Page last updated: 2024-08-16

pyrimethamine and thiabendazole

pyrimethamine has been researched along with thiabendazole in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19902 (9.52)18.7374
1990's13 (61.90)18.2507
2000's1 (4.76)29.6817
2010's5 (23.81)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Afzelius, L; Andersson, TB; Baroni, M; Cruciani, G; Karlén, A; Masimirembwa, CM; Mecucci, S; Zamora, I1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Gozalbes, R; Pineda-Lucena, A1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Carere, A; Conti, G; Conti, L; Crebelli, R1
Coulaud, JP; Pasticier, A; Payet, M; Saimot, G1
Barrett-Connor, E1
Natarajan, AT1
Bassani, B; Leopardi, P; Pacchierotti, F; Zijno, A1
Adler, ID1
Hartley-Asp, B; Wallin, M1
Parry, JM1
Parry, EM; Parry, JM; Warr, TJ1
Parry, JM; Sors, A1
Duivenvoorden, WC; Meijers, M; Natarajan, AT; Zwanenburg, TS1
Di Sibio, A; Lomi, A; Sbrana, I; Scarcelli, V1
Lynch, AM; Parry, JM1
Aardema, MJ; Brauninger, RM; Carr, GJ; Gibson, DP; Kerckaert, GA; LeBoeuf, RA1
Barale, R; Barrai, I; Bernacchi, F; Betti, C; Marrazzini, A1

Reviews

4 review(s) available for pyrimethamine and thiabendazole

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Drugs for the treatment of parasitic infection.
    The Medical clinics of North America, 1982, Volume: 66, Issue:1

    Topics: Antimony; Bithionol; Chloroquine; Diethylcarbamazine; Humans; Mebendazole; Melarsoprol; Metronidazole; Niclosamide; Niridazole; Oxamniquine; Parasitic Diseases; Pentamidine; Piperazines; Primaquine; Pyrantel Pamoate; Pyrimethamine; Suramin; Thiabendazole; Trichlorfon

1982
Synopsis of the in vivo results obtained with the 10 known or suspected aneugens tested in the CEC collaborative study.
    Mutation research, 1993, Volume: 287, Issue:1

    Topics: Aneuploidy; Animals; Cadmium; Cadmium Chloride; Cells, Cultured; Chloral Hydrate; Chlorides; Chromosome Aberrations; Colchicine; Diazepam; Econazole; Europe; European Union; Hydroquinones; Male; Mice; Micronucleus Tests; Mitotic Index; Mutagenicity Tests; Mutagens; Ploidies; Pyrimethamine; Spermatocytes; Thiabendazole; Thimerosal; Vinblastine

1993
The detection and assessment of the aneugenic potential of environmental chemicals: the European Community Aneuploidy Project.
    Mutation research, 1993, Volume: 287, Issue:1

    Topics: Aneuploidy; Animals; Aspergillus; Cadmium; Cadmium Chloride; Cell Cycle; Cells, Cultured; Chloral Hydrate; Chlorides; Colchicine; Diazepam; Econazole; Environmental Pollutants; Europe; European Union; Hydroquinones; Mammals; Mutagenicity Tests; Mutagens; Pyrimethamine; Salmonella typhimurium; Thiabendazole; Thimerosal; Vinblastine

1993

Other Studies

17 other study(ies) available for pyrimethamine and thiabendazole

ArticleYear
Conformer- and alignment-independent model for predicting structurally diverse competitive CYP2C9 inhibitors.
    Journal of medicinal chemistry, 2004, Feb-12, Volume: 47, Issue:4

    Topics: Amino Acids; Aryl Hydrocarbon Hydroxylases; Binding Sites; Cytochrome P-450 CYP2C9; Enzyme Inhibitors; Models, Molecular; Molecular Conformation; Molecular Structure; Quantitative Structure-Activity Relationship

2004
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
QSAR-based solubility model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2010, Oct-01, Volume: 18, Issue:19

    Topics: Databases, Factual; Models, Molecular; Pharmaceutical Preparations; Quantitative Structure-Activity Relationship; Solubility; Water

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
In vitro studies with nine known or suspected spindle poisons: results in tests for chromosome malsegregation in Aspergillus nidulans.
    Mutagenesis, 1991, Volume: 6, Issue:2

    Topics: Aneuploidy; Aspergillus nidulans; Cadmium; Cadmium Chloride; Chloral Hydrate; Chromosomes, Fungal; Colchicine; Crossing Over, Genetic; Diazepam; Econazole; Hydroquinones; Mitosis; Pyrimethamine; Spindle Apparatus; Thiabendazole; Thimerosal

1991
[Tropical and parasitic diseases].
    La Revue du praticien, 1974, Nov-11, Volume: 24, Issue:51

    Topics: Acute Kidney Injury; Amebiasis; Antimalarials; Cholera; Drug Resistance, Microbial; Encephalitis; Glomerulonephritis; Helminthiasis; Hepatitis B Antigens; Humans; Leprosy; Malaria; Neurologic Manifestations; Parasitic Diseases; Pyrimethamine; Rifampin; Sulfonamides; Thiabendazole; Tropical Medicine; Trypanosomiasis, African

1974
An overview of the results of testing of known or suspected aneugens using mammalian cells in vitro.
    Mutation research, 1993, Volume: 287, Issue:1

    Topics: Aneuploidy; Animals; Cadmium; Cadmium Chloride; Cell Division; Cell Line; Cells, Cultured; Chloral Hydrate; Chlorides; Chromosome Aberrations; Colchicine; Cricetinae; Cricetulus; Diazepam; Econazole; Fibroblasts; Humans; Hydroquinones; Lymphocytes; Micronucleus Tests; Mitosis; Mutagenicity Tests; Mutagens; Pyrimethamine; Thiabendazole; Thimerosal; Vinblastine

