatho-adrenomedullary outflow in rats.
Topics: Analysis of Variance; Animals; Arachidonic Acid; Brain; Corticotropin-Releasing Hormone; Epinephrine; Injections, Intraventricular; Male; Norepinephrine; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Urocortins | 2001 |
Involvement of corticotropin-releasing factor subtype 1 receptor in the acquisition phase of learned helplessness in rats.
Topics: Animals; Behavior, Animal; Dose-Response Relationship, Drug; Imipramine; Learning; Male; Pyridines; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone | 2001 |
Anxiolytic properties of the selective, non-peptidergic CRF(1) antagonists, CP154,526 and DMP695: a comparison to other classes of anxiolytic agent.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Dopamine; Dose-Response Relationship, Drug; Extracellular Space; Interpersonal Relations; Male; Norepinephrine; Postural Balance; Pyridines; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Serotonin; Vocalization, Animal | 2001 |
Divergent effects of corticotropin releasing hormone on endothelial cell nitric oxide synthase are associated with different expression of CRH type 1 and 2 receptors.
Topics: Animals; Blotting, Western; Cell Line; Cell Line, Transformed; Corticotropin-Releasing Hormone; Endothelium, Vascular; Gene Expression Regulation; Humans; Interleukin-1; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Nitrites; Peptide Fragments; Protein Isoforms; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Time Factors; Tumor Necrosis Factor-alpha | 2001 |
Peripheral urocortin inhibits gastric emptying and food intake in mice: differential role of CRF receptor 2.
Topics: Animals; Anti-Anxiety Agents; Capsaicin; Corticotropin-Releasing Hormone; Eating; Fasting; Gastric Emptying; Humans; Male; Mice; Mice, Inbred C57BL; Peptide Fragments; Pyrazoles; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Urocortins | 2001 |
Effects of CP-154,526 on responding during extinction from cocaine self-administration in rats.
Topics: Animals; Behavior, Animal; Cocaine; Extinction, Psychological; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Reinforcement Schedule; Self Administration | 2001 |
Human urocortin II, a new CRF-related peptide, displays selective CRF(2)-mediated action on gastric transit in rats.
Topics: Animals; Colon; Corticotropin-Releasing Hormone; Gastric Emptying; Humans; Male; Mammals; Peptide Fragments; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Restraint, Physical; Stress, Physiological; Urocortins | 2002 |
Brain pharmacokinetics of a nonpeptidic corticotropin-releasing factor receptor antagonist.
Topics: Animals; Blood-Brain Barrier; Brain; Male; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone | 2002 |
Peripheral CRF activates myenteric neurons in the proximal colon through CRF(1) receptor in conscious rats.
Topics: Acetylcholine; Animals; Colon; Consciousness; Corticotropin-Releasing Hormone; Injections, Intraperitoneal; Male; Myenteric Plexus; NADPH Dehydrogenase; Neurons; Proto-Oncogene Proteins c-fos; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone | 2002 |
Potential role for the hypothalamo-pituitary-adrenal axis in the conditioned reinforcer-induced reinstatement of extinguished cocaine seeking in rats.
Topics: Analysis of Variance; Animals; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Corticosterone; Extinction, Psychological; Hypothalamo-Hypophyseal System; Ketoconazole; Male; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Reinforcement Schedule; Reinforcement, Psychology; Self Administration; Stress, Psychological | 2002 |
The corticotropin-releasing factor receptor 1 antagonist CP-154,526 reverses stress-induced learning deficits in mice.
Topics: Animals; Arousal; Calcium-Calmodulin-Dependent Protein Kinases; Conditioning, Classical; Culture Techniques; Fear; Hippocampus; Hypothalamo-Hypophyseal System; Injections, Intraperitoneal; Long-Term Potentiation; Male; Mice; Mice, Inbred BALB C; Neuronal Plasticity; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Stress, Psychological | 2003 |
CRF1-receptor antagonist CP-154526 reduces alerting-related cutaneous vasoconstriction in conscious rabbits.
Topics: Animals; Arousal; Blood Flow Velocity; Ear; Laser-Doppler Flowmetry; Male; Pain Measurement; Physical Stimulation; Pyrimidines; Pyrroles; Rabbits; Receptors, Corticotropin-Releasing Hormone; Vasoconstriction | 2003 |
Dopamine-dependent responses to cocaine depend on corticotropin-releasing factor receptor subtypes.
Topics: Animals; Behavior, Animal; Cocaine; Corticotropin-Releasing Hormone; Dopamine; Extracellular Space; Hormone Antagonists; Male; Microdialysis; Motor Activity; Nucleus Accumbens; Peptide Fragments; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Spatial Behavior; Ventral Tegmental Area | 2003 |
Extrahypothalamic corticotropin-releasing hormone mediates (-)-nicotine-induced elevation of plasma corticosterone in rats.
