Page last updated: 2024-08-16

pyrilamine and leukotriene d4

pyrilamine has been researched along with leukotriene d4 in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (61.54)18.2507
2000's3 (23.08)29.6817
2010's2 (15.38)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K1
Carmody, LC; Dandapani, S; Donckele, E; Feng, Y; Fernandez, C; Germain, AR; Gupta, PB; Lander, ES; Morgan, B; Munoz, B; Nag, PP; Palmer, M; Perez, JR; Schreiber, SL; Verplank, L1
Ellis, JL; Hubbard, WC; Lichtenstein, LM; Meeker, S; Undem, BJ1
Sato, F; Timmerman, H; Wada, Y; Zhang, MQ1
Langer, JC; Liebman, SM; Monk, PK; Pelletier, GJ1
Bochnowicz, S; Underwood, DC1
Brideau, C; Chan, CC; Ho, E; Rodger, IW; Savoie, C; Tousignant, C1
Kadowaki, S; Nakao, E; Takahashi, K; Umezu, K; Yamada, K; Yamada, N1
Ellis, JL; Undem, BJ1
Takami, M; Tsukada, W1
Belvisi, MG; Birrell, MA; Foster, ML; Hele, DJ; Webber, SE1
Kohno, S; Mizutani, N; Nabe, T; Osaki, S; Sugahara, S; Takenaka, H1
Dahlén, SE; Låstbom, L; Ryrfeldt, A; Sundström, E1

Other Studies

13 other study(ies) available for pyrilamine and leukotriene d4

ArticleYear
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship

2010
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.
    Bioorganic & medicinal chemistry letters, 2013, Mar-15, Volume: 23, Issue:6

    Topics: Amides; Breast Neoplasms; Cell Line, Tumor; Drug Screening Assays, Antitumor; Female; Humans; Neoplastic Stem Cells; Small Molecule Libraries; Structure-Activity Relationship

2013
Recombinant stem cell factor-induced mast cell activation and smooth muscle contraction in human bronchi.
    American journal of respiratory cell and molecular biology, 1994, Volume: 11, Issue:6

    Topics: Antibodies, Anti-Idiotypic; Autacoids; Bronchi; Carbachol; Dicarboxylic Acids; Hematopoietic Cell Growth Factors; Histamine Antagonists; Humans; Immunoglobulin E; In Vitro Techniques; Leukotriene D4; Mast Cells; Muscle Contraction; Muscle, Smooth; Pyrilamine; Recombinant Proteins; Stem Cell Factor

1994
(Piperidinylalkoxy)chromones: novel antihistamines with additional antagonistic activity against leukotriene D4.
    Journal of medicinal chemistry, 1995, Jun-23, Volume: 38, Issue:13

    Topics: Animals; Capillary Permeability; Cerebral Cortex; Chromones; Drug Antagonism; Guinea Pigs; Histamine H1 Antagonists; Ileum; In Vitro Techniques; Leukotriene D4; Lung; Mice; Muscle Contraction; Pyrilamine

1995
Mast cell mediators and peritoneal adhesion formation in the rat.
    The Journal of surgical research, 1995, Volume: 59, Issue:3

    Topics: Animals; Azepines; Disease Models, Animal; Histamine Antagonists; Leukotriene D4; Male; Mast Cells; Methysergide; Ondansetron; Peritoneal Diseases; Platelet Activating Factor; Propionates; Pyrilamine; Quinolines; Ranitidine; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Tissue Adhesions; Triazoles

1995
Dose-dependent mediation of leukotriene D4-induced airway microvascular leakage and bronchoconstriction in the guinea pig.
    Prostaglandins, leukotrienes, and essential fatty acids, 1995, Volume: 52, Issue:6

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Bridged Bicyclo Compounds, Heterocyclic; Bronchi; Bronchoconstriction; Capillary Permeability; Chromones; Fatty Acids, Unsaturated; Furans; Guinea Pigs; Hydrazines; Hydroxyurea; Leukotriene D4; Lipoxygenase Inhibitors; Lung; Male; Meclofenamic Acid; Plasma; Prostaglandin Endoperoxides, Synthetic; Pyrilamine; Receptors, Thromboxane; SRS-A; Thromboxane A2; Trachea; Vasoconstrictor Agents

1995
Evaluation of bronchoconstriction induced by neurokinins and its inhibition by selective nonpeptide antagonists in conscious guinea pigs, using a double-chamber plethysmograph technique.
    Canadian journal of physiology and pharmacology, 1994, Volume: 72, Issue:1

    Topics: Airway Resistance; Animals; Benzamides; Bronchoconstriction; Bronchodilator Agents; Guinea Pigs; Histamine; Indomethacin; Leukotriene D4; Male; Neurokinin A; Parasympatholytics; Piperidines; Plethysmography; Propionates; Pyrilamine; Quinolines

1994
Pharmacological profile of the novel, potent and selective peptide leukotriene antagonist (E)-2,2-diethyl-3'-[2-[2-(4-isopropyl)thiazolyl]ethenyl]succinanilic acid.
    Arzneimittel-Forschung, 1994, Volume: 44, Issue:6

    Topics: Acetylcholine; Animals; Bronchodilator Agents; Dose-Response Relationship, Drug; Guinea Pigs; Histamine Antagonists; Ileum; In Vitro Techniques; Leukotriene Antagonists; Leukotriene C4; Leukotriene D4; Male; Muscle Contraction; Muscle, Smooth; Penicillin G; Pyrilamine; Thiazoles; Trachea

1994
Role of cysteinyl-leukotrienes and histamine in mediating intrinsic tone in isolated human bronchi.
    American journal of respiratory and critical care medicine, 1994, Volume: 149, Issue:1

    Topics: Bronchi; Chlorpheniramine; Dicarboxylic Acids; Female; Histamine; Humans; Hydroxyurea; In Vitro Techniques; Indazoles; Isometric Contraction; Isotonic Solutions; Leukotriene D4; Lipoxygenase Inhibitors; Male; Middle Aged; Muscle Tonus; Muscle, Smooth; Pyrilamine; SRS-A

1994
Effect of DP-1904, a thromboxane synthetase inhibitor, on antigen- and spasmogen-induced bronchoconstriction in rodents.
    European journal of pharmacology, 1999, Feb-05, Volume: 366, Issue:2-3

    Topics: Acetylcholine; Animals; Antigens; Arachidonic Acid; Bradykinin; Bronchoconstriction; Bronchoconstrictor Agents; Enzyme Inhibitors; Guinea Pigs; Histamine; Histamine H1 Antagonists; Imidazoles; Indomethacin; Leukotriene D4; Male; Methacrylates; Platelet Activating Factor; Pyrilamine; Rats; Rats, Sprague-Dawley; Tetrahydronaphthalenes; Thromboxane-A Synthase

1999
Mediator involvement in antigen-induced bronchospasm and microvascular leakage in the airways of ovalbumin sensitized Brown Norway rats.
    British journal of pharmacology, 2001, Volume: 132, Issue:2

    Topics: Acetates; Animals; Anti-Asthmatic Agents; Bronchi; Bronchial Spasm; Capillary Permeability; Cyclopropanes; Histamine; Histamine H1 Antagonists; Leukotriene D4; Male; Methysergide; Ovalbumin; Pyrilamine; Quinolines; Rats; Rats, Inbred BN; Respiratory Hypersensitivity; Serotonin; Serotonin Antagonists; Sulfides; Trachea

2001
Comparison of cedar pollen-induced allergic rhinitis in passively and actively sensitized guinea pigs.
    Japanese journal of pharmacology, 2001, Volume: 85, Issue:4

    Topics: Airway Resistance; Animals; Guinea Pigs; Histamine; Histamine H1 Antagonists; Immunization, Passive; Leukotriene D4; Male; Nasal Provocation Tests; Pollen; Pyrilamine; Rhinitis, Allergic, Seasonal; Sneezing; Trees; Vaccination

2001
Interactions among three classes of mediators explain antigen-induced bronchoconstriction in the isolated perfused and ventilated guinea pig lung.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 307, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Bronchoconstriction; Cysteine; Drug Interactions; Guinea Pigs; Histamine; Histamine Antagonists; Leukotriene D4; Leukotrienes; Lung; Male; Ovalbumin; Perfusion; Pyrilamine; Thromboxanes

2003