Page last updated: 2024-08-16

pyrilamine and thioperamide

pyrilamine has been researched along with thioperamide in 48 studies

Research

Studies (48)

TimeframeStudies, this research(%)All Research%
pre-19901 (2.08)18.7374
1990's25 (52.08)18.2507
2000's19 (39.58)29.6817
2010's3 (6.25)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Timmerman, H1
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM1
Frymarkiewicz, A; Walczyński, K1
Adem, A; Kieć-Kononowicz, K; Sadek, B; Shafiullah, M; Shehab, S; Subramanian, D; Więcek, M1
Fogel, WA; Karcz, T; Kieć-Kononowicz, K; Leurs, R; McNaught Flores, D; Stasiak, A; Staszewski, M; Walczyński, K1
Clapham, J; Kilpatrick, GJ2
Maeyama, K; Onodera, K; Sakai, N; Watanabe, T; Yanai, K1
Fukui, H; Inagaki, N; Kanamura, A; Kondou, H; Koyama, Y; Wada, H1
Barnes, PJ; Ichinose, M1
Garbarg, M; Gros, C; Schwartz, JC; Tuong, MD1
Kohno, S; Nabe, T; Nakao, S; Ogawa, K; Ohata, K; Yamamura, H1
Ballabeni, V; Barocelli, E; Chiavarini, M; Impicciatore, M1
Kohno, S; Nabe, T; Ogawa, K; Ohata, K; Yamamura, H1
Carson, CC; Davies, MG; Hagen, PO; Kim, YC; Lee, TH1
Kamondi, A; Reiner, PB1
Bristow, DR; Zamani, MR1
Kamei, C; Tasaka, K1
Konno, K; Nakata, J; Takeyama, K; Tamaoki, J1
KAMEI, CH1
Akiyama, K; Maeda, Y; Mita, H; Saito, H; Shimizu, H1
Davison, JS; Jennings, LJ; Pariente, JA; Salido, GM; Sharkey, KA; Singh, J1
Eaton, SJ; Eoh, S; Harrington, ME; Hoque, S; Meyer, J1
Chiyotani, A; Konno, K; Nakata, J; Takeyama, K; Tamaoki, J1
Hayashi, Y; Kagawa, K; Mammoto, T; Mashimo, T; Yamamoto, Y; Yamatodani, A; Yoshiya, I1
Bivalacqua, TJ; Champion, HC; Czapla, MA; Ilgenfritz, C; Kadowitz, PJ; Santiago, JA1
Lecklin, A; Tuomisto, L1
Acuña, Y; Campos, HA; Israel, A; Mathison, Y1
Jokinen, M; Laitinen, JT1
Grundy, D; Haupt, W; Kirkup, AJ; Kreis, ME1
Anichtchik, OV; Panula, P; Peitsaro, N1
Hishinuma, S; Ogura, K1
Ikarashi, Y; Ishige, A; Kuribara, H; Maruyama, Y; Sasaki, H; Yuzurihara, M1
Attoub, S; Bado, A; Laigneau, JP; Lewin, MJ; Moizo, L; Sobhani, I1
Ghosh, AK; Hirasawa, N; Ohuchi, K1
Chen, Z; Li, WD; Shen, YJ; Wei, EQ; Zhu, LJ1
Bischoff, AM; Büsselberg, D; Dutschmann, M; Richter, DW1
Bacon, KB; Gantner, F; Sakai, K; Takeshita, K1
Brzozowski, T; Ceranowicz, P; Dembiński, A; Dembiński, M; Konturek, SJ; Pawlik, WW; Warzecha, Z1
Eckman, JR; Wagner, MC; Wick, TM1
Holopainen, IE; Kukko-Lukjanov, TK; Michelsen, KA; Panula, P; Soini, S; Taira, T1
Gálfi, M; Juhász, A; László, F; László, FA; Molnár, A; Radács, M; Varga, C1
Adachi, N; Arai, T; Hiraga, N; Liu, K; Nagaro, T1
Dutschmann, M; Gratzl, M; Lazarov, N; Reindl, S; Rey-Ares, V; Rozloznik, M1
Krishna, DR; Kumar, KV; Palit, G1
Alcayaga, J; Del Rio, R; Fujiwara, K; Iturriaga, R; Koenig, CS; Moya, EA1
Hirasawa, N; Hong, J; Ishihara, K; Katoh, G; Ohsawa, Y; Ohuchi, K; Seyama, T; Shibata, K; Tamura, S1
Hirasawa, N; Ohuchi, K1

