Page last updated: 2024-08-16

pyrilamine and impromidine

pyrilamine has been researched along with impromidine in 29 studies

Research

Studies (29)

TimeframeStudies, this research(%)All Research%
pre-199022 (75.86)18.7374
1990's5 (17.24)18.2507
2000's2 (6.90)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Timmerman, H1
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM1
Anjelkovic, IZ; Collis, CS; Djuric, D; Rosic, M; Segal, MB; Zlokovic, BV1
Arrang, JM; Garbarg, M; Schwartz, JC1
Edvinsson, L; Jansen, I; Ottosson, A1
Trzeciakowski, JP1
Männistö, PT; Mattila, J; Tuominen, RK2
Ledgard, SE; Nieves, AL; Woodward, DF1
Bugajski, J; Gadek, A1
Iwata, M; Kohno, S; Shigei, T; Tsuru, H1
Abacioğlu, N; Demiryürek, T; Ercan, ZS; Kanzik, L; Türker, RK; Zengil, H1
Dhawan, KN; Gulati, A; Gupta, GP; Nath, C1
Ea-Kim, L; Oudart, N1
Donaldson, J; Hill, SJ1
Bohm, U; Falus, A; Fekete, MI; Meretey, K1
Oriowo, MA1
Heldsinger, AA; Skoglund, ML; Vinik, AI1
Koo, A1
Guth, PH; Hirabayashi, K1
Bugajski, J; Janusz, Z1
Bank, L; Bortz, D; Lipschitz, E; Marks, IN1
Kusunoki, M; Tanaka, C; Taniyama, K1
Arrang, JM; Duchemin, AM; Garbarg, M; Quach, TT; Rose, C; Schwartz, JC1
Curwain, BP; Turner, NC1
Akaike, N; Munakata, M1
Jouvet, M; Lin, JS; Sakai, K1
Jafri, MS; Moore, KA; Taylor, GE; Weinreich, D1
Buschauer, A; Schalkhausser, F; Seifert, R; Xie, SX; Ye, QZ1

Reviews

1 review(s) available for pyrilamine and impromidine

ArticleYear
Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:1

    Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship

1990

Trials

1 trial(s) available for pyrilamine and impromidine

ArticleYear
Effect of mepyramine on the untoward side-effects of impromidine.
    South African medical journal = Suid-Afrikaanse tydskrif vir geneeskunde, 1984, Aug-18, Volume: 66, Issue:7

    Topics: Aminopyridines; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Drug Interactions; Female; Flushing; Gastric Acid; Humans; Imidazoles; Impromidine; Male; Middle Aged; Pulse; Pyrilamine; Random Allocation; Receptors, Histamine; Receptors, Histamine H2

1984

Other Studies

27 other study(ies) available for pyrilamine and impromidine

ArticleYear
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4

2005
The effects of (R) alpha-methyl histamine on the isolated guinea pig aorta.
    Agents and actions. Supplements, 1991, Volume: 33

    Topics: Animals; Aorta; Cimetidine; Female; Guanidines; Guinea Pigs; Histamine; Histamine Antagonists; Imidazoles; Impromidine; Male; Methylhistamines; Muscle, Smooth, Vascular; Potassium; Pyrilamine; Receptors, Histamine; Receptors, Histamine H3; Vasoconstriction; Vasodilation

1991
Autoinhibition of histamine synthesis mediated by presynaptic H3-receptors.
    Neuroscience, 1987, Volume: 23, Issue:1

    Topics: Animals; Burimamide; Cerebral Cortex; Cimetidine; Histamine; Histamine Release; Hypothalamus; Hypothalamus, Posterior; Imidazoles; Impromidine; Male; Potassium; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H3; Synaptosomes; Thiazoles

1987
Pharmacological characterization of histamine receptors in the human temporal artery.
    British journal of clinical pharmacology, 1989, Volume: 27, Issue:2

    Topics: Adult; Cimetidine; Dinoprost; Female; Histamine; Humans; Imidazoles; Impromidine; In Vitro Techniques; Male; Methylhistamines; Middle Aged; Pyridines; Pyrilamine; Receptors, Histamine; Temporal Arteries; Thiazoles; Vasoconstriction; Vasodilation

1989
Inhibition of guinea pig ileum contractions mediated by a class of histamine receptor resembling the H3 subtype.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 243, Issue:3

    Topics: Animals; Dose-Response Relationship, Drug; Electric Stimulation; Female; Guinea Pigs; Histamine; Ileum; Imidazoles; Impromidine; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Pyrilamine; Receptors, Histamine; Receptors, Histamine H3

1987
Studies on the site and mechanism of the inhibitory action of intracerebral histamine on the cold-stimulated thyrotropin secretion in male rats.
    Brain research, 1985, Sep-23, Volume: 343, Issue:2

    Topics: Animals; Brain Mapping; Cimetidine; Cold Temperature; Histamine; Hypothalamus; Imidazoles; Impromidine; Injections, Intraventricular; Male; Pyridines; Pyrilamine; Rats; Thyrotropin

1985
Conjunctival immediate hypersensitivity: re-evaluation of histamine involvement in the vasopermeability response.
    Investigative ophthalmology & visual science, 1986, Volume: 27, Issue:1

    Topics: Albumins; Animals; Capillary Permeability; Cimetidine; Conjunctiva; Dimaprit; Dose-Response Relationship, Drug; Drug Combinations; Eyelids; Guinea Pigs; Histamine; Histamine Antagonists; Hypersensitivity, Immediate; Imidazoles; Impromidine; Male; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1986
Hyperlipemic responses induced by centrally administered histamine H1- and H2-receptor agonists in rats.
    Agents and actions, 1987, Volume: 20, Issue:3-4

    Topics: Animals; Brain; Cimetidine; Dimaprit; Fatty Acids, Nonesterified; Hyperlipidemias; Imidazoles; Impromidine; Injections, Intraventricular; Male; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Thiourea

1987
Characterization of histamine receptors in isolated rabbit veins.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 243, Issue:2

    Topics: Animals; Cimetidine; Endothelium, Vascular; Female; Histamine; Imidazoles; Impromidine; Male; Pyrilamine; Rabbits; Ranitidine; Receptors, Histamine; Receptors, Histamine H2; Species Specificity; Vasoconstriction; Veins

1987
Endothelium-dependent relaxing effect of histamine on the isolated guinea-pig main pulmonary artery strips.
    Agents and actions, 1987, Volume: 22, Issue:1-2

    Topics: Animals; Cimetidine; Endothelium, Vascular; Female; Guinea Pigs; Histamine; Imidazoles; Impromidine; In Vitro Techniques; Male; Muscle Relaxation; Pulmonary Artery; Pyrilamine; Receptors, Histamine H2

1987
Role of central histaminergic mechanism in behavioural depression (swimming despair) in mice.
    Life sciences, 1988, Volume: 42, Issue:24

    Topics: Animals; Atropine; Central Nervous System; Cimetidine; Depression; Desipramine; Disease Models, Animal; Histamine; Imidazoles; Imipramine; Impromidine; Male; Mice; Motor Activity; Pyrilamine; Receptors, Histamine H2

1988
A highly potent and selective H3 agonist relaxes rabbit middle cerebral artery, in vitro.
    European journal of pharmacology, 1988, Jun-10, Volume: 150, Issue:3

    Topics: Animals; Cerebral Arteries; Cimetidine; Histamine; Imidazoles; Impromidine; In Vitro Techniques; Male; Methylhistamines; Muscle Relaxation; Muscle, Smooth, Vascular; Potassium; Pyrilamine; Rabbits; Receptors, Histamine

1988
Histamine-induced inositol phospholipid breakdown in the longitudinal smooth muscle of guinea-pig ileum.
    British journal of pharmacology, 1985, Volume: 85, Issue:2

    Topics: Animals; Cerebellum; Cimetidine; Female; Guinea Pigs; Histamine; Ileum; Imidazoles; Impromidine; In Vitro Techniques; Inositol Phosphates; Kinetics; Male; Muscle Contraction; Phosphatidylinositols; Pyrilamine

1985
Effect of H1 and H2 agonists on the chemiluminescence of human blood mononuclear cells induced by phytohaemagglutinin.
    Immunopharmacology, 1985, Volume: 9, Issue:3

    Topics: Cimetidine; Histamine; Humans; Imidazoles; Impromidine; Luminescent Measurements; Methylhistamines; Monocytes; Phytohemagglutinins; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Structure-Activity Relationship

1985
An inhibitory effect of histamine on the rat anococcygeus muscle.
    The Journal of pharmacy and pharmacology, 1982, Volume: 34, Issue:3

    Topics: Acetylcholine; Animals; Carbachol; Cimetidine; Dimaprit; Drug Interactions; Guanidines; Histamine; Imidazoles; Impromidine; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Pyrilamine; Rats; Thiourea

1982
Evidence for histamine H1 and H2 receptors in guinea-pig oxyntic cells.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:1

    Topics: Animals; Carbonic Anhydrases; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Impromidine; In Vitro Techniques; Methylhistamines; Parietal Cells, Gastric; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1983
In vivo characterization of histamine H1- and H2-receptors in the rat stomach microcirculation.
    British journal of pharmacology, 1983, Volume: 78, Issue:1

    Topics: Animals; Cimetidine; Imidazoles; Impromidine; Kinetics; Male; Microcirculation; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Stomach

1983
The effect of histamine on microvascular permeability in the muscularis externa of rat small intestine.
    Microvascular research, 1983, Volume: 25, Issue:3

    Topics: Animals; Capillary Permeability; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Imidazoles; Impromidine; Intestine, Small; Male; Microscopy, Fluorescence; Muscle, Smooth; Pyrilamine; Rats; Rats, Inbred Strains

1983
Inhibition of the TSH secretion by histamine in male rats.
    Acta endocrinologica, 1983, Volume: 103, Issue:1

    Topics: Animals; Cimetidine; Cold Temperature; Histamine; Histamine Antagonists; Histidine; Imidazoles; Impromidine; Male; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thyrotropin; Thyrotropin-Releasing Hormone

1983
Central histaminergic stimulation of pituitary--adrenocortical response in the rat.
    Life sciences, 1983, Sep-19, Volume: 33, Issue:12

    Topics: Animals; Cimetidine; Corticosterone; Dimaprit; Dose-Response Relationship, Drug; Histamine; Imidazoles; Impromidine; Male; Pituitary-Adrenal System; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1983
Inhibitory histamine H2-receptor in the guinea-pig urinary bladder.
    European journal of pharmacology, 1984, Oct-01, Volume: 105, Issue:1-2

    Topics: Acetylcholine; Animals; Calcium; Choline; Cimetidine; Diphenhydramine; Electric Stimulation; Female; Guinea Pigs; Histamine; Imidazoles; Impromidine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nicotine; Norepinephrine; Pyrilamine; Receptors, Histamine; Receptors, Histamine H2; Scopolamine; Tetrodotoxin; Urinary Bladder

1984
Histamine-induced responses in mammalian brain slices: characterization of H1 and H2 receptors.
    Advances in biochemical psychopharmacology, 1983, Volume: 37

    Topics: Animals; Brain; Chlorpheniramine; Cyclic AMP; Glycogen; Guinea Pigs; Hippocampus; Imidazoles; Impromidine; In Vitro Techniques; Kinetics; Mice; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2

1983
Comparison of the agonist activity of impromidine (SK & F 92676) in anaesthetized rabbits and on the rabbit isolated fundic mucosa.
    British journal of pharmacology, 1981, Volume: 73, Issue:4

    Topics: Animals; Dose-Response Relationship, Drug; Gastric Acid; Gastric Fundus; Gastric Mucosa; Guanidines; Histamine; Imidazoles; Impromidine; Male; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H2

1981
Regulation of K+ conductance by histamine H1 and H2 receptors in neurones dissociated from rat neostriatum.
    The Journal of physiology, 1994, Oct-15, Volume: 480 ( Pt 2)

    Topics: Animals; Cimetidine; Dose-Response Relationship, Drug; Famotidine; Female; Histamine; Histamine Agonists; Impromidine; In Vitro Techniques; Ion Transport; Male; Membrane Potentials; Methylhistamines; Neostriatum; Potassium; Potassium Channels; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Triprolidine

1994
Hypothalamo-preoptic histaminergic projections in sleep-wake control in the cat.
    The European journal of neuroscience, 1994, Apr-01, Volume: 6, Issue:4

    Topics: Animals; Brain; Cats; Dose-Response Relationship, Drug; Electroencephalography; Female; Histamine; Histidine Decarboxylase; Hypothalamus, Anterior; Impromidine; Male; Methylhistidines; Microinjections; Preoptic Area; Pyrilamine; Sleep; Sleep, REM; Time Factors; Wakefulness

1994
Histamine H1 receptor activation blocks two classes of potassium current, IK(rest) and IAHP, to excite ferret vagal afferents.
    The Journal of physiology, 1997, Sep-15, Volume: 503 ( Pt 3)

    Topics: Action Potentials; Animals; Diphenhydramine; Electric Conductivity; Ferrets; Histamine; Histamine Agonists; Histamine H1 Antagonists; Impromidine; Male; Methylhistamines; Neurons, Afferent; Nodose Ganglion; Patch-Clamp Techniques; Potassium; Potassium Channel Blockers; Pyrilamine; Receptors, Histamine H1; Thiazoles; Vagus Nerve

1997
Effects of impromidine- and arpromidine-derived guanidines on recombinant human and guinea pig histamine H1 and H2 receptors.
    Archiv der Pharmazie, 2007, Volume: 340, Issue:1

    Topics: Animals; Binding, Competitive; Cell Line; GTP Phosphohydrolases; GTP-Binding Protein alpha Subunits, Gq-G11; GTP-Binding Protein alpha Subunits, Gs; Guanidines; Guinea Pigs; Histamine Agonists; Histamine H1 Antagonists; Humans; Imidazoles; Impromidine; Insecta; Molecular Structure; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Recombinant Fusion Proteins; Structure-Activity Relationship; Transfection

2007