pyrilamine has been researched along with ranitidine in 92 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 20 (21.74) | 18.7374 |
1990's | 41 (44.57) | 18.2507 |
2000's | 23 (25.00) | 29.6817 |
2010's | 8 (8.70) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Timmerman, H | 1 |
Brown, TH; Ganellin, CR; Griffiths, R; Jones, M; Mitchell, RC; Rana, KK; Saunders, D; Smith, IR; Sore, NE; Young, RC | 1 |
Carrupt, PA; Crivori, P; Cruciani, G; Testa, B | 1 |
Ahman, M; Holmén, AG; Wan, H | 1 |
Ambroso, JL; Ayrton, AD; Baines, IA; Bloomer, JC; Chen, L; Clarke, SE; Ellens, HM; Harrell, AW; Lovatt, CA; Reese, MJ; Sakatis, MZ; Taylor, MA; Yang, EY | 1 |
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM | 1 |
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
Chirtel, SJ; Field, RB | 1 |
Clapham, J; Kilpatrick, GJ | 1 |
Boura, AL; King, RG; Leitch, IM | 1 |
Hiyoshi, Y; Iguchi, A; Li, X; Nonogaki, K; Sakamoto, N; Tamagawa, T; Watanabe, G | 1 |
Bani Sacchi, T; Gambassi, F; Giannella, E; Mannaioni, PF; Masini, E; Palmerani, B; Pistelli, A | 1 |
Blanco, I; Rodriguez, J; Rodriguez, R; Sabriá, J; Toledo, A | 1 |
Bairy, KL; Kulkarni, DR; Ramesh, KV; Rao, CM | 1 |
Heim, HK; Oestmann, A; Sewing, KF | 1 |
Guidobono, F; Netti, C; Pagani, F; Pecile, A; Sibilia, V; Villa, I | 1 |
Ezeamuzie, CI; Umezurike, CC | 1 |
Nicholson, AN; Pascoe, PA; Stone, BM | 1 |
Alvarez, EO; Banzan, AM | 4 |
Iwata, M; Kohno, S; Shigei, T; Tsuru, H | 1 |
Donoso, AO; Podestá, E; Seltzer, AM | 1 |
Knigge, U; Matzen, S; Warberg, J | 1 |
Bommer, M; Herz, A; Kley, N; Liebisch, D; Noble, E | 1 |
Owman, C; Schmidt, G; Sjöberg, NO | 1 |
Barontini, M; Donoso, AO | 1 |
Marshall, K; Senior, J | 1 |
Kume, S; Ohashi, T; Ozaki, Y | 1 |
Daly, MJ; Humphray, JM; Stables, R | 1 |
Bunce, KT; Daly, MJ; Humphray, JM; Stables, R | 2 |
Christiansen, PM; Dejgaard, A; Knigge, U; Larsen, K; Wollesen, F | 1 |
Aghajanian, GK; Lakoski, JM | 1 |
Donoso, AO; Seltzer, A; Zárate, MB | 1 |
Del Soldato, P | 1 |
Barak, V; Fabian, I; Geller-Bernstein, C; Handzel, ZT; Mor, S; Nagler, A | 1 |
Langer, JC; Liebman, SM; Monk, PK; Pelletier, GJ | 1 |
Akaike, N; Munakata, M | 1 |
Hiyoshi, Y; Iguchi, A; Li, X; Nonogaki, K; Ozawa, K; Sakamoto, N; Tamagawa, T; Watanabe, G | 1 |
Iguchi, A; Kunoh, Y; Nonogaki, K; Sakamoto, N; Tamagawa, T; Zhu, LX | 1 |
Holm, L; Jägare, A | 1 |
Langer, JC; Marshall, J; Sohal, SS | 1 |
Bristow, DR; Zamani, MR | 1 |
Onaka, T; Yagi, K | 1 |
Abrahám, CS; Deli, MA; Joó, F; Krizbai, I; Szabó, CA | 1 |
Nowak, JZ; Sek, B; Zawilska, JB | 1 |
KAMEI, CH | 1 |
Hanai, N; Kusano, A; Masaki, S; Miki, I; Ohmori, K; Ohta, S; Otoshi, M; Sato, S | 1 |
Andrysiak, PK; Kmieć, BL | 2 |
Agut, J; Ortiz, JA; Sacristán, A; Sánchez, JC | 1 |
Murakami, Y; Okuma, Y; Osumi, Y; Yokotani, K | 1 |
Ito, Y; Kashiwagi, S; Kimura, C; Oike, M | 1 |
Lecklin, A; Tuomisto, L | 1 |
Alvarez, EO; Orofino, AG; Ruarte, MB | 2 |
Fan, DS; Liu, T; Yang, PC; Zhang, TY | 1 |
Grundy, D; Haupt, W; Kirkup, AJ; Kreis, ME | 1 |
Allescher, HD; Hahn, A; Huber, A; Neumayer, N | 1 |
Akiba, Y; Kaunitz, JD; Tanaka, S | 1 |
Danowski, J; Kmieć, BL | 3 |
Al-Rashood, KA; Al-Sayed, MI; Bakheet, DM; El Tahir, KE; El-Obeid, HA | 1 |
Hishinuma, S; Ogura, K | 1 |
Firth, TA; Guarraci, FA; Hemming, JM; Jennings, LJ; Mawe, GM; Nelson, MT | 1 |
Harasawa, K | 1 |
Jørgensen, H; Kjaer, A; Knigge, U; Warberg, J | 1 |
Ishinaga, H; Kishioka, C; Majima, Y; Sakakura, Y; Takeuchi, K | 1 |
Kolaczkowska, E; Plytycz, B; Seljelid, R | 1 |
Al Obaid, AR; Al Rasheed, NM; Al Sayed, MI; Al Zuhair, HH; Fatani, AJ | 1 |
Attoub, S; Bado, A; Laigneau, JP; Lewin, MJ; Moizo, L; Sobhani, I | 1 |
Liu, T; Wang, B; Yang, P | 1 |
Bernsand, M; Bjorkqvist, M; Ericsson, P; Hakanson, R; Norlen, P; Zhao, CM | 1 |
Adachi, N; Arai, T; Liu, K | 2 |
Farahmanfar, M; Fazli-Tabaei, S; Khalilzadeh, A; Yahyavi, SH; Zarrindast, MR | 1 |
