pyrilamine has been researched along with cimetidine in 399 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 202 (50.63) | 18.7374 |
1990's | 126 (31.58) | 18.2507 |
2000's | 54 (13.53) | 29.6817 |
2010's | 16 (4.01) | 24.3611 |
2020's | 1 (0.25) | 2.80 |
Authors | Studies |
---|---|
Timmerman, H | 1 |
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET | 1 |
Brown, TH; Ganellin, CR; Griffiths, R; Jones, M; Mitchell, RC; Rana, KK; Saunders, D; Smith, IR; Sore, NE; Young, RC | 1 |
Blake, JF; Curatolo, WJ; Lombardo, F | 1 |
Nezu, J; Oku, A; Sai, Y; Sakamoto, K; Shimane, M; Tamai, I; Tsuji, A; Yabuuchi, H | 1 |
Nezu, JI; Ohashi, R; Oku, A; Sai, Y; Shimane, M; Tamai, I; Tsuji, A; Yabuuchi, H | 1 |
Carrupt, PA; Crivori, P; Cruciani, G; Testa, B | 1 |
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM | 1 |
Axe, FU; Bembenek, SD; Butler, CR; Coles, F; Dunford, PJ; Edwards, JP; Fourie, AM; Grice, CA; Karlsson, L; Lundeen, K; Riley, JP; Savall, BM; Tays, KL; Wei, J; Williams, KN; Xue, X | 1 |
Altenbach, RJ; Brioni, JD; Carr, TL; Chandran, P; Cowart, MD; Esbenshade, TA; Honore, P; Hsieh, GC; Lewis, LG; Liu, H; Manelli, AM; Marsh, KC; Milicic, I; Miller, TR; Strakhova, MI; Vortherms, TA; Wakefield, BD; Wetter, JM; Witte, DG | 1 |
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K | 1 |
Ambroso, JL; Ayrton, AD; Baines, IA; Bloomer, JC; Chen, L; Clarke, SE; Ellens, HM; Harrell, AW; Lovatt, CA; Reese, MJ; Sakatis, MZ; Taylor, MA; Yang, EY | 1 |
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ | 1 |
Anzini, M; Brogi, S; Butini, S; Campiani, G; Cappelli, A; Caselli, G; Castriconi, F; Gemma, S; Giordani, A; Giorgi, G; Giuliani, G; Lanza, M; Letari, O; Makovec, F; Manini, M; Mennuni, L; Valenti, S | 1 |
Belyakov, S; Dambrova, M; Kazoka, H; Kuznecovs, J; Lebedev, A; Liepinsh, E; Mishnev, A; Orlova, N; Ponomaryov, Y; Vavers, E; Veinberg, G; Vikainis, S; Vilskersts, R; Vorona, M; Zvejniece, L | 1 |
Bednarski, M; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pękala, E; Powroźnik, B; Słoczyńska, K; Walczak, M; Waszkielewicz, AM; Żesławska, E | 1 |
Filipek, B; Gunia-Krzyżak, A; Marona, H; Nitek, W; Pańczyk, K; Pękala, E; Rapacz, A; Słoczyńska, K; Waszkielewicz, AM; Żelaszczyk, D; Żesławska, E | 1 |
Abdel-Hamid, MK; Andersson, S; Chau, N; Daniel, JA; Deane, FM; Hill, TA; McCluskey, A; Odell, LR; Robinson, PJ; Sakoff, JA; Young, KA | 1 |
Kuschinsky, W; Wahl, M | 1 |
Bommelaer, G; Guth, PH | 1 |
Bruggeman, TM; Davenport, HW; Wood, JG | 1 |
Cheung, LY; Porterfield, G | 1 |
Kaliner, M | 1 |
Grönneberg, R; Hägermark, O; Strandberg, K | 1 |
Behsudi, FM; Bruce, LA; Fawcett, CP | 1 |
Becker, M; Malchow, H; Painz, B; Rack, M; Ruoff, HJ; Sewing, KF | 1 |
De Cock, W; De Cree, J; Verhaegen, H | 1 |
Al-Haboubi, HA; Zeitlin, IJ | 2 |
Gerner, T; Haffner, JF; Norstein, J | 1 |
Harvey, CA; Owen, DA; Shaw, KD | 1 |
Vohra, MM | 1 |
Casteels, R; Suzuki, H | 1 |
Bertaccini, G; Coruzzi, G; Musso, E | 1 |
Bertaccini, G; Impicciatore, M; Morini, G | 1 |
Chand, N; Eyre, P | 1 |
Barkla, DH; Tutton, PJ | 1 |
Bertaccini, G; Coruzzi, G; Vitali, T | 1 |
Carter, DC; Grossman, MI; Impicciatore, M | 1 |
Chirtel, SJ; Field, RB | 1 |
Code, CF; Nakaya, N; Tasaka, K | 1 |
Brandes, LJ; LaBella, FS | 1 |
Balster, RL; Beardsley, PM | 1 |
Bach, FW; Knigge, U; Matzen, S; Secher, NH; Warberg, J | 1 |
Bagavandoss, P; Mitchell, MA; Wilks, JW | 1 |
Alada, AR; Oyebola, DD | 1 |
Cervos-Navarro, J; Dey, PK; Nyberg, F; Sharma, HS | 1 |
Bailly, DA; Gruetter, CA; Stewart, NL; Szarek, JL | 1 |
Imamura, T; Kawasaki, H; Taguchi, T; Takasaki, K | 1 |
Anjelkovic, IZ; Collis, CS; Djuric, D; Rosic, M; Segal, MB; Zlokovic, BV | 1 |
Endou, M; Gando, S; Hattori, Y; Kanno, M | 2 |
Corfield, DR; Webber, SE; Widdicombe, JG | 1 |
Chan, CC; Foster, A | 1 |
Nowak, JZ; Sek, B | 1 |
Bogdanovic, RP; Brandes, LJ; Sukhu, B | 1 |
Ahmad, Z; Baumann, G; Berdel, WE; Felix, SB; Hashemi, T; Niemczyk, M | 1 |
Holtzman, MJ; Jacobs, SC; Mahoney, M; Pentland, AP | 1 |
Gabel, RA; Macia, RA; Matthews, WD; Reginato, MJ | 1 |
Ishikawa, T; Sato, M; Shiosaka, S; Tani, E; Tohyama, M | 1 |
Edvinsson, L; Jansen, I; Langemark, M; Olesen, J; Ottosson, AL | 1 |