1993
In vivo studies on chemically induced aneuploidy in mouse somatic and germinal cells.
    Mutation research, 1993, Volume: 287, Issue:1

    Topics: Aneuploidy; Animals; Bone Marrow; Cadmium; Cadmium Chloride; Chloral Hydrate; Chlorides; Colchicine; Diazepam; Econazole; Hydroquinones; Male; Mice; Mice, Inbred Strains; Micronucleus Tests; Mutagenicity Tests; Mutagens; Ploidies; Pyrimethamine; Spermatocytes; Testis; Thiabendazole; Thimerosal

1993
Effects of potential aneuploidy inducing agents on microtubule assembly in vitro.
    Mutation research, 1993, Volume: 287, Issue:1

    Topics: Aneuploidy; Animals; Brain; Cadmium; Cadmium Chloride; Cattle; Chloral Hydrate; Chlorides; Colchicine; Diazepam; Econazole; Hydroquinones; Microtubule Proteins; Microtubules; Mutagens; Pyrimethamine; Thiabendazole; Thimerosal; Vinblastine

1993
An evaluation of the use of in vitro tubulin polymerisation, fungal and wheat assays to detect the activity of potential chemical aneugens.
    Mutation research, 1993, Volume: 287, Issue:1

    Topics: Aneuploidy; Animals; Aspergillus nidulans; Cadmium; Cadmium Chloride; Chloral Hydrate; Chlorides; Colchicine; Diazepam; Econazole; Fungi; Hydroquinones; Mammals; Microtubules; Mutagenicity Tests; Mutagens; Pyrimethamine; Saccharomyces cerevisiae; Thiabendazole; Thimerosal; Triticum; Tubulin; Vinblastine

1993
A comparison of two in vitro mammalian cell cytogenetic assays for the detection of mitotic aneuploidy using 10 known or suspected aneugens.
    Mutation research, 1993, Volume: 287, Issue:1

    Topics: Aneuploidy; Animals; Cadmium; Cadmium Chloride; Cell Division; Cell Line; Centromere; Chloral Hydrate; Chlorides; Colchicine; Cricetinae; Cricetulus; Diazepam; Econazole; Hydroquinones; Karyotyping; Mutagenicity Tests; Mutagens; Pyrimethamine; Thiabendazole; Thimerosal; Vinblastine

1993
Induction of mitotic aneuploidy using Chinese hamster primary embryonic cells. Test results of 10 chemicals.
    Mutation research, 1993, Volume: 287, Issue:1

    Topics: Aneuploidy; Animals; Cadmium; Cadmium Chloride; Cells, Cultured; Chloral Hydrate; Chlorides; Colchicine; Cricetinae; Cricetulus; Diazepam; Dose-Response Relationship, Drug; Econazole; Embryo, Mammalian; Female; Hydroquinones; Male; Mitosis; Mutagenicity Tests; Mutagens; Pyrimethamine; Thiabendazole; Thimerosal; Vincristine

1993
C-mitosis and numerical chromosome aberration analyses in human lymphocytes: 10 known or suspected spindle poisons.
    Mutation research, 1993, Volume: 287, Issue:1

    Topics: Cadmium; Cadmium Chloride; Cells, Cultured; Chloral Hydrate; Chlorides; Chromosome Aberrations; Colchicine; Diazepam; Diploidy; Dose-Response Relationship, Drug; Econazole; Humans; Hydroquinones; Lymphocytes; Mitosis; Mutagenicity Tests; Mutagens; Ploidies; Polyploidy; Pyrimethamine; Spindle Apparatus; Thiabendazole; Thimerosal; Vinblastine

1993
The cytochalasin-B micronucleus/kinetochore assay in vitro: studies with 10 suspected aneugens.
    Mutation research, 1993, Volume: 287, Issue:1

    Topics: Aneuploidy; Animals; Cadmium; Cadmium Chloride; Cell Division; Cell Line; Centromere; Chloral Hydrate; Chlorides; Colchicine; Cricetinae; Cricetulus; Cytochalasin B; Diazepam; Dose-Response Relationship, Drug; Econazole; Humans; Hydroquinones; Micronucleus Tests; Mitomycin; Mutagens; Pyrimethamine; Thiabendazole; Thimerosal; Vinblastine

1993
Detection of aneuploidy-inducing carcinogens in the Syrian hamster embryo (SHE) cell transformation assay.
    Mutation research, 1995, Volume: 343, Issue:1

    Topics: Aneuploidy; Animals; Asbestos; Benomyl; Cadmium; Cadmium Chloride; Carcinogenicity Tests; Carcinogens; Cells, Cultured; Chloral Hydrate; Chlorides; Cricetinae; Demecolcine; Diazepam; Diethylstilbestrol; Econazole; Embryo, Mammalian; Evaluation Studies as Topic; Griseofulvin; Mesocricetus; Pyrimethamine; Thiabendazole

1995
Micronucleus test and metaphase analyses in mice exposed to known and suspected spindle poisons.
    Mutagenesis, 1994, Volume: 9, Issue:6

    Topics: Animals; Bone Marrow Cells; Cadmium; Cadmium Chloride; Cells, Cultured; Chloral Hydrate; Chlorides; Chromosome Aberrations; Colchicine; Diazepam; Econazole; Hydroquinones; Male; Metaphase; Mice; Micronucleus Tests; Pyrimethamine; Spindle Apparatus; Thiabendazole; Thimerosal; Vinblastine

1994