Reviews

2 review(s) available for pyrilamine and thioperamide

ArticleYear
Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:1

    Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship

1990
[Roles of histamine in the exacerbated allergic dermatitis].
    Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan, 2011, Volume: 131, Issue:2

    Topics: Animals; Cyclosporine; Dermatitis, Atopic; Disease Models, Animal; Drug Therapy, Combination; Histamine; Histamine Antagonists; Humans; Mice; Picryl Chloride; Piperidines; Pyrilamine; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H3; Receptors, Histamine H4; Tetradecanoylphorbol Acetate

2011

Other Studies

46 other study(ies) available for pyrilamine and thioperamide

ArticleYear
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4

2005
Non-imidazole histamine H3 ligands, part IV: SAR of 1-[2-thiazol-5-yl-(2-aminoethyl)]-4-n-propylpiperazine derivatives.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:4

    Topics: Animals; Guinea Pigs; Histamine H1 Antagonists; Histamine H3 Antagonists; Imidazoles; Jejunum; Male; Piperazine; Piperazines; Receptors, Histamine H3; Structure-Activity Relationship

2009
Anticonvulsant properties of histamine H3 receptor ligands belonging to N-substituted carbamates of imidazopropanol.
    Bioorganic & medicinal chemistry letters, 2013, Sep-01, Volume: 23, Issue:17

    Topics: 1-Propanol; Animals; Anticonvulsants; Carbamates; Electroshock; Histamine Agonists; Histamine Antagonists; Imidazoles; Ligands; Rats; Rats, Wistar; Receptors, Histamine H3; Seizures

2013
Design, synthesis, and
    MedChemComm, 2019, Feb-01, Volume: 10, Issue:2

    Topics:

2019
Histamine H3 receptors modulate the release of [3H]-acetylcholine from slices of rat entorhinal cortex: evidence for the possible existence of H3 receptor subtypes.
    British journal of pharmacology, 1992, Volume: 107, Issue:4

    Topics: Acetylcholine; Animals; Dose-Response Relationship, Drug; Hippocampus; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Piperidines; Potassium; Pyrilamine; Ranitidine; Rats; Receptors, Histamine; Receptors, Histamine H3

1992
Effects of thioperamide, a histamine H3 receptor antagonist, on locomotor activity and brain histamine content in mast cell-deficient W/Wv mice.
    Life sciences, 1991, Volume: 48, Issue:25

    Topics: Animals; Benzothiazoles; Brain Chemistry; Dopamine; Histamine; Histamine Antagonists; Histamine H2 Antagonists; Mast Cells; Methylhistamines; Mice; Mice, Mutant Strains; Motor Activity; Phenoxypropanolamines; Piperidines; Pyrilamine; Receptors, Histamine H3; Thiazoles

1991
Histamine-induced inositol phosphate accumulation in type-2 astrocytes.
    Biochemical and biophysical research communications, 1991, Jun-14, Volume: 177, Issue:2

    Topics: Animals; Astrocytes; Cells, Cultured; Chlorpheniramine; Famotidine; Histamine; Inositol Phosphates; Piperidines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine

1991
Histamine H3 receptors modulate antigen-induced bronchoconstriction in guinea pigs.
    The Journal of allergy and clinical immunology, 1990, Volume: 86, Issue:4 Pt 1

    Topics: Animals; Antigens; Bronchoconstriction; Cimetidine; Dose-Response Relationship, Drug; Dose-Response Relationship, Immunologic; Guinea Pigs; Histamine; Immunization; Male; Ovalbumin; Piperidines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Skin Tests

1990
Effects of histamine H3-receptor ligands on various biochemical indices of histaminergic neuron activity in rat brain.
    European journal of pharmacology, 1989, May-02, Volume: 164, Issue:1

    Topics: Animals; Brain; Brain Chemistry; Cyclic AMP; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine Decarboxylase; In Vitro Techniques; Male; Methylhistamines; Neurons; Piperidines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H3

1989
Possible participation of histamine H3-receptors in the regulation of anaphylactic histamine release from isolated rat peritoneal mast cells.
    Japanese journal of pharmacology, 1994, Volume: 66, Issue:2

    Topics: Anaphylaxis; Animals; Anticonvulsants; Chromatography, High Pressure Liquid; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Histamine; Histamine Agonists; Histamine Antagonists; Histamine Release; In Vitro Techniques; L-Lactate Dehydrogenase; Male; Mast Cells; Methylhistamines; p-Methoxy-N-methylphenethylamine; Peritoneal Cavity; Peritoneum; Piperidines; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H3

1994
R-alpha-methylhistamine-induced inhibition of gastric acid secretion in pylorus-ligated rats via central histamine H3 receptors.
    British journal of pharmacology, 1995, Volume: 115, Issue:7

    Topics: Animals; Cimetidine; Female; Gastric Acid; Gastric Mucosa; Histamine Agonists; Histamine Antagonists; Injections, Intraventricular; Methylhistamines; Piperidines; Pylorus; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H3

1995
Dimaprit, a histamine H2-agonist, inhibits anaphylactic histamine release from mast cells and the decreased release is restored by thioperamide (H3-antagonist), but not by cimetidine (H2-antagonist).
    Japanese journal of pharmacology, 1993, Volume: 62, Issue:1

    Topics: Anaphylaxis; Animals; Anticonvulsants; Betahistine; Cimetidine; Dimaprit; Histamine H2 Antagonists; Histamine Release; In Vitro Techniques; Indicators and Reagents; Male; Mast Cells; Piperidines; Pyrilamine; Rats; Rats, Wistar

1993
Characterization and function of histamine receptors in corpus cavernosum.
    The Journal of urology, 1995, Volume: 153, Issue:2

    Topics: Acetylcholine; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Papaverine; Penis; Piperidines; Pyrilamine; Rabbits; Receptors, Histamine; Thiazoles

1995
Mechanisms of antihistamine-induced sedation in the human brain: H1 receptor activation reduces a background leakage potassium current.
    Neuroscience, 1994, Volume: 59, Issue:3

    Topics: Cerebral Cortex; Cimetidine; Evoked Potentials; Histamine; Histamine Antagonists; Humans; Hypnotics and Sedatives; Membrane Potentials; Neurons; Piperidines; Potassium Channels; Pyrilamine; Receptors, Histamine H1

1994
Desensitization of histamine H1 receptor-mediated inositol phosphate production in HeLa cells.
    British journal of pharmacology, 1993, Volume: 109, Issue:2

    Topics: Bradykinin; HeLa Cells; Histamine; Humans; Inositol; Inositol Phosphates; Piperidines; Pyrilamine; Ranitidine; Receptors, Histamine H1; Sodium Fluoride

1993
Effect of histamine on memory retrieval in old rats.
    Biological & pharmaceutical bulletin, 1993, Volume: 16, Issue:2

    Topics: Acetylcholine; Aging; Animals; Anticonvulsants; Avoidance Learning; Cerebrovascular Circulation; Cimetidine; Dose-Response Relationship, Drug; Exploratory Behavior; Histamine; Histamine Agonists; Injections, Intraventricular; Male; Memory; Methylhistamines; Motor Activity; Piperidines; Pyrilamine; Rats; Rats, Wistar

1993
Histamine H3 receptor-mediated modulation of water consumption in the rat.
    European journal of pharmacology, 1993, Feb-23, Volume: 232, Issue:1

    Topics: Animals; Drinking; Histamine; Histamine Antagonists; Male; Methylhistamines; Nicotinic Acids; Piperidines; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H3; Tetrazoles; Triazoles

1993
Effect of oxitropium bromide on histamine-induced airway goblet cell secretion.
    American journal of respiratory and critical care medicine, 1996, Volume: 154, Issue:1

    Topics: Administration, Inhalation; Aerosols; Animals; Atropine; Cimetidine; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine Antagonists; Histocytochemistry; Injections, Intravenous; Male; Mucus; Muscarinic Antagonists; Piperidines; Pyrilamine; Receptors, Histamine; Scopolamine Derivatives; Trachea; Vagus Nerve

1996
EFFECTS OF HISTAMINE AND RELATED COMPOUNDS ON THE BOVINE IRIS DILATOR.
    Methods and findings in experimental and clinical pharmacology, 1996, Volume: 18, Issue:4

    Topics: Analysis of Variance; Animals; Cattle; Chlorpheniramine; Cimetidine; Diphenhydramine; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Ileum; Iris; Lethal Dose 50; Male; Methylhistamines; Muscle Contraction; Muscle, Smooth; p-Methoxy-N-methylphenethylamine; Piperidines; Potassium; Pyrilamine; Ranitidine; Receptors, Histamine H1; Substance P

1996
Histamine augments VCAM-1 expression on IL-4- and TNF-alpha-stimulated human umbilical vein endothelial cells.
    International archives of allergy and immunology, 1996, Volume: 111, Issue:2

    Topics: Amanitins; Antibodies, Blocking; Antigens, CD; Cell Adhesion; Cells, Cultured; Cimetidine; Eosinophils; Histamine; Histamine Antagonists; Humans; Immunohistochemistry; Integrin alpha4; Interleukin-4; Piperidines; Platelet Activating Factor; Pyrilamine; Tumor Necrosis Factor-alpha; Umbilical Veins; Vascular Cell Adhesion Molecule-1

1996
Control of exocrine secretion in the guinea-pig pancreas by histamine H3 receptors.
    Canadian journal of physiology and pharmacology, 1996, Volume: 74, Issue:6

    Topics: alpha-Amylases; Animals; Choline; Electric Stimulation; Female; Guinea Pigs; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Pancreas; Piperidines; Pyrilamine; Receptors, Histamine H3; Tritium

1996
Circadian rhythm photic phase shifts are not altered by histamine receptor antagonists.
    Brain research bulletin, 1996, Volume: 41, Issue:4

    Topics: Animals; Benzothiazoles; Cimetidine; Circadian Rhythm; Cricetinae; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Mesocricetus; Phenoxypropanolamines; Photoperiod; Piperidines; Pyrilamine; Receptors, Histamine H3; Thiazoles

1996
Histamine H2 receptor-mediated airway goblet cell secretion and its modulation by histamine-degrading enzymes.
    The Journal of allergy and clinical immunology, 1997, Volume: 99, Issue:2

    Topics: Amine Oxidase (Copper-Containing); Animals; Asthma; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glycoproteins; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine N-Methyltransferase; Male; Methylhistamines; Mucus; Piperidines; Pyrilamine; Recombinant Proteins; Trachea

1997
Interactions between neuronal histamine and halothane anesthesia in rats.
    Journal of neurochemistry, 1997, Volume: 69, Issue:1

    Topics: Anesthetics, Inhalation; Animals; Benzothiazoles; Drug Interactions; Enzyme Inhibitors; Halothane; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine Release; Male; Methylhistidines; Microdialysis; Neurons; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Rats, Sprague-Dawley; Thiazoles

1997
Comparison of responses to T-kinin and bradykinin in the mesenteric vascular bed of the cat.
    Peptides, 1997, Volume: 18, Issue:9

    Topics: Adamantane; Analysis of Variance; Animals; Bradykinin; Bradykinin Receptor Antagonists; Cats; Cimetidine; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Female; Histamine Antagonists; Male; Meclofenamic Acid; Mesentery; Morpholines; NG-Nitroarginine Methyl Ester; Piperidines; Potassium Channels; Pyrilamine

1997
The blockade of H1 receptors attenuates the suppression of feeding and diuresis induced by inhibition of histamine catabolism.
    Pharmacology, biochemistry, and behavior, 1998, Volume: 59, Issue:3

    Topics: Animals; Brain Chemistry; Diuresis; Enzyme Inhibitors; Feeding Behavior; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Piperidines; Pyrilamine; Pyrimethamine; Ranitidine; Rats; Rats, Wistar; Water-Electrolyte Balance

1998
Thioperamide, a histamine H3-receptor blocker, facilitates vasopressor response to footshocks.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1998, Volume: 47, Issue:3

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Cimetidine; Electric Stimulation; Enzyme Inhibitors; Heart Rate; Hindlimb; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistidines; Norepinephrine; Phentolamine; Piperidines; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Vasoconstrictor Agents

1998
Guanosine 5'-(gamma-[35S]thio)triphosphate autoradiography allows selective detection of histamine H3 receptor-dependent G protein activation in rat brain tissue sections.
    Journal of neurochemistry, 1998, Volume: 71, Issue:2

    Topics: Adenosine; Animals; Autoradiography; Basal Ganglia; Brain Chemistry; Cerebral Cortex; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Male; Piperidines; Protein Binding; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H3; Signal Transduction; Substantia Nigra; Sulfur Radioisotopes; Xanthines

1998
Histamine sensitivity of mesenteric afferent nerves in the rat jejunum.
    The American journal of physiology, 1998, Volume: 275, Issue:4

    Topics: Afferent Pathways; Animals; Blood Pressure; Dimaprit; Histamine; Histamine Agonists; Histamine Antagonists; Jejunum; Muscle, Smooth; Nifedipine; Piperidines; Pyrilamine; Ranitidine; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Splanchnic Circulation

1998
Identification of a histamine H(3)-like receptor in the zebrafish (Danio rerio) brain.
    Journal of neurochemistry, 2000, Volume: 75, Issue:2

    Topics: Animals; Autoradiography; Brain; Cimetidine; Female; Guanosine 5'-O-(3-Thiotriphosphate); Histamine Agonists; Histamine Antagonists; Imidazoles; Kinetics; Male; Methylhistamines; Piperidines; Pyrilamine; Radioligand Assay; Receptors, Histamine H3; Sulfur Radioisotopes; Thiourea; Tritium; Zebrafish

2000
Ca(2+)/calmodulin-mediated regulation of the desensitizing process in G(q) protein-coupled histamine H(1) receptor-mediated Ca(2+) responses in human U373 MG astrocytoma cells.
    Journal of neurochemistry, 2000, Volume: 75, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Astrocytoma; Calcineurin Inhibitors; Calcium; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Cyclosporine; Enzyme Inhibitors; GTP-Binding Protein alpha Subunits, Gq-G11; GTP-Binding Proteins; Histamine; Histamine H1 Antagonists; Humans; Kinetics; Okadaic Acid; Piperidines; Pyrilamine; Ranitidine; Receptors, Histamine H1; Sulfonamides; Tacrolimus; Tumor Cells, Cultured

2000
Effects of drugs acting as histamine releasers or histamine receptor blockers on an experimental anxiety model in mice.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 67, Issue:1