Ishikawa, E; Matsukura, S; Nakatsuru, K; Ohgo, S | 1 |
Stehle, J | 1 |
Benedito, S; Nielsen, PJ; Nyborg, NC; Prieto, D | 1 |
Arima, N; Chiba, T; Fujita, T; Morishita, T; Nakamura, A; Nakata, H; Yamashita, Y | 1 |
Bugajski, J; Chłap, Z; Fogel, WA; Gadek-Michalska, A; Turoń, M | 1 |
Bairy, KL; Kulkarni, DR; Ramesh, KV; Rao, CM | 1 |
Cooke, HJ; Fertel, R; Su, HC; Wang, YZ | 1 |
Dolata, J; Lindberg, S; Mercke, U | 1 |
Hill, SJ; Iredale, PA; Kendall, DA; Martin, KF; Ruck, A | 1 |
Bugajski, J; Turon, M; Tyton, J | 1 |
Cervós-Navarro, J; Sharma, HS | 1 |
Cruz, MA; González, C; Rudolph, MI; Sepúlveda, WH | 1 |
Northover, AM | 1 |
Cooke, HJ; Wang, YZ | 1 |
Młynarska, MS | 1 |
Brown, LA; Chen, M | 1 |
Barnes, PJ; Ichinose, M | 1 |
Edvinsson, L; Hill, SJ; Ottosson, A | 1 |
Leathard, HL; Norman, BJ | 1 |
Keitoku, M; Maruyama, Y; Takishima, T | 1 |
Cheung, LY; Wicina, GM; Wood, JG | 1 |
Banks, BE; Dempsey, CE; Vernon, CA; Warner, JA; Yamey, J | 1 |
Johnson, CG; Johnson, CL | 1 |
Barnes, PJ; Liu, SF; Yacoub, M | 1 |
Gamse, R; Saria, A | 2 |
Cho, CH; Dai, S; Ogle, CW | 1 |
Ledgard, SE; Owen, DA; Pipkin, MA; Woodward, DF | 1 |
Feniuk, W; Humphrey, PP; Trevethick, MA | 1 |
Burtin, C; Eschalier, A; Lavarenne, J; Tounissou, P | 1 |
Braimbridge, MV; Erol, C; Hearse, DJ; Maxwell, MP; Saldanha, C; Sonmez, B | 1 |
Holzer, P; Holzer-Petsche, U; Leander, S | 1 |
Abdullah, NA; Assem, ES | 1 |
Hurwitz, A; Innis, JD | 1 |
Arrang, JM; Garbarg, M; Schwartz, JC | 1 |
Bakich, V; Brown, JC; Kwok, YN; McIntosh, CH; Wong, J | 1 |
Clough, GF; Noor, NM; Smaje, LH | 1 |
Hirasawa, N; Kamo, I; Tsurufuji, S | 1 |
Buck, M; Goswami, S; Marom, Z; Schachter, EN; Witek, T | 1 |
Dann, O; Estler, CJ; Steinmann, U | 1 |
Edvinsson, L; Jansen, I; Ottosson, A | 1 |
Gupta, GP; Tangri, KK; Vrat, S | 1 |
Guo, ZG; Luo, WS | 1 |
Bugajski, J; Gadek-Michalska, A | 1 |
Khan, MA; Sen, PC | 1 |
Fujimoto, K; Fukagawa, K; Ookuma, K; Sakata, T; Shiraishi, T; Wada, H; Yoshimatsu, H | 1 |
Bach, FW; Bang, P; Knigge, U; Matzen, S; Warberg, J | 1 |
Akamine, M; Kitazawa, T; Kondo, H; Ohta, T; Shimizu, T; Temma, K | 1 |
Ezeamuzie, CI; Umezurike, CC | 1 |
Dailey, RA; Hall, JA; Lewis, PE; Meisterling, EM | 1 |
Hazama, A; Okada, Y; Yada, T | 1 |
Bhandari, P; Bhargava, KP; Chugh, A; Dixit, KS; Gupta, YK; Seth, SD | 1 |
Chansouria, JP; Dey, PK; Mohanty, S; Olsson, Y; Sharma, HS; Singh, S | 1 |
Gary, RK; Gleason, JG; Nieves, AL; Wasserman, MA; Williams, LS; Woodward, DF | 1 |
Kanaide, H; Kobayashi, S; Kuga, T; Matsumoto, T; Nakamura, M; Nishimura, J | 1 |
Bunn, SJ; Livett, BG; Wan, DC | 1 |
Acevedo, CG; Cruz, MA; Gonzalez, C; Rudolph, MI; Sepulveda, WH | 1 |
Guo, ZG; Qiu, R | 1 |
Adaikan, PG; Lau, LC; Ratnam, SS | 1 |
Jorgenson, KL; Kow, LM; Pfaff, DW | 1 |
Ono, H; Suzuki, H | 1 |
Nishimura, H; Yamaguchi, K | 1 |
Nicholson, AN; Pascoe, PA; Stone, BM | 1 |
Trzeciakowski, JP | 1 |
Heldsinger, AA; Pittenger, GL; Seino, S; Vinik, AI | 1 |
Banks, RO; Jacobson, ED | 1 |
Foreman, JC; Norris, DB; Rising, TJ; Webber, SE | 1 |
Hawley, SB; Nieves, AL; Spada, CS; Woodward, DF | 2 |
Hutchison, VH; Spriestersbach, KK | 1 |
Knigge, U; Matzen, S; Warberg, J | 2 |
Cordeiro, RS; Corrêa, FM; Henriques, MG; Martins, MA; Silva, PM | 1 |
Fu, SX; Li, CG; Li, YS | 1 |
Clerici, C; Franco-Montoya, ML; Harf, A; Macquin-Mavier, I | 1 |
Honda, K; Kaneko, K; Komatsu, H; Nakamura, M; Oda, M; Tsuchiya, M | 1 |
Männistö, PT; Mattila, J; Tuominen, RK | 2 |
Ledgard, SE; Nieves, AL; Woodward, DF | 1 |
Barker, LA; Winbery, SL | 1 |
Kim, LE; Oudart, N; Sercombe, R; Teste, JF | 1 |
Bugajski, J; Gadek, A | 1 |
Iwata, M; Kohno, S; Shigei, T; Tsuru, H | 1 |
Abacioğlu, N; Demiryürek, T; Ercan, ZS; Kanzik, L; Türker, RK; Zengil, H | 1 |
Dhawan, KN; Gulati, A; Gupta, GP; Nath, C | 1 |
Ea-Kim, L; Oudart, N | 1 |
Donaldson, J; Hill, SJ | 1 |
Kawasaki, H; Takasaki, K | 1 |
Fromm, D; Furukawa, T; Olender, EJ; Woods, DJ | 1 |
Hunt, WA; Kandasamy, SB | 1 |
Bohm, U; Falus, A; Fekete, MI; Meretey, K | 1 |
Allescher, HD; Berezin, I; Daniel, EE; Jury, J | 1 |
Guo, ZG; Zhou, CJ | 1 |
Itowi, N; Nagai, K; Nakagawa, H; Wada, H; Watanabe, T | 1 |
Palmer, JM; Tamura, K; Wood, JD | 1 |