Roohbakhsh, A; Rostami, P; Zarei, M; Zarrindast, MR | 1 |
Moghadam, AH; Roohbakhsh, A; Rostami, P; Zarrindast, MR | 1 |
Hajizadeh-Moghaddam, A; Rostami, P; Zarrindast, MR | 1 |
Moghimi, M; Rezayof, A; Rostami, P; Zarrindast, MR | 1 |
Fazli-Tabaei, S; Rostami, P; Torabi, M; Zarrindast, MR | 1 |
Adachi, N; Arai, T; Hiraga, N; Liu, K; Nagaro, T | 1 |
Rezayof, A; Rostami, P; Valizadegan, F; Zarrindast, MR | 1 |
Bina, P; Nasehi, M; Piri, M; Zarrindast, MR | 1 |
Erfanparast, A; Farshid, AA; Khalilzadeh, E; Tamaddonfard, E | 1 |
Khodarahmi, P; Oryan, S; Rezayof, A; Zarrindast, MR | 1 |
Ghasri, S; Hamzely, A; Khoshkholgh Sima, B; Mobarakeh, JI; Nezhad, RM; Nunoki, K; Rahimi, AA; Takahashi, K; Torkaman-Boutorabi, A; Yanai, K | 1 |
Asgariyan, M; Nasehi, M; Piri, M; Zarrindast, MR | 1 |
Jimenez-Gomez, C; Podlesnik, CA | 1 |
1 review(s) available for pyrilamine and ranitidine
Article | Year |
---|---|
Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship | 1990 |
1 trial(s) available for pyrilamine and ranitidine
Article | Year |
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Dehydration-induced vasopressin secretion in humans: involvement of the histaminergic system.
Topics: Adult; Aldosterone; Cimetidine; Cross-Over Studies; Dehydration; Double-Blind Method; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Male; Osmolar Concentration; Placebos; Pyrilamine; Ranitidine; Receptors, Histamine H1; Receptors, Histamine H2; Vasopressins; Water-Electrolyte Balance | 2000 |
90 other study(ies) available for pyrilamine and ranitidine
Article | Year |
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Development of a new physicochemical model for brain penetration and its application to the design of centrally acting H2 receptor histamine antagonists.
Topics: Algorithms; Animals; Blood-Brain Barrier; Brain; Chemical Phenomena; Chemistry, Physical; Clonidine; Guinea Pigs; Histamine H2 Antagonists; Imipramine; Pyrilamine; Structure-Activity Relationship | 1988 |
Predicting blood-brain barrier permeation from three-dimensional molecular structure.
Topics: Blood-Brain Barrier; Databases, Factual; Models, Chemical; Molecular Conformation; Multivariate Analysis; Permeability; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship | 2000 |
Relationship between brain tissue partitioning and microemulsion retention factors of CNS drugs.
Topics: Brain; Central Nervous System; Chromatography, Liquid; Emulsions; Mass Spectrometry | 2009 |
Preclinical strategy to reduce clinical hepatotoxicity using in vitro bioactivation data for >200 compounds.
Topics: Chemical and Drug Induced Liver Injury; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Decision Trees; Drug Evaluation, Preclinical; Drug-Related Side Effects and Adverse Reactions; Glutathione; Humans; Liver; Pharmaceutical Preparations; Protein Binding | 2012 |
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4 | 2005 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |
The effects of histamine, pyrilamine, cimetidine, and ranitidine on secretion of lingual lipase and amylase from rat von Ebner's glands.
Topics: Amylases; Animals; Cimetidine; Exocytosis; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Lipase; Male; Pyrilamine; Ranitidine; Rats; Rats, Sprague-Dawley; Salivary Glands | 1992 |
Histamine H3 receptors modulate the release of [3H]-acetylcholine from slices of rat entorhinal cortex: evidence for the possible existence of H3 receptor subtypes.
Topics: Acetylcholine; Animals; Dose-Response Relationship, Drug; Hippocampus; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Piperidines; Potassium; Pyrilamine; Ranitidine; Rats; Receptors, Histamine; Receptors, Histamine H3 | 1992 |
Pharmacological evaluation of the histamine H1 and 5-HT blocking properties of 2-N-(carboxamidinonormianserin) (FCC5): in-vitro studies.
