Page last updated: 2024-08-16

pyrimethamine and emetine

pyrimethamine has been researched along with emetine in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19904 (36.36)18.7374
1990's0 (0.00)18.2507
2000's2 (18.18)29.6817
2010's5 (45.45)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Adrián, F; Anderson, P; Brinker, A; Caldwell, JS; Chatterjee, A; Gray, NS; Henson, K; Janes, J; Kato, N; Kuhen, K; Matzen, JT; McNamara, C; Nagle, A; Nam, TG; Plouffe, D; Schultz, PG; Trager, R; Winzeler, EA; Yan, SF; Zhou, Y1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Barnes, SW; Bonamy, GM; Bopp, SE; Borboa, R; Bright, AT; Chatterjee, A; Che, J; Cohen, S; Dharia, NV; Diagana, TT; Fidock, DA; Froissard, P; Gagaring, K; Gettayacamin, M; Glynne, RJ; Gordon, P; Groessl, T; Kato, N; Kuhen, KL; Lee, MC; Mazier, D; McNamara, CW; Meister, S; Nagle, A; Nam, TG; Plouffe, DM; Richmond, W; Roland, J; Rottmann, M; Sattabongkot, J; Schultz, PG; Tuntland, T; Walker, JR; Winzeler, EA; Wu, T; Zhou, B; Zhou, Y1
Breytenbach, WJ; de Kock, C; N'Da, DD; Pretorius, SI; Smith, PJ1
Cloete, TT; de Kock, C; N'Da, DD; Smith, PJ1
Barnard, L; Birkholtz, LM; Botha, M; Brunschwig, C; Burrows, JN; Chibale, K; Churchyard, A; Coetzer, TL; Denti, P; Egan, TJ; Laing, L; Lauterbach, S; Machado, M; Ndubi, F; Njogu, PM; Njoroge, M; Nondaba, S; Okombo, J; Prudêncio, M; Reader, J; Singh, K; Wiesner, L; Wilkinson, C; Wittlin, S; Yeates, C1
Fernex, M1
Brossi, A1
Baden, HP; Clendenning, W; Cornell, RC; Deneau, DD; Eaglstein, WH; Golub, A; King, L; Kulp, KR; Maibach, H; McCullough, JL; Stoughton, RB; Taylor, JS; Weinstein, GD; Zackheim, H1
Nakajima, Y1
NEAL, RA1

Reviews

1 review(s) available for pyrimethamine and emetine

ArticleYear
[Antiprotozoal drugs].
    Nihon rinsho. Japanese journal of clinical medicine, 2003, Volume: 61 Suppl 2

    Topics: Animals; Antiprotozoal Agents; Drug Combinations; Emetine; Humans; Mefloquine; Metronidazole; Phenanthrenes; Primaquine; Protozoan Infections; Pyrimethamine; Quinine; Sulfadoxine; Tinidazole

2003

Trials

1 trial(s) available for pyrimethamine and emetine

ArticleYear
A clinical screening program for topical chemotherapeutic drugs in psoriasis.
    Archives of dermatology, 1981, Volume: 117, Issue:7

    Topics: Adult; Animals; Clinical Trials as Topic; Cycloheximide; Dermatologic Agents; Double-Blind Method; Drug Evaluation, Preclinical; Emetine; Fluorouracil; Humans; Mitoguazone; Psoriasis; Pyrimethamine; Rabbits; Skin; Thiotepa

1981

Other Studies

9 other study(ies) available for pyrimethamine and emetine

ArticleYear
In silico activity profiling reveals the mechanism of action of antimalarials discovered in a high-throughput screen.
    Proceedings of the National Academy of Sciences of the United States of America, 2008, Jul-01, Volume: 105, Issue:26

    Topics: Animals; Antimalarials; Cluster Analysis; Computational Biology; Drug Evaluation, Preclinical; Drug Resistance; Folic Acid Antagonists; Malaria; Models, Molecular; Parasites; Plasmodium falciparum; Reproducibility of Results; Structure-Activity Relationship; Tetrahydrofolate Dehydrogenase

2008
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Imaging of Plasmodium liver stages to drive next-generation antimalarial drug discovery.
    Science (New York, N.Y.), 2011, Dec-09, Volume: 334, Issue:6061

    Topics: Animals; Antimalarials; Cell Line, Tumor; Drug Discovery; Drug Evaluation, Preclinical; Drug Resistance; Erythrocytes; Humans; Imidazoles; Liver; Malaria; Mice; Mice, Inbred BALB C; Molecular Structure; Piperazines; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Plasmodium yoelii; Polymorphism, Single Nucleotide; Protozoan Proteins; Random Allocation; Small Molecule Libraries; Sporozoites

2011
Synthesis, characterization and antimalarial activity of quinoline-pyrimidine hybrids.
    Bioorganic & medicinal chemistry, 2013, Jan-01, Volume: 21, Issue:1

    Topics: Animals; Antimalarials; Cell Survival; CHO Cells; Cricetinae; Inhibitory Concentration 50; Malaria, Falciparum; Plasmodium falciparum; Pyrimidines; Quinolines

2013
Synthesis, in vitro antiplasmodial activity and cytotoxicity of a series of artemisinin-triazine hybrids and hybrid-dimers.
    European journal of medicinal chemistry, 2014, Apr-09, Volume: 76

    Topics: Antimalarials; Artemisinins; Dimerization; Inhibitory Concentration 50; Magnetic Resonance Spectroscopy; Mass Spectrometry; Plasmodium falciparum; Spectrophotometry, Infrared; Triazines

2014
Antimalarial Pyrido[1,2-a]benzimidazoles: Lead Optimization, Parasite Life Cycle Stage Profile, Mechanistic Evaluation, Killing Kinetics, and in Vivo Oral Efficacy in a Mouse Model.
    Journal of medicinal chemistry, 2017, 02-23, Volume: 60, Issue:4

    Topics: Animals; Antimalarials; Benzimidazoles; Life Cycle Stages; Malaria; Male; Mice; Plasmodium berghei; Structure-Activity Relationship

2017
[Prevention and therapy of malaria and amebiasis].
    Schweizerische medizinische Wochenschrift, 1977, May-07, Volume: 107, Issue:18

    Topics: Acetamides; Amebiasis; Chloroquine; Drug Combinations; Drug Resistance, Microbial; Emetine; Humans; Malaria; Nitroimidazoles; Protective Devices; Pyrimethamine; Sulfadoxine; Tetracycline

1977
Some recent results on the chemotherapy of amebiasis, coccidiosis, and malaria.
    Pure and applied chemistry. Chimie pure et appliquee, 1969, Volume: 19, Issue:1

    Topics: Amebiasis; Animals; Animals, Domestic; Anti-Bacterial Agents; Coccidiosis; Emetine; Malaria; Pyrimethamine; Quinine; Sulfadimethoxine

1969
CHEMOTHERAPY OF CUTANEOUS LEISHMANIASIS: LEISHMANIA TROPICA INFECTIONS IN MICE.
    Annals of tropical medicine and parasitology, 1964, Volume: 58

    Topics: Amidines; Animals; Antimony; Antiprotozoal Agents; Chloroquine; Chlortetracycline; Dapsone; Deoxyribonuclease I; Emetine; Hyaluronoglucosaminidase; Hydrastis; Leishmania tropica; Leishmaniasis; Leishmaniasis, Cutaneous; Leishmaniasis, Mucocutaneous; Mice; Pathology; Pharmacology; Primaquine; Pyrimethamine; Quinacrine; Research; Streptodornase and Streptokinase; Streptokinase; Sulfonamides; Surface-Active Agents; Toxicology

1964