Cross, KS; el-Sanadiki, MN; Hagen, PO; McCann, RL; Mikat, EM; Murray, JJ | 1 |
Xu, YH; Yi, SN | 1 |
Kitamura, K; Yamanaka, K | 1 |
Dveksler, G; Franchi, AM; Gimeno, AL; Gimeno, MF; Viggiano, M | 1 |
Chen, J; Johnson, L; Spada, C; Woodward, DF | 1 |
Charap, A; Duzman, E; Leon, J; Shen, CD | 1 |
Kannisto, P; Owman, C; Schmidt, G; Sjöberg, NO | 1 |
Kotlikoff, MI; Murray, RK; Reynolds, EE | 1 |
Fan, TP; Lo, WW | 1 |
Harvey, MH; Reber, HA; Wedgwood, KR | 1 |
Bommer, M; Herz, A; Kley, N; Liebisch, D; Noble, E | 1 |
Bugajski, J; Cetera, B; Gadek, A | 1 |
Jantos, H; Monti, JM; Pellejero, T | 1 |
Kakimoto, M; Kurokawa, K; Nakayama, Y; Tasaka, K | 1 |
Owman, C; Schmidt, G; Sjöberg, NO | 1 |
Ledgard, SE; Woodward, DF | 1 |
Barrett, RJ; Kau, ST | 1 |
Gerdin, B; Sandler, H | 1 |
Cirino, M; Letts, LG | 1 |
Christiansen, PM; Knigge, U; Thuesen, B | 1 |
Bogdanovic, RP; Brandes, LJ | 1 |
Fedan, JS; Hogaboom, GK; Horstemeyer, DL; Ice, KS; O'donnell, JP; Smith, DJ | 1 |
Kanaide, H; Kobayashi, S; Matsumoto, T; Nakamura, M; Nishimura, J; Shogakiuchi, Y | 1 |
Bommer, M; Costa, T; Herz, A; Noble, EP; Sincini, E | 1 |
Owen, DA; Pipkin, MA | 1 |
Kauffman, GL; Kleibeuker, JH; Walsh, JH | 1 |
Kikuchi, M; Oh-ishi, S | 1 |
Banning, JW; Dipietro, RA; Griffith, RK | 1 |
Kume, S; Ohashi, T; Ozaki, Y | 1 |
Gristwood, RW; Lincoln, JC; Owen, DA | 1 |
Daniel, D; Owen, DA; Poy, E; Woodward, DF | 1 |
Fischer, J; Fromm, D; Kolis, M; Shang, A | 1 |
Daly, MJ; Humphray, JM; Stables, R | 1 |
Bunce, KT; Daly, MJ; Humphray, JM; Stables, R | 2 |
Cade, JF; Clancy, RL; Pain, MC; Walker, SE | 1 |
Coupet, J; Szuchs-Myers, VA | 1 |
Owen, DA; Woodward, DF | 1 |
Oriowo, MA | 1 |
Maśliński, S; Stochla, K | 1 |
Owen, DA; Pipkin, MA; Raval, P; Woodward, DF | 1 |
Robinson, BV | 1 |
Kaminka, ME; Mashkovskiĭ, MD; Tupikina, SM | 1 |
Heldsinger, AA; Skoglund, ML; Vinik, AI | 1 |
Aghajanian, GK; Lakoski, JM | 1 |
Hoffman, LH; Hoos, PC | 1 |
Langwiński, R; Malec, D | 1 |
Guldvog, I; Linnestad, P; Schrumpf, E | 1 |
Black, J; Shaw, J; Vincenc, K | 1 |
Hösli, E; Hösli, L; Schneider, U; Wiget, W | 1 |
Nemeth, PR; Ort, CA; Wood, JD | 1 |
Obel, AO | 1 |
Andersen, V; Geisler, A; Klysner, R; Manthorpe, R; Nielsen, H; Norn, S; Permin, H; Petersen, J; Skov, PS; Wiik, A | 1 |
Franklin, JE; Liebow, C | 1 |
Gazelius, B; Olgart, L; Panopoulos, P | 1 |
Folkers, K; Lundberg, JM; Rosell, S; Saria, A | 1 |
Koo, A | 1 |
Bugajski, J; Janusz, Z | 1 |
Owen, DA; Pipkin, MA; Woodward, DF | 1 |
Kusunoki, M; Tanaka, C; Taniyama, K | 1 |
Binderup, L | 1 |
Chand, N; DeRoth, L | 1 |
Abbound, HE; Dousa, TP; Edis, AJ; Heath, H; Zimmerman, D | 1 |
Chader, GJ; Koh, SW | 1 |
Kandasamy, SB; Williams, BA | 1 |
Chiou, GC; Miyano, K | 1 |
Christiansen, PM; Dejgaard, A; Knigge, U; Thuesen, B; Wollesen, F | 2 |
Christiansen, PM; Dejgaard, A; Knigge, U; Larsen, K; Wollesen, F | 1 |
Alphin, RS; Callaham, EM; Foxwell, MH; Smith, WL; Yanni, JM | 1 |
Di Donato, M; Mantovani, P; Santicioli, P | 1 |
Gerdin, B; Lundberg, C | 1 |
Rothwell, NJ; Stock, MJ; Wyllie, MG | 1 |
Chung, YH; Kamei, C; Miyake, H; Tasaka, K | 1 |
Ertresvaag, K; Gerner, T; Haffner, JF; Norstein, J | 1 |
Kou, K; Suzuki, H | 1 |
Godfraind, T; Miller, RC | 1 |
Mészáros, J; Szegi, J | 1 |
Coffman, JD; Cohen, RA; Rasmussen, HM | 1 |
Hui, HW; Robinson, JR; Zeleznick, L | 1 |
Crassaris, LG; Fidani, V; Papadopoulos, AG; Paradelis, AG; Stavrakis, AO; Triantaphyllidis, CJ | 1 |
Gajtkowski, GA; Norris, DB; Rising, TJ | 1 |
Leusen, I; Van de Voorde, J | 3 |
Tayal, G; Tripathi, KD | 2 |
Carter, DC; Lewi, HJ | 1 |
Iwata, M; Shigei, T; Tsuru, H | 1 |
Askenase, PW; Nordlund, JJ | 1 |
Baenziger, NL; Becherer, PR; Force, LE | 1 |
Davenport, HW; Wood, JG | 1 |
Rand, MJ; Story, DF; Wong-Dusting, HK | 1 |
Singh, KP; Tayal, G; Tripathi, KD | 1 |
Boyce, MJ; Harvey, CA; Owen, DA | 1 |
Hunt, WA; Kaliner, M; Wescott, SL | 1 |
Fosbraey, P; Johnson, ES; Mckay, FF | 1 |
Verma, SC; Vyas, S | 1 |
Casteels, R | 1 |
Ichikawa, T; Naito, Y; Nakazawa, S; Tsukamoto, Y | 1 |
Argenbright, LW; Forbes, PD; Stewart, GJ | 2 |
Arnold, G; Reinhardt, D; Walkenhorst, R | 1 |
Knight, SE; McIsaac, RL; Rennie, CD | 1 |
Brown, PA; Vernikos, J | 1 |
Krabbe, AA; Olesen, J | 1 |
