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pyrimethamine and chloroquine diphosphate

pyrimethamine has been researched along with chloroquine diphosphate in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19905 (38.46)18.7374
1990's1 (7.69)18.2507
2000's2 (15.38)29.6817
2010's5 (38.46)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bertaux, L; Bogreau, H; Bouchiba, H; Garnotel, E; Kraemer, P; Parzy, D; Pradines, B; Rogier, C; Savini, H; Simon, F1
Che, P; Cong, X; Huang, H; Huang, J; Jiang, H; Li, H; Li, X; Liu, X; Lu, W; Ma, H; Ma, R; Shen, X; Zhang, Y; Zhu, J1
Cloete, TT; de Kock, C; N'Da, DD; Smith, PJ1
Bekhit, AA; Bekhit, AEA; El-Seidy, AM; Fahmy, SM; Ghareeb, D; Hassan, AMM; Ibrahim, TM; Nasralla, SN; Saudi, MN1
Beale, GH; Chutmongkonkul, M; Thaithong, S1
Davidson, DE; Gwadz, RW; Koontz, LC; Miller, LH1
Howells, RE; Judge, BM1
Belda Mira, A; Díaz Sánchez, F; Michavila Gómez, J; Rovira Daudí, E1
APPEL, B; BALER, GR; COLLINS, SF; SCHIFF, BL; TYE, MJ1
SRIVASTAVA, JR1
El-Qudaby, HM; Khalil, SM; Zayed, MA1
Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ1
Ekins, S; Williams, AJ; Xu, JJ1

Other Studies

13 other study(ies) available for pyrimethamine and chloroquine diphosphate

ArticleYear
First case of emergence of atovaquone-proguanil resistance in Plasmodium falciparum during treatment in a traveler in Comoros.
    Antimicrobial agents and chemotherapy, 2008, Volume: 52, Issue:6

    Topics: Animals; Antimalarials; Atovaquone; Comoros; Drug Resistance; France; Genotype; Humans; Malaria, Falciparum; Male; Parasitic Sensitivity Tests; Plasmodium falciparum; Proguanil; Travel; Treatment Failure

2008
Design and synthesis of small molecular dual inhibitor of falcipain-2 and dihydrofolate reductase as antimalarial agent.
    Bioorganic & medicinal chemistry letters, 2012, Jan-15, Volume: 22, Issue:2

    Topics: Animals; Antimalarials; Cysteine Endopeptidases; Dose-Response Relationship, Drug; Enzyme Inhibitors; Malaria; Mice; Mice, Inbred Strains; Models, Molecular; Molecular Weight; Plasmodium berghei; Structure-Activity Relationship; Tetrahydrofolate Dehydrogenase

2012
Synthesis, in vitro antiplasmodial activity and cytotoxicity of a series of artemisinin-triazine hybrids and hybrid-dimers.
    European journal of medicinal chemistry, 2014, Apr-09, Volume: 76

    Topics: Antimalarials; Artemisinins; Dimerization; Inhibitory Concentration 50; Magnetic Resonance Spectroscopy; Mass Spectrometry; Plasmodium falciparum; Spectrophotometry, Infrared; Triazines

2014
Synthesis, in silico experiments and biological evaluation of 1,3,4-trisubstituted pyrazole derivatives as antimalarial agents.
    European journal of medicinal chemistry, 2019, Feb-01, Volume: 163

    Topics: Animals; Anti-Inflammatory Agents; Antimalarials; Computer Simulation; Hemolysis; Humans; Inhibitory Concentration 50; Molecular Docking Simulation; Plasmodium berghei; Plasmodium falciparum; Pyrazoles; Structure-Activity Relationship

2019
Susceptibility of Plasmodium falciparum to five drugs: an in vitro study of isolates mainly from Thailand.
    Transactions of the Royal Society of Tropical Medicine and Hygiene, 1983, Volume: 77, Issue:2

    Topics: Amodiaquine; Antimalarials; Chloroquine; Drug Resistance, Microbial; Humans; In Vitro Techniques; Mefloquine; Plasmodium falciparum; Pyrimethamine; Quinine; Quinolines; Thailand

1983
Plasmodium gallinaceum: avian screen for drugs with radical curative properties.
    Experimental parasitology, 1983, Volume: 55, Issue:2

    Topics: Animals; Antimalarials; Chickens; Chloroquine; Drug Evaluation, Preclinical; Malaria, Avian; Plasmodium; Primaquine; Pyrimethamine

1983
Sustained-release implants in the chemotherapy of experimental rodent malaria I. A comparison of the effects of some antimalarials in polydimethylsiloxane matrices.
    Annals of tropical medicine and parasitology, 1981, Volume: 75, Issue:5

    Topics: Animals; Antimalarials; Chloroquine; Dimethylpolysiloxanes; Drug Implants; Malaria; Male; Mefloquine; Mice; Mice, Inbred Strains; Naphthoquinones; Piperidines; Plasmodium berghei; Primaquine; Proguanil; Pyrimethamine; Quinolines; Silicone Elastomers; Sulfadiazine; Triazines

1981
[Porphyria cutanea tarda and human immunodeficiency virus infection. Apropos of 2 further cases].
    Revista clinica espanola, 1994, Volume: 194, Issue:7

    Topics: Adult; Anti-Inflammatory Agents, Non-Steroidal; Chloroquine; Drug Therapy, Combination; HIV Infections; Humans; Male; Porphyria Cutanea Tarda; Pyrimethamine; Substance-Related Disorders; Zidovudine

1994
Chronic discoid lupus erythematosus: treatment with daraprim and chloroquine diphosphate (aralen).
    The New England journal of medicine, 1954, Jul-08, Volume: 251, Issue:2

    Topics: Antimalarials; Chloroquine; Humans; Lupus Erythematosus, Discoid; Lupus Erythematosus, Systemic; Pyrimethamine

1954
Therapeutic trials with pyrimethamine (daraprim), resochin, amodiaquin (camoquin) and quinine.
    Indian journal of malariology, 1953, Volume: 7, Issue:4

    Topics: Amodiaquine; Antimalarials; Chloroquine; Humans; Malaria; Pyrimethamine; Quinine

1953
Spectrophotometric study of the reaction mechanism between DDQ Pi- and iodine sigma-acceptors and chloroquine and pyrimethamine drugs and their determination in pure and in dosage forms.
    Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy, 2005, Volume: 62, Issue:1-3

    Topics: Antimalarials; Chloroquine; Dosage Forms; Iodine; Kinetics; Pyrimethamine; Spectrophotometry; Thermodynamics

2005
Developing structure-activity relationships for the prediction of hepatotoxicity.
    Chemical research in toxicology, 2010, Jul-19, Volume: 23, Issue:7

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes

2010
A predictive ligand-based Bayesian model for human drug-induced liver injury.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands

2010