Topics: Animals; Corticosterone; Corticotropin-Releasing Hormone; Cyclooxygenase Inhibitors; Indomethacin; Male; Microdialysis; Nicotine; Norepinephrine; Paraventricular Hypothalamic Nucleus; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Time Factors | 2003 |
Corticotropin-releasing factor (CRF) and related peptides confer neuroprotection via type 1 CRF receptors.
Topics: 1-Methyl-3-isobutylxanthine; Amphibian Proteins; Amyloid beta-Peptides; Animals; Animals, Newborn; Apoptosis; Blotting, Western; Cell Survival; Cells, Cultured; Cerebellum; Cerebral Cortex; Chromatin; Chromones; Colforsin; Corticotropin-Releasing Hormone; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Glycogen Synthase Kinase 3; Hippocampus; In Situ Nick-End Labeling; Inhibitory Concentration 50; L-Lactate Dehydrogenase; Mitogen-Activated Protein Kinase Kinases; Morpholines; Neurons; Neuroprotective Agents; Peptide Fragments; Peptide Hormones; Peptides; Phosphorylation; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Thionucleotides; Time Factors; Urocortins; Urotensins; Vasodilator Agents | 2003 |
Delayed stress-induced colonic hypersensitivity in male Wistar rats: role of neurokinin-1 and corticotropin-releasing factor-1 receptors.
Topics: Animals; Colon; Electromyography; Fear; Hypersensitivity, Delayed; Immunohistochemistry; Indoles; Isoindoles; Male; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Nociceptors; Physical Stimulation; Piperidines; Pyrimidines; Pyrroles; Quinuclidines; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Receptors, Neurokinin-1; Stress, Psychological; Sympathectomy, Chemical; Sympathetic Nervous System | 2004 |
Effect of long-term blockade of CRF(1) receptors on exploratory behaviour, monoamines and transcription factor AP-2.
Topics: Animals; Biogenic Monoamines; Brain; DNA-Binding Proteins; Exploratory Behavior; Male; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Transcription Factor AP-2; Transcription Factors | 2004 |
CRF-receptor 1 blockade attenuates acute posttraumatic hyperglycemia in rats.
Topics: Acute Disease; Adrenocorticotropic Hormone; Animals; Biological Transport; Blood Glucose; Corticosterone; Dexamethasone; Glucocorticoids; Glucose; Hyperglycemia; Insulin; Male; Muscle, Skeletal; Phosphatidylinositol 3-Kinases; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Wounds and Injuries | 2004 |
Antidepressant effects of citalopram and CRF receptor antagonist CP-154,526 in a rat model of depression.
Topics: Animals; Antidepressive Agents; Behavior, Animal; Citalopram; Depression; Disease Models, Animal; Dose-Response Relationship, Drug; Pyrimidines; Pyrroles; Rats; Rats, Inbred Strains; Receptors, Corticotropin-Releasing Hormone; Social Behavior; Swimming | 2004 |
Transcriptional regulation of the CART promoter in CATH.a cells.
Topics: Animals; Cell Line; Colforsin; Corticotropin-Releasing Hormone; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Gene Expression Regulation; Locus Coeruleus; Mice; Mutagenesis, Site-Directed; Nerve Tissue Proteins; Neurotransmitter Agents; Promoter Regions, Genetic; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; RNA, Messenger; Transcription, Genetic | 2004 |
Does amygdaloid corticotropin-releasing hormone (CRH) mediate anxiety-like behaviors? Dissociation of anxiogenic effects and CRH release.
Topics: Amygdala; Animals; Anti-Anxiety Agents; Anxiety; Avoidance Learning; Behavior, Animal; Bombesin; Brain Chemistry; Corticotropin-Releasing Hormone; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Eating; Electroshock; Environment; Glutamic Acid; Hormone Antagonists; Male; Microdialysis; Peptide Fragments; Pyrimidines; Pyrroles; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone | 2004 |
CRF1 receptor antagonist CP-154,526 reduces cardiovascular responses during acute psychological stress in rabbits.
Topics: Adrenergic beta-Antagonists; Animals; Blood Pressure; Electroencephalography; Heart Rate; Propranolol; Pyrimidines; Pyrroles; Rabbits; Receptors, Corticotropin-Releasing Hormone; Stress, Psychological | 2004 |
The effects of CRF antagonists, antalarmin, CP154,526, LWH234, and R121919, in the forced swim test and on swim-induced increases in adrenocorticotropin in rats.
Topics: Adrenocorticotropic Hormone; Animals; Antidepressive Agents; Corticotropin-Releasing Hormone; Hypothalamo-Hypophyseal System; Male; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Restraint, Physical; Stress, Psychological; Swimming; Triazoles | 2005 |
Prior multiple ethanol withdrawals enhance stress-induced anxiety-like behavior: inhibition by CRF1- and benzodiazepine-receptor antagonists and a 5-HT1a-receptor agonist.
Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Buspirone; Central Nervous System Depressants; Drug Interactions; Ethanol; Flumazenil; Food, Formulated; GABA Modulators; Interpersonal Relations; Male; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Restraint, Physical; Serotonin Receptor Agonists; Stress, Psychological; Substance Withdrawal Syndrome; Time Factors | 2005 |
CRF receptor type 1 mediates continual hypoxia-induced CRF peptide and CRF mRNA expression increase in hypothalamic PVN of rats.
Topics: Adrenocorticotropic Hormone; Animals; Cell Hypoxia; Corticosterone; Gene Expression Regulation; Immunohistochemistry; In Situ Hybridization; Male; Paraventricular Hypothalamic Nucleus; Pituitary Gland; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger | 2005 |
Corticotropin-releasing factor receptor subtypes mediating nutritional suppression of estrous behavior in Syrian hamsters.
Topics: Animal Nutritional Physiological Phenomena; Animals; Corticotropin-Releasing Hormone; Cricetinae; Estrus; Female; Food Deprivation; Mesocricetus; Neuropeptide Y; Peptide Fragments; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Sexual Behavior, Animal; Urocortins | 2005 |
Comparison of the effects of diazepam, the CRF1 antagonist CP-154,526 and the group II mGlu receptor agonist LY379268 on stress-evoked extracellular norepinephrine levels.
Topics: Amino Acids; Animals; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; Extracellular Fluid; Male; Norepinephrine; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Receptors, Metabotropic Glutamate; Stress, Physiological | 2005 |
Effects of corticotropin-releasing hormone receptor antagonists on cocaine-induced dopamine overflow in the medial prefrontal cortex and nucleus accumbens of rats.
Topics: Animals; Chromatography, High Pressure Liquid; Cocaine; Corticotropin-Releasing Hormone; Dopamine; Dopamine Uptake Inhibitors; Male; Microdialysis; Nucleus Accumbens; Prefrontal Cortex; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone | 2005 |
CRH receptor type 1 mediates continual hypoxia-induced changes of immunoreactive prolactin and prolactin mRNA expression in rat pituitary.
Topics: Adrenalectomy; Adrenocorticotropic Hormone; Animals; Cold Temperature; Corticotropin-Releasing Hormone; Hypoxia; Immunohistochemistry; Male; Paraventricular Hypothalamic Nucleus; Peptide Fragments; Pituitary Gland; Prolactin; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Restraint, Physical; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Stress, Psychological | 2006 |
Effects of CP 154,526, a CRF1 receptor antagonist, on behavioral responses to cocaine in rats.
Topics: Animals; Behavior, Animal; Cocaine; Discrimination, Psychological; Dose-Response Relationship, Drug; Male; Motor Activity; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Reinforcement, Psychology; Self Administration | 2005 |
The CRH1 antagonist CP154,526 failed to alter ischemia-induced neurodegeneration and spatial memory deficits in rats but inhibited behavioral activity in the novel open field.
Topics: Animals; Behavior, Animal; Cell Count; Dose-Response Relationship, Drug; Exploratory Behavior; Hippocampus; Ischemia; Male; Memory Disorders; Nerve Degeneration; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Spatial Behavior; Time Factors | 2006 |
Endogenous expression and in vitro study of CRF-related peptides and CRF receptors in the rat gastric antrum.
Topics: Animals; Corticotropin-Releasing Hormone; DNA Primers; Gastric Emptying; Gene Expression Regulation; Immunohistochemistry; Male; Neurons; Pyloric Antrum; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Urocortins | 2006 |
Region-specific effects of brain corticotropin-releasing factor receptor type 1 blockade on footshock-stress- or drug-priming-induced reinstatement of morphine conditioned place preference in rats.
Topics: Amygdala; Animals; Behavior, Animal; Brain; Central Nervous System Agents; Cocaine; Conditioning, Operant; Extinction, Psychological; Heroin; Injections, Intraventricular; Learning; Male; Morphine; Nucleus Accumbens; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Reinforcement, Psychology; Septal Nuclei; Stress, Psychological | 2006 |
The corticotropin-releasing factor (CRF)(1) receptor antagonists CP154,526 and DMP695 inhibit light-induced phase advances of hamster circadian activity rhythms.
Topics: Animals; Circadian Rhythm; Corticotropin-Releasing Hormone; Cricetinae; Depressive Disorder; Dose-Response Relationship, Drug; Hypothalamo-Hypophyseal System; Jet Lag Syndrome; Light; Male; Mesocricetus; Pituitary-Adrenal System; Pyridines; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Stress, Psychological; Suprachiasmatic Nucleus | 2006 |
Anxiogenic and aversive effects of corticotropin-releasing factor (CRF) in the bed nucleus of the stria terminalis in the rat: role of CRF receptor subtypes.
Topics: Animals; Anxiety; Avoidance Learning; Behavior, Animal; Conditioning, Psychological; Corticotropin-Releasing Hormone; Male; Peptide Fragments; Pyrimidines; Pyrroles; Rats; Rats, Long-Evans; Receptors, Corticotropin-Releasing Hormone; Septal Nuclei | 2006 |
CP-154,526, a CRF type-1 receptor antagonist, attenuates the cue-and methamphetamine-induced reinstatement of extinguished methamphetamine-seeking behavior in rats.
Topics: Amphetamine-Related Disorders; Animals; Corticotropin-Releasing Hormone; Cues; Dose-Response Relationship, Drug; Extinction, Psychological; Hypothalamo-Hypophyseal System; Infusions, Intravenous; Injections, Intraperitoneal; Injections, Intraventricular; Ketoconazole; Male; Methamphetamine; Motivation; Pituitary-Adrenal System; Premedication; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Self Administration | 2007 |
Suppression of adrenocorticotrophic hormone secretion by simultaneous antagonism of vasopressin 1b and CRH-1 receptors on three different stress models.
Topics: Adrenocorticotropic Hormone; Animals; Antidiuretic Hormone Receptor Antagonists; Drug Administration Routes; Drug Administration Schedule; Drug Combinations; Drug Evaluation, Preclinical; Ether; Indoles; Male; Pyrimidines; Pyrroles; Pyrrolidines; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Restraint, Physical; Stress, Psychological; Swimming | 2006 |
An arginine vasopressin V1b antagonist, SSR149415 elicits antidepressant-like effects in an olfactory bulbectomy model.
Topics: Animals; Antidepressive Agents; Depression; Disease Models, Animal; Drug Administration Schedule; Indoles; Male; Olfactory Bulb; Pyrimidines; Pyrroles; Pyrrolidines; Rats; Rats, Wistar; Statistics, Nonparametric | 2007 |
Comparison of the V1b antagonist, SSR149415, and the CRF1 antagonist, CP-154,526, in rodent models of anxiety and depression.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Anxiety; Conditioning, Psychological; Depression; Female; Guinea Pigs; Humans; Indoles; Male; Maze Learning; Mice; Pyrimidines; Pyrroles; Pyrrolidines; Rats; Receptors, Corticotropin-Releasing Hormone; Receptors, Vasopressin; Vocalization, Animal | 2007 |
Effects of hypoxia on glucose, insulin, glucagon, and modulation by corticotropin-releasing factor receptor type 1 in the rat.
Topics: Altitude; Animals; Blood Glucose; Body Weight; Corticosterone; Eating; Glucagon; Hypoxia; Insulin; Leptin; Liver Glycogen; Male; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone | 2007 |
Corticotropin releasing factor-1 receptor antagonist, CP-154,526, blocks the expression of ethanol-induced behavioral sensitization in DBA/2J mice.
Topics: Analysis of Variance; Animals; Behavior, Animal; Central Nervous System Depressants; Dose-Response Relationship, Drug; Drug Interactions; Ethanol; Hormone Antagonists; Male; Mice; Mice, Inbred DBA; Motor Activity; Pyrimidines; Pyrroles; Time Factors | 2007 |
Blockade of the corticotropin releasing factor type 1 receptor attenuates elevated ethanol drinking associated with drinking in the dark procedures.
Topics: Alcohol Drinking; Alcoholism; Animals; Association Learning; Circadian Rhythm; Darkness; Dose-Response Relationship, Drug; Ethanol; Hypothalamo-Hypophyseal System; Injections, Intraperitoneal; Male; Mice; Mice, Inbred C57BL; Motor Activity; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone | 2008 |
The CRF-1 receptor antagonist, CP-154,526, attenuates stress-induced increases in ethanol consumption by BALB/cJ mice.
Topics: Alcohol Drinking; Alcoholism; Animals; Brain; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Signal Transduction; Species Specificity; Stress, Psychological | 2008 |
Corticotropin-releasing factor type 1 receptors mediate the visceral hyperalgesia induced by repeated psychological stress in rats.
Topics: Animals; Blood-Brain Barrier; Chronic Disease; Colon; Corticotropin-Releasing Hormone; Disease Models, Animal; Hyperalgesia; Infusion Pumps, Implantable; Injections, Subcutaneous; Male; Mechanotransduction, Cellular; Peptide Fragments; Pressure; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Rectum; Stress, Psychological | 2008 |
Corticotropin-releasing hormone receptor 1 coexists with endothelin-1 and modulates its mRNA expression and release in rat paraventricular nucleus during hypoxia.
Topics: Animals; Corticosterone; Endothelin-1; Gene Expression Regulation; Hypoxia; Male; Paraventricular Hypothalamic Nucleus; Pyrimidines; Pyrroles; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; RNA, Messenger; Time Factors | 2008 |
Corticotropin-releasing factor-1 receptor involvement in behavioral neuroadaptation to ethanol: a urocortin1-independent mechanism.
Topics: Adaptation, Biological; Adrenocorticotropic Hormone; Animals; Behavior, Animal; Ethanol; Gene Deletion; Mice; Mice, Inbred C57BL; Mice, Knockout; Mifepristone; Nervous System Physiological Phenomena; Psychomotor Performance; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Urocortins | 2008 |
Corticotropin-releasing hormone receptor 1 antagonist blocks colonic hypersensitivity induced by a combination of inflammation and repetitive colorectal distension.
Topics: Animals; Colitis; Colon; Dilatation, Pathologic; Electromyography; Humans; Inflammation; Irritable Bowel Syndrome; Male; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Trinitrobenzenesulfonic Acid | 2008 |
The alcohol deprivation effect in C57BL/6J mice is observed using operant self-administration procedures and is modulated by CRF-1 receptor signaling.
Topics: Alcoholism; Animals; Conditioning, Operant; Ethanol; Male; Mice; Mice, Inbred C57BL; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Self Administration; Signal Transduction; Substance Withdrawal Syndrome | 2009 |
Social subordination and polymorphisms in the gene encoding the serotonin transporter enhance estradiol inhibition of luteinizing hormone secretion in female rhesus monkeys.
Topics: Analysis of Variance; Animals; Body Weight; Dominance-Subordination; Estradiol; Female; Hydrocortisone; Hypothalamo-Hypophyseal System; Individuality; Luteinizing Hormone; Macaca mulatta; Pituitary-Adrenal System; Polymorphism, Genetic; Pyrimidines; Pyrroles; Radioimmunoassay; Receptors, Corticotropin-Releasing Hormone; Serotonin Plasma Membrane Transport Proteins; Social Environment; Stress, Psychological | 2009 |
The alarm pheromone in male rats as a unique anxiety model: psychopharmacological evidence using anxiolytics.
Topics: Administration, Inhalation; Animals; Anti-Anxiety Agents; Anxiety; Buspirone; Clonidine; Disease Models, Animal; Male; Midazolam; Phenelzine; Pheromones; Propranolol; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Reflex, Startle | 2010 |
CRF-1 antagonist and CRF-2 agonist decrease binge-like ethanol drinking in C57BL/6J mice independent of the HPA axis.
Topics: Alcohol-Induced Disorders, Nervous System; Animals; Corticotropin-Releasing Hormone; Disease Models, Animal; Hormone Antagonists; Hypothalamo-Hypophyseal System; Injections, Intraperitoneal; Injections, Intraventricular; Male; Mice; Mice, Inbred C57BL; Mifepristone; Peptide Fragments; Pyridines; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Signal Transduction; Urocortins | 2010 |
Pain is a salient "stressor" that is mediated by corticotropin-releasing factor-1 receptors.
Topics: Aniline Compounds; Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Corticotropin-Releasing Hormone; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Hyperalgesia; Indomethacin; Inflammation; Male; Mice; Pain; Pain Threshold; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Spinal Cord Injuries; Stomach Ulcer; Stress, Psychological | 2010 |
Blocking corticotropin-releasing factor-2 receptors, but not corticotropin-releasing factor-1 receptors or glucocorticoid feedback, disrupts the development of conditioned defeat.
Topics: Aggression; Analysis of Variance; Animals; Antimetabolites; Association Learning; Conditioning, Classical; Cricetinae; Dominance-Subordination; Feedback, Physiological; Glucocorticoids; Hormone Antagonists; Hypothalamo-Hypophyseal System; Male; Mesocricetus; Metyrapone; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone | 2010 |
Stress-induced priming of glutamate synapses unmasks associative short-term plasticity.
Topics: Animals; Biophysical Phenomena; Biophysics; Chelating Agents; Corticotropin-Releasing Hormone; Dizocilpine Maleate; Drug Interactions; Egtazic Acid; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Exocytosis; Freezing Reaction, Cataleptic; Glutamic Acid; In Vitro Techniques; Male; Neuronal Plasticity; Neurons; Paraventricular Hypothalamic Nucleus; Patch-Clamp Techniques; Pyrimidines; Pyrroles; Quinoxalines; Rats; Rats, Sprague-Dawley; SNARE Proteins; Stress, Physiological; Synapses; Time Factors | 2010 |
Restraint stress-induced reduction in prepulse inhibition in Brown Norway rats: role of the CRF2 receptor.
Topics: Acoustic Stimulation; Analysis of Variance; Animals; Grooming; Male; Pyrimidines; Pyrroles; Rats; Receptors, Corticotropin-Releasing Hormone; Reflex, Startle; Restraint, Physical; Sensory Gating; Stress, Physiological | 2011 |
[(76) Br]BMK-152, a nonpeptide analogue, with high affinity and low nonspecific binding for the corticotropin-releasing factor type 1 receptor.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Autoradiography; Barium Radioisotopes; Binding Sites; Binding, Competitive; Brain; In Vitro Techniques; Ligands; Macaca mulatta; Male; Mice; Mice, Knockout; Protein Binding; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Triazines | 2011 |
Prevention of social stress-escalated cocaine self-administration by CRF-R1 antagonist in the rat VTA.
Topics: Animals; Cocaine; Cocaine-Related Disorders; Locomotion; Male; Neurons; Pyrimidines; Pyrroles; Rats; Rats, Long-Evans; Receptors, Corticotropin-Releasing Hormone; Reinforcement Schedule; Self Administration; Stress, Psychological; Ventral Tegmental Area | 2011 |
Pretreatment with CP-154526 blocks the modifying effects of alarm pheromone on components of sexual behavior in male, but not in female, rats.
Topics: Animals; Female; Male; Pheromones; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Sex Characteristics; Sexual Behavior, Animal | 2011 |
Effects of acute stress on acquisition of nicotine conditioned place preference in adolescent rats: a role for corticotropin-releasing factor 1 receptors.
Topics: Acute Disease; Age Factors; Animals; Conditioning, Psychological; Dose-Response Relationship, Drug; Male; Nicotine; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Stress, Psychological | 2012 |
α(2) Adrenergic and imidazoline receptor agonists prevent cue-induced cocaine seeking.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Cocaine; Cues; Dose-Response Relationship, Drug; Drug Interactions; Drug-Seeking Behavior; Extinction, Psychological; Guanfacine; Imidazoles; Imidazoline Receptors; Isoquinolines; Male; Motor Activity; Naphthyridines; Prazosin; Propranolol; Pyrimidines; Pyrroles; Quinoxalines; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology; Self Administration | 2011 |
Lifelong CRF overproduction is associated with altered gene expression and sensitivity of discrete GABA(A) and mGlu receptor subtypes.
Topics: Animals; Corticotropin-Releasing Hormone; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Agonists; Gene Expression Regulation; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Pyridines; Pyrimidines; Pyrroles; Rats; Receptors, GABA-A; Receptors, Metabotropic Glutamate | 2012 |
Alcohol in excess: CRF₁ receptors in the rat and mouse VTA and DRN.
Topics: Alcohol Drinking; Animals; Dose-Response Relationship, Drug; Drinking; Ethanol; Male; Mice; Mice, Inbred C57BL; Pyrimidines; Pyrroles; Raphe Nuclei; Rats; Rats, Long-Evans; Receptors, Corticotropin-Releasing Hormone; Species Specificity; Ventral Tegmental Area | 2013 |
Role of corticotropin-releasing factor (CRF) receptor-1 on the catecholaminergic response to morphine withdrawal in the nucleus accumbens (NAc).
Topics: Animals; Corticosterone; Dopamine; Male; Morphine; Morphine Dependence; Naloxone; Neurons; Norepinephrine; Nucleus Accumbens; Phosphorylation; Proto-Oncogene Proteins c-fos; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Serine; Substance Withdrawal Syndrome; Tyrosine 3-Monooxygenase; Ventral Tegmental Area | 2012 |
Long-term loss of dopamine release mediated by CRF-1 receptors in the rat lateral septum after repeated cocaine administration.
Topics: Animals; Cocaine; Corticotropin-Releasing Hormone; Dopamine; Dopamine Uptake Inhibitors; Drug Administration Schedule; Drug Interactions; Male; Microdialysis; Peptides, Cyclic; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Septum of Brain; Time Factors | 2013 |
Differential effect of orexin-1 and CRF-1 antagonism on stress circuits: a fMRI study in the rat with the pharmacological stressor Yohimbine.
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Aminopyridines; Amygdala; Animals; Benzazepines; Corpus Striatum; Corticosterone; Dopamine Antagonists; Functional Neuroimaging; Gyrus Cinguli; Male; Medetomidine; Neural Pathways; Orexin Receptor Antagonists; Piperidines; Pyrimidines; Pyrroles; Rats; Receptors, Corticotropin-Releasing Hormone; Stress, Psychological; Yohimbine | 2013 |
CRF1 receptor antagonists do not reverse pharmacological disruption of prepulse inhibition in rodents.
Topics: Acoustic Stimulation; Animals; Corticotropin-Releasing Hormone; Dextroamphetamine; Dizocilpine Maleate; Dopamine; Dose-Response Relationship, Drug; Hydrocarbons, Halogenated; Ketamine; Male; Mice; Mice, Transgenic; Nucleus Accumbens; Prefrontal Cortex; Prepulse Inhibition; Pyridines; Pyrimidines; Pyrroles; Rats; Receptors, Corticotropin-Releasing Hormone; Reflex, Startle; Thiazines | 2014 |
Drug-induced suppression of ACTH secretion does not promote anti-depressive or anxiolytic effects.
Topics: Adrenocorticotropic Hormone; Analysis of Variance; Animals; Anti-Anxiety Agents; Anxiety; Disease Models, Animal; Dose-Response Relationship, Drug; Indoles; Interpersonal Relations; Male; Maze Learning; Pyrimidines; Pyrroles; Pyrrolidines; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Swimming | 2014 |
Neurokinin B signaling in the female rat: a novel link between stress and reproduction.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arcuate Nucleus of Hypothalamus; Corticosterone; Corticotropin-Releasing Hormone; Female; Gonadotropin-Releasing Hormone; Injections, Intraventricular; Lipopolysaccharides; Luteinizing Hormone; Neurokinin B; Neurons; Ovariectomy; Peptide Fragments; Pyrimidines; Pyrroles; Quinolines; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Receptors, Neurokinin-3; Receptors, Vasopressin; Reproduction; Signal Transduction; Stress, Physiological; Substance P | 2014 |
Epigenetic upregulation of corticotrophin-releasing hormone mediates postnatal maternal separation-induced memory deficiency.
Topics: Acetylation; Animals; Animals, Newborn; Corticotropin-Releasing Hormone; Electric Stimulation; Epigenesis, Genetic; Hippocampus; Histones; Long-Term Potentiation; Maternal Deprivation; Maze Learning; Memory Disorders; Methyl-CpG-Binding Protein 2; Neuronal Plasticity; Phosphorylation; Promoter Regions, Genetic; Pyrimidines; Pyrroles; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; RNA, Messenger; Up-Regulation | 2014 |
Prevention of alcohol-heightened aggression by CRF-R1 antagonists in mice: critical role for DRN-PFC serotonin pathway.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aggression; Alcohol Drinking; Animals; Central Nervous System Agents; Central Nervous System Depressants; Dorsal Raphe Nucleus; Ethanol; Mice; Neural Pathways; Prefrontal Cortex; Pyridazines; Pyrimidines; Pyrroles; Receptor, Serotonin, 5-HT1A; Receptors, Corticotropin-Releasing Hormone; Self Administration; Serotonin; Serotonin 5-HT1 Receptor Agonists; Thiazoles | 2014 |
Dissociation of μ-opioid receptor and CRF-R1 antagonist effects on escalated ethanol consumption and mPFC serotonin in C57BL/6J mice.
Topics: Alcohol Drinking; Aminopyridines; Animals; Behavior, Animal; Central Nervous System Depressants; Dorsal Raphe Nucleus; Ethanol; Immunohistochemistry; Infusions, Intraventricular; Male; Mice; Mice, Inbred C57BL; Microdialysis; Naltrexone; Narcotic Antagonists; Prefrontal Cortex; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Receptors, Opioid, mu; Self Administration; Serotonin; Tryptophan Hydroxylase | 2016 |
Injection of corticotropin-releasing hormone into the amygdala aggravates visceral nociception and induces noradrenaline release in rats.
Topics: Amygdala; Animals; Colon; Corticotropin-Releasing Hormone; Dilatation, Pathologic; Dopamine; Male; Nociception; Norepinephrine; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Rectum; Serotonin | 2015 |
Corticotropin-releasing factor 1 receptor mediates the activity of the reward system evoked by morphine-induced conditioned place preference.
Topics: Animals; Conditioning, Operant; Hormone Antagonists; Locus Coeruleus; Male; Mice; Morphine; Morphine Dependence; Narcotics; Neurons; Nucleus Accumbens; Pyrimidines; Pyrroles; Random Allocation; Receptors, Corticotropin-Releasing Hormone; Reward; Spatial Behavior; Ventral Tegmental Area | 2015 |
Reduction of ethanol intake by corticotropin-releasing factor receptor-1 antagonist in "heavy-drinking" mice in a free-choice paradigm.
Topics: Alcohol Drinking; Amygdala; Animals; Choice Behavior; Drinking; Ethanol; Male; Mice; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone | 2015 |
Long-term effects of early adolescent stress: dysregulation of hypothalamic-pituitary-adrenal axis and central corticotropin releasing factor receptor 1 expression in adult male rats.
Topics: Animals; Anxiety; Corticosterone; Depression; Disease Models, Animal; Electroshock; Exercise Therapy; Foot; Hypothalamo-Hypophyseal System; Male; Maze Learning; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Random Allocation; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Running; Stress Disorders, Post-Traumatic; Stress, Psychological | 2015 |
Lifelong disturbance of serotonin transporter functioning results in fear learning deficits: Reversal by blockade of CRF1 receptors.
Topics: Animals; Basolateral Nuclear Complex; Disease Models, Animal; Dorsal Raphe Nucleus; Fear; Gene Knockout Techniques; Learning; Learning Disabilities; Male; Neurotransmitter Agents; Paroxetine; Prepulse Inhibition; Pyrimidines; Pyrroles; Rats, Transgenic; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Reflex, Startle; RNA-Binding Proteins; RNA, Messenger | 2015 |
CP-154,526 Modifies CREB Phosphorylation and Thioredoxin-1 Expression in the Dentate Gyrus following Morphine-Induced Conditioned Place Preference.
Topics: Animals; Blotting, Western; Cells, Cultured; Conditioning, Psychological; Cyclic AMP Response Element-Binding Protein; Dentate Gyrus; Fluorescent Antibody Technique; Immunoenzyme Techniques; Male; Mice; Morphine; Morphine Dependence; Narcotics; Neurons; Phosphorylation; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Thioredoxins | 2015 |
Role of Corticotropin Releasing Factor 1 Signaling in Cocaine Seeking during Early Extinction in Female and Male Rats.