Seidler, FJ; Slotkin, TA; Subramanian, N; Whitmore, WL | 1 |
Boe, J; Boe, MA; Simonsson, BG | 1 |
Bos, E; Du, XY; Saxena, PR; Schoemaker, RG | 1 |
Evans, TW; Griffiths, MJ; MacAllister, RJ; Messent, M | 1 |
Akerström, G; Lisander, B | 1 |
Kohno, S; Nabe, T; Nakao, S; Ogawa, K; Ohata, K; Yamamura, H | 1 |
Barak, V; Fabian, I; Geller-Bernstein, C; Handzel, ZT; Mor, S; Nagler, A | 1 |
Ballabeni, V; Barocelli, E; Chiavarini, M; Impicciatore, M | 1 |
Hashioka, T | 1 |
Brown, RE; Fedorov, NB; Haas, HL; Reymann, KG | 1 |
Fischer, Y; Hirsch, B; Kammermeier, H; Linssen, M; Rösen, P; Thomas, J; van der Vusse, GJ | 1 |
Homma, I; Iwase, M; Kanamaru, M | 2 |
Kohno, S; Nabe, T; Ogawa, K; Ohata, K; Yamamura, H | 1 |
Choi, AY; Fukui, H; Perlman, RL | 1 |
Carson, CC; Davies, MG; Hagen, PO; Kim, YC; Lee, TH | 1 |
Akaike, N; Munakata, M | 1 |
Edvinsson, L; Hedner, T; Sun, X | 1 |
Fischer, R; Pavenstädt, H; Schlunck, G; Schollmeyer, P; Späth, MM; Wanner, C | 1 |
Gando, S; Hattori, Y; Kanno, M; Nagashima, M | 1 |
Kamondi, A; Reiner, PB | 1 |
Chen, YL; Guo, ZG; Xie, DN | 1 |
Garbarg, M; Kjaer, A; Knigge, U; Rouleau, A; Warberg, J | 1 |
Dalton, TK; Harris, AH; Hunt, WA; Joseph, JA; Kandasamy, SB; Rabin, BM | 1 |
Shibata, S; Watanabe, S | 1 |
Kamei, C; Tasaka, K; Tsujimoto, S; Yoshida, T | 1 |
Kondratenko, TY; Kornilova, ZCh; Kuzina, NV; Perelman, MI; Severin, ES; Zacharova, IV | 1 |
Desautels, M; Halvorson, I; Muralidhara, DV; Thornhill, J; Wollin, A | 1 |
Banchelli, G; Buffoni, F; Conforti, L; Ignesti, G; Pirisino, R; Raimondi, L | 1 |
Maeda, K; Tagami, H; Tomita, Y | 1 |
Kamei, C; Tasaka, K | 1 |
Bach, FW; Kjaer, A; Knigge, U; Madsen, EL; Søe-Jensen, P; Warberg, J | 1 |
Finlay-Jones, JJ; Hart, PH; Jones, CA; Jones, KL; Santucci, I; Spencer, LK; Watson, CJ | 1 |
Fukui, M; Ikezaki, K; Natori, Y; Nomura, T | 1 |
Miyamoto, A; Nishio, A | 1 |
Cheung, LY; Darnell, MP; Wood, JG | 1 |
Gonzalez, R; Reinicke, K; Rudolph, GM | 1 |
Everaert, E; Germonpré, PR; Joos, GF; Kips, JC; Pauwels, RA | 1 |
Borda, ES; Goren, N; Leiros, CP; Sterin-Borda, L | 1 |
Endo, Y; Kuroda, H; Nakamura, M; Narita, K | 1 |
Assenmacher, I; Barbanel, G; Givalois, L; Ixart, G; Malaval, F; Mekaouche, M; Siaud, P | 1 |
Konno, K; Nakata, J; Takeyama, K; Tamaoki, J | 1 |
Arilla, E; Puebla, L; Rodríguez-Martín, E | 1 |
KAMEI, CH | 1 |
Clark, EA; Hill, SJ | 1 |
Akiyama, K; Maeda, Y; Mita, H; Saito, H; Shimizu, H | 1 |
Barzanti, F; Gruenert, DC; Hrelia, S; Rugolo, M | 1 |
Larmark, M; Lisander, B | 1 |
Eaton, SJ; Eoh, S; Harrington, ME; Hoque, S; Meyer, J | 1 |
Anesini, C; Boccio, J; Borda, E; Cremaschi, G; Genaro, A; Sterin-Borda, L; Zubillaga, M | 1 |
Fertel, RH; Wood, JD; Xia, Y | 1 |
Chiyotani, A; Konno, K; Nakata, J; Takeyama, K; Tamaoki, J | 1 |
Amann, R; Donnerer, J; Peskar, BA; Schuligoi, R | 1 |
Kandasamy, SB | 1 |
He, S; Walls, AF | 1 |
Agut, J; Ortiz, JA; Sacristán, A; Sánchez, JC | 1 |
Larsen, PJ; Luckman, SM | 1 |
Branum, JC; Kline, RS; Whisnant, CS | 1 |
Bergoc, R; Cricco, G; Davio, C; Duran, H; Fitzsimons, C; Molinari, B; Palmieri, M; Rivera, E | 1 |
Dobigny, C; Saffar, JL | 1 |
Khodorova, AB; Nechaeva, MV; Turpaev, TM | 1 |
Arisawa, T; Asai, J; Goto, H; Hase, S; Hayakawa, T; Takeda, T | 1 |
Easton, AS; Fraser, PA; Sarker, MH | 2 |
Bivalacqua, TJ; Champion, HC; Czapla, MA; Ilgenfritz, C; Kadowitz, PJ; Santiago, JA | 1 |
Agustí, C; Cardell, LO; Nadel, JA; Stjärne, P; Wagstaff, SJ | 1 |
Ito, Y; Kashiwagi, S; Kimura, C; Oike, M | 1 |
Barnes, PJ; Dupont, LJ; Mak, JC; Pype, JL; Verleden, GM | 1 |
Bizot-Espiard, JG; Caignard, DH; Guillaumet, G; Pfeiffer, B; Renard, P; Savelon, L; Viaud, MC | 1 |
Carman-Krzan, M; Juric, DM; Lipnik-Stangelj, M | 1 |
Bergoc, R; Davio, C; Legnazzi, BL; Monczor, F; Rivera, E | 1 |
Durán, H; Fitzsimons, C; Labombarda, F; Molinari, B; Rivera, E | 1 |
Acuña, Y; Campos, HA; Israel, A; Mathison, Y | 1 |
Fukuoka, M; Haraguchi, R; Iwanaga, T; Kubo, H; Nakajima, S; Tohda, Y | 1 |
Miller, DJ; O'Dowd, A | 1 |
Capasso, F; Costa, M; Izzo, AA; Mascolo, N | 1 |
Delaey, C; Depypere, H; Van de Voorde, J; Vanheel, B | 1 |
Jørgensen, H; Kjaer, A; Knigge, U; Warberg, J; Willems, E | 1 |
Carman-Krzan, M; Lipnik-Stangelj, M | 1 |
