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pyro(l-alpha-aminoadipyl)-l-histidyl-l-thiazolidine-4-carboxamide and thiazolidines

pyro(l-alpha-aminoadipyl)-l-histidyl-l-thiazolidine-4-carboxamide has been researched along with thiazolidines in 38 studies

Compound Research Comparison

Studies
(pyro(l-alpha-aminoadipyl)-l-histidyl-l-thiazolidine-4-carboxamide)
Trials
(pyro(l-alpha-aminoadipyl)-l-histidyl-l-thiazolidine-4-carboxamide)
Recent Studies (post-2010)
(pyro(l-alpha-aminoadipyl)-l-histidyl-l-thiazolidine-4-carboxamide)
Studies
(thiazolidines)
Trials
(thiazolidines)
Recent Studies (post-2010) (thiazolidines)
47003,5441601,407

Research

Studies (38)

TimeframeStudies, this research(%)All Research%
pre-199034 (89.47)18.7374
1990's4 (10.53)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Singh, DK; Yarbrough, GG1
Sharif, NA; To, ZP; Whiting, RL1
Hutson, PH; Middlemiss, DN; Semark, JE1
Barrett, JE; Brady, LS1
Michel, AD; Sharif, NA; To, Z; Whiting, RL1
Helke, CJ; Phillips, ET1
Dailey, A; Markush, S; Pranzatelli, MR1
Pranzatelli, MR1
Bansinath, M; Bhargava, HN1
Horita, A; Simasko, SM1
Bhargava, HN; Matwyshyn, GA1
Faden, AI1
Ambrose, F; Barbaz, B; Bittiger, H; Iyengar, S; Neale, RF; Petrack, B; Rinehart, RK; Steel, DJ; Williams, M; Wood, PL1
Jacobowitz, DM; Sills, MA1
Carino, MA; Horita, A; Lai, H1
Jacobowitz, DM; Mellow, AM; Sills, MA; Sunderland, T1
Bergmann, F; Elam, R; Feuerstein, G1
Schechter, LE; Simansky, KJ1
Bhargava, HN; Das, S1
Faden, AI; Jacobs, TP1
Funatsu, K; Inanaga, K; Teshima, S1
Ogawa, N1
Horita, A; Kalivas, PW; Santori, EM; Schmidt, DE1
Rastogi, RB; Singhal, RL1
Hichens, M1
Moore, KE; Nielsen, JA1
Barrett, JE; Brady, LS; Valentine, JO1
Ezra, D; Faden, AI; Feuerstein, G; Lux, WE; Snyder, F1
Demarest, KT; Moore, KE; Yamada, K1
Fadok, VA; Lothrop, CD; Tamas, PM1
Clineschmidt, BV; Lotti, VJ; Yarbrough, GG1
Arison, BH; Hirschmann, R; Holly, FW; Homnick, C; Nutt, RF; Veber, DF1
Carino, MA; Horita, A1
Delarue, C; Jegou, S; Kupryszewski, G; Leboulenger, F; Leroux, P; Netchitailo, P; Perroteau, I; Tonon, MC; Vaudry, H1
Horita, A1
Antolik, EK; Faison, EP; Yarbrough, GG1
Deshpande, SB; Warnick, JE1
Handley, SL; McCreary, AC1

Other Studies

38 other study(ies) available for pyro(l-alpha-aminoadipyl)-l-histidyl-l-thiazolidine-4-carboxamide and thiazolidines

ArticleYear
Effects of MK-771 on the isolated amphibian spinal cord: comparison with thyrotropin-releasing hormone.
    Canadian journal of physiology and pharmacology, 1979, Volume: 57, Issue:8

    Topics: Animals; Bufonidae; Dipeptides; In Vitro Techniques; Membrane Potentials; Spinal Cord; Thiazoles; Thiazolidines; Thyrotropin-Releasing Hormone

1979
Analogs of thyrotropin-releasing hormone (TRH): receptor affinities in brains, spinal cords, and pituitaries of different species.
    Neurochemical research, 1991, Volume: 16, Issue:2