Topics: Animals; Electric Stimulation; Guinea Pigs; Heart Rate; Histamine; Histamine H1 Antagonists; Ileum; In Vitro Techniques; Male; Mianserin; Muscle Contraction; Muscle, Smooth; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Serotonin Antagonists; Stomach | 1992 |
Role of brain histamine H1- and H2-receptors in neostigmine-induced hyperglycemia in rats.
Topics: Animals; Blood Glucose; Brain; Hyperglycemia; Male; Neostigmine; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2 | 1992 |
Histamine release by platelet aggregation.
Topics: Animals; Arachidonic Acids; Blood Platelets; Histamine Release; In Vitro Techniques; L-Lactate Dehydrogenase; Male; Mast Cells; Platelet Aggregation; Pyridines; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains | 1990 |
A comparative study of histamine and K+ effects on (Ca(2+)-Mg2+)-ATPase activity in synaptosomes.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Ca(2+) Mg(2+)-ATPase; Calcium Chloride; Calcium-Transporting ATPases; Cell Membrane; Choline; Diltiazem; Dose-Response Relationship, Drug; Histamine; Potassium; Pyrilamine; Ranitidine; Rats; Sodium; Synapses; Synaptosomes; Verapamil | 1991 |
Effects of antihistamines on wound healing.
Topics: Animals; Cimetidine; Female; Histamine Antagonists; Male; Promethazine; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Wound Healing | 1991 |
Effects of histamine on protein and glycoprotein production of isolated pig gastric mucosal cells.
Topics: 16,16-Dimethylprostaglandin E2; Acetylglucosamine; Animals; Colforsin; Gastric Mucosa; Glycoproteins; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Leucine; Protein Biosynthesis; Pyrilamine; Ranitidine; Receptors, Histamine H1; Receptors, Histamine H2; Swine; Tritium | 1990 |
A selective role for brain histamine in prolactin release induced by opiates.
Topics: Animals; beta-Endorphin; Brain Chemistry; Histamine; Injections, Intraventricular; Male; Methylhistidines; Prolactin; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains | 1990 |
Effect of histamine H2-receptor antagonists on acute inflammatory of the rat paw oedema.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Cimetidine; Edema; Freund's Adjuvant; Histamine; Histamine H2 Antagonists; Male; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Triazoles | 1989 |
Histaminergic systems and sleep. Studies in man with H1 and H2 antagonists.
Topics: Adolescent; Adult; Brompheniramine; Cimetidine; Electroencephalography; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Male; Phenothiazines; Psychomotor Performance; Pyrilamine; Ranitidine; Sleep; Sleep Stages; Sleep, REM; Triprolidine | 1985 |
Histamine sensitive sites in hippocampus: their probable role on prolactin release in male rats.
Topics: Animals; Hippocampus; Histamine; Histamine H1 Antagonists; Male; Methylhistidines; Microinjections; Prolactin; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Stress, Physiological | 1987 |
Characterization of histamine receptors in isolated rabbit veins.
Topics: Animals; Cimetidine; Endothelium, Vascular; Female; Histamine; Imidazoles; Impromidine; Male; Pyrilamine; Rabbits; Ranitidine; Receptors, Histamine; Receptors, Histamine H2; Species Specificity; Vasoconstriction; Veins | 1987 |
Restraint stress stimulation of prolactin and ACTH secretion: role of brain histamine.
Topics: Adrenocorticotropic Hormone; Animals; Corticosterone; Histamine; Hypothalamo-Hypophyseal System; Male; Methylhistidines; Pituitary-Adrenal System; Prolactin; Pyrilamine; Ranitidine; Rats; Synaptic Transmission | 1986 |
Histamine in dorsal and ventral hippocampus. II. Effects of H1 and H2 histamine antagonists on exploratory behavior in male rats.
Topics: Aminopyridines; Animals; Brain Mapping; Exploratory Behavior; Hippocampus; Histamine; Histidine Decarboxylase; Male; Methylhistidines; Motor Activity; Neural Inhibition; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Synaptic Transmission | 1986 |
Histaminergic mediation of the stress-induced release of prolactin in male rats.
Topics: Animals; Cimetidine; Ether; Histamine; Injections, Intravenous; Injections, Intraventricular; Male; Prolactin; Pyrilamine; Pyrimidinones; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine; Restraint, Physical; Stress, Physiological | 1988 |
Histamine affects release and biosynthesis of opioid peptides primarily via H1-receptors in bovine chromaffin cells.
Topics: Adrenal Glands; Animals; Calcium; Cattle; Cells, Cultured; Chromaffin System; Cimetidine; Clemastine; Cobalt; Enkephalin, Leucine; Enkephalin, Methionine; Enkephalins; Gallopamil; Histamine; Histamine Antagonists; Nifedipine; Protein Precursors; Pyrilamine; Ranitidine; Receptors, Histamine; Receptors, Histamine H1; RNA, Messenger | 1987 |
Histamine induces ovulation in the isolated perfused rat ovary.
Topics: Animals; Cimetidine; Female; Gonadotropins, Equine; Histamine; Luteinizing Hormone; Ovary; Ovulation Induction; Perfusion; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains | 1986 |
Increase in plasma catecholamines by intraventricular injection of histamine in conscious rats.
Topics: Animals; Brain; Epinephrine; Histamine; Injections, Intraventricular; Male; Norepinephrine; Pyrilamine; Ranitidine; Rats | 1986 |
The effect of mepyramine and ranitidine on the oestrogen and anti-oestrogen stimulated rat uterus.
Topics: Aminopyridines; Animals; Estrogen Antagonists; Estrogens; Female; Organ Size; Pyrilamine; Ranitidine; Rats; Receptors, Histamine; Regional Blood Flow; Tamoxifen; Uterine Contraction; Uterus | 1986 |
Effects of histamine agonists and antagonists on luminol-dependent chemiluminescence of granulocytes.
Topics: Cimetidine; Dimaprit; Granulocytes; Histamine; Histamine Antagonists; Humans; In Vitro Techniques; Luminescent Measurements; Luminol; Pyridazines; Pyridines; Pyrilamine; Ranitidine; Thiourea | 1984 |
Antagonism of vasodepressor and gastric secretory responses to histamine by the H2-receptor antagonists, ranitidine and cimetidine, in the anaesthetized dog.
Topics: Anesthesia; Animals; Blood Pressure; Cimetidine; Dogs; Dose-Response Relationship, Drug; Female; Furans; Gastric Acid; Guanidines; Histamine; Histamine H2 Antagonists; Male; Pyrilamine; Ranitidine | 1981 |
The effect of ranitidine on gastric acid secretory response curves to histamine, pentagastrin or bethanechol in the dog with a Heidenhain pouch.
Topics: Animals; Bethanechol Compounds; Cimetidine; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Furans; Gastric Acid; Histamine; Histamine H2 Antagonists; Male; Pentagastrin; Pyrilamine; Ranitidine | 1981 |
H2-receptor antagonists protect against aspirin-induced gastric lesions in the rat.
Topics: Animals; Aspirin; Cimetidine; Female; Furans; Gastric Mucosa; Histamine H2 Antagonists; Pyrilamine; Ranitidine; Rats; Stomach Ulcer | 1981 |
The effect of histamine stimulation and H2 -receptor inhibition on the pituitary prolactin and ACTH release and on cortisol secretion in human males.
Topics: Adrenocorticotropic Hormone; Adult; Aged; Furans; Histamine; Histamine H2 Antagonists; Humans; Hydrocortisone; Male; Middle Aged; Pituitary Gland, Anterior; Prolactin; Pyrilamine; Ranitidine | 1983 |
Effects of histamine, H1- and H2-receptor antagonists on the activity of serotonergic neurons in the dorsal raphe nucleus.
Topics: Animals; Brain Stem; Cimetidine; Diphenhydramine; gamma-Aminobutyric Acid; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Metiamide; Neurons; Pyrilamine; Ranitidine; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Serotonin; Synaptic Transmission | 1983 |
Histamine-induced prolactin release: pharmacological characterization of receptors in male rats.
Topics: Anesthesia; Animals; Furans; Histamine; Male; Methylhistamines; Metiamide; Prolactin; Pyrilamine; Ranitidine; Rats; Receptors, Histamine | 1983 |
Studies with specific agonists and antagonists of the role of histamine H1- and H2-receptor activation in the pathogenesis of gastric lesions in rats.
Topics: Aminopyridines; Animals; Atropine; Dimaprit; Drug Interactions; Female; Histamine; Pyridines; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Stomach Ulcer; Thiourea | 1984 |
Histamine enhances granulocyte-macrophage colony-stimulating factor and interleukin-6 production by human peripheral blood mononuclear cells.
Topics: Antibodies; Cell Adhesion; Cells, Cultured; Cimetidine; Enzyme-Linked Immunosorbent Assay; Granulocyte-Macrophage Colony-Stimulating Factor; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Interleukin-3; Interleukin-6; Kinetics; Leukocytes, Mononuclear; Pyrilamine; Radioimmunoassay; Ranitidine; Stem Cells; Stimulation, Chemical; Terfenadine | 1995 |
Mast cell mediators and peritoneal adhesion formation in the rat.
Topics: Animals; Azepines; Disease Models, Animal; Histamine Antagonists; Leukotriene D4; Male; Mast Cells; Methysergide; Ondansetron; Peritoneal Diseases; Platelet Activating Factor; Propionates; Pyrilamine; Quinolines; Ranitidine; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Tissue Adhesions; Triazoles | 1995 |
Regulation of K+ conductance by histamine H1 and H2 receptors in neurones dissociated from rat neostriatum.
Topics: Animals; Cimetidine; Dose-Response Relationship, Drug; Famotidine; Female; Histamine; Histamine Agonists; Impromidine; In Vitro Techniques; Ion Transport; Male; Membrane Potentials; Methylhistamines; Neostriatum; Potassium; Potassium Channels; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Triprolidine | 1994 |
Histamine-induced, central nervous system-mediated hyperglycemia is suppressed by atropine in the brain.
Topics: Animals; Atropine; Brain; Central Nervous System; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Hyperglycemia; Injections, Intraventricular; Male; Neurotransmitter Agents; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Receptors, Muscarinic | 1993 |
Involvement of central cholinergic muscarinic receptors and histamine H1 receptors in hyperglycemia induced by prostaglandin F2 alpha in rats.
Topics: Animals; Atropine; Dinoprost; Diphenhydramine; Histamine H1 Antagonists; Hyperglycemia; Injections, Intraventricular; Male; Muscarinic Antagonists; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Receptors, Muscarinic | 1993 |
Histamine is not involved in pentagastrin-induced gastric mucosal vasodilation in the rat.
Topics: Animals; Blood Flow Velocity; Blood Vessels; Erythrocytes; Gastric Acid; Gastric Mucosa; Histamine; Injections, Intra-Arterial; Injections, Intravenous; Laser-Doppler Flowmetry; Male; Pentagastrin; Pyrilamine; Ranitidine; Rats; Rats, Sprague-Dawley; Vasodilation | 1994 |
Histamine does not mediate mucosal permeability changes after subclinical intestinal ischemia-reperfusion injury.
Topics: Animals; Chromium Radioisotopes; Edetic Acid; Enterocolitis, Pseudomembranous; Histamine; Ileum; Intestinal Absorption; Intestinal Mucosa; Male; Pyrilamine; Ranitidine; Rats; Rats, Sprague-Dawley; Reperfusion Injury; Weaning | 1993 |
Desensitization of histamine H1 receptor-mediated inositol phosphate production in HeLa cells.
Topics: Bradykinin; HeLa Cells; Histamine; Humans; Inositol; Inositol Phosphates; Piperidines; Pyrilamine; Ranitidine; Receptors, Histamine H1; Sodium Fluoride | 1993 |
Suppressive vasopressin response to emotional stress: the neuroactive substance that may be involved.
Topics: Animals; Benzazepines; Naloxone; Prolactin; Pyrilamine; Ranitidine; Rats; Stress, Psychological; Vasopressins | 1993 |
Receptor-mediated regulation by histamine of the acid phosphatase activity in cultured cerebral endothelial cells.
Topics: Acid Phosphatase; Animals; Cell Line; Cerebral Cortex; Endothelium; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Indicators and Reagents; Molecular Weight; Nitrophenols; Organophosphorus Compounds; Pyrilamine; Ranitidine; Rats | 1996 |
A bizarre receptor mediating stimulatory effect of histamine on cyclic AMP formation in duck pineal gland.
Topics: Animals; Cyclic AMP; Ducks; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Methylhistamines; Pineal Gland; Pyrilamine; Ranitidine; Receptors, Histamine | 1995 |
EFFECTS OF HISTAMINE AND RELATED COMPOUNDS ON THE BOVINE IRIS DILATOR.
Topics: Analysis of Variance; Animals; Cattle; Chlorpheniramine; Cimetidine; Diphenhydramine; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Ileum; Iris; Lethal Dose 50; Male; Methylhistamines; Muscle Contraction; Muscle, Smooth; p-Methoxy-N-methylphenethylamine; Piperidines; Potassium; Pyrilamine; Ranitidine; Receptors, Histamine H1; Substance P | 1996 |
Histamine enhanced the TNF-alpha-induced expression of E-selectin and ICAM-1 on vascular endothelial cells.
Topics: Animals; Cells, Cultured; CHO Cells; Cricetinae; Dibenzoxepins; Diphenhydramine; Drug Interactions; E-Selectin; Endothelium, Vascular; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Intercellular Adhesion Molecule-1; Ketotifen; Olopatadine Hydrochloride; Pyrilamine; Ranitidine; Tumor Necrosis Factor-alpha; Umbilical Veins | 1996 |
Hippocampus and learning: possible role of histamine receptors.
Topics: Animals; Evoked Potentials, Auditory; Hippocampus; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Learning; Male; Memory; Pyrilamine; Ranitidine; Rats; Rats, Sprague-Dawley; Reaction Time | 1996 |
Hippocampal histamine receptors: possible role on the mechanisms of memory in the rat, II.
Topics: Animals; Avoidance Learning; Electroshock; Hippocampus; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Memory; Microinjections; Pyrilamine; Ranitidine; Rats; Receptors, Histamine | 1996 |
Morphobiochemical studies on alpha-amylase secretion by pancreatic follicles of guinea pigs after the application of exogenous histamine.
Topics: alpha-Amylases; Animals; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; L-Lactate Dehydrogenase; Male; Pancreas; Pyrilamine; Ranitidine | 1997 |
Action of ebrotidine, ranitidine and cimetidine on the specific binding to histamine H1- and H2-receptors.
Topics: Animals; Benzenesulfonates; Cell Membrane; Cerebellum; Cerebral Cortex; Cimetidine; Depression, Chemical; Guinea Pigs; Histamine H2 Antagonists; In Vitro Techniques; Isotope Labeling; Male; Protein Binding; Pyrilamine; Ranitidine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Tritium | 1997 |
Brain histamine mediates the bombesin-induced central activation of sympatho-adrenomedullary outflow.
Topics: Adrenal Medulla; Animals; Bombesin; Brain; Epinephrine; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Hypothalamus; Injections, Intraventricular; Male; Norepinephrine; Pargyline; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Sympathetic Nervous System | 1997 |
Effects of acute glucose overload on histamine H2 receptor-mediated Ca2+ mobilization in bovine cerebral endothelial cells.
Topics: Animals; Bradykinin; Brain; Bucladesine; Calcium; Cattle; Cells, Cultured; Cimetidine; Cyclic AMP; Dose-Response Relationship, Drug; Endothelium, Vascular; Glucose; Histamine; Histamine Antagonists; Homeostasis; Microcirculation; Neomycin; Neurotransmitter Agents; Protein Kinase C; Pyrilamine; Ranitidine; Receptors, Histamine H2; Staurosporine | 1998 |
The blockade of H1 receptors attenuates the suppression of feeding and diuresis induced by inhibition of histamine catabolism.
Topics: Animals; Brain Chemistry; Diuresis; Enzyme Inhibitors; Feeding Behavior; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Piperidines; Pyrilamine; Pyrimethamine; Ranitidine; Rats; Rats, Wistar; Water-Electrolyte Balance | 1998 |
Hippocampal histamine receptors and conflictive exploration in the rat: studies using the elevated asymmetric plus-maze.
Topics: Animals; Exploratory Behavior; Hippocampus; Histamine; Male; Maze Learning; Pyrilamine; Ranitidine; Rats; Rats, Sprague-Dawley; Receptors, Histamine | 1997 |
Effect of substance P on the short-circuit current of rat nasal mucosal epithelium.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Biphenyl Compounds; Disease Models, Animal; Electric Stimulation; Epithelium; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine Release; Male; Mast Cells; Nasal Mucosa; Pyrilamine; Ranitidine; Rats; Rats, Sprague-Dawley; Rhinitis, Allergic, Seasonal; Substance P | 1998 |
Histamine sensitivity of mesenteric afferent nerves in the rat jejunum.
Topics: Afferent Pathways; Animals; Blood Pressure; Dimaprit; Histamine; Histamine Agonists; Histamine Antagonists; Jejunum; Muscle, Smooth; Nifedipine; Piperidines; Pyrilamine; Ranitidine; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Splanchnic Circulation | 1998 |
Effect of interleukin-1beta on the ascending and descending reflex in rat small intestine.
Topics: Animals; Cyclooxygenase Inhibitors; Electric Stimulation; Histamine Antagonists; Imidazoles; In Vitro Techniques; Indomethacin; Interleukin-1; Interleukin-2; Intestine, Small; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Muscles; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Interleukin-1; Reflex; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiourea; Tumor Necrosis Factor-alpha | 1998 |
Pentagastrin gastroprotection against acid is related to H2 receptor activation but not acid secretion.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Aspirin; Gastric Acid; Gastric Mucosa; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Hydrogen-Ion Concentration; Male; Omeprazole; Pentagastrin; Perfusion; Pyrilamine; Ranitidine; Rats; Rats, Sprague-Dawley; Stomach Ulcer | 1998 |
Morphobiochemical investigations of the thyroid gland of the guinea pig after the application of some receptor antagonists and histamine.
Topics: Animals; Ca(2+) Mg(2+)-ATPase; Guinea Pigs; Histamine; Histamine Antagonists; Ipratropium; L-Lactate Dehydrogenase; Male; Monoamine Oxidase; Muscarinic Antagonists; Pyrilamine; Ranitidine; Receptors, Histamine H1; Receptors, Histamine H2; Sodium-Potassium-Exchanging ATPase; Thyroid Gland; Thyroxine; Triiodothyronine | 1999 |
Histoenzymatic investigations of the thyroid gland of guinea pig after the application of some receptor antagonists and histamine.
Topics: Animals; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Histocytochemistry; L-Lactate Dehydrogenase; Male; Pyrilamine; Ranitidine; Receptors, Histamine; Shock; Thyroid Gland | 1999 |
Morphobiochemical studies on alpha-amylase secretion by parotid gland acini of guinea pigs after the application of exogenous histamine.
Topics: alpha-Amylases; Animals; Cytoplasmic Granules; Enzyme Precursors; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Histocytochemistry; L-Lactate Dehydrogenase; Male; Parotid Gland; Pyrilamine; Ranitidine | 1999 |
Exploratory behaviour after intra-accumbens histamine and/or histamine antagonists injection in the rat.
Topics: Animals; Arousal; Brain Mapping; Exploratory Behavior; Fear; Histamine; Histamine Antagonists; Injections; Male; Maze Learning; Motivation; Nucleus Accumbens; Pyrilamine; Ranitidine; Rats; Rats, Sprague-Dawley; Reaction Time; Social Environment | 1999 |
Studies on the cardiovascular depressant effects of N-ethyl- and N-benzyl-1,2-diphenylethanolamines in the rat: elucidation of the mechanisms of action.
Topics: Animals; Arrhythmias, Cardiac; Blood Pressure; Calcium Chloride; Cardiovascular Agents; Cardiovascular Diseases; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Ethanolamines; Heart Rate; Histamine H1 Antagonists; Histamine H2 Antagonists; Indomethacin; Male; Pyrilamine; Ranitidine; Rats; Rats, Wistar | 1999 |
Ca(2+)/calmodulin-mediated regulation of the desensitizing process in G(q) protein-coupled histamine H(1) receptor-mediated Ca(2+) responses in human U373 MG astrocytoma cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Astrocytoma; Calcineurin Inhibitors; Calcium; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Cyclosporine; Enzyme Inhibitors; GTP-Binding Protein alpha Subunits, Gq-G11; GTP-Binding Proteins; Histamine; Histamine H1 Antagonists; Humans; Kinetics; Okadaic Acid; Piperidines; Pyrilamine; Ranitidine; Receptors, Histamine H1; Sulfonamides; Tacrolimus; Tumor Cells, Cultured | 2000 |
Actions of histamine on muscle and ganglia of the guinea pig gallbladder.
Topics: Adenosine Triphosphate; Animals; Dimaprit; Excitatory Postsynaptic Potentials; Female; Gallbladder; Gallbladder Emptying; Ganglia, Autonomic; Guinea Pigs; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Mast Cells; Membrane Potentials; Muscle, Smooth; p-Methoxy-N-methylphenethylamine; Patch-Clamp Techniques; Potassium Channels; Pyrilamine; Ranitidine; Receptors, Histamine H1; Receptors, Histamine H2 | 2000 |
Does the histaminergic system play a role in spinal nociception?
Topics: Animals; Dose-Response Relationship, Drug; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Methylhistamines; Motor Neurons; Pain; Pyrilamine; Ranitidine; Rats; Spinal Cord; Synaptic Transmission | 2000 |
Histamine alters gene expression in cultured human nasal epithelial cells.
Topics: Cells, Cultured; Epithelial Cells; Gene Expression; Histamine; Histamine H2 Antagonists; Humans; Nasal Mucosa; Pyrilamine; Ranitidine; Receptors, Histamine H1; RNA, Messenger; Tumor Necrosis Factor-alpha | 2001 |
Role of mast cells in zymosan-induced peritoneal inflammation in Balb/c and mast cell-deficient WBB6F1 mice.
Topics: Animals; Anti-Asthmatic Agents; Cimetidine; Cromolyn Sodium; Histamine Antagonists; Hypoglycemic Agents; Mast Cells; Mice; Mice, Inbred BALB C; Mice, Knockout; Peritonitis; Pyrilamine; Ranitidine; Receptors, Histamine; Triprolidine; Zymosan | 2001 |
Effects of two newly synthesized analogues of lidocaine on rat arterial blood pressure and heart rate.
Topics: Anesthetics, Local; Animals; Anti-Arrhythmia Agents; Antihypertensive Agents; Atropine; Benzoates; Blood Pressure; Calcium Chloride; Cyproheptadine; Enzyme Inhibitors; Heart Rate; Hexamethonium; Histamine Agonists; Indomethacin; Lidocaine; Male; Monitoring, Physiologic; NG-Nitroarginine Methyl Ester; Pyrilamine; Quinacrine; Ranitidine; Rats; Rats, Wistar; Vasodilator Agents | 2001 |
The H3 receptor is involved in cholecystokinin inhibition of food intake in rats.
Topics: Animals; Brain; Cholecystokinin; Dose-Response Relationship, Drug; Eating; Gastric Mucosa; Histamine; Histamine Agonists; Histamine Antagonists; Injections, Intraperitoneal; Male; Methylhistamines; Piperidines; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Receptors, Histamine H3; Sincalide; Stomach | 2001 |
[Effect of substance P on the short-circuit current of nasal mucosal epithelium].
Topics: Animals; Biphenyl Compounds; Electrophysiology; Epithelium; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Nasal Mucosa; Ovalbumin; Pyrilamine; Ranitidine; Rats; Rats, Sprague-Dawley; Rhinitis, Allergic, Perennial; Substance P; Tetrodotoxin | 1998 |
Histochemical and biochemical studies on the secretory mechanisms of some glands of guinea-pigs treated with histamine.
Topics: Adrenal Glands; Animals; Endocrine Glands; Exocrine Glands; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Ipratropium; Male; Muscarinic Antagonists; Pancreas; Parotid Gland; Pyrilamine; Ranitidine; Thyroid Gland; Tissue Fixation | 2002 |
Submucosal microinfusion of endothelin and adrenaline mobilizes ECL-cell histamine in rat stomach, and causes mucosal damage: a microdialysis study.
Topics: Animals; Cells, Cultured; Endothelins; Enterochromaffin-like Cells; Epinephrine; Female; Gastric Mucosa; Gastrins; Histamine; Histamine Release; Histidine Decarboxylase; Infusions, Parenteral; Male; Methylhistidines; Microdialysis; Microinjections; Misoprostol; Omeprazole; Parietal Cells, Gastric; Pyrilamine; Ranitidine; Rats; Rats, Sprague-Dawley; Somatostatin; Time Factors | 2003 |
Alleviation of ischemic neuronal damage by postischemic loading with histidine in the rat striatum.
Topics: Animals; Brain Ischemia; Cell Count; Corpus Striatum; Drug Interactions; Functional Laterality; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Infarction, Middle Cerebral Artery; Male; Neurons; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Reperfusion; Reperfusion Injury; Time Factors | 2004 |
Prevention of brain infarction by postischemic administration of histidine in rats.
Topics: Animals; Brain Ischemia; Disease Models, Animal; Functional Laterality; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Infarction, Middle Cerebral Artery; Injections, Intraperitoneal; Injections, Intraventricular; Male; Motor Activity; Neurons; Neuroprotective Agents; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Statistics, Nonparametric | 2005 |
Cross state-dependent retrieval between histamine and lithium.
Topics: Analysis of Variance; Animals; Avoidance Learning; Behavior, Animal; Dose-Response Relationship, Drug; Drug Interactions; Histamine; Histamine H1 Antagonists; Injections, Intraventricular; Lithium; Male; Memory; Mice; Mice, Inbred Strains; Pyrilamine; Ranitidine; Time Factors | 2005 |
Intracerebroventricular effects of histaminergic agents on morphine-induced anxiolysis in the elevated plus-maze in rats.
Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Drug Interactions; Histamine; Histamine Agents; Histamine H1 Antagonists; Histamine H2 Antagonists; Injections, Intraventricular; Male; Microinjections; Morphine; Narcotics; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Stereotaxic Techniques | 2005 |
The effects of histaminergic agents in the central amygdala of rats in the elevated plus-maze test of anxiety.
Topics: Amygdala; Animals; Anxiety; Histamine; Histamine Agents; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Microinjections; Pyrilamine; Ranitidine; Rats; Stereotaxic Techniques | 2005 |
The effects of histaminergic agents in the ventral hippocampus of rats in the plus-maze test of anxiety-like behaviours.
Topics: Analysis of Variance; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Hippocampus; Histamine; Histamine Agents; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Maze Learning; Microinjections; Pyrilamine; Ranitidine; Rats; Rats, Wistar | 2006 |
Histaminergic receptors of medial septum and conditioned place preference: D1 dopamine receptor mechanism.
Topics: Analysis of Variance; Animals; Behavior, Animal; Benzazepines; Conditioning, Psychological; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Motor Activity; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Reaction Time; Receptors, Dopamine; Receptors, Histamine; Septum of Brain; Sulpiride | 2006 |
The effects of histaminergic agents in the dorsal hippocampus of rats in the elevated plus-maze test of anxiety.
Topics: Animals; Anxiety; Hippocampus; Histamine; Male; Maze Learning; Motor Activity; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H2 | 2006 |
Suppression of inflammatory cell recruitment by histamine receptor stimulation in ischemic rat brains.
Topics: Animals; Antigens, CD; Brain Ischemia; CD4-Positive T-Lymphocytes; Cell Count; Drug Combinations; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Immunohistochemistry; Infarction, Middle Cerebral Artery; Male; Neutrophils; Peroxidase; Piperidines; Pyrilamine; Random Allocation; Ranitidine; Rats; Rats, Wistar; Receptors, Histamine; Reperfusion; Time Factors | 2007 |
Histaminergic system of the lateral septum in the modulation of anxiety-like behaviour in rats.
Topics: Animals; Anxiety; Behavior, Animal; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Microinjections; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Septum of Brain; Stereotaxic Techniques | 2008 |
Anxiety-like behavior induced by histaminergic agents can be prevented by cannabinoidergic WIN55,212-2 injected into the dorsal hippocampus in mice.
Topics: Animals; Anxiety; Benzoxazines; Exploratory Behavior; Hippocampus; Histamine; Histamine Antagonists; Male; Mice; Morpholines; Naphthalenes; Piperidines; Pyrazoles; Pyrilamine; Ranitidine | 2010 |
Effect of microinjection of histamine into the dorsal hippocampus on the orofacial formalin-induced pain in rats.
Topics: Analgesics; Animals; Behavior, Animal; Facial Pain; Formaldehyde; Hippocampus; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Injections, Subcutaneous; Lip; Male; Microinjections; Pain Measurement; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H2 | 2010 |
Withdrawal from repeated administration of morphine alters histamine-induced anxiogenic effects produced by intra-ventral hippocampal microinjection.
Topics: Analysis of Variance; Animals; Anxiety; Behavior, Animal; Hippocampus; Histamine; Histamine Antagonists; Imidazoles; Male; Microinjections; Morphine; Motor Activity; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Substance Withdrawal Syndrome; Thiourea | 2010 |
Interaction of histamine and calcitonin gene-related peptide in the formalin induced pain perception in rats.
Topics: Analgesics; Animals; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Drug Interactions; Drug Therapy, Combination; Formaldehyde; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Hyperalgesia; Male; Pain; Pain Perception; Peptide Fragments; Pyrilamine; Ranitidine; Rats; Rats, Wistar | 2011 |
Influence of nitric oxide agents in the dorsal hippocampus of mice on anxiogenic-like effect induced by histamine.
Topics: Animals; Anxiety; Arginine; CA1 Region, Hippocampal; Enzyme Inhibitors; Hippocampus; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Mice; Microinjections; Motor Activity; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase Type I; Pyrilamine; Ranitidine | 2012 |
Punishing and cardiovascular effects of intravenous histamine in rats: pharmacological selectivity.
Topics: Animals; Cardiovascular System; Conditioning, Operant; Dose-Response Relationship, Drug; Heart Rate; Histamine; Histamine Antagonists; Injections, Intravenous; Ketotifen; Male; Punishment; Pyrilamine; Ranitidine; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology | 2013 |