de Wildt, DJ; Hendriksen, CF; van de Kuil, A; van den Hout, JW; Vleeming, W | 1 |
Akaishi, Y; Hattori, Y; Kanno, M; Kitabatake, A; Yasuda, K; Yoshimoto, K | 1 |
Anichtchik, OV; Panula, P; Peitsaro, N | 1 |
Nakazato, E; Ohno, M; Watanabe, S; Yamamoto, T | 1 |
Jørgensen, H; Kjaer, A; Knigge, U; Warberg, J | 1 |
Ikarashi, Y; Ishige, A; Kuribara, H; Maruyama, Y; Sasaki, H; Yuzurihara, M | 1 |
Hidaka, Y; Itadani, H; Nakamura, T; Ohta, M; Tanaka, K | 1 |
Cunha, FQ; Ferreira, SH; Parada, CA; Tambeli, CH | 1 |
Kolaczkowska, E; Plytycz, B; Seljelid, R | 1 |
Hardwick, JC; Peterson, BA; Powers, MJ | 1 |
Cheng, JS; Chou, KJ; Jan, CR; Lee, KC; Tang, KY; Tseng, LL; Wang, JL | 1 |
Masuyama, K; Minoda, R; Toriya, T; Yumoto, E | 1 |
Chang, HT; Cheng, JS; Chou, KJ; Jan, CR; Lee, KC; Tang, KY; Wang, JL | 1 |
Ghosh, AK; Hirasawa, N; Ohuchi, K | 1 |
Furue, M; Koga, T; Kohda, F; Uchi, H; Urabe, K | 1 |
Fogel, WA; Stasiak, A; Wagner, W | 1 |
Arias-Montaño, JA; García, L; Guerrero-Hernández, A; Rueda, A; Soria-Jasso, LE | 1 |
Adachi, T; Hori, Y; Ishigaki-Suzuki, S; Kagaya, Y; Kikuchi, Y; Makabe-Kobayashi, Y; Nagy, A; Ohtsu, H; Shirato, K; Takai, T; Ujike, A; Watanabe, T | 1 |
Bacon, KB; Center, DM; Cruikshank, WW; Gantner, F; Sakai, K; Tusche, MW | 1 |
Aceves, J; Arias-Montaño, JA; Bárbara, A | 1 |
Anisman, H; Hayley, S; Kelly, O | 1 |
Bischoff, AM; Büsselberg, D; Dutschmann, M; Richter, DW | 1 |
Eidi, A; Eidi, M; Oryan, S; Parivar, K; Zarrindast, MR | 1 |
Madri, JA; Payne, GW; Segal, SS; Sessa, WC | 1 |
Assadi, E; Oryan, S; Sahebgharani, M; Torkaman-Boutorabi, A; Zarrindast, MR | 1 |
Nakamura, T; Ueno, K; Yamaura, K; Yano, S; Yonekawa, T | 1 |
Araújo Palmeira, CC; Ashmawi, HA; Chambergo, FS; Posso, IP | 1 |
Jørgensen, H; Kjaer, A; Knigge, U; Kristoffersen, U; Madsen, K; Toftegaard, C; Warberg, J | 1 |
Bacon, KB; Gantner, F; Sakai, K; Takeshita, K | 1 |
Atwell, R; Brown, L; Campbell, F; Fenning, A; Hoey, A | 1 |
Athanazio, R; Barbetta, M; de Castro e Silva, E; Duarte, G; Fregoneze, JB; Luz, P; Magrani, J; Ramos, AC; Varjão, B | 1 |
Athanazio, R; Barbetta, M; de Castro e Silva, E; Fregoneze, JB; Magrani, J; Ramos, AC | 1 |
Tsuruki, T; Yoshikawa, M | 1 |
Cheung, JH; Lam, FY; Ng, SC; Yeung, JH | 1 |
Benedito, S; García-Sacristán, A; Hernández, M; Martínez, AC; Pagán, RM; Prieto, D; Raposo, R | 1 |
Chen, Z; Hu, WW; Liu, LY; Ma, L; Wei, EQ; Xu, LS; Yang, LX; Yu, X | 1 |
Carlos, D; de Paula, L; Faccioli, LH; Malheiro, A; Santos, WF | 1 |
Gálfi, M; Juhász, A; László, F; László, FA; Molnár, A; Radács, M; Varga, C | 1 |
Carlos, D; de Paula, L; Faccioli, LH; Jamur, MC; Martins, MA; Matias-Peres, C; Oliver, C; Sá-Nunes, A; Serra, MF | 1 |
Dube, PH; Handley, SA; Miller, VL | 1 |
Bennett, T; Gardiner, SM; Kemp, PA; March, JE | 1 |
Bai, ZT; Chai, ZF; Ji, YH; Jiang, F; Liu, T; Pang, XY | 1 |
Baldo, CF; Capellini, VK; Celotto, AC; Evora, PR; Rodrigues, AJ; Viaro, F; Vicente, WV | 1 |
Fukino, K; Ikawa, Y; Kuribayashi, M; Ohkuni, Y; Ueno, K; Yonekawa, T | 1 |
Decaluwé, K; Nimmegeers, S; Van de Voorde, J | 1 |
Qi, Y; Qian, ZB; Wu, ZH | 1 |
Hirasawa, N; Hong, J; Ishihara, K; Katoh, G; Ohsawa, Y; Ohuchi, K; Seyama, T; Shibata, K; Tamura, S | 1 |
Chen, Z; Fan, YY; He, P; Hu, WW; Xu, LS; Zhang, WP | 1 |
Arias, K; Baig, M; Chu, D; Colangelo, M; Coyle, A; Goncharova, S; Jordana, M; Vadas, P; Walker, T; Waserman, S | 1 |
Maslinski, S; Mittal, TK; Rongies, W; Szewczyk, G; Szukiewicz, D | 1 |
Halliwill, JR; Maclean, DA; Pellinger, TK; Simmons, GH | 1 |
Alisch, R; Buschauer, A; Elz, S; Sadek, B | 1 |
Breslin, JW; Kurtz, KH; Moor, AN; Souza-Smith, FM | 1 |
Chen, J; Deng, L; Ding, S; Ge, J; Hong, T; Huang, Z; Jia, J; Lin, J; Wang, TC; Yang, X; Zou, Y | 1 |
Chen, Z; Hou, WW; Hu, TT; Lou, GD; Ohtsu, H; Shi, LY; Tang, YY; Wang, RR; Yu, J; Yue, JX; Zhang, SH | 1 |
Lkhagvasuren, B; Oka, T | 1 |
Lafuente, JV; Muresanu, DF; Nozari, A; Ozkizilcik, A; Patnaik, R; Sharma, A; Sharma, HS; Tian, ZR | 1 |
Aneesha, VA; Gopi, RP; Kumar, D; Kumawat, S; Susanth, VS; Vineetha, S | 1 |
2 review(s) available for pyrilamine and cimetidine
Article | Year |
---|---|
Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship | 1990 |
Vascular actions of leukotrienes.
