Page last updated: 2024-08-16

pyrilamine and promethazine

pyrilamine has been researched along with promethazine in 30 studies

Research

Studies (30)

TimeframeStudies, this research(%)All Research%
pre-199023 (76.67)18.7374
1990's3 (10.00)18.2507
2000's4 (13.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Strassburg, CP; Tukey, RH1
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J1
Cooper, A; Jones, D; Major, J; Scholes, P; Walters, M; Wilde, C1
Hill, SJ; Marrian, DH; Young, JM1
Emson, PC; Hill, SJ; Young, JM1
Gárdos, G; Lassen, UV; Pape, L1
Baldo, BA; Fletcher, TC1
Bairy, KL; Kulkarni, DR; Ramesh, KV; Rao, CM1
Fujimoto, K; Fukagawa, K; Ookuma, K; Sakata, T; Shiraishi, T; Wada, H; Yoshimatsu, H1
Foxwell, MH; Johnson, DN; Kilpatrick, BF; Leonard, CA; Nolan, JC; Proakis, AG; Stephens, DJ; Yanni, JM1
Katona, PG; Rigel, DF1
Calcutt, CR; Ganellin, CR; Jackson, B; Leigh, BK; Owen, DA; Smith, IR1
Fleisch, JH; Haisch, KD; Rinkema, LE; Whitesitt, CA1
Blahd, WH; Tyan, ML1
Delini-Stula, A; Radeke, E; van Riezen, H1
Itoh, Y; Nishibori, M; Oishi, R; Saeki, K1
Katayama, S; Tasaka, K1
Wallace, RM; Young, JM1
Daum, PR; Hill, SJ; Young, JM1
Chung, YH; Kamei, C; Miyake, H; Tasaka, K1
Brown, PA; Vernikos, J1
Khodorova, AB; Nechaeva, MV; Turpaev, TM1
Bartolini, A; Galeotti, N; Ghelardini, C2
Merk, HF1
BETTINI, S; CANTORE, G1
DAS, PC; GOSWAMI, R; PHUKAN, D1
HALPERN, BN; NEVEU, T; SPECTOR, S1
BAIN, WA; BROADBENT, JL; WARIN, RP1

Reviews

2 review(s) available for pyrilamine and promethazine

ArticleYear
Human UDP-glucuronosyltransferases: metabolism, expression, and disease.
    Annual review of pharmacology and toxicology, 2000, Volume: 40

    Topics: Autoimmunity; Chromosome Mapping; Glucuronides; Glucuronosyltransferase; Humans; Hyperbilirubinemia; Neoplasms; Steroids; Terminology as Topic

2000
Standard treatment: the role of antihistamines.
    The journal of investigative dermatology. Symposium proceedings, 2001, Volume: 6, Issue:2

    Topics: Cyclizine; Cytochrome P-450 Enzyme System; Diphenhydramine; Electrocardiography; Histamine H1 Antagonists; Humans; Promethazine; Pyrilamine; Urticaria

2001

Other Studies

28 other study(ies) available for pyrilamine and promethazine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
    Journal of medicinal chemistry, 2008, Jan-24, Volume: 51, Issue:2

    Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase

2008
Characterization of an adenylate cyclase system sensitive to histamine H2-receptor excitation in cells from dog gastric mucosa.
    Agents and actions, 1976, Volume: 6, Issue:6

    Topics: Adenylyl Cyclase Inhibitors; Animals; Burimamide; Cells; Chlorpheniramine; Cyclic AMP; Dogs; Gastric Mucosa; Histamine; Histamine Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Kinetics; Methylhistamines; Metiamide; Promethazine; Pyrilamine

1976
Specific binding of 3H-mepyramine to histamine H1 receptors in intestinal smooth muscle.
    Nature, 1977, Nov-24, Volume: 270, Issue:5635

    Topics: Animals; Binding, Competitive; Chlorpheniramine; Guinea Pigs; In Vitro Techniques; Intestine, Small; Kinetics; Muscle, Smooth; Promethazine; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Triprolidine

1977
The binding of [3H]mepyramine to histamine H1 receptors in guinea-pig brain.
    Journal of neurochemistry, 1978, Volume: 31, Issue:4

    Topics: Aminopyridines; Animals; Brain; Cerebellum; Guinea Pigs; Promethazine; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1

1978
Effect of antihistamines and chlorpromazine on the calcium-induced hyperpolarization of the Amphiuma red cell membrane.
    Biochimica et biophysica acta, 1976, Nov-02, Volume: 448, Issue:4

    Topics: Animals; Biological Transport, Active; Calcimycin; Calcium; Cell Membrane Permeability; Chlorpromazine; Erythrocyte Membrane; Erythrocytes; Histamine; Membrane Potentials; Potassium; Promethazine; Pyridines; Pyrilamine; Urodela

