Page last updated: 2024-08-16

pyrilamine and temelastine

pyrilamine has been researched along with temelastine in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19906 (66.67)18.7374
1990's1 (11.11)18.2507
2000's2 (22.22)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Carrupt, PA; Crivori, P; Cruciani, G; Testa, B1
Caron, G; Ermondi, G1
Bach, FW; Bang, P; Knigge, U; Matzen, S; Warberg, J1
Malo, PE; Muccitelli, R; Tucker, SS; Wasserman, MA1
Knigge, U; Matzen, S; Warberg, J2
Brown, EA; Griffiths, R; Harvey, CA; Owen, DA1
Calcutt, CR; Ganellin, CR; Jackson, B; Leigh, BK; Owen, DA; Smith, IR1
Bach, FW; Kjaer, A; Knigge, U; Madsen, EL; Søe-Jensen, P; Warberg, J1

Other Studies

9 other study(ies) available for pyrilamine and temelastine

ArticleYear
Predicting blood-brain barrier permeation from three-dimensional molecular structure.
    Journal of medicinal chemistry, 2000, Jun-01, Volume: 43, Issue:11

    Topics: Blood-Brain Barrier; Databases, Factual; Models, Chemical; Molecular Conformation; Multivariate Analysis; Permeability; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Calculating virtual log P in the alkane/water system (log P(N)(alk)) and its derived parameters deltalog P(N)(oct-alk) and log D(pH)(alk).
    Journal of medicinal chemistry, 2005, May-05, Volume: 48, Issue:9

    Topics: 1-Octanol; Alkanes; Hydrogen-Ion Concentration; Least-Squares Analysis; Mathematics; Models, Chemical; Models, Molecular; Solvents; Water

2005
Involvement of histaminergic neurons in the stress-induced release of pro-opiomelanocortin-derived peptides in rats.
    Acta endocrinologica, 1989, Volume: 120, Issue:4

    Topics: Adrenocorticotropic Hormone; Animals; beta-Endorphin; beta-Lipotropin; Chromatography, Gel; Cimetidine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Pyrilamine; Pyrimidinones; Rats; Rats, Inbred Strains; Stress, Physiological

1989
Effects of SK&F 93944 (Temelastine), a potent histamine H1-receptor antagonist in pharmacologic and antigen-induced bronchoconstriction.
    Methods and findings in experimental and clinical pharmacology, 1986, Volume: 8, Issue:8

    Topics: Animals; Antigens; Bronchi; Dogs; Female; Guinea Pigs; Histamine; Histamine H1 Antagonists; In Vitro Techniques; Male; Muscle Contraction; Ovalbumin; Pyrilamine; Pyrimidinones; Trachea

1986
Histaminergic stimulation of prolactin secretion mediated via H1- or H2-receptors: dependence on routes of administration.
    Neuroendocrinology, 1986, Volume: 44, Issue:1

    Topics: Animals; Cimetidine; Dimaprit; Histamine; Histamine H1 Antagonists; Male; Methylhistamines; Pituitary Gland, Anterior; Prolactin; Pyrilamine; Pyrimidinones; Rats; Receptors, Histamine; Thiazoles; Thiourea

1986
Pharmacological studies with SK&F 93944 (temelastine), a novel histamine H1-receptor antagonist with negligible ability to penetrate the central nervous system.
    British journal of pharmacology, 1986, Volume: 87, Issue:3

    Topics: Animals; Autonomic Nervous System; Central Nervous System; Cerebrovascular Circulation; Female; Guinea Pigs; Hemodynamics; Histamine; Histamine H1 Antagonists; Male; Parasympatholytics; Pyrilamine; Pyrimidinones; Skin Absorption; Sympathetic Nervous System

1986
Evidence for low brain penetration by the H1-receptor antagonist temelastine (SK&F 93944).
    European journal of pharmacology, 1987, Jan-06, Volume: 133, Issue:1

    Topics: Animals; Brain; Dose-Response Relationship, Drug; Histamine H1 Antagonists; In Vitro Techniques; Male; Mice; Motor Activity; Promethazine; Pyrilamine; Pyrimidinones; Receptors, Histamine H1; Tritium

1987
Histaminergic mediation of the stress-induced release of prolactin in male rats.
    Neuroendocrinology, 1988, Volume: 47, Issue:1

    Topics: Animals; Cimetidine; Ether; Histamine; Injections, Intravenous; Injections, Intraventricular; Male; Prolactin; Pyrilamine; Pyrimidinones; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine; Restraint, Physical; Stress, Physiological

1988
Insulin/hypoglycemia-induced adrenocorticotropin and beta-endorphin release: involvement of hypothalamic histaminergic neurons.
    Endocrinology, 1993, Volume: 132, Issue:5

    Topics: Adrenocorticotropic Hormone; Animals; beta-Endorphin; Cetirizine; Cimetidine; Histamine; Histamine Agonists; Histamine Antagonists; Hypoglycemia; Hypothalamus; Insulin; Male; Methylhistamines; Neurons; Pyrilamine; Pyrimidinones; Rats; Rats, Wistar

1993