Topics: Aminophylline; Animals; Atropine; Blood Platelets; Blood Vessels; Capillary Permeability; Cimetidine; Guanethidine; Hexamethonium Compounds; Humans; Indomethacin; Methysergide; Muscle Contraction; Muscle, Smooth, Vascular; Propranolol; Pyrilamine; Regional Blood Flow; Skin; SRS-A; Vasoconstriction | 1985 |
6 trial(s) available for pyrilamine and cimetidine
Article | Year |
---|---|
Human gastric mucosal adenylate cyclase: activation by histamine-H2-receptor stimulation and inhibition by cimetidine in vitro and in peptic ulcer patients.
Topics: Adenylyl Cyclases; Cimetidine; Clinical Trials as Topic; Enzyme Activation; Female; Gastric Mucosa; Guanidines; Histamine; Humans; Male; Middle Aged; Peptic Ulcer; Phenethylamines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H2; Thiourea | 1979 |
Efficacy of cimetidine/pyrilamine eyedrops. A dose response study with histamine challenge.
Topics: Adult; Aminopyridines; Cimetidine; Clinical Trials as Topic; Dose-Response Relationship, Drug; Drug Combinations; Eye; Eye Diseases; Female; Histamine; Humans; Hyperemia; Hypersensitivity; Male; Ophthalmic Solutions; Pyrilamine | 1986 |
The effect of histamine on the human fingertip circulation.
Topics: Cimetidine; Cold Temperature; Fingers; Histamine; Humans; Norepinephrine; Pyrilamine; Regional Blood Flow; Vascular Resistance; Vasoconstriction | 1984 |
Headache provocation by continuous intravenous infusion of histamine. Clinical results and receptor mechanisms.
Topics: Aminopyridines; Cimetidine; Headache; Histamine; Humans; Migraine Disorders; Pyrilamine | 1980 |
Dehydration-induced vasopressin secretion in humans: involvement of the histaminergic system.
Topics: Adult; Aldosterone; Cimetidine; Cross-Over Studies; Dehydration; Double-Blind Method; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Male; Osmolar Concentration; Placebos; Pyrilamine; Ranitidine; Receptors, Histamine H1; Receptors, Histamine H2; Vasopressins; Water-Electrolyte Balance | 2000 |
Local histamine H(1-) and H(2)-receptor blockade reduces postexercise skeletal muscle interstitial glucose concentrations in humans.
Topics: Adult; Cimetidine; Ethanol; Exercise; Extracellular Space; Female; Glucose; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Hyperemia; Male; Microdialysis; Pyrilamine; Quadriceps Muscle; Receptors, Histamine H1; Receptors, Histamine H2; Tritium; Young Adult | 2010 |
391 other study(ies) available for pyrilamine and cimetidine
Article | Year |
---|---|
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium | 1985 |
Development of a new physicochemical model for brain penetration and its application to the design of centrally acting H2 receptor histamine antagonists.
Topics: Algorithms; Animals; Blood-Brain Barrier; Brain; Chemical Phenomena; Chemistry, Physical; Clonidine; Guinea Pigs; Histamine H2 Antagonists; Imipramine; Pyrilamine; Structure-Activity Relationship | 1988 |
Computation of brain-blood partitioning of organic solutes via free energy calculations.
Topics: Animals; Blood-Brain Barrier; Brain; Cattle; Cells, Cultured; Endothelium, Vascular; Membrane Lipids; Microcirculation; Molecular Conformation; Molecular Structure; Monte Carlo Method; Permeability; Pharmaceutical Preparations; Software; Solubility; Thermodynamics | 1996 |
Novel membrane transporter OCTN1 mediates multispecific, bidirectional, and pH-dependent transport of organic cations.
Topics: Animals; Biological Transport, Active; Carrier Proteins; Cell Line; Gene Expression; Humans; Hydrogen-Ion Concentration; Membrane Potentials; Membrane Proteins; Membrane Transport Proteins; Oocytes; Organic Cation Transport Proteins; Quinidine; RNA, Messenger; Symporters; Tetraethylammonium Compounds; Xenopus laevis | 1999 |
Na(+)-dependent carnitine transport by organic cation transporter (OCTN2): its pharmacological and toxicological relevance.
Topics: Biological Transport, Active; Carnitine; Carrier Proteins; Cations; Cells, Cultured; Dose-Response Relationship, Drug; Embryo, Mammalian; Humans; Hydrogen-Ion Concentration; Kidney; Membrane Proteins; Organic Cation Transport Proteins; Sodium; Solute Carrier Family 22 Member 5; Stereoisomerism | 1999 |
Predicting blood-brain barrier permeation from three-dimensional molecular structure.
Topics: Blood-Brain Barrier; Databases, Factual; Models, Chemical; Molecular Conformation; Multivariate Analysis; Permeability; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship | 2000 |
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4 | 2005 |
Identification of a potent, selective, and orally active leukotriene a4 hydrolase inhibitor with anti-inflammatory activity.
Topics: Administration, Oral; Animals; Anti-Inflammatory Agents; Catalysis; Dogs; Drug Evaluation, Preclinical; Enzyme Inhibitors; Epoxide Hydrolases; Humans; Magnetic Resonance Spectroscopy; Mice; Structure-Activity Relationship | 2008 |
cis-4-(Piperazin-1-yl)-5,6,7a,8,9,10,11,11a-octahydrobenzofuro[2,3-h]quinazolin-2-amine (A-987306), a new histamine H4R antagonist that blocks pain responses against carrageenan-induced hyperalgesia.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzofurans; Carrageenan; Disease Models, Animal; Drug Design; Drug Evaluation, Preclinical; Humans; Hyperalgesia; Ligands; Mice; Molecular Structure; Pain; Peritonitis; Quinazolines; Rats; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Stereoisomerism; Structure-Activity Relationship | 2008 |
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship | 2010 |
Preclinical strategy to reduce clinical hepatotoxicity using in vitro bioactivation data for >200 compounds.
Topics: Chemical and Drug Induced Liver Injury; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Decision Trees; Drug Evaluation, Preclinical; Drug-Related Side Effects and Adverse Reactions; Glutathione; Humans; Liver; Pharmaceutical Preparations; Protein Binding | 2012 |
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship | 2012 |
Synthesis and structure-activity relationship studies in serotonin 5-HT(1A) receptor agonists based on fused pyrrolidone scaffolds.
Topics: Animals; Area Under Curve; Humans; Intestinal Absorption; Ligands; Male; Metabolic Clearance Rate; Models, Chemical; Models, Molecular; Molecular Structure; Protein Binding; Protein Structure, Tertiary; Pyrrolidinones; Radioligand Assay; Receptor, Serotonin, 5-HT1A; Receptors, Serotonin, 5-HT3; Serotonin 5-HT1 Receptor Agonists; Structure-Activity Relationship | 2013 |
Synthesis and biological evaluation of 2-(5-methyl-4-phenyl-2-oxopyrrolidin-1-yl)-acetamide stereoisomers as novel positive allosteric modulators of sigma-1 receptor.