    Topics: Animals; Anxiety; Cimetidine; Disease Models, Animal; Histamine Antagonists; Histamine Release; Injections, Intraperitoneal; Injections, Intraventricular; Male; Mice; p-Methoxy-N-methylphenethylamine; Piperidines; Pyrilamine

2000
The H3 receptor is involved in cholecystokinin inhibition of food intake in rats.
    Life sciences, 2001, Jun-15, Volume: 69, Issue:4

    Topics: Animals; Brain; Cholecystokinin; Dose-Response Relationship, Drug; Eating; Gastric Mucosa; Histamine; Histamine Agonists; Histamine Antagonists; Injections, Intraperitoneal; Male; Methylhistamines; Piperidines; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Receptors, Histamine H3; Sincalide; Stomach

2001
Enhancement by histamine of vascular endothelial growth factor production in granulation tissue via H(2) receptors.
    British journal of pharmacology, 2001, Volume: 134, Issue:7

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Cells, Cultured; Cimetidine; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Endothelial Growth Factors; Enzyme Inhibitors; Fibroblasts; Gene Expression Regulation; Granulation Tissue; Histamine; Histamine Antagonists; Immunohistochemistry; Indoles; Indomethacin; Inflammation; Isoquinolines; Lymphokines; Macrophages, Peritoneal; Male; Maleimides; Naphthalenes; Neovascularization, Pathologic; Piperidines; Protein Kinase C; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine H2; RNA, Messenger; Specific Pathogen-Free Organisms; Sulfonamides; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors

2001
Effects of histidine, a precursor of histamine, on pentylenetetrazole-induced seizures in rats.
    Acta pharmacologica Sinica, 2002, Volume: 23, Issue:4

    Topics: Animals; Drug Synergism; Epilepsy; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histidine; Kindling, Neurologic; Male; Pentylenetetrazole; Piperidines; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine H1; Receptors, Histamine H3

2002
Histaminergic modulation of the intact respiratory network of adult mice.
    Pflugers Archiv : European journal of physiology, 2003, Volume: 445, Issue:5

    Topics: Animals; Cimetidine; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Hypoxia; Medulla Oblongata; Mice; Mice, Inbred C57BL; Nerve Net; Neurons; Phrenic Nerve; Piperidines; Pons; Pyrilamine; Receptors, Histamine H3; Respiratory System

2003
Critical role of histamine H4 receptor in leukotriene B4 production and mast cell-dependent neutrophil recruitment induced by zymosan in vivo.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 307, Issue:3

    Topics: Animals; Bone Marrow Cells; Carrageenan; Cimetidine; Cytokines; Dose-Response Relationship, Drug; Enzyme-Linked Immunosorbent Assay; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine Release; Leukotriene B4; Mast Cells; Mice; Mice, Inbred BALB C; Neutrophil Infiltration; Piperidines; Pleurisy; Pyrilamine; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H3; Receptors, Histamine H4; Zymosan

2003
Role of capsaicin-sensitive nerves and histamine H1, H2, and H3 receptors in the gastroprotective effect of histamine against stress ulcers in rats.
    European journal of pharmacology, 2005, Jan-31, Volume: 508, Issue:1-3

    Topics: Animals; Capsaicin; DNA; Gastric Mucosa; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Immersion; Interleukin-1; Male; Neurons, Afferent; Piperidines; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Regional Blood Flow; Restraint, Physical; Stomach Ulcer; Stress, Physiological

2005
Histamine increases sickle erythrocyte adherence to endothelium.
    British journal of haematology, 2006, Volume: 132, Issue:4

    Topics: Analysis of Variance; Anemia, Sickle Cell; Cell Adhesion; Cells, Cultured; Endothelial Cells; Endothelium, Vascular; Erythrocytes; Famotidine; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Imidazoles; Methylhistamines; P-Selectin; Piperidines; Pyrilamine; Stimulation, Chemical; Thiazoles; Thiourea; Venules

2006
Histaminergic neurons protect the developing hippocampus from kainic acid-induced neuronal damage in an organotypic coculture system.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2006, Jan-25, Volume: 26, Issue:4

    Topics: Animals; Cell Death; Cells, Cultured; Coculture Techniques; Convulsants; Hippocampus; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Hypothalamus, Anterior; Hypothalamus, Posterior; Imidazoles; Kainic Acid; Methylhistidines; Microscopy, Confocal; Neurons; Neuroprotective Agents; Organ Culture Techniques; Piperidines; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine H1; Receptors, Histamine H3; Thiourea; Triprolidine

2006
Histamine-induced enhancement of vasopressin and oxytocin secretion in rat neurohypophyseal tissue cultures.
    Regulatory peptides, 2006, May-15, Volume: 134, Issue:2-3

    Topics: Animals; Cimetidine; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Kinetics; Male; Oxytocin; Piperidines; Pituitary Gland, Posterior; Pyrilamine; Rats; Tissue Culture Techniques; Vasopressins

2006
Suppression of inflammatory cell recruitment by histamine receptor stimulation in ischemic rat brains.
    European journal of pharmacology, 2007, Feb-28, Volume: 557, Issue:2-3

    Topics: Animals; Antigens, CD; Brain Ischemia; CD4-Positive T-Lymphocytes; Cell Count; Drug Combinations; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Immunohistochemistry; Infarction, Middle Cerebral Artery; Male; Neutrophils; Peroxidase; Piperidines; Pyrilamine; Random Allocation; Ranitidine; Rats; Rats, Wistar; Receptors, Histamine; Reperfusion; Time Factors

2007
Expression of histamine receptors and effect of histamine in the rat carotid body chemoafferent pathway.
    The European journal of neuroscience, 2006, Volume: 24, Issue:12

    Topics: Afferent Pathways; Amidines; Animals; Blotting, Northern; Carotid Body; Chemoreceptor Cells; Female; Gene Expression; Histamine; Histamine Antagonists; Histidine Decarboxylase; Immunohistochemistry; Male; Medulla Oblongata; Microscopy, Immunoelectron; Phrenic Nerve; Piperidines; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine; Respiration; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sodium Cyanide

2006
Histaminergic H1 receptors mediate L-histidine-induced anxiety in elevated plus-maze test in mice.
    Behavioural pharmacology, 2007, Volume: 18, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Benzothiazoles; Diazepam; Dose-Response Relationship, Drug; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Male; Mice; Phenoxypropanolamines; Piperidines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H3

2007
Modulatory effects of histamine on cat carotid body chemoreception.
    Respiratory physiology & neurobiology, 2008, Dec-31, Volume: 164, Issue:3

    Topics: Acetylcholine; Action Potentials; Animals; Carotid Body; Cats; Chemoreceptor Cells; Dose-Response Relationship, Drug; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H3 Antagonists; Hypoxia; In Vitro Techniques; Male; Microscopy, Immunoelectron; Nicotine; Nicotinic Agonists; Piperidines; Pyrilamine; Tyrosine 3-Monooxygenase

2008
Modification of the picryl chloride-induced allergic dermatitis model in mouse ear lobes by 12-O-tetradecanoylphorbol 13-acetate, and analysis of the role of histamine in the modified model.
    International archives of allergy and immunology, 2009, Volume: 148, Issue:4

    Topics: Animals; Cell Count; Cimetidine; Cyclophosphamide; Cyclosporine; Cytokines; Dermatitis, Allergic Contact; Disease Models, Animal; Ear Auricle; Eosinophil Peroxidase; Eosinophils; Gene Expression; Histamine; Histamine Antagonists; Immunoglobulin E; Interferon-gamma; Interleukin-4; Male; Mast Cells; Mice; Mice, Inbred BALB C; Picryl Chloride; Piperidines; Pyrilamine; Tetradecanoylphorbol Acetate; Thymic Stromal Lymphopoietin

2009