    Topics: Animals; Binding, Competitive; Brain; Cattle; Dogs; Pituitary Gland, Anterior; Pyrrolidonecarboxylic Acid; Rabbits; Rats; Receptors, Neurotransmitter; Receptors, Thyrotropin-Releasing Hormone; Sheep; Species Specificity; Spinal Cord; Thiazolidines; Thyrotropin-Releasing Hormone

1991
The TRH analogue MK-771, increases acetylcholine release in hippocampus but not striatum of the conscious rat.
    Neuroscience letters, 1990, Aug-14, Volume: 116, Issue:1-2

    Topics: Acetylcholine; Animals; Antidepressive Agents; Chromatography, High Pressure Liquid; Corpus Striatum; Hippocampus; Kinetics; Male; Organ Specificity; Rats; Rats, Inbred Strains; Thiazolidines; Thyrotropin-Releasing Hormone

1990
Neuropeptide modulation of the behavioral effects of drugs.
    Progress in clinical and biological research, 1985, Volume: 192

    Topics: Animals; Chlordiazepoxide; Columbidae; Conditioning, Psychological; Drug Interactions; Electroshock; Haloperidol; Neurotensin; Pentobarbital; Rabbits; Reinforcement, Psychology; Saimiri; Substance P; Thiazolidines; Thyrotropin-Releasing Hormone

1985
Differential affinities of TRH analogs at the mammalian spinal cord TRH receptor: implications for therapy in spinal injuries.
    Neuroscience letters, 1989, Sep-25, Volume: 104, Issue:1-2

    Topics: Animals; Binding, Competitive; Guinea Pigs; Pyrrolidonecarboxylic Acid; Rabbits; Rats; Receptors, Neurotransmitter; Receptors, Thyrotropin-Releasing Hormone; Spinal Cord; Spinal Injuries; Thiazolidines; Thyrotropin-Releasing Hormone

1989
Thyrotropin-releasing hormone receptor activation in the spinal cord increases blood pressure and sympathetic tone to the vasculature and the adrenals.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:1

    Topics: Adrenal Glands; Adrenalectomy; Animals; Autonomic Nerve Block; Blood Pressure; Cardiovascular System; Heart Rate; Hemodynamics; Injections, Spinal; Male; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Thyrotropin-Releasing Hormone; Regional Blood Flow; Spinal Cord; Sympathetic Nervous System; Thiazolidines; Thyrotropin-Releasing Hormone; Vascular Resistance

1988
The regulation of TRH and serotonin receptors: chronic TRH and analog administration in the rat.
    Journal of receptor research, 1988, Volume: 8, Issue:5

    Topics: Animals; Behavior, Animal; Binding, Competitive; Biogenic Amines; Brain Stem; Cerebral Cortex; Chromatography, High Pressure Liquid; Hypothalamus; In Vitro Techniques; Locomotion; Male; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Receptors, Serotonin; Receptors, Thyrotropin-Releasing Hormone; Spinal Cord; Thiazolidines; Thyrotropin-Releasing Hormone

1988
The comparative pharmacology of the behavioral syndromes induced by TRH and by 5-HT in the rat.
    General pharmacology, 1988, Volume: 19, Issue:2

    Topics: 5-Hydroxytryptophan; 5,7-Dihydroxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Antidepressive Agents; Behavior, Animal; Body Temperature; Cisterna Magna; Injections; Male; Pyrimidines; Rats; Rats, Inbred Strains; Serotonin; Tetrahydronaphthalenes; Thiazolidines; Thyrotropin-Releasing Hormone

1988
Evidence for a peripheral action of thyrotropin releasing hormone on gastrointestinal transit in mice.
    Neuropharmacology, 1988, Volume: 27, Issue:4

    Topics: Animals; Antidepressive Agents; Antipsychotic Agents; Drug Synergism; Gastrointestinal Transit; Loperamide; Male; Mice; Mice, Inbred Strains; Morphine; Naltrexone; Narcotic Antagonists; Quaternary Ammonium Compounds; Thiazolidines; Thyrotropin-Releasing Hormone

1988
Treatment of rats with the TRH analog MK-771. Down-regulation of TRH receptors and behavioral tolerance.
    Neuropharmacology, 1985, Volume: 24, Issue:2

    Topics: Animals; Body Temperature; Depression, Chemical; Drug Tolerance; Injections, Intraventricular; Male; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Thyrotropin-Releasing Hormone; Thiazolidines; Thyrotropin-Releasing Hormone

1985
Comparative effects of thyrotropin releasing hormone, MK-771 and DN-1417 on morphine abstinence syndrome.
    Psychopharmacology, 1985, Volume: 87, Issue:2

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Anticonvulsants; Body Temperature; Body Weight; Male; Mice; Morphine Dependence; Naloxone; Substance Withdrawal Syndrome; Thiazolidines; Thyrotropin-Releasing Hormone; Time Factors

1985
New pharmacologic approaches to spinal cord injury: opiate antagonists and thyrotropin-releasing hormone.
    Central nervous system trauma : journal of the American Paralysis Association, 1985,Spring, Volume: 2, Issue:1

    Topics: Animals; Azocines; Cats; Endorphins; Enkephalin, Leucine; Humans; Naloxone; Narcotic Antagonists; Rabbits; Receptors, Opioid; Spinal Cord Injuries; Thiazolidines; Thyrotropin-Releasing Hormone

1985
Benzodiazepine interactions with central thyroid-releasing hormone binding sites: characterization and physiological significance.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:1

    Topics: Amygdala; Animals; Benzodiazepines; Brain; Cerebral Cortex; Chlordiazepoxide; Corpus Striatum; Cyclic GMP; Flunitrazepam; Kinetics; Male; Membranes; Midazolam; Pentobarbital; Pyrazoles; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Thyrotropin-Releasing Hormone; Sleep; Thiazolidines; Thyrotropin; Thyrotropin-Releasing Hormone

1986
Chronic administration of desipramine or nialamide decreases wet-dog shakes in rats produced by the TRH-analog MK-771.
    Brain research, 1987, Jan-13, Volume: 401, Issue:1

    Topics: Animals; Desipramine; Drug Synergism; Male; Motor Activity; Nialamide; Rats; Rats, Inbred Strains; Stereotyped Behavior; Thiazolidines; Thyrotropin-Releasing Hormone

1987
Preliminary studies on the effects of a TRH analog, MK-771, in an animal model of Alzheimer's disease.
    Proceedings of the Western Pharmacology Society, 1987, Volume: 30

    Topics: Alzheimer Disease; Animals; Antidepressive Agents; Disease Models, Animal; Rats; Thiazolidines; Thyrotropin-Releasing Hormone

1987
Central muscarinic cholinergic antagonists block wet-dog shakes produced by the TRH analog MK-771 in the rat.
    Brain research, 1988, Jun-21, Volume: 453, Issue:1-2

    Topics: Animals; Atropine; Dose-Response Relationship, Drug; Injections, Intraperitoneal; Male; Movement Disorders; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine; Thiazolidines; Thyrotropin-Releasing Hormone

1988
Interaction of thyrotropin-releasing hormone (TRH) and serotonin in cardiovascular control.
    European journal of pharmacology, 1988, Sep-01, Volume: 154, Issue:1

    Topics: Animals; Blood Pressure; Catecholamines; Cats; Female; Heart Rate; Hemorrhage; Male; Methysergide; Serotonin; Thiazolidines; Thyrotropin-Releasing Hormone

1988
Properties of some 1-arylpiperazines as antagonists of stereotyped behaviors mediated by central serotonergic receptors in rodents.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 247, Issue:3

    Topics: Animals; Brain; Dose-Response Relationship, Drug; Male; Metergoline; Mice; Motor Activity; Piperazines; Rats; Receptors, Serotonin; Serotonin Antagonists; Stereotyped Behavior; Syndrome; Thiazolidines; Thyrotropin-Releasing Hormone

1988
Lack of interaction between thyrotropin releasing hormone and its analogs with 3H-quinuclidinyl benzilate recognition sites in the rat striatum.
    Neuropharmacology, 1985, Volume: 24, Issue:7

    Topics: Animals; Anticonvulsants; Corpus Striatum; In Vitro Techniques; Male; Rats; Rats, Inbred Strains; Receptors, Cholinergic; Receptors, Muscarinic; Thiazolidines; Thyrotropin-Releasing Hormone

1985
Effect of TRH analogs on neurologic recovery after experimental spinal trauma.
    Neurology, 1985, Volume: 35, Issue:9

    Topics: Animals; Cats; Spinal Cord Injuries; Thiazolidines; Thyrotropin-Releasing Hormone

1985
Binding of TRH, DN-1417 and MK-771 to TRH receptors in the rat brain. Relationship to their central actions.
    The Kurume medical journal, 1983, Volume: 30 Suppl

    Topics: Animals; Binding Sites; Brain; Guanosine Triphosphate; Male; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, Thyrotropin-Releasing Hormone; Thiazolidines; Thyrotropin-Releasing Hormone

1983
Biochemical properties of TRH receptors in the rat central nervous system.
    The Kurume medical journal, 1983, Volume: 30 Suppl

    Topics: Animals; Brain; Cations; Dithiothreitol; Ethylmaleimide; Radioligand Assay; Rats; Receptors, Cell Surface; Receptors, Thyrotropin-Releasing Hormone; Synaptic Membranes; Thiazolidines; Thyrotropin-Releasing Hormone

1983
Failure of muscarinic blockade to antagonize analepsis induced by thyrotropin-releasing hormone and MK-771 in the rat.
    Psychopharmacology, 1981, Volume: 74, Issue:1

    Topics: Animals; Central Nervous System Stimulants; Hippocampus; Male; Mice; Parasympatholytics; Phenobarbital; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Species Specificity; Thiazolidines; Thyrotropin-Releasing Hormone

1981
MK-771 enhances the turnover of norepinephrine in brain.
    Research communications in chemical pathology and pharmacology, 1981, Volume: 33, Issue:1

    Topics: Animals; Brain; Corpus Striatum; Male; Norepinephrine; Olfactory Bulb; Rats; Stimulation, Chemical; Thiazolidines; Thyrotropin-Releasing Hormone; Tyrosine 3-Monooxygenase

1981
A comparison of thyrotropin-releasing hormone with analogs: influence of disposition upon pharmacology.
    Drug metabolism reviews, 1983, Volume: 14, Issue:1

    Topics: Animals; Brain; Central Nervous System; Drug Stability; Humans; Intestinal Absorption; Pituitary Gland; Receptors, Cell Surface; Receptors, Thyrotropin-Releasing Hormone; Thiazolidines; Thyrotropin-Releasing Hormone

1983
Thyrotropin-releasing hormone and its analog MK-771 increase the cerebroventricular perfusate content of dihydroxyphenylacetic acid.
    Journal of neurochemistry, 1984, Volume: 43, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Cerebral Ventricles; Dose-Response Relationship, Drug; Male; Perfusion; Phenylacetates; Rats; Rats, Inbred Strains; Thiazolidines; Thyrotropin-Releasing Hormone

1984
Effects of thyrotropin-releasing hormone (TRH) and a TRH analogue, MK-771, on punished responding of squirrel monkeys.
    Psychopharmacology, 1984, Volume: 83, Issue:2

    Topics: Animals; Conditioning, Psychological; Food; Male; Punishment; Saimiri; Thiazolidines; Thyrotropin-Releasing Hormone

1984
Hypotension produced by platelet-activating factor is reversed by thyrotropin-releasing hormone.
    Circulatory shock, 1984, Volume: 13, Issue:3

    Topics: Animals; Blood Pressure; Guinea Pigs; Hypotension; Male; Naloxone; Platelet Activating Factor; Thiazolidines; Thyrotropin-Releasing Hormone; Time Factors

1984
Effects of behaviorally active doses of thyrotropin-releasing hormone and its analog MK-771 on dopaminergic neuronal systems in the brain of the rat.
    Neuropharmacology, 1984, Volume: 23, Issue:7A

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Behavior, Animal; Brain; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Dose-Response Relationship, Drug; Limbic System; Male; Mesencephalon; Muscle Contraction; Neurons; Rats; Receptors, Dopamine; Substantia Nigra; Thiazolidines; Thyrotropin-Releasing Hormone

1984
Canine and feline thyroid function assessment with the thyrotropin-releasing hormone response test.
    American journal of veterinary research, 1984, Volume: 45, Issue:11

    Topics: Animals; Cats; Dogs; Dose-Response Relationship, Drug; Stimulation, Chemical; Thiazolidines; Thyroid Function Tests; Thyroid Gland; Thyrotropin-Releasing Hormone; Thyroxine; Triiodothyronine

1984
Investigations on the interaction of thyrotropin-releasing hormone (TRH) and MK-771 with central noradrenergic mechanisms.
    Psychopharmacology, 1980, Volume: 70, Issue:2

    Topics: Animals; Brain Chemistry; Catecholamines; Central Nervous System; Dipeptides; Female; Methazolamide; Methyltyrosines; Norepinephrine; Rats; Reflex; Thiazolidines; Thyrotropin-Releasing Hormone

1980
Synthesis of thyrotropin-releasing hormone analogues with selective central nervous system effects.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:6

    Topics: Central Nervous System; Pyrrolidonecarboxylic Acid; Structure-Activity Relationship; Thiazolidines; Thyrotropin-Releasing Hormone; Thyroxine; Triiodothyronine

1981
A comparison of the pharmacological properties of TRH and MK-771.
    Proceedings of the Western Pharmacology Society, 1981, Volume: 24

    Topics: Animals; Blood Pressure; Gastrointestinal Motility; Injections, Intraventricular; Male; Pentobarbital; Rabbits; Thiazolidines; Thyrotropin-Releasing Hormone

1981
In vitro study of frog (Rana ridibunda Pallas) neurointermediate lobe secretion by use of a simplified perifusion system. I. Effect of TRH analogs upon alpha-MSH release.
    General and comparative endocrinology, 1982, Volume: 46, Issue:1

    Topics: Animals; Brain; Male; Melanocyte-Stimulating Hormones; Rana ridibunda; Ranidae; Thiazolidines; Thyrotropin-Releasing Hormone

1982
Peptides in central regulation of the parasympathetic nervous system.
    Proceedings of the Western Pharmacology Society, 1982, Volume: 25

    Topics: Animals; Digestive System Physiological Phenomena; Parasympathetic Nervous System; Peptides; Rabbits; Thiazolidines; Thyrotropin-Releasing Hormone

1982
MK-771 antagonizes the enhanced response to apomorphine in rats treated chronically with haloperidol - implications for tardive dyskinesia.
    Neuroscience letters, 1982, Dec-31, Volume: 34, Issue:3

    Topics: Animals; Apomorphine; Disease Models, Animal; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Female; Haloperidol; Humans; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereotyped Behavior; Thiazolidines; Thyrotropin-Releasing Hormone

1982
Analogs of thyrotropin-releasing hormone in potentiating the spinal monosynaptic reflex in vitro.
    European journal of pharmacology, 1994, Dec-27, Volume: 271, Issue:2-3

    Topics: Animals; In Vitro Techniques; Pyrrolidonecarboxylic Acid; Rats; Reflex, Monosynaptic; Spinal Cord; Structure-Activity Relationship; Thiazolidines; Thyrotropin-Releasing Hormone

1994
The thyrotrophin-releasing hormone analogue MK771 induces tic-like behaviours: the effects of dopamine D1 and D2 receptor antagonists.
    European journal of pharmacology, 1999, Mar-12, Volume: 369, Issue:1

    Topics: Animals; Antidepressive Agents; Behavior, Animal; Behavioral Symptoms; Benzazepines; Blinking; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Male; Mice; Raclopride; Receptors, Dopamine D1; Salicylamides; Sulpiride; Thiazolidines; Thyrotropin-Releasing Hormone; Tic Disorders

1999