Topics: Acetamides; Allosteric Regulation; Animals; Rats; Rats, Wistar; Receptors, sigma; Sigma-1 Receptor; Stereoisomerism; Structure-Activity Relationship | 2013 |
Design, physico-chemical properties and biological evaluation of some new N-[(phenoxy)alkyl]- and N-{2-[2-(phenoxy)ethoxy]ethyl}aminoalkanols as anticonvulsant agents.
Topics: Amino Alcohols; Animals; Anticonvulsants; Chemistry, Physical; Dose-Response Relationship, Drug; Drug Design; Epilepsy; Male; Mice; Microsomes, Liver; Molecular Structure; Pilocarpine | 2016 |
Structure-anticonvulsant activity studies in the group of (E)-N-cinnamoyl aminoalkanols derivatives monosubstituted in phenyl ring with 4-Cl, 4-CH
Topics: Amino Alcohols; Animals; Anticonvulsants; Crystallography, X-Ray; Disease Models, Animal; Dose-Response Relationship, Drug; Electroshock; Mice; Models, Molecular; Molecular Structure; Rats; Seizures; Structure-Activity Relationship | 2017 |
Pyrimidine-Based Inhibitors of Dynamin I GTPase Activity: Competitive Inhibition at the Pleckstrin Homology Domain.
Topics: Binding, Competitive; Carbon-13 Magnetic Resonance Spectroscopy; Cell Line, Tumor; Drug Screening Assays, Antitumor; Dynamin I; Enzyme Inhibitors; Humans; Mass Spectrometry; Pleckstrin Homology Domains; Proton Magnetic Resonance Spectroscopy; Pyrimidines | 2017 |
The dilating effect of histamine on pial arteries of cats and its mediation by H2 receptors.
Topics: Animals; Arteries; Cats; Cimetidine; Dose-Response Relationship, Drug; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Pia Mater; Pyrilamine; Receptors, Histamine; Receptors, Histamine H2 | 1979 |
Protection by histamine receptor antagonists and prostaglandin against gastric mucosal barrier disruption in the rat.
Topics: Administration, Topical; Animals; Aspirin; Cimetidine; Drug Combinations; Gastric Juice; Gastric Mucosa; Histamine H2 Antagonists; Injections, Intraperitoneal; Membrane Potentials; Potassium; Prostaglandins E, Synthetic; Pyrilamine; Rats; Sodium; Stomach Ulcer | 1979 |
Local control of blood flow in the dog's stomach: vasodilatation caused by acid back-diffusion following topical application of salicylic acid.
Topics: Animals; Atropine; Capillary Permeability; Cimetidine; Diffusion; Dogs; Histamine; Hydrochloric Acid; Hydrogen-Ion Concentration; Papaverine; Perfusion; Pyrilamine; Salicylates; Stomach; Vasodilation | 1979 |
Is histamine a mediator in bile-induced gastric mucosal injury?
Topics: Animals; Bile; Cimetidine; Disease Models, Animal; Dogs; Gastric Mucosa; Histamine; Histamine Release; Humans; Hydrogen-Ion Concentration; Membrane Potentials; Permeability; Pyrilamine; Sodium; Stomach Diseases; Taurocholic Acid | 1978 |
Human lung tissue and anaphylaxis: the effects of histamine on the immunologic release of mediators.
Topics: Antigens; Biological Assay; Cimetidine; Cyclic AMP; Cyclic GMP; Diphenhydramine; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine Release; Humans; Lung; Methylhistamines; Metiamide; Pyrilamine; SRS-A | 1978 |
Effects of histamine receptor antagonists on histamine-induced responses in human skin.
Topics: Adult; Axons; Cimetidine; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Injections, Intradermal; Lidocaine; Metiamide; Pyrilamine; Reflex; Skin | 1979 |
Histaminergic involvement in thyrotropin-releasing hormone stimulation of antral tissue in the rat.
Topics: Animals; Atropine; Bethanechol Compounds; Cimetidine; Histamine; In Vitro Techniques; Male; Muscle Contraction; Pyloric Antrum; Pyrilamine; Rats; Thyrotropin-Releasing Hormone | 1979 |
Histamine receptor-bearing T lymphocytes in patients with allergy, autoimmune disease, or recurrent infection.
Topics: Adolescent; Adult; Aged; Autoimmune Diseases; Child; Child, Preschool; Cimetidine; Female; Humans; Hypersensitivity; Infant; Infections; Male; Middle Aged; Pyrilamine; Receptors, Histamine; Recurrence; Rosette Formation; T-Lymphocytes | 1978 |
The actions of cimetidine, mepyramine, indomethacin and aprotinin (Trasylol) on the inflammatory response in adjuvant rats [proceedings].
Topics: Aminopyridines; Animals; Aprotinin; Arthritis; Arthritis, Experimental; Cimetidine; Guanidines; Indomethacin; Male; Pyrilamine; Rats | 1979 |
The effects of mepyramine and cimetidine on the motor responses to histamine, cholecystokinin, and gastrin in the fundus and antrum of isolated guinea-pig stomachs.
Topics: Acetylcholine; Aminopyridines; Animals; Cholecystokinin; Cimetidine; Female; Gastrins; Gastrointestinal Motility; Guanidines; Guinea Pigs; Histamine; Histamine Antagonists; In Vitro Techniques; Male; Pressure; Pyloric Antrum; Pyrilamine | 1979 |
Histamine-induced increases in gastric blood flow in rats.
Topics: Animals; Blood Flow Velocity; Cimetidine; Histamine; Pyrilamine; Rats; Regional Blood Flow; Stomach; Vasodilator Agents | 1979 |
An inhibitory action of histamine on the rat isolated vas deferens.
Topics: Animals; Cimetidine; Drug Interactions; Electric Stimulation; Histamine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Pyrilamine; Rats; Vas Deferens | 1979 |
Effect of histamine on the small arteries in the gracilis muscle of the rabbit.
Topics: Animals; Arteries; Cimetidine; Female; Histamine; Male; Membrane Potentials; Muscle Contraction; Muscle, Smooth, Vascular; Muscles; Norepinephrine; Pyrilamine; Rabbits; Receptors, Histamine H1; Receptors, Histamine H2 | 1979 |
[Histamine receptors in the guinea pig papillary muscle].
Topics: Animals; Cimetidine; Epinephrine; Female; Guinea Pigs; Histamine; Male; Papillary Muscles; Pyrilamine; Receptors, Histamine; Thiazoles; Thiourea | 1977 |
The effects of stimulants and inhibitors of histamine receptors on acid secretion from guinea pig gastric fundus.
