Page last updated: 2024-08-16

pyrilamine and dizocilpine maleate

pyrilamine has been researched along with dizocilpine maleate in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (12.50)18.2507
2000's3 (37.50)29.6817
2010's4 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Anzini, M; Brogi, S; Butini, S; Campiani, G; Cappelli, A; Caselli, G; Castriconi, F; Gemma, S; Giordani, A; Giorgi, G; Giuliani, G; Lanza, M; Letari, O; Makovec, F; Manini, M; Mennuni, L; Valenti, S1
Belyakov, S; Dambrova, M; Kazoka, H; Kuznecovs, J; Lebedev, A; Liepinsh, E; Mishnev, A; Orlova, N; Ponomaryov, Y; Vavers, E; Veinberg, G; Vikainis, S; Vilskersts, R; Vorona, M; Zvejniece, L1
Díaz-Trelles, R; Fernández-Sánchez, MT; Novelli, A; Puia, G1
Fujii, Y; Kamei, C; Nishiga, M; Sugimoto, Y; Taga, C1
Chen, Z; Hu, WW; Liu, LY; Ma, L; Wei, EQ; Xu, LS; Yang, LX; Yu, X1
Hao, X; Levin, ED; Perraut, C; Roegge, CS1
Arrang, JM; Burban, A; Davenas, E; Motawaj, M1
Darras, FH; Decker, M; Khan, N; Nurulain, SM; Saad, A; Sadek, B1

Other Studies

8 other study(ies) available for pyrilamine and dizocilpine maleate

ArticleYear
Synthesis and structure-activity relationship studies in serotonin 5-HT(1A) receptor agonists based on fused pyrrolidone scaffolds.
    European journal of medicinal chemistry, 2013, Volume: 63

    Topics: Animals; Area Under Curve; Humans; Intestinal Absorption; Ligands; Male; Metabolic Clearance Rate; Models, Chemical; Models, Molecular; Molecular Structure; Protein Binding; Protein Structure, Tertiary; Pyrrolidinones; Radioligand Assay; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin, 5-HT3; Serotonin 5-HT1 Receptor Agonists; Structure-Activity Relationship

2013
Synthesis and biological evaluation of 2-(5-methyl-4-phenyl-2-oxopyrrolidin-1-yl)-acetamide stereoisomers as novel positive allosteric modulators of sigma-1 receptor.
    Bioorganic & medicinal chemistry, 2013, May-15, Volume: 21, Issue:10

    Topics: Acetamides; Allosteric Regulation; Animals; Rats; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism; Structure-Activity Relationship

2013
Terfenadine prevents NMDA receptor-dependent and -independent toxicity following sodium channel activation.
    Brain research, 1999, Sep-25, Volume: 842, Issue:2

    Topics: Animals; Cell Survival; Cells, Cultured; Cerebellum; Dizocilpine Maleate; Glutamic Acid; Neurons; Pyrilamine; Rats; Receptors, N-Methyl-D-Aspartate; Saxitoxin; Sodium Channels; Terfenadine; Tetrodotoxin; Veratridine

1999
Effects of the NMDA antagonist MK-801 on radial maze performance in histidine-deficient rats.
    Life sciences, 2002, Mar-22, Volume: 70, Issue:18

    Topics: Amino Acids; Animals; Brain; Diet; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Histamine H1 Antagonists; Histidine; Male; Maze Learning; Memory Disorders; Pyrilamine; Rats; Rats, Wistar; Scopolamine

2002
Histamine ameliorates spatial memory deficits induced by MK-801 infusion into ventral hippocampus as evaluated by radial maze task in rats.
    Acta pharmacologica Sinica, 2005, Volume: 26, Issue:12

    Topics: Animals; Cimetidine; Dizocilpine Maleate; Dose-Response Relationship, Drug; Hippocampus; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Injections, Intraventricular; Male; Maze Learning; Memory Disorders; Pyrilamine; Rats; Rats, Sprague-Dawley

2005
Histamine H1 receptor involvement in prepulse inhibition and memory function: relevance for the antipsychotic actions of clozapine.
    Pharmacology, biochemistry, and behavior, 2007, Volume: 86, Issue:4

    Topics: Animals; Antipsychotic Agents; Clozapine; Dizocilpine Maleate; Drug Interactions; Female; Histamine H1 Antagonists; Maze Learning; Memory; Nicotine; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine H1; Reflex, Startle

2007
Activation of brain histaminergic neurotransmission: a mechanism for cognitive effects of memantine in Alzheimer's disease.
    The Journal of pharmacology and experimental therapeutics, 2011, Volume: 336, Issue:2

    Topics: Alzheimer Disease; Animals; Brain; Brain-Derived Neurotrophic Factor; Calcium; Cognition; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Histamine; Humans; Male; Memantine; Methylhistamines; Mice; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission

2011
The dual-acting H3 receptor antagonist and AChE inhibitor UW-MD-71 dose-dependently enhances memory retrieval and reverses dizocilpine-induced memory impairment in rats.
    Behavioural brain research, 2016, Jan-15, Volume: 297

    Topics: Animals; Avoidance Learning; Benzothiazoles; Cholinesterase Inhibitors; Disease Models, Animal; Dizocilpine Maleate; Donepezil; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Histamine H3 Antagonists; Indans; Male; Memory; Memory Disorders; Nootropic Agents; Phenoxypropanolamines; Piperidines; Pyrilamine; Pyrroles; Quinazolines; Random Allocation; Rats, Wistar; Receptors, Histamine H3

2016