pyrilamine has been researched along with thiourea in 71 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 51 (71.83) | 18.7374 |
1990's | 11 (15.49) | 18.2507 |
2000's | 8 (11.27) | 29.6817 |
2010's | 1 (1.41) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bunce, KT; Parsons, ME | 1 |
Becker, M; Malchow, H; Painz, B; Rack, M; Ruoff, HJ; Sewing, KF | 1 |
Allouche, G; Foussard, C; Parrot, JL; Ruff, F; Santais, MC | 1 |
Cho, CH; Ogle, CW | 1 |
Bertaccini, G; Coruzzi, G; Musso, E | 1 |
Bertaccini, G; Impicciatore, M; Morini, G | 1 |
Barbezat, GO; Bowey, FS; Hickman, R; Kaplan, ER | 1 |
Barkla, DH; Tutton, PJ | 1 |
Carter, DC; Grossman, MI; Impicciatore, M | 1 |
Giles, RW; Heise, G; Wilcken, DE | 1 |
Czerwińska, U; Kazimierczak, W; Maśliński, C; Wyczólkowska, J | 1 |
Adamas, B; Kazimierczak, W; Lewa, A; Maśliński, C; Peret, M | 1 |
Brandon, JM; Wallis, RM | 1 |
Johnston, BM; Owen, DA | 1 |
Goadby, P; Little, MA | 1 |
Ruoff, HJ; Sewing, KF | 1 |
Meek, ME; Newcombe, RG; Rees, WD; Rhodes, J; Wheeler, MH | 1 |
Nowak, JZ; Sek, B | 1 |
Benedito, S; Nielsen, PJ; Nyborg, NC; Prieto, D | 1 |
Dolata, J; Lindberg, S; Mercke, U | 1 |
Almeida, L; Figueiredo, A; Gonçalo, M; Poiares-Baptista, A; Ribeiro, CA; Teixeira, F | 1 |
Cooke, HJ; Wang, YZ | 1 |
Młynarska, MS | 1 |
Matsuki, T; Ohhashi, T | 1 |
Bugajski, J; Gadek-Michalska, A | 1 |
Girard, A; Marche, P | 1 |
Hutchison, VH; Spriestersbach, KK | 1 |
Knigge, U; Matzen, S; Warberg, J | 1 |
Baker, CH; Davis, DL; Lindsey, BG; Sutton, ET | 1 |
Akahori, H; Kamei, C; Kitazumi, K; Tasaka, K | 1 |
Ledgard, SE; Nieves, AL; Woodward, DF | 1 |
Barker, LA; Winbery, SL | 1 |
Donaldson, J; Hill, SJ | 1 |
Kim, LE; Oudart, N; Sercombe, R; Teste, JF | 1 |
Bugajski, J; Gadek, A | 1 |
Jouvet, M; Lin, JS; Sakai, K | 1 |
Fromm, D; Furukawa, T; Olender, EJ; Woods, DJ | 1 |
Kume, S; Ohashi, T; Ozaki, Y | 1 |
Gristwood, RW; Lincoln, JC; Owen, DA | 1 |
Daniel, D; Owen, DA; Poy, E; Woodward, DF | 1 |
Oriowo, MA | 1 |
Heldsinger, AA; Skoglund, ML; Vinik, AI | 1 |
Donoso, AO; Zárate, MB | 1 |
Guldvog, I; Linnestad, P; Schrumpf, E | 1 |
Nemeth, PR; Ort, CA; Wood, JD | 1 |
Bugajski, J; Janusz, Z | 1 |
Owen, DA; Pipkin, MA; Woodward, DF | 1 |
Bottomley, KM; Lewis, S; Rising, TJ; Steward, A | 1 |
Jespersen, LT; Mikkelsen, E; Sakr, AM | 1 |
Cooke, HJ; Nemeth, PR; Wood, JD | 1 |
Bordi, F; Chiavarini, M; Impicciatore, M; Morini, G; Plazzi, PV; Vitali, F | 1 |
Binderup, L | 1 |
Chand, N; DeRoth, L | 1 |
Del Soldato, P | 1 |
Alvarez, EO | 1 |
Harvey, CA; Owen, DA; Shaw, KD | 1 |
Di Donato, M; Mantovani, P; Santicioli, P | 1 |
Duchemin, AM; Quach, TT; Rose, C; Schwartz, JC | 1 |
Imaizumi, M; Miyazaki, S; Onodera, K; Timmerman, H | 1 |
Hemedah, M; Mitchelson, F | 1 |
Allescher, HD; Hahn, A; Huber, A; Neumayer, N | 1 |
Jørgensen, H; Kjaer, A; Knigge, U; Warberg, J; Willems, E | 1 |
de Wildt, DJ; Hendriksen, CF; van de Kuil, A; van den Hout, JW; Vleeming, W | 1 |
Anichtchik, OV; Panula, P; Peitsaro, N | 1 |
Chen, Z; Hu, WW; Huang, YW; Wei, EQ; Yanai, K; Zhang, LS | 1 |
Djahanguiri, B; Khalilzadeh, A; Zarrindast, MR | 1 |
Eckman, JR; Wagner, MC; Wick, TM | 1 |
Holopainen, IE; Kukko-Lukjanov, TK; Michelsen, KA; Panula, P; Soini, S; Taira, T | 1 |
Chen, Z; Hu, DN; Liu, CQ; Liu, FX; Luo, JH | 1 |
Kamei, C; Masuoka, T | 1 |
Khodarahmi, P; Oryan, S; Rezayof, A; Zarrindast, MR | 1 |
1 trial(s) available for pyrilamine and thiourea
Article | Year |
---|---|
Human gastric mucosal adenylate cyclase: activation by histamine-H2-receptor stimulation and inhibition by cimetidine in vitro and in peptic ulcer patients.
Topics: Adenylyl Cyclases; Cimetidine; Clinical Trials as Topic; Enzyme Activation; Female; Gastric Mucosa; Guanidines; Histamine; Humans; Male; Middle Aged; Peptic Ulcer; Phenethylamines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H2; Thiourea | 1979 |
70 other study(ies) available for pyrilamine and thiourea
Article | Year |
---|---|
Investigation of the role of histamine H1-receptors in the control of gastric acid secretion in the rat.
Topics: Animals; Dose-Response Relationship, Drug; Ethylamines; Female; Gastric Juice; Histamine; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1978 |
Role of H2-receptor antagonists in the feedback of histamine [proceedings].
Topics: Amine Oxidase (Copper-Containing); Anaphylaxis; Animals; Burimamide; Cyclic AMP; Feedback; Guinea Pigs; Histamine; Lung; Metiamide; Pyridines; Pyrilamine; Thiourea | 1977 |
Histamine H1- and H2-receptor-mediated gastric microcirculatory effects in the aetiology of stress ulceration in the rat stomach.
Topics: Aminopyridines; Animals; Dose-Response Relationship, Drug; Gastric Mucosa; Humans; Male; Mast Cells; Metiamide; Microcirculation; Pyrilamine; Rats; Receptors, Histamine; Stomach Ulcer; Stress, Psychological; Thiourea | 1978 |
[Histamine receptors in the guinea pig papillary muscle].
Topics: Animals; Cimetidine; Epinephrine; Female; Guinea Pigs; Histamine; Male; Papillary Muscles; Pyrilamine; Receptors, Histamine; Thiazoles; Thiourea | 1977 |
The effects of stimulants and inhibitors of histamine receptors on acid secretion from guinea pig gastric fundus.
Topics: Animals; Cimetidine; Female; Gastric Mucosa; Guinea Pigs; Histamine; In Vitro Techniques; Male; Methylhistamines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea; Time Factors | 1978 |
Effect of histamine H1- and H2-receptor blockade on canine gastric acid secretion.
Topics: Animals; Dogs; Gastric Juice; Metiamide; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Secretory Rate; Stomach; Thiourea | 1978 |
Stimulation of cell proliferation by histamine H2 receptors in dimethylhdrazine-induced adenocarcinomata.
Topics: Adenocarcinoma; Animals; Cell Division; Cimetidine; Colon; Colonic Neoplasms; Dimethylhydrazines; Histamine; Intestinal Mucosa; Male; Metiamide; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H2; Stimulation, Chemical; Thiourea | 1978 |
Effect of dimaprit on gastric acid secretion in conscious cats.
Topics: Animals; Cats; Cimetidine; Gastric Juice; Histamine; Methylhistamines; Pentagastrin; Pyrilamine; Receptors, Histamine H2; Thiourea; Time Factors | 1978 |
Histamine receptors in the coronary circulation of the dog. Effects of mepyramine and metiamide on responses to histamine infusions.
Topics: Animals; Coronary Circulation; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Histamine; Injections, Intra-Arterial; Metiamide; Myocardial Contraction; Pyridines; Pyrilamine; Receptors, Histamine; Thiourea; Time Factors | 1977 |
The pharmacological inhibition of the heterologous PCA reaction by histamine antagonists and chloropromazine [proceedings].
Topics: Animals; Chlorpromazine; Immune Sera; Immunoglobulin E; Metiamide; Mice; Passive Cutaneous Anaphylaxis; Pyridines; Pyrilamine; Rats; Thiourea | 1977 |
The participation of H1 and H2 histamine receptors in vascular skin permeability induced by some imidazoles [proceedings].
Topics: Animals; Burimamide; Guinea Pigs; Imidazoles; Male; Metiamide; Permeability; Pyridines; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Skin; Skin Physiological Phenomena; Thiourea | 1977 |
Effect of mepyramine, a histamine H1-, and burimamide, a histamine H2-receptor antagonist, on ovum implantation in the rat.
Topics: Animals; Blastocyst; Burimamide; Embryo Implantation; Female; Pyridines; Pyrilamine; Rats; Thiourea | 1977 |
Histamine, histamine antagonists and regional blood flow.
Topics: Animals; Blood Pressure; Cats; Drug Interactions; Female; Hemodynamics; Histamine; Male; Metiamide; Pyridines; Pyrilamine; Regional Blood Flow; Thiourea; Vascular Resistance | 1977 |
The action of metiamide in anaphylaxis in vivo in the guinea-pig [proceedings].
Topics: Anaphylaxis; Animals; Guinea Pigs; Lung Volume Measurements; Metiamide; Pyrilamine; Thiourea | 1976 |
Adenylate cyclase of the dog gastric mucosa: stimulation by histamine and inhibition by metiamide.
Topics: Adenylyl Cyclases; Animals; Dogs; Female; Gastric Mucosa; Histamine; In Vitro Techniques; Metiamide; Pyrilamine; Thiourea | 1976 |
Proceedings: Role of histamine receptors in the pathophysiology of gastric mucosal damage.
Topics: Animals; Dogs; Gastric Mucosa; Metiamide; Pyridines; Pyrilamine; Receptors, Drug; Sodium; Taurocholic Acid; Thiourea | 1976 |
Cyclic AMP generating systems in vertebrate retina: effects of histamine and an established retinal modulator, dopamine.
Topics: Adenylyl Cyclases; Animals; Cerebral Cortex; Chickens; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dopamine; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Retina; Thiazoles; Thiourea | 1991 |
Histamine induces endothelium-dependent relaxation of bovine retinal arteries.
Topics: Acetylcholine; Animals; Cattle; Cimetidine; Dimaprit; Endothelium, Vascular; Histamine; Muscle Relaxation; Pyridines; Pyrilamine; Receptors, Histamine; Retinal Artery; Tachyphylaxis; Thiourea | 1991 |
Histamine stimulation of mucociliary activity in the rabbit maxillary sinus.
Topics: Animals; Atropine; Cilia; Cimetidine; Dimaprit; Female; Histamine; Histamine H2 Antagonists; Male; Maxillary Sinus; Mucociliary Clearance; Pyrilamine; Rabbits; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Muscarinic; Thiourea | 1990 |
Mechanism of action of doxepin in the treatment of chronic urticaria.
Topics: Adult; Aged; Animals; Atropine; Carbachol; Chronic Disease; Dimaprit; Doxepin; Female; Gastric Juice; Guinea Pigs; Heart; Histamine; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Pylorus; Pyrilamine; Rats; Thiourea; Urticaria | 1990 |
H2 receptors mediate cyclical chloride secretion in guinea pig distal colon.
Topics: Animals; Bumetanide; Chlorides; Cimetidine; Colon; Dimaprit; Guinea Pigs; Histamine; In Vitro Techniques; Intestinal Mucosa; Kinetics; Male; Muscle, Smooth; Pyrilamine; Receptors, Histamine H2; Tetrodotoxin; Thiourea | 1990 |
Antagonistic effect of naloxone on the hypertensive response of intraventricularly administered histamine.
Topics: Animals; Blood Pressure; Cimetidine; Dimaprit; Hemodynamics; Histamine; In Vitro Techniques; Injections, Intraventricular; Male; Naloxone; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Thiourea | 1990 |
Endothelium and mechanical responses of isolated monkey pulmonary veins to histamine.
Topics: Animals; Dimaprit; Endothelium, Vascular; Famotidine; Hemoglobins; Histamine; In Vitro Techniques; Macaca; Methylene Blue; Pulmonary Veins; Pyridines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Vasoconstriction; Vasodilation | 1990 |
Antagonistic action of naloxone on central histamine receptors-stimulated corticosterone secretion in rats under stress.
Topics: Animals; Cimetidine; Corticosterone; Dimaprit; Histamine; Male; Methylhistamines; Naloxone; Pituitary-Adrenal System; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Restraint, Physical; Stress, Physiological; Thiourea | 1989 |
Phosphoinositides and cicletanine.
Topics: Angiotensin II; Animals; Antihypertensive Agents; Aorta, Thoracic; Cells, Cultured; Dimaprit; Diuretics; Guinea Pigs; Histamine; Male; Muscle, Smooth, Vascular; Phenylephrine; Phosphatidylinositols; Pyridines; Pyrilamine; Thiourea | 1988 |
Histamine and histamine receptors: behavioral thermoregulation in the salamander Necturus maculosus.
Topics: Animals; Body Temperature Regulation; Cimetidine; Dimaprit; Histamine; Histidine; Necturus; Pyridines; Pyrilamine; Receptors, Histamine; Thiourea | 1986 |
Histaminergic stimulation of prolactin secretion mediated via H1- or H2-receptors: dependence on routes of administration.
Topics: Animals; Cimetidine; Dimaprit; Histamine; Histamine H1 Antagonists; Male; Methylhistamines; Pituitary Gland, Anterior; Prolactin; Pyrilamine; Pyrimidinones; Rats; Receptors, Histamine; Thiazoles; Thiourea | 1986 |
Adrenergic and histaminergic neural interactions in dog paws.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Aminopyridines; Animals; Blood Pressure; Blood Volume; Capillaries; Dogs; Electric Stimulation; Hindlimb; Metiamide; Pyrilamine; Reference Values; Regional Blood Flow; Sciatic Nerve; Thiourea; Vascular Resistance | 1988 |
The effects of histamine and some related compounds on conditioned avoidance response in rats.
Topics: Acetylcholine; Animals; Avoidance Learning; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Hypothalamus; Injections, Intraventricular; Kinetics; Male; Methylhistamines; Pyrilamine; Rats; Rats, Inbred Strains; Scopolamine; Thiazoles; Thiourea | 1985 |
Conjunctival immediate hypersensitivity: re-evaluation of histamine involvement in the vasopermeability response.
Topics: Albumins; Animals; Capillary Permeability; Cimetidine; Conjunctiva; Dimaprit; Dose-Response Relationship, Drug; Drug Combinations; Eyelids; Guinea Pigs; Histamine; Histamine Antagonists; Hypersensitivity, Immediate; Imidazoles; Impromidine; Male; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1986 |
Metronidazole and 5-aminosalicylic acid enhance the contractile activity of histaminergic agonists on the guinea-pig isolated ileum.
Topics: Aminosalicylic Acids; Animals; Cimetidine; Computers; Dimaprit; Dose-Response Relationship, Drug; Drug Synergism; Duodenum; Female; Guinea Pigs; Heart; Histamine; Ileum; In Vitro Techniques; Jejunum; Male; Mesalamine; Metronidazole; Muscle Contraction; Myenteric Plexus; Pyrilamine; Receptors, Histamine; Scopolamine; Tetrodotoxin; Thiourea | 1986 |
Selective enhancement of histamine H1-receptor responses in guinea-pig ileal smooth muscle by 1,4-dithiothreitol.
Topics: Acetylcholine; Animals; Dimaprit; Dithionitrobenzoic Acid; Dithiothreitol; Dose-Response Relationship, Drug; Female; Guanidines; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Thiourea | 1986 |
Participation of vascular H1-receptors in histaminergic relaxation of rabbit middle cerebral artery in vitro.
Topics: Animals; Cerebral Arteries; Cimetidine; Dimaprit; Drug Interactions; Histamine; In Vitro Techniques; Methylhistamines; Muscle Relaxation; Muscle, Smooth, Vascular; Phenethylamines; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Thiourea | 1986 |
Hyperlipemic responses induced by centrally administered histamine H1- and H2-receptor agonists in rats.
Topics: Animals; Brain; Cimetidine; Dimaprit; Fatty Acids, Nonesterified; Hyperlipidemias; Imidazoles; Impromidine; Injections, Intraventricular; Male; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Thiourea | 1987 |
Evidence for histaminergic arousal mechanisms in the hypothalamus of cat.
Topics: Animals; Arousal; Cats; Dimaprit; Female; Histamine; Histamine Antagonists; Histidine Decarboxylase; Hypothalamus; Hypothalamus, Posterior; Injections; Injections, Intraperitoneal; Male; Methylhistidines; Pyrilamine; Thiourea | 1988 |
Histamine receptor effects on dissipation of an intracellular proton gradient of isolated gastric mucosal surface cells.
Topics: Animals; Bicarbonates; Chlorides; Cimetidine; Dimaprit; Diphenhydramine; Gastric Acid; Gastric Mucosa; Histamine; Protons; Pyridines; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Sodium; Thiourea | 1987 |
Effects of histamine agonists and antagonists on luminol-dependent chemiluminescence of granulocytes.
Topics: Cimetidine; Dimaprit; Granulocytes; Histamine; Histamine Antagonists; Humans; In Vitro Techniques; Luminescent Measurements; Luminol; Pyridazines; Pyridines; Pyrilamine; Ranitidine; Thiourea | 1984 |
Effects of histamine on human isolated heart muscle: comparison with effects of noradrenaline.
Topics: Cimetidine; Dimaprit; Heart; Histamine; Humans; In Vitro Techniques; Myocardial Contraction; Norepinephrine; Propranolol; Pyrilamine; Receptors, Histamine H2; Thiourea | 1980 |
Evaluation of the role of Histamine H1- and H2-receptors in cutaneous inflammation in the guinea-pig produced by histamine and mast cell degranulation.
Topics: Animals; Cimetidine; Dimaprit; Guinea Pigs; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Inflammation; Male; Mast Cells; Mathematics; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Skin; Thiourea; Vasodilation | 1980 |
An inhibitory effect of histamine on the rat anococcygeus muscle.
Topics: Acetylcholine; Animals; Carbachol; Cimetidine; Dimaprit; Drug Interactions; Guanidines; Histamine; Imidazoles; Impromidine; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Pyrilamine; Rats; Thiourea | 1982 |
Evidence for histamine H1 and H2 receptors in guinea-pig oxyntic cells.
Topics: Animals; Carbonic Anhydrases; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Impromidine; In Vitro Techniques; Methylhistamines; Parietal Cells, Gastric; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1983 |
Release of prolactin and luteinizing hormone by histamine agonists in ovariectomized, steroid-treated rats under ether anesthesia.
Topics: Animals; Castration; Dimaprit; Female; Histamine; Histamine H1 Antagonists; Luteinizing Hormone; Methylhistamines; Metiamide; Pituitary Gland, Anterior; Prolactin; Pyridines; Pyrilamine; Rats; Thiourea | 1983 |
The effect of histamine, H1 and H2 agonists, and H1 and H2 antagonists on postprandial pancreatic polypeptide release in dogs.
Topics: Animals; Cimetidine; Dimaprit; Dogs; Food; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Pancreatic Polypeptide; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Secretory Rate; Thiazoles; Thiourea | 1983 |
Intracellular study of effects of histamine on electrical behaviour of myenteric neurones in guinea-pig small intestine.
Topics: Action Potentials; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine Antagonists; In Vitro Techniques; Intestine, Small; Membrane Potentials; Myenteric Plexus; Neurons; Neurotransmitter Agents; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Serotonin; Thiourea | 1984 |
Central histaminergic stimulation of pituitary--adrenocortical response in the rat.
Topics: Animals; Cimetidine; Corticosterone; Dimaprit; Dose-Response Relationship, Drug; Histamine; Imidazoles; Impromidine; Male; Pituitary-Adrenal System; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1983 |
Studies on cutaneous vascular permeability in the rat: increases caused by histamine and histamine-like agents.
Topics: Animals; Capillary Permeability; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Histamine; Microcirculation; Pyrilamine; Rats; Regional Blood Flow; Skin; Thiourea | 1984 |
A new in vivo method for the measurement of repetitive anaphylactic responses in the guinea-pig.
Topics: Albuterol; Anaphylaxis; Animals; Antibodies; Cromolyn Sodium; Dimaprit; Guinea Pigs; Male; Pyrilamine; Theophylline; Thiourea | 1984 |
Studies on the effect of histamine in isolated human pulmonary arteries and veins.
Topics: Aged; Dimaprit; Female; Histamine; Humans; In Vitro Techniques; Male; Methylhistamines; Middle Aged; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phentolamine; Potassium; Pulmonary Artery; Pulmonary Veins; Pyrilamine; Thiourea | 1984 |
Histamine action on guinea pig ileal mucosa.
Topics: Animals; Bicarbonates; Biological Transport, Active; Chlorides; Dimaprit; Electric Conductivity; Female; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Intestinal Mucosa; Male; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1984 |
[Imidazolic H2-agonists: importance of 2-amino substitution for pharmacological activity].
Topics: Animals; Biological Assay; Cats; Dimaprit; Gastric Acid; Guinea Pigs; Histamine; Methylhistamines; Muscle Relaxation; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Structure-Activity Relationship; Thiourea; Urinary Bladder | 1984 |
Effects of the H2-receptor agonist dimaprit on lymphocyte responsiveness in vitro.
Topics: Animals; Cells, Cultured; Cimetidine; Dimaprit; Ephedrine; Female; Glucosamine; In Vitro Techniques; Lymphocyte Activation; Lymphocytes; Metoprolol; Phagocytosis; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H2; T-Lymphocytes; T-Lymphocytes, Regulatory; Thiourea; Thymidine | 1984 |
Acute systemic anaphylaxis in adult domestic fowl: evidence for the protective role of H2-histaminergic and beta 2-adrenergic receptors.
Topics: Anaphylaxis; Animals; Blood Pressure; Carotid Arteries; Chickens; Chromones; Cimetidine; Dimaprit; Ethers; Heart Rate; Metiamide; Poultry Diseases; Propranolol; Pyrilamine; Receptors, Adrenergic; Receptors, Adrenergic, beta; Receptors, Histamine; Receptors, Histamine H2; Terbutaline; Thiourea | 1980 |
Studies with specific agonists and antagonists of the role of histamine H1- and H2-receptor activation in the pathogenesis of gastric lesions in rats.
Topics: Aminopyridines; Animals; Atropine; Dimaprit; Drug Interactions; Female; Histamine; Pyridines; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Stomach Ulcer; Thiourea | 1984 |
Effects of histamine antagonists injected in the preoptic-anterior hypothalamic area on the prolactin surge induced by estrogen in ovariectomized rats.
Topics: Aminopyridines; Animals; Castration; Circadian Rhythm; Drug Implants; Estrogens; Female; Hypothalamus, Anterior; Metiamide; Preoptic Area; Prolactin; Pyrilamine; Rats; Rats, Inbred Strains; Thiourea | 1984 |
Evidence for both histamine H1- and H2-receptors in the gastric vasculature of the cat.
Topics: Animals; Cats; Celiac Artery; Dimaprit; Gastric Juice; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Regional Blood Flow; Stomach; Thiourea; Time Factors | 1980 |
Further experiments on the pharmacological actions of ergometrine.
Topics: Animals; Cattle; Cimetidine; Coronary Vessels; Dimaprit; Ergonovine; Gastric Acid; Guinea Pigs; Histamine; Muscle Contraction; Pyrilamine; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1981 |
Specific desensitization of histamine H1 receptor-mediated [3H]glycogen hydrolysis in brain slices.
Topics: Adult; Animals; Brain; Cerebral Cortex; Cycloheximide; Dimaprit; Glycogen; Humans; Hydrolysis; In Vitro Techniques; Kinetics; Male; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Thiourea | 1981 |
Effects of clobenpropit (VUF-9153), a histamine H3-receptor antagonist, on learning and memory, and on cholinergic and monoaminergic systems in mice.
Topics: Acetylcholine; Animals; Avoidance Learning; Benzothiazoles; Biogenic Monoamines; Brain; Drug Interactions; Histamine Antagonists; Histamine H2 Antagonists; Imidazoles; Male; Memory; Methylhistamines; Mice; Mice, Inbred ICR; Phenoxypropanolamines; Piperidines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H3; Scopolamine; Thiazoles; Thiourea | 1997 |
Comparison of the effects of histamine and N(alpha)-methylhistamine on neuronal function in the guinea-pig oesophagus and ileum.
Topics: Acetylcholine; Animals; Atropine; Dose-Response Relationship, Drug; Electric Stimulation; Esophagus; Guinea Pigs; Histamine; Histamine Antagonists; Ileum; Imidazoles; In Vitro Techniques; Methylhistamines; Muscle, Skeletal; Muscle, Smooth; Neurons; Neurons, Afferent; Pyrilamine; Receptors, Cholinergic; Receptors, Neurokinin-1; Receptors, Neurokinin-3; Substance P; Tetrodotoxin; Thiourea; Vagus Nerve | 1997 |
Effect of interleukin-1beta on the ascending and descending reflex in rat small intestine.
Topics: Animals; Cyclooxygenase Inhibitors; Electric Stimulation; Histamine Antagonists; Imidazoles; In Vitro Techniques; Indomethacin; Interleukin-1; Interleukin-2; Intestine, Small; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Muscles; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Interleukin-1; Reflex; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiourea; Tumor Necrosis Factor-alpha | 1998 |
Histaminergic and catecholaminergic interactions in the central regulation of vasopressin and oxytocin secretion.
Topics: Animals; Arginine Vasopressin; Blood Pressure; Cerebral Ventricles; Cimetidine; Epinephrine; Histamine; Histamine Agonists; Hypothalamus; Imidazoles; Infusions, Parenteral; Male; Methylhistamines; Norepinephrine; Oxytocin; Pituitary Gland, Posterior; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H2; Thiazoles; Thiourea | 1999 |
Mepyramine but not cimetidine or clobenpropit blocks pertussis toxin-induced histamine sensitization in rats.
Topics: Animals; Blood Gas Analysis; Blood Pressure; Cimetidine; Drug Interactions; Histamine; Histamine Antagonists; Imidazoles; Male; Pertussis Toxin; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine; Thiourea; Virulence Factors, Bordetella | 2000 |
Identification of a histamine H(3)-like receptor in the zebrafish (Danio rerio) brain.
Topics: Animals; Autoradiography; Brain; Cimetidine; Female; Guanosine 5'-O-(3-Thiotriphosphate); Histamine Agonists; Histamine Antagonists; Imidazoles; Kinetics; Male; Methylhistamines; Piperidines; Pyrilamine; Radioligand Assay; Receptors, Histamine H3; Sulfur Radioisotopes; Thiourea; Tritium; Zebrafish | 2000 |
Effects of endogenous histamine on seizure development of pentylenetetrazole-induced kindling in rats.
Topics: Animals; Dose-Response Relationship, Drug; Drug Synergism; Histamine; Histamine Release; Histidine; Imidazoles; Injections, Intraventricular; Kindling, Neurologic; Male; Methylhistidines; Pentylenetetrazole; Piperidines; Pyrilamine; Rats; Rats, Sprague-Dawley; Seizures; Thiourea | 2003 |
Effects of intracerebroventricular administration of ultra low doses of histaminergic drugs on morphine state-dependent memory of passive avoidance in mice.
Topics: Analgesics, Opioid; Animals; Avoidance Learning; Behavior, Animal; Dose-Response Relationship, Drug; Drug Interactions; Histamine; Histamine Agents; Imidazoles; Injections, Intraventricular; Male; Memory; Mice; Morphine; Morphine Dependence; Pyrilamine; Reaction Time; Thiourea | 2006 |
Histamine increases sickle erythrocyte adherence to endothelium.
Topics: Analysis of Variance; Anemia, Sickle Cell; Cell Adhesion; Cells, Cultured; Endothelial Cells; Endothelium, Vascular; Erythrocytes; Famotidine; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Imidazoles; Methylhistamines; P-Selectin; Piperidines; Pyrilamine; Stimulation, Chemical; Thiazoles; Thiourea; Venules | 2006 |
Histaminergic neurons protect the developing hippocampus from kainic acid-induced neuronal damage in an organotypic coculture system.
Topics: Animals; Cell Death; Cells, Cultured; Coculture Techniques; Convulsants; Hippocampus; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Hypothalamus, Anterior; Hypothalamus, Posterior; Imidazoles; Kainic Acid; Methylhistidines; Microscopy, Confocal; Neurons; Neuroprotective Agents; Organ Culture Techniques; Piperidines; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine H1; Receptors, Histamine H3; Thiourea; Triprolidine | 2006 |
Apomorphine-induced turning behavior in 6-hydroxydopamine lesioned rats is increased by histidine and decreased by histidine decarboxylase, histamine H1 and H2 receptor antagonists, and an H3 receptor agonist.
Topics: Animals; Apomorphine; Basal Ganglia; Enzyme Inhibitors; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Histidine Decarboxylase; Imidazoles; Injections, Intraventricular; Male; Methylhistidines; Narcotic Antagonists; Oxidopamine; Piperidines; Pyrilamine; Rats; Rats, Sprague-Dawley; Stereotyped Behavior; Sympatholytics; Synapses; Thiourea | 2008 |
The ameliorating effects of NMDA receptor agonists on histamine H1 antagonist-induced memory and hippocampal theta disruptions are prevented by the H3 receptor agonist in rats.
Topics: Animals; Cycloserine; Excitatory Amino Acid Agonists; Hippocampus; Histamine Agonists; Histamine H1 Antagonists; Imidazoles; Male; Maze Learning; Memory; Memory Disorders; Pyrilamine; Random Allocation; Rats; Receptors, N-Methyl-D-Aspartate; Space Perception; Spermidine; Theta Rhythm; Thiourea | 2009 |
Withdrawal from repeated administration of morphine alters histamine-induced anxiogenic effects produced by intra-ventral hippocampal microinjection.
Topics: Analysis of Variance; Animals; Anxiety; Behavior, Animal; Hippocampus; Histamine; Histamine Antagonists; Imidazoles; Male; Microinjections; Morphine; Motor Activity; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Substance Withdrawal Syndrome; Thiourea | 2010 |