pyrroles has been researched along with aprikalim in 33 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 5 (15.15) | 18.7374 |
1990's | 28 (84.85) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Berry, JL; Foster, RW; Small, RC | 1 |
Downing, SJ; Hollingsworth, M; Piper, I | 1 |
Ashford, ML; Ben-Ari, Y; Zini, S | 1 |
Berry, JL; Elliott, KR; Foster, RW; Green, KA; Murray, MA; Small, RC | 1 |
Longmore, J; Newgreen, DT; Weston, AH | 1 |
Berry, JL; Cook, SJ; Foster, RW; Green, KA; Murray, MA; Small, RC | 1 |
Hood, JS; Kadowitz, PJ; McMahon, TJ | 1 |
Bray, KM; Longmore, J; Weston, AH | 1 |
Brown, TJ; Raeburn, D | 1 |
Cavero, I; Mondot, S; Montier, F; Pratz, J | 1 |
Franke, C; Hatt, H; Quasthoff, S; Richter-Turtur, M | 1 |
Downing, SJ; Hollingsworth, M; Minshall, E; Piper, I; Sadraei, H | 1 |
Lederer, WJ; Nichols, CG; Ripoll, C | 1 |
Neumcke, B; Weik, R | 1 |
Cavero, I; Courteix, J; Escande, D; Laville, M; Le Guern, S; Thuringer, D | 1 |
Hollingsworth, M; Piper, I | 1 |
Eltze, M | 1 |
Grafe, P; Lehmann-Horn, F; Quasthoff, S; Spuler, A | 1 |
Brown, TJ; Raeburn, D; Sweetland, J | 1 |
Hollingsworth, M; Piper, IT | 1 |
Atwal, KS | 1 |
Grover, GJ | 2 |
Edwards, G; Weston, AH | 1 |
Cavero, I; Premmereur, J | 1 |
Mayhan, WG | 2 |
Bowring, NE; Clapham, JC; Fuller, DA; Good, DM; Trail, BK | 1 |
Advenier, C; Dumas, JP; Dumas, M; Giudicelli, JF | 1 |
Ha, JH; Kim, WJ; Lee, KY | 1 |
Fattaccini, CM; Haj-Dahmane, S; Hamon, M; Lanfumey, L; Laporte, AM; Vantalon, V | 1 |
Greenwood, IA; Weston, AH | 1 |
Cheuk, JM; Hollingsworth, M; Hughes, SJ; Maresh, MJ; Piper, IT | 1 |
3 review(s) available for pyrroles and aprikalim
Article | Year |
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Pharmacology and structure-activity relationships for KATP modulators: tissue-selective KATP openers.
Topics: Action Potentials; Adenosine Triphosphate; Animals; Antihypertensive Agents; Benzopyrans; Cardiovascular Diseases; Cromakalim; Diazoxide; Guanidines; Guinea Pigs; Minoxidil; Muscle Relaxation; Muscle, Smooth, Vascular; Niacinamide; Nicorandil; Picolines; Pinacidil; Potassium Channels; Pyrans; Pyrroles; Radioligand Assay; Rats; Structure-Activity Relationship; Vasodilator Agents | 1994 |
Protective effects of ATP-sensitive potassium-channel openers in experimental myocardial ischemia.
Topics: Action Potentials; Adenosine Triphosphate; Animals; Benzopyrans; Cromakalim; Dihydropyridines; Disease Models, Animal; Dogs; Guanidines; Guinea Pigs; Myocardial Contraction; Myocardial Infarction; Myocardial Ischemia; Picolines; Pinacidil; Potassium Channels; Pyrans; Pyrroles; Rats; Vasodilator Agents | 1994 |
Pharmacology of ATP-sensitive potassium channel (KATP) openers in models of myocardial ischemia and reperfusion.
Topics: Animals; ATP-Binding Cassette Transporters; Benzopyrans; Cromakalim; Guanidines; Humans; Ischemic Preconditioning, Myocardial; KATP Channels; Mitochondria, Heart; Models, Cardiovascular; Myocardial Ischemia; Myocardial Reperfusion; Niacinamide; Nicorandil; Picolines; Pinacidil; Potassium Channels; Potassium Channels, Inwardly Rectifying; Pyrans; Pyrroles; Rats | 1997 |
30 other study(ies) available for pyrroles and aprikalim
Article | Year |
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Tracheal relaxation induced by potassium channel opening drugs: its antagonism by adrenergic neurone blocking agents.
Topics: Adrenergic Antagonists; Animals; Benzopyrans; Cromakalim; Dose-Response Relationship, Drug; Female; Guanidines; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Relaxation; Parasympatholytics; Picolines; Pinacidil; Potassium Channels; Pyrans; Pyrroles; Rubidium Radioisotopes; Stereoisomerism; Theophylline; Trachea | 1992 |
Cross tolerance between cromakalim and RP49356 in the uterus of the rat in vivo and in vitro.
Topics: Animals; Benzopyrans; Cromakalim; Drug Tolerance; Female; In Vitro Techniques; Infusions, Intravenous; Picolines; Potassium Channels; Pyrans; Pyrroles; Rats; Uterine Contraction; Uterus | 1992 |
Characterization of sulfonylurea receptors and the action of potassium channel openers on cholinergic neurotransmission in guinea pig isolated small intestine.
Topics: Adenosine Triphosphate; Animals; ATP-Binding Cassette Transporters; Benzopyrans; Choline; Cromakalim; Electric Stimulation; Glyburide; Guinea Pigs; Intestine, Small; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Picolines; Potassium Channels; Potassium Channels, Inwardly Rectifying; Pyrans; Pyrroles; Receptors, Drug; Sulfonylurea Receptors; Synaptic Transmission; Tritium | 1991 |
Mechanical, biochemical and electrophysiological studies of RP 49356 and cromakalim in guinea-pig and bovine trachealis muscle.
Topics: 2',3'-Cyclic-Nucleotide Phosphodiesterases; Animals; Benzopyrans; Bronchodilator Agents; Calcium; Cattle; Cromakalim; Cyclic AMP; Electrophysiology; Guinea Pigs; In Vitro Techniques; Intracellular Fluid; Kinetics; Membrane Potentials; Muscle Relaxation; Muscle, Smooth; Picolines; Potassium Channels; Pyrans; Pyrroles; Trachea | 1991 |
Effects of cromakalim, RP49356, diazoxide, glibenclamide and galanin in rat portal vein.
Topics: Adenosine Triphosphate; Animals; Benzopyrans; Cromakalim; Diazoxide; Galanin; Glyburide; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Peptides; Picolines; Portal Vein; Potassium Channels; Pyrans; Pyrroles; Rats; Rats, Inbred Strains; Rubidium Radioisotopes; Vasodilator Agents | 1990 |
Guinea-pig isolated trachealis: the effects of charybdotoxin on mechanical activity, membrane potential changes and the activity of plasmalemmal K(+)-channels.
Topics: Adrenergic beta-Agonists; Animals; Benzopyrans; Calcium; Cell Membrane; Charybdotoxin; Cromakalim; Guinea Pigs; In Vitro Techniques; Isoproterenol; Membrane Potentials; Muscle Relaxation; Muscle, Smooth; Picolines; Potassium Channels; Pyrans; Pyrroles; Scorpion Venoms; Theophylline; Trachea; Vasodilator Agents | 1991 |
Pulmonary vasodilator responses to RP 52891 are mediated by activation of a glibenclamide-sensitive K+ATP channel.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetylcholine; Adenosine Triphosphate; Animals; Benzopyrans; Blood Gas Analysis; Blood Pressure; Cats; Cromakalim; Female; Glyburide; Guanidines; Hydrogen-Ion Concentration; Isoproterenol; Male; Nitroprusside; Picolines; Pinacidil; Potassium Channels; Prostaglandin Endoperoxides, Synthetic; Pulmonary Circulation; Pyrans; Pyrroles; Vasodilation; Vasodilator Agents | 1991 |
The contribution of Rb-permeable potassium channels to the relaxant and membrane hyperpolarizing actions of cromakalim, RP49356 and diazoxide in bovine tracheal smooth muscle.
Topics: Animals; Benzopyrans; Cattle; Cromakalim; Diazoxide; Electrophysiology; In Vitro Techniques; Isometric Contraction; Muscle, Smooth; Picolines; Potassium Channels; Potassium Radioisotopes; Pyrans; Pyrroles; Rubidium; Rubidium Radioisotopes; Trachea | 1991 |
RP 49356 and cromakalim relax airway smooth muscle in vitro by opening a sulphonylurea-sensitive K+ channel: a comparison with nifedipine.
Topics: Animals; Benzopyrans; Calcium; Cromakalim; Glipizide; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Nifedipine; Picolines; Potassium Channels; Pyrans; Pyrroles; Trachea | 1991 |
Effects of the K+ channel activators, RP 52891, cromakalim and diazoxide, on the plasma insulin level, plasma renin activity and blood pressure in rats.
Topics: Animals; Antihypertensive Agents; Benzopyrans; Blood Glucose; Blood Pressure; Cromakalim; Diazoxide; Drug Interactions; Glucose; Glyburide; Infusions, Intravenous; Insulin; Male; Membrane Potentials; Picolines; Potassium Channels; Pyrans; Pyrroles; Rats; Renin | 1991 |
Two different types of potassium channels in human skeletal muscle activated by potassium channel openers.
Topics: Adenosine Triphosphate; Benzopyrans; Cromakalim; Dihydropyridines; Electrophysiology; Glyburide; Humans; Muscles; Picolines; Potassium Channels; Pyrans; Pyrroles | 1990 |
Effects of several potassium channel openers and glibenclamide on the uterus of the rat.
Topics: Animals; Benzopyrans; Blood Pressure; Cromakalim; Female; Glyburide; Guanidines; Heart Rate; Hemodynamics; In Vitro Techniques; Oxytocin; Parasympatholytics; Picolines; Pinacidil; Potassium Channels; Potassium Chloride; Pregnancy; Pyrans; Pyrroles; Rats; Rats, Inbred Strains; Uterus; Vasodilator Agents | 1990 |
Modulation of ATP-sensitive K+ channel activity and contractile behavior in mammalian ventricle by the potassium channel openers cromakalim and RP49356.
Topics: Adenosine Triphosphate; Animals; Benzopyrans; Cromakalim; Dose-Response Relationship, Drug; Glucose; Guinea Pigs; In Vitro Techniques; Myocardial Contraction; Picolines; Potassium Channels; Pyrans; Pyrroles; Rats | 1990 |
Effects of potassium channel openers on single potassium channels in mouse skeletal muscle.
Topics: Adenosine Triphosphate; Animals; Benzopyrans; Calcium; Cromakalim; Female; Guanidines; In Vitro Techniques; Membrane Potentials; Mice; Muscles; Organ Specificity; Picolines; Pinacidil; Potassium Channels; Pyrans; Pyrroles | 1990 |
Potassium channel openers act through an activation of ATP-sensitive K+ channels in guinea-pig cardiac myocytes.
Topics: Adenosine Triphosphate; Animals; Benzopyrans; Cromakalim; Electrophysiology; Glyburide; Guanidines; Guinea Pigs; Heart; In Vitro Techniques; Ion Channel Gating; Muscle, Smooth, Vascular; Picolines; Pinacidil; Potassium Channels; Pyrans; Pyrroles; Subtraction Technique | 1989 |
Cromakalim, RP49356, pinacidil and minoxidil sulphate in the rat uterus and their antagonism by glibenclamide. Smooth Muscle Research Group.
Topics: Animals; Benzopyrans; Cromakalim; Female; Glyburide; Guanidines; In Vitro Techniques; Minoxidil; Parasympatholytics; Picolines; Pinacidil; Pyrans; Pyrroles; Rats; Rats, Inbred Strains; Uterine Contraction | 1989 |
Glibenclamide is a competitive antagonist of cromakalim, pinacidil and RP 49356 in guinea-pig pulmonary artery.
Topics: Animals; Benzopyrans; Cromakalim; Glyburide; Guanidines; Guinea Pigs; In Vitro Techniques; Male; Methylene Blue; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Niacinamide; Nicorandil; Picolines; Pinacidil; Potassium Channels; Potassium Chloride; Pulmonary Artery; Purinones; Pyrans; Pyrroles; Tetraethylammonium Compounds | 1989 |
Cromakalim, pinacidil and RP 49356 activate a tolbutamide-sensitive K+ conductance in human skeletal muscle fibres.
Topics: Benzopyrans; Cromakalim; Guanidines; Humans; In Vitro Techniques; Membrane Potentials; Muscles; Picolines; Pinacidil; Potassium Channels; Pyrans; Pyrroles; Tolbutamide; Vasodilator Agents | 1989 |
Comparison of the effects of RP 49356, cromakalim and nifedipine on guinea-pig trachea in vitro.
Topics: Animals; Benzopyrans; Cromakalim; Guinea Pigs; In Vitro Techniques; Male; Muscle, Smooth; Nifedipine; Picolines; Potassium Channels; Pyrans; Pyrroles; Trachea | 1989 |
Cromakalim- and RP 49356-induced 42K+ and 86Rb+ efflux in rat myometrium.
Topics: Animals; Benzopyrans; Cromakalim; Female; Ion Transport; Myometrium; Oxytocin; Picolines; Potassium; Potassium Channels; Potassium Chloride; Pregnancy; Pyrans; Pyrroles; Rats; Rubidium; Time Factors; Vasodilator Agents | 1995 |
KATP--fact or artefact? New thoughts on the mode of action of the potassium channel openers.
Topics: Animals; Benzopyrans; Cromakalim; Electrophysiology; Guanidines; Insulinoma; Ion Channel Gating; Muscle, Smooth, Vascular; Pancreatic Neoplasms; Phosphorylation; Picolines; Potassium Channels; Pyrans; Pyrroles; Rats; Tumor Cells, Cultured; Vasodilator Agents | 1994 |
ATP sensitive potassium channel openers are of potential benefit in ischaemic heart disease.
Topics: Benzopyrans; Cromakalim; Dihydropyridines; Guanidines; Humans; Myocardial Ischemia; Myocardium; Niacinamide; Nicorandil; Picolines; Pinacidil; Potassium Channels; Pyrans; Pyrroles; Sodium-Potassium-Exchanging ATPase; Vasodilator Agents | 1994 |
Effect of diabetes mellitus on response of the basilar artery to activation of ATP-sensitive potassium channels.
Topics: Adenosine Triphosphate; Animals; Basilar Artery; Benzopyrans; Blood Pressure; Cromakalim; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Male; Nitroglycerin; Picolines; Potassium Channels; Pyrans; Pyrroles; Rats; Rats, Sprague-Dawley; Vasodilator Agents | 1994 |
Effects of levcromakalim and RP52891 on NANCe nerve-mediated changes in pulmonary dynamics evoked by vagal stimulation in the guinea-pig.
Topics: Airway Resistance; Animals; Autonomic Nervous System; Benzopyrans; Bronchoconstriction; Bronchodilator Agents; Cromakalim; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Lung; Male; Picolines; Potassium Channels; Pyrans; Pyrroles; Respiration; Respiratory Function Tests; Vagus Nerve | 1993 |
Effects of three K+ channel openers on airways and pulmonary circulation in the isolated guinea-pig lung.
Topics: Animals; Benzopyrans; Bronchoconstriction; Cromakalim; Dose-Response Relationship, Drug; Guanidines; Guinea Pigs; In Vitro Techniques; Lung; Male; Muscle Contraction; Muscle, Smooth, Vascular; Picolines; Pinacidil; Potassium; Potassium Channels; Pulmonary Circulation; Pyrans; Pyrroles | 1993 |
In vivo reactivity of resistance arterioles to activation of ATP-sensitive K+ channels.
Topics: Animals; Antihypertensive Agents; Arginine; Benzopyrans; Cheek; Cricetinae; Cromakalim; Male; Mesocricetus; Microcirculation; Muscle, Smooth, Vascular; Nitric Acid; omega-N-Methylarginine; Picolines; Potassium Channels; Pyrans; Pyrroles | 1993 |
Actions of potassium channel openers in rat detrusor urinae.
Topics: Animals; Benzopyrans; Cromakalim; Guanidines; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Picolines; Potassium Channels; Pyrans; Pyrroles; Rats; Rats, Sprague-Dawley; Urinary Bladder | 1993 |
Possible involvement of K(ATP) channels in the control of 5-HT neurons.
Topics: Adenosine Triphosphate; Animals; Autoradiography; Benzopyrans; Cromakalim; Electrophysiology; GABA-A Receptor Antagonists; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Male; Neurons; Picolines; Potassium Channels; Pyrans; Pyrroles; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Sulfonylurea Compounds | 1993 |
Effects of rubidium on responses to potassium channel openers in rat isolated aorta.
Topics: Animals; Antihypertensive Agents; Aorta, Thoracic; Benzopyrans; Cromakalim; In Vitro Techniques; Male; Microelectrodes; Muscle Relaxation; Muscle, Smooth, Vascular; Picolines; Portal Vein; Potassium Channels; Potassium Chloride; Potassium Radioisotopes; Pyrans; Pyrroles; Rats; Rats, Sprague-Dawley; Rubidium; Rubidium Radioisotopes; Tachyphylaxis; Vasodilator Agents | 1993 |
Inhibition of contractions of the isolated human myometrium by potassium channel openers.
Topics: Benzopyrans; Cromakalim; Female; Glyburide; Humans; Ion Channel Gating; Oxytocin; Parasympatholytics; Picolines; Potassium Channels; Potassium Chloride; Potassium Radioisotopes; Pregnancy; Pyrans; Pyrroles; Uterine Contraction | 1993 |