Topics: Animals; Cimetidine; Female; Gastric Mucosa; Guinea Pigs; Histamine; In Vitro Techniques; Male; Methylhistamines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea; Time Factors | 1978 |
Spasmolytic action of histamine in airway smooth muscle of horse.
Topics: Animals; Atropine; Bronchi; Burimamide; Cimetidine; Histamine; Horses; In Vitro Techniques; Indomethacin; Metiamide; Muscle Contraction; Muscle, Smooth; Propranolol; Pyrilamine; Respiratory System; Trachea | 1978 |
Stimulation of cell proliferation by histamine H2 receptors in dimethylhdrazine-induced adenocarcinomata.
Topics: Adenocarcinoma; Animals; Cell Division; Cimetidine; Colon; Colonic Neoplasms; Dimethylhydrazines; Histamine; Intestinal Mucosa; Male; Metiamide; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H2; Stimulation, Chemical; Thiourea | 1978 |
Effect of histamine and related compounds on the papillary muscle of the guinea pig.
Topics: Animals; Chlorpheniramine; Cimetidine; Female; Guinea Pigs; Histamine; In Vitro Techniques; Male; Metiamide; Myocardial Contraction; Papillary Muscles; Pyrilamine; Structure-Activity Relationship; Verapamil | 1978 |
Effect of dimaprit on gastric acid secretion in conscious cats.
Topics: Animals; Cats; Cimetidine; Gastric Juice; Histamine; Methylhistamines; Pentagastrin; Pyrilamine; Receptors, Histamine H2; Thiourea; Time Factors | 1978 |
The effects of histamine, pyrilamine, cimetidine, and ranitidine on secretion of lingual lipase and amylase from rat von Ebner's glands.
Topics: Amylases; Animals; Cimetidine; Exocytosis; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Lipase; Male; Pyrilamine; Ranitidine; Rats; Rats, Sprague-Dawley; Salivary Glands | 1992 |
Histamine leukocytosis. I. Effect of histamine on peripheral leukocyte counts.
Topics: Animals; Cimetidine; Dogs; Erythrocyte Count; Guanidines; Guinea Pigs; Histamine; Leukocyte Count; Leukocytosis; Osmolar Concentration; Pyrilamine; Rabbits; Waxes | 1992 |
Histamine and calcium are independently regulated intracellular mediators of lymphocyte mitogenesis.
Topics: Animals; Calcium; Calcium Channels; Cell Membrane; Cells, Cultured; Cerebral Cortex; Cimetidine; Concanavalin A; DNA Replication; Histamine; Histamine Antagonists; Kinetics; Lymphocytes; Mice; Mice, Inbred BALB C; Phenyl Ethers; Pyrilamine; Rats; Receptors, Histamine H1; Receptors, Nicotinic; Spleen; Verapamil | 1992 |
The intravenous self-administration of antihistamines by rhesus monkeys.
Topics: Animals; Benzhydryl Compounds; Chlorpheniramine; Cimetidine; Dose-Response Relationship, Drug; Histamine H1 Antagonists; Hydroxyzine; Macaca mulatta; Male; Motivation; Pyrilamine; Self Administration; Substance-Related Disorders; Tripelennamine | 1992 |
Pituitary-adrenal responses to head-up tilt in humans: effect of H1- and H2-receptor blockade.
Topics: Adult; Blood Pressure; Cardiovascular Physiological Phenomena; Cardiovascular System; Cimetidine; Head; Histamine H1 Antagonists; Histamine H2 Antagonists; Hormones; Humans; Hypotension; Male; Pituitary-Adrenal System; Posture; Pyrilamine; Supine Position; Time Factors | 1992 |
Visualization of histamine binding to nuclei.
Topics: Animals; Binding Sites; Cell Membrane; Cell Nucleus; Cimetidine; Corpus Luteum; Endothelium, Vascular; Female; Granulosa Cells; Histamine; Microscopy, Fluorescence; Oocytes; Ovary; Pyrilamine; Rabbits; Staining and Labeling | 1992 |
High dose of histamine required for gastric acid secretion in the common African toad, Bufo regularis.
Topics: Animals; Bufonidae; Carbachol; Cimetidine; Evaluation Studies as Topic; Gastric Acid; Gastric Acidity Determination; Histamine; Injections, Intramuscular; Pyrilamine; Time Factors | 1992 |
Histamine modulates heat stress-induced changes in blood-brain barrier permeability, cerebral blood flow, brain oedema and serotonin levels: an experimental study in conscious young rats.
Topics: Animals; Blood-Brain Barrier; Brain; Brain Edema; Cimetidine; Histamine; Hot Temperature; Male; Organ Specificity; Pyrilamine; Rats; Rats, Wistar; Regional Blood Flow; Serotonin; Stress, Physiological | 1992 |
Histamine H1-receptors mediate endothelium-dependent relaxation of rat isolated pulmonary arteries.
Topics: Animals; Cimetidine; Endothelium, Vascular; Histamine; Indomethacin; Male; Muscle, Smooth, Vascular; Nitric Oxide; Phenylephrine; Pulmonary Artery; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Vasodilation | 1992 |
Endogenous calcitonin gene-related peptide mediates nonadrenergic noncholinergic depressor response to spinal cord stimulation in the pithed rat.
Topics: Animals; Atropine; Blood Pressure; Calcitonin Gene-Related Peptide; Capsaicin; Cimetidine; Electric Stimulation; Male; Peptide Fragments; Propranolol; Pyrilamine; Rats; Rats, Inbred Strains; Spinal Cord; Stimulation, Chemical; Vasodilation | 1992 |
The effects of (R) alpha-methyl histamine on the isolated guinea pig aorta.
Topics: Animals; Aorta; Cimetidine; Female; Guanidines; Guinea Pigs; Histamine; Histamine Antagonists; Imidazoles; Impromidine; Male; Methylhistamines; Muscle, Smooth, Vascular; Potassium; Pyrilamine; Receptors, Histamine; Receptors, Histamine H3; Vasoconstriction; Vasodilation | 1991 |
Characterization of histamine receptors modulating inotropic and biochemical activities in rabbit left atria.
Topics: Animals; Atrial Function; Cardiotonic Agents; Cimetidine; Female; Heart; Heart Atria; Histamine; Hydrolysis; Inositol Phosphates; Male; Myocardial Contraction; Phosphatidylinositols; Pyrilamine; Rabbits; Receptors, Histamine H1; Receptors, Histamine H2; Stimulation, Chemical; Tritium | 1991 |
Mechanisms of platelet activating factor-induced changes in sheep tracheal blood flow.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Azepines; Chromones; Cimetidine; Dose-Response Relationship, Drug; Female; Indomethacin; Methacholine Compounds; Muscle Tonus; Muscle, Smooth; Nedocromil; Platelet Activating Factor; Pyrilamine; Quinolones; Regional Blood Flow; Sheep; Trachea; Triazoles; Vascular Resistance | 1991 |
Peptide leukotriene involvement in pulmