Page last updated: 2024-08-18

pyrroles and bisindolylmaleimide i

pyrroles has been researched along with bisindolylmaleimide i in 19 studies

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (10.53)18.2507
2000's13 (68.42)29.6817
2010's4 (21.05)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bonev, AD; Nelson, MT1
Goekjian, PG; Jirousek, MR1
Aravamudan, B; Broadie, K1
Larsson, C; Svensson, K1
Abe, K; Misawa, M1
Dewey, WL; Elzey, MJ; Javed, RR; Smith, FL1
Calixto, JB; El Sayah, M1
Han, JS; Kim, DS; Kim, TW; Yoon, MS1
Dewey, WL; Javed, RR; Smith, FL; Smith, PA1
Bowman, L; Castranova, V; Ding, M; Huang, C; Lu, Y; Vallyathan, V1
Nuwayhid, SJ; Werling, LL1
Dewey, WL; Gabra, BH; Javed, RR; Smith, FL; Smith, PA1
Bartlett, SR; Bennett, PR; Duggan, SV; Iglesias, T; Lindstrom, T; Mann, GE1
Eggo, MC; Susarla, R; Watkinson, JC1
Adwanikar, H; Fu, Y; Han, J; Ishola, T; Neugebauer, V; Ramsey, C; Scerbo, M1
Azuma, M; Morimoto-Tochigi, A; Nakajima, E; Shearer, TR; Walkup, RD1
Chang, Y; Lin, YW; Wang, SJ1
Dai, Y; Kobayashi, K; Kogure, Y; Noguchi, K; Wan, Y; Wang, S; Yamanaka, H; Zhang, W; Zhu, W1
Berrout, J; Boukelmoune, N; Mamenko, M; O'Neil, RG; Pochynyuk, O; Zaika, OL1

Reviews

1 review(s) available for pyrroles and bisindolylmaleimide i

ArticleYear
Protein kinase C in the treatment of disease: signal transduction pathways, inhibitors, and agents in development.
    Current medicinal chemistry, 1999, Volume: 6, Issue:9

    Topics: Azepines; Bryostatins; Carbazoles; Enzyme Inhibitors; Humans; Hydroxybenzoates; Indoles; Lactones; Macrolides; Maleimides; Oligodeoxyribonucleotides, Antisense; Protein Kinase C; Pyrroles; Signal Transduction; Thionucleotides

1999

Other Studies

18 other study(ies) available for pyrroles and bisindolylmaleimide i

ArticleYear
Muscarinic inhibition of ATP-sensitive K+ channels by protein kinase C in urinary bladder smooth muscle.
    The American journal of physiology, 1993, Volume: 265, Issue:6 Pt 1

    Topics: Adenosine Triphosphate; Animals; Benzopyrans; Carbachol; Cromakalim; Diglycerides; Glyburide; Guanosine Diphosphate; Guinea Pigs; In Vitro Techniques; Indoles; Maleimides; Membrane Potentials; Muscarinic Antagonists; Muscle, Smooth; Potassium Channels; Protein Kinase C; Pyrroles; Receptors, Muscarinic; Tetradecanoylphorbol Acetate; Thionucleotides; Urinary Bladder

1993
Synaptic Drosophila UNC-13 is regulated by antagonistic G-protein pathways via a proteasome-dependent degradation mechanism.
    Journal of neurobiology, 2003, Feb-15, Volume: 54, Issue:3

    Topics: Acetylcysteine; Animals; Antibodies; Blotting, Western; Caenorhabditis elegans Proteins; Carbazoles; Carrier Proteins; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cysteine Endopeptidases; Drosophila; Drosophila Proteins; Drug Interactions; Enzyme Inhibitors; Estrenes; GTP-Binding Proteins; Helminth Proteins; Horseradish Peroxidase; Immunohistochemistry; Indoles; Insect Proteins; Maleimides; Microscopy, Confocal; Multienzyme Complexes; Mutation; Neomycin; Neuromuscular Junction; Oligopeptides; Phorbol Esters; Phospholipid Ethers; Presynaptic Terminals; Proteasome Endopeptidase Complex; Pyrroles; Pyrrolidinones; Synapses; Tumor Suppressor Proteins; Type C Phospholipases

2003
A protein kinase Cbeta inhibitor attenuates multidrug resistance of neuroblastoma cells.
    BMC cancer, 2003, Mar-26, Volume: 3

    Topics: Carboplatin; Cell Line, Tumor; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Synergism; Humans; Indoles; Maleimides; Mesylates; Neuroblastoma; Paclitaxel; Peripheral Nervous System Neoplasms; Protein Kinase C; Pyrroles; Tumor Cells, Cultured; Vincristine

2003
Astrocyte stellation induced by Rho kinase inhibitors in culture.
    Brain research. Developmental brain research, 2003, Jun-12, Volume: 143, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Actins; Amides; Animals; Astrocytes; Carbazoles; Cell Size; Cells, Cultured; Cerebral Cortex; Colchicine; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Gout Suppressants; Indoles; Intracellular Signaling Peptides and Proteins; Maleimides; Phalloidine; Protein Serine-Threonine Kinases; Pyridines; Pyrroles; Rats; rho-Associated Kinases

2003
The expression of a high level of morphine antinociceptive tolerance in mice involves both PKC and PKA.
    Brain research, 2003, Sep-19, Volume: 985, Issue:1

    Topics: Analgesics; Animals; Brain; Carbazoles; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Drug Interactions; Drug Therapy, Combination; Drug Tolerance; Enzyme Inhibitors; Indoles; Injections, Intraventricular; Isoquinolines; Male; Maleimides; Mice; Morphine; Morphine Dependence; Pain; Protein Kinase C; Protein Serine-Threonine Kinases; Pyrroles

2003
New evidence on the mechanisms underlying bradykinin-mediated contraction of the pig iris sphincter in vitro.
    Peptides, 2003, Volume: 24, Issue:7

    Topics: Animals; Benzamides; Bradykinin; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Calcium; Calcium Channels; Capsaicin; Carbazoles; Conotoxins; Dipeptides; Dose-Response Relationship, Drug; Egtazic Acid; In Vitro Techniques; Indoles; Iris; Maleimides; Muscle Contraction; Nicardipine; omega-Agatoxin IVA; Peptide Fragments; Piperidines; Protein Kinase Inhibitors; Protein Kinases; Pyrroles; Receptors, Calcitonin Gene-Related Peptide; Receptors, Drug; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Swine; Tachykinins

2003
Thyrotropin-releasing hormone increases phospholipase D activity through stimulation of protein kinase C in GH3 cells.
    Endocrine, 2004, Volume: 23, Issue:1

    Topics: Animals; Calcium; Cell Line, Tumor; Diglycerides; Enzyme Activation; Enzyme Inhibitors; Estrenes; Indoles; Isoenzymes; Maleimides; Phospholipase D; Protein Kinase C; Protein Transport; Pyrroles; Pyrrolidinones; Rats; Thyrotropin-Releasing Hormone

2004
PKC and PKA inhibitors reverse tolerance to morphine-induced hypothermia and supraspinal analgesia in mice.
    European journal of pharmacology, 2004, May-25, Volume: 492, Issue:2-3

    Topics: Analgesics, Opioid; Animals; Carbazoles; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Drug Tolerance; Hypothermia, Induced; Indoles; Injections, Intraventricular; Injections, Spinal; Male; Maleimides; Mice; Morphine; Pain Measurement; Protein Kinase C; Pyrroles; Tail

2004
Involvement of protein kinase C in crystalline silica-induced activation of the MAP kinase and AP-1 pathway.
    American journal of physiology. Lung cellular and molecular physiology, 2006, Volume: 290, Issue:2

    Topics: Animals; Cell Line; Crystallization; Enzyme Activation; Enzyme Inhibitors; Indoles; Maleimides; MAP Kinase Signaling System; Mice; Naphthalenes; Protein Kinase C; Protein Kinase C-alpha; Protein Kinase C-epsilon; Protein Transport; Pyrroles; Silicon Dioxide; Transcription Factor AP-1; Transfection

2006
Sigma2 (sigma2) receptors as a target for cocaine action in the rat striatum.
    European journal of pharmacology, 2006, Mar-27, Volume: 535, Issue:1-3

    Topics: Animals; Benzylamines; Calcium; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Enzyme Inhibitors; In Vitro Techniques; Indoles; Male; Maleimides; Mesylates; N-Methylaspartate; Nomifensine; Pentazocine; Piperidines; Protein Kinase C; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, sigma; Sigma-1 Receptor; Spiro Compounds; Sulfonamides; Tritium

2006
PKC and PKA inhibitors reinstate morphine-induced behaviors in morphine tolerant mice.
    Pharmacological research, 2006, Volume: 54, Issue:6

    Topics: Analgesics, Opioid; Animals; Behavior, Animal; Body Temperature; Carbazoles; Cyclic AMP-Dependent Protein Kinases; Drug Implants; Drug Tolerance; Enzyme Inhibitors; Hot Temperature; Hypothermia; Indoles; Injections, Intraventricular; Isoquinolines; Male; Maleimides; Mice; Morphine; Pain; Protein Kinase C; Pyrroles; Reaction Time

2006
Role of atypical protein kinase C isozymes and NF-kappaB in IL-1beta-induced expression of cyclooxygenase-2 in human myometrial smooth muscle cells.
    Journal of cellular physiology, 2007, Volume: 210, Issue:3

    Topics: Cells, Cultured; Cyclooxygenase 2; Enzyme Inhibitors; Female; Gene Expression Regulation; Gene Expression Regulation, Enzymologic; Humans; Indoles; Interleukin-1; Isoenzymes; Maleimides; Mesylates; Myocytes, Smooth Muscle; Myometrium; NF-kappa B; p38 Mitogen-Activated Protein Kinases; Protein Kinase C; Pyrroles; RNA, Messenger

2007
Regulation of plasminogen activators in human thyroid follicular cells and their relationship to differentiated function.
    Journal of cellular physiology, 2007, Volume: 212, Issue:3

    Topics: Adenylyl Cyclases; Aprotinin; Cell Differentiation; Cells, Cultured; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Activators; Epidermal Growth Factor; Fibroblast Growth Factors; Flavonoids; Humans; Indoles; Insulin; Iodine; Iodine Radioisotopes; Maleimides; Mesylates; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Plasminogen Inactivators; Protein Kinase C; Protein Kinase C beta; Protein Kinase Inhibitors; Pyrroles; RNA, Messenger; Serine Proteinase Inhibitors; Signal Transduction; Tetradecanoylphorbol Acetate; Thyroid Gland; Thyrotropin; Time Factors; Tissue Plasminogen Activator; Urokinase-Type Plasminogen Activator

2007
PKA and ERK, but not PKC, in the amygdala contribute to pain-related synaptic plasticity and behavior.
    Molecular pain, 2008, Jul-16, Volume: 4

    Topics: Amygdala; Animals; Arthritis; Behavior; Butadienes; Carbazoles; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Disease Models, Animal; Enzyme Activation; Extracellular Signal-Regulated MAP Kinases; Indoles; Male; Maleimides; Neuronal Plasticity; Neurons; Nitriles; Pain; Protein Kinase C; Protein Kinase Inhibitors; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Thionucleotides

2008
Mechanism for carbachol-induced secretion of lacritin in cultured monkey lacrimal acinar cells.
    Investigative ophthalmology & visual science, 2010, Volume: 51, Issue:9

    Topics: Anilides; Animals; Calcium; Carbachol; Cells, Cultured; Cholinergic Agonists; Enzyme Inhibitors; Eye Proteins; Gene Expression Profiling; Glycoproteins; Immunohistochemistry; Indoles; Lacrimal Apparatus; Macaca mulatta; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Oligonucleotide Array Sequence Analysis; Protein Kinase C; Pyrroles; RNA, Messenger; Signal Transduction; Thiadiazoles

2010
Idebenone inhibition of glutamate release from rat cerebral cortex nerve endings by suppression of voltage-dependent calcium influx and protein kinase A.
    Naunyn-Schmiedeberg's archives of pharmacology, 2011, Volume: 384, Issue:1

    Topics: 4-Aminopyridine; Animals; Aspartic Acid; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium Signaling; Carbazoles; Cerebral Cortex; Clonazepam; Cyclic AMP-Dependent Protein Kinases; Dantrolene; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glutamate Plasma Membrane Transport Proteins; Glutamic Acid; Indoles; Isoquinolines; Macrolides; Male; Maleimides; Membrane Potentials; Nerve Endings; omega-Conotoxins; Potassium; Protein Kinase C; Protein Kinase Inhibitors; Pyrroles; Rats; Rats, Sprague-Dawley; Sodium-Calcium Exchanger; Sulfonamides; Synaptosomes; Thiazepines; Ubiquinone

2011
Potentiation of the P2X3 ATP receptor by PAR-2 in rat dorsal root ganglia neurons, through protein kinase-dependent mechanisms, contributes to inflammatory pain.
    The European journal of neuroscience, 2012, Volume: 36, Issue:3

    Topics: Adenosine Triphosphate; Animals; Carbazoles; Colforsin; Cyclic AMP-Dependent Protein Kinases; Ganglia, Spinal; Indoles; Inflammation; Male; Maleimides; MAP Kinase Signaling System; Membrane Potentials; Neurons; Pain; Phosphorylation; Protein Kinase C; Protein Transport; Purinergic P2X Receptor Agonists; Purinergic P2X Receptor Antagonists; Pyrroles; Rats, Sprague-Dawley; Receptor, PAR-2; Receptors, Purinergic P2X3; Tetradecanoylphorbol Acetate

2012
Discrete control of TRPV4 channel function in the distal nephron by protein kinases A and C.
    The Journal of biological chemistry, 2013, Jul-12, Volume: 288, Issue:28

    Topics: Animals; Calcium; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Fura-2; In Vitro Techniques; Indoles; Isoquinolines; Kidney Tubules, Collecting; Maleimides; Mice; Mice, Inbred C57BL; Microscopy, Fluorescence; Morpholines; Nephrons; Perfusion; Phorbol Esters; Protein Kinase C; Protein Kinase Inhibitors; Protein Transport; Pyrroles; Signal Transduction; Sulfonamides; TRPV Cation Channels

2013