Topics: Animals; Cocaine; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Extinction, Psychological; Female; Male; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; Self Administration; Signal Transduction | 2016 |
CRF
Topics: Animals; Anti-Anxiety Agents; Benzodioxoles; Corticotropin-Releasing Hormone; Dose-Response Relationship, Drug; Drug Interactions; Guinea Pigs; Maternal Deprivation; Mice; Mice, Transgenic; Mifepristone; Paroxetine; Pyridines; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Receptors, Glucocorticoid; Steroids; Vocalization, Animal | 2017 |
The non-peptide CRH1-antagonist CP-154,526 elicits a paradoxical route-dependent activation of the HPA axis.
Topics: Adrenocorticotropic Hormone; Animals; Arterial Pressure; Heart Rate; Hypothalamo-Hypophyseal System; Injections, Intra-Arterial; Injections, Intraperitoneal; Male; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone | 2017 |
The effects of enhancing endocannabinoid signaling and blocking corticotrophin releasing factor receptor in the amygdala and hippocampus on the consolidation of a stressful event.
Topics: Amidohydrolases; Animals; Anxiety; Basolateral Nuclear Complex; Benzamides; CA1 Region, Hippocampal; Carbamates; Disease Models, Animal; Endocannabinoids; Male; Memory Consolidation; Nootropic Agents; Pyrimidines; Pyrroles; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Corticotropin-Releasing Hormone; Reflex, Startle; RNA, Messenger; Stress Disorders, Post-Traumatic; Stress, Psychological | 2017 |
Chondroprotection by urocortin involves blockade of the mechanosensitive ion channel Piezo1.
Topics: Autocrine Communication; Calcium; Cartilage, Articular; Cell Survival; Cells, Cultured; Chondrocytes; Cyclic AMP; Humans; Ion Channels; Paracrine Communication; Peptide Fragments; Peptides, Cyclic; Protein Conformation; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Signal Transduction; Urocortins | 2017 |
Early adolescent stress-induced changes in prefrontal cortex miRNA-135a and hippocampal miRNA-16 in male rats.
Topics: Age Factors; Animals; Anxiety; Disease Models, Animal; Hippocampus; Male; MicroRNAs; Paroxetine; Prefrontal Cortex; Pyrimidines; Pyrroles; Rats; Receptor, Serotonin, 5-HT1A; Receptors, Corticotropin-Releasing Hormone; Selective Serotonin Reuptake Inhibitors; Spatial Memory; Stress, Psychological | 2017 |
Maternal stress and the MPOA: Activation of CRF receptor 1 impairs maternal behavior and triggers local oxytocin release in lactating rats.
Topics: Analysis of Variance; Animals; Animals, Newborn; Carrier Proteins; Corticotropin-Releasing Hormone; Female; Gene Expression Regulation; Hormone Antagonists; Lactation; Male; Maternal Behavior; Maze Learning; Microdialysis; Oxytocin; Preoptic Area; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Corticotropin-Releasing Hormone; RNA, Messenger | 2018 |
Conditioned aversive memory associated with morphine withdrawal increases brain-derived neurotrophic factor in dentate gyrus and basolateral amygdala.
Topics: Affect; Analgesics, Opioid; Animals; Basolateral Nuclear Complex; Brain-Derived Neurotrophic Factor; Conditioning, Classical; Corticosterone; Corticotropin-Releasing Hormone; Cyclic AMP Response Element-Binding Protein; Dentate Gyrus; Extinction, Psychological; Male; Memory; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Morphine; Naloxone; Narcotic Antagonists; Protein Precursors; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Substance Withdrawal Syndrome | 2020 |
Central angiotensin II type 1 receptor as a therapeutic target against frequent urination.
Topics: Amphibian Proteins; Angiotensin II; Angiotensin II Type 1 Receptor Blockers; Animals; Male; Peptide Hormones; Pyrimidines; Pyrroles; Rats; Rats, Wistar; Receptors, Corticotropin-Releasing Hormone; Telmisartan; Urination | 2019 |
Naloxone-induced conditioned place aversion score and extinction period are higher in C57BL/6J morphine-dependent mice than in Swiss: Role of HPA axis.
Topics: Animals; Avoidance Learning; Conditioning, Operant; Extinction, Psychological; Hypothalamo-Hypophyseal System; Male; Memory; Mice; Mice, Inbred C57BL; Morphine; Morphine Dependence; Naloxone; Narcotic Antagonists; Narcotics; Pituitary-Adrenal System; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Substance Withdrawal Syndrome | 2021 |
Sex-specific plasticity in CRF regulation of inhibitory control in central amygdala CRF1 neurons after chronic voluntary alcohol drinking.
Topics: Alcohol Drinking; Animals; Central Amygdaloid Nucleus; Corticotropin-Releasing Hormone; Ethanol; Female; gamma-Aminobutyric Acid; Male; Mice; Neurons; Pyrimidines; Pyrroles; Receptors, Corticotropin-Releasing Hormone; Receptors, GABA-A; Sex Characteristics; Synaptic Transmission | 2022 |