1976
Phylogenetic aspects of hypersensitivity: immediate hypersensitivity reactions in flatfish.
    Advances in experimental medicine and biology, 1975, Volume: 64

    Topics: Animals; Antibody Formation; Biological Assay; Biological Evolution; Cromolyn Sodium; Diethylcarbamazine; Fishes; Guinea Pigs; Hypersensitivity, Immediate; Methysergide; Phylogeny; Promethazine; Pyrilamine; Rats; Species Specificity

1975
Effects of antihistamines on wound healing.
    Indian journal of experimental biology, 1991, Volume: 29, Issue:4

    Topics: Animals; Cimetidine; Female; Histamine Antagonists; Male; Promethazine; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Wound Healing

1991
Neuronal histamine modulates feeding behavior through H1-receptor in rat hypothalamus.
    The American journal of physiology, 1989, Volume: 256, Issue:3 Pt 2

    Topics: Animals; Chlorpheniramine; Cimetidine; Drinking Behavior; Famotidine; Feeding Behavior; Histamine; Histamine H2 Antagonists; Hypothalamus; Injections, Intraventricular; Male; Motor Activity; Neurons; Promethazine; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Reference Values; Thiazoles

1989
Rocastine (AHR-11325), a rapid acting, nonsedating antihistamine.
    Agents and actions, 1989, Volume: 28, Issue:1-2

    Topics: Anaphylaxis; Animals; Astemizole; Azepines; Benzhydryl Compounds; Benzimidazoles; Brompheniramine; Cats; Chlorpheniramine; Diphenhydramine; Electroencephalography; Female; Guinea Pigs; Histamine; Histamine H1 Antagonists; Ileum; Kinetics; Male; Mice; Mice, Inbred ICR; Muscle Contraction; Oxazepines; Piperazines; Promethazine; Pyrilamine; Terfenadine; Yohimbine

1989
Effects of antihistamines and local anesthetics on excess tachycardia in conscious dogs.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:1

    Topics: Anesthetics, Local; Animals; Atropine; Chlorpheniramine; Diphenhydramine; Dogs; Dose-Response Relationship, Drug; Histamine; Histamine H1 Antagonists; Lidocaine; Male; Procaine; Promethazine; Pyrilamine; Tachycardia

1986
Evidence for low brain penetration by the H1-receptor antagonist temelastine (SK&F 93944).
    European journal of pharmacology, 1987, Jan-06, Volume: 133, Issue:1

    Topics: Animals; Brain; Dose-Response Relationship, Drug; Histamine H1 Antagonists; In Vitro Techniques; Male; Mice; Motor Activity; Promethazine; Pyrilamine; Pyrimidinones; Receptors, Histamine H1; Tritium

1987
Pharmacologic analysis of LY188695 (KB-2413), 1-(2-ethoxyethyl)-2-(4-methyl-1-homopiperazinyl)-benzimidazole difumarate, a potent histamine1 receptor antagonist.
    Agents and actions, 1987, Volume: 20, Issue:1-2

    Topics: Animals; Benzhydryl Compounds; Benzimidazoles; Bronchial Provocation Tests; Chlorpheniramine; Diphenhydramine; Guinea Pigs; Histamine H1 Antagonists; Lung; Male; Muscle, Smooth; Promethazine; Pyrilamine; Terfenadine; Triprolidine

1987
Effects of H1 blocking agents on age-related osteopenia in the mouse.
    Mechanisms of ageing and development, 1987, Volume: 38, Issue:3

    Topics: Aging; Animals; Bone and Bones; Bone Diseases, Metabolic; Dimenhydrinate; Female; Histamine H1 Antagonists; Meclizine; Mice; Mice, Inbred Strains; Promethazine; Pyrilamine

1987
Enhanced functional responsiveness of the dopaminergic system--the mechanism of anti-immobility effects of antidepressants in the behavioural despair test in the rat.
    Neuropharmacology, 1988, Volume: 27, Issue:9

    Topics: Animals; Antidepressive Agents; Immobilization; Male; Motor Activity; Prazosin; Promethazine; Pyrilamine; Rats; Sulpiride

1988
Mechanism of the central hyperglycemic action of histamine in mice.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:2

    Topics: Adrenalectomy; Animals; Blood Glucose; Chlorpheniramine; Chromatography, High Pressure Liquid; Corticosterone; Dose-Response Relationship, Drug; Epinephrine; Histamine; Hyperglycemia; Mice; Norepinephrine; Phentolamine; Promethazine; Propranolol; Pyrilamine; Pyrimethamine; Receptors, Histamine H1; Receptors, Histamine H2; Time Factors

1987
Effects of H1-receptor blocking drugs on the frog sartorius neuromuscular junction.
    British journal of pharmacology, 1985, Volume: 85, Issue:4

    Topics: Action Potentials; Aminopyridines; Animals; Diphenhydramine; Dose-Response Relationship, Drug; Electric Conductivity; Electrophysiology; Membrane Potentials; Neuromuscular Junction; Perfusion; Promethazine; Pyrilamine; Ranidae; Receptors, Histamine; Receptors, Histamine H1; Time Factors

1985
Temperature dependence of the binding of [3H]mepyramine and related compounds to the histamine H1 receptor.
    Molecular pharmacology, 1983, Volume: 23, Issue:1

    Topics: Aminopyridines; Animals; Cerebellum; Chlorpromazine; Guinea Pigs; Histamine H1 Antagonists; Kinetics; Male; Phenothiazines; Promethazine; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Temperature; Tripelennamine

1983
Histamine H1-agonist potentiation of adenosine-stimulated cyclic AMP accumulation in slices of guinea-pig cerebral cortex: comparison of response and binding parameters.
    British journal of pharmacology, 1982, Volume: 77, Issue:2

    Topics: Adenosine; Animals; Brain; Cyclic AMP; Female; Guinea Pigs; Histamine; In Vitro Techniques; Male; Promethazine; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2

1982
Analgesic effect of histamine induced by intracerebral injection into mice.
    Agents and actions, 1984, Volume: 15, Issue:3-4

    Topics: Analgesics; Animals; Benzoquinones; Cimetidine; Diphenhydramine; Electric Stimulation; Enkephalin, Leucine; Histamine; Histamine Antagonists; Male; Mice; Mice, Inbred Strains; Morphine; Naloxone; Promethazine; Pyrilamine; Quinones; Reaction Time

1984
Antihistamine effect on synaptosomal uptake of serotonin, norepinephrine and dopamine.
    European journal of pharmacology, 1980, Jul-11, Volume: 65, Issue:1

    Topics: Animals; Cimetidine; Diphenhydramine; Dopamine; Female; Histamine Antagonists; In Vitro Techniques; Kinetics; Norepinephrine; Promethazine; Pyrilamine; Rats; Serotonin; Synaptosomes

1980
[Possible involvement of histamine in humoral regulation of the spontaneous contractile activity of the chick embryo amnion].
    Doklady Akademii nauk, 1997, Volume: 355, Issue:2

    Topics: Amnion; Animals; Chick Embryo; Cimetidine; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Muscle Contraction; Muscle, Smooth; Promethazine; Pyrilamine

1997
The role of potassium channels in antihistamine analgesia.
    Neuropharmacology, 1999, Volume: 38, Issue:12

    Topics: Animals; Diphenhydramine; Drug Synergism; Histamine H1 Antagonists; Ion Channel Gating; Male; Mice; Oligonucleotides, Antisense; Pain Measurement; Pertussis Toxin; Potassium Channels; Promethazine; Pyrilamine; Virulence Factors, Bordetella

1999
Antihistamine antinociception is mediated by Gi-protein activation.
    Neuroscience, 2002, Volume: 109, Issue:4

    Topics: Analgesics; Animals; Behavior, Animal; Central Nervous System; Diphenhydramine; Dose-Response Relationship, Drug; Drug Interactions; GTP-Binding Protein alpha Subunits, Gi-Go; Histamine H1 Antagonists; Male; Mice; Motor Activity; Neurons; Nociceptors; Oligodeoxyribonucleotides, Antisense; Pain; Pain Threshold; Promethazine; Pyrilamine; Receptors, Histamine H1; Synaptic Transmission

2002
[Protective action of ACTH, cortisone, calcium gluconate, pyrilamine (neoantergan), promethazine (fargan), and chlorpromazine (largactil) against experimental poisoning with Latrodectus venom in guinea pigs].
    Rendiconti - Istituto superiore di sanita, 1955, Volume: 18, Issue:6

    Topics: Adrenocorticotropic Hormone; Antipsychotic Agents; Calcium Gluconate; Chlorpromazine; Cortisone; Gluconates; Guinea Pigs; Phenothiazines; Poisoning; Promethazine; Pyrilamine; Venoms

1955
Local anesthetic action of antihistaminics (promethazine hydrochloride and mepyramine maleate).
    Indian journal of medical sciences, 1958, Volume: 12, Issue:2

    Topics: Anesthetics, Local; Histamine H1 Antagonists; Promethazine; Pyrilamine

1958
On the nature of the chemical mediators involved in anaphylactic reactions in mice.
    British journal of pharmacology and chemotherapy, 1963, Volume: 20

    Topics: Anaphylaxis; Animals; Anti-Allergic Agents; Capillary Permeability; Chlorpromazine; Histamine; Histamine H1 Antagonists; Lysergic Acid Diethylamide; Mice; Passive Cutaneous Anaphylaxis; Promethazine; Pyrilamine; Serotonin

1963
Comparison of anthisan (mepyramine maleate) and phenergan as histamine antagonists.
    Lancet (London, England), 1949, Jul-09, Volume: 2, Issue:6567

    Topics: Histamine; Histamine Antagonists; Promethazine; Pyrilamine

1949