Page last updated: 2024-08-16

pyrilamine and procaine

pyrilamine has been researched along with procaine in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19908 (61.54)18.7374
1990's1 (7.69)18.2507
2000's3 (23.08)29.6817
2010's1 (7.69)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Caron, G; Ermondi, G1
Ahman, M; Holmén, AG; Wan, H1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Gupta, VD; Shek, OH1
Finch, L; Hicks, PE1
Haranath, PS; Indira-Narayan, G; Venkatakrishna-Bhatt, H1
Amann, R; Barthó, L; Lembeck, F1
White, JM1
Katona, PG; Rigel, DF1
Kawasaki, H; Takasaki, K1
Horio, S; Ishida, Y; Moritoki, H; Nagare, T1
Fu, LW; Longhurst, JC; Phan, A1

Other Studies

13 other study(ies) available for pyrilamine and procaine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Calculating virtual log P in the alkane/water system (log P(N)(alk)) and its derived parameters deltalog P(N)(oct-alk) and log D(pH)(alk).
    Journal of medicinal chemistry, 2005, May-05, Volume: 48, Issue:9

    Topics: 1-Octanol; Alkanes; Hydrogen-Ion Concentration; Least-Squares Analysis; Mathematics; Models, Chemical; Models, Molecular; Solvents; Water

2005
Relationship between brain tissue partitioning and microemulsion retention factors of CNS drugs.
    Journal of medicinal chemistry, 2009, Mar-26, Volume: 52, Issue:6

    Topics: Brain; Central Nervous System; Chromatography, Liquid; Emulsions; Mass Spectrometry

2009
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Comparison of stability-indicating assay methods: ultraviolet, high pressure liquid chromatography and acid dye.
    American journal of hospital pharmacy, 1976, Volume: 33, Issue:10

    Topics: Chromatography, High Pressure Liquid; Codeine; Coloring Agents; Drug Stability; Ephedrine; Fluorometry; Methods; Morphine; Procaine; Pyrilamine; Spectrophotometry, Ultraviolet; Thiamine

1976
No evidence for central histamine-receptor involvement with the hypotensive effect of clonidine in cats.
    European journal of pharmacology, 1976, Volume: 40, Issue:2

    Topics: Animals; Behavior, Animal; Blood Pressure; Cats; Clonidine; Injections, Intraventricular; Metiamide; Phentolamine; Procaine; Pyrilamine; Receptors, Histamine; Tolazoline

1976
Pressor response induced by local anaesthetics perfused through the cerebral ventricles of dogs.
    British journal of pharmacology, 1975, Volume: 55, Issue:1

    Topics: Adrenal Glands; Adrenalectomy; Anesthetics, Local; Animals; Blood Pressure; Carotid Sinus; Denervation; Dogs; Ethylenediamines; Hexamethonium Compounds; Injections, Intraventricular; Perfusion; Phentolamine; Procaine; Pyridines; Pyrilamine; Time Factors

1975
Studies on effects of the substance P analogues [D-Pro2, D-Trp7,9]-substance P and [D-Arg1, D-Trp7,9, L-Leu11]-substance P not related to their antagonist action.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 333, Issue:3

    Topics: Acetylcholine; Animals; Blood Pressure; Guinea Pigs; Histamine Release; In Vitro Techniques; Muscle Contraction; Neuropeptides; Nociceptors; Procaine; Pyrilamine; Rabbits; Regional Blood Flow; Substance P; Tachykinins

1986
The discriminative stimulus properties of mepyramine.
    Life sciences, 1985, Sep-23, Volume: 37, Issue:12

    Topics: Aminopyridines; Animals; Chlorpheniramine; Discrimination, Psychological; Histamine H1 Antagonists; Imipramine; Male; Procaine; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Scopolamine

1985
Effects of antihistamines and local anesthetics on excess tachycardia in conscious dogs.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:1

    Topics: Anesthetics, Local; Animals; Atropine; Chlorpheniramine; Diphenhydramine; Dogs; Dose-Response Relationship, Drug; Histamine; Histamine H1 Antagonists; Lidocaine; Male; Procaine; Promethazine; Pyrilamine; Tachycardia

1986
Central alpha-2 adrenoceptor-mediated hypertensive response to clonidine in conscious, normotensive rats.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 236, Issue:3

    Topics: Animals; Azepines; Blood Pressure; Brain; Cimetidine; Clonidine; Hydroxydopamines; Injections, Intraventricular; Ketanserin; Male; Methoxamine; Oxidopamine; Piperidines; Prazosin; Procaine; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1986
Interaction of local anaesthetics with histamine H1 receptors in guinea-pig ileum.
    The Journal of pharmacy and pharmacology, 1997, Volume: 49, Issue:7

    Topics: Anesthetics, Local; Animals; Binding, Competitive; Chloroquine; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine H1 Antagonists; Ileum; Isotope Labeling; Male; Muscle Contraction; Muscle, Smooth; Procaine; Pyrilamine; Quinacrine; Receptors, Histamine H1; Structure-Activity Relationship; Tetracaine

1997
Myocardial ischemia-mediated excitatory reflexes: a new function for thromboxane A2?
    American journal of physiology. Heart and circulatory physiology, 2008, Volume: 295, Issue:6

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Anesthetics, Local; Animals; Cats; Disease Models, Animal; Dose-Response Relationship, Drug; Female; Heart; Hemodynamics; Histamine H1 Antagonists; Indoles; Kidney; Male; Myocardial Ischemia; Pressoreceptors; Procaine; Pyrilamine; Receptors, Thromboxane; Reflex; Serotonin Antagonists; Sulfonamides; Sympathetic Nervous System; Thromboxane A2; Tropisetron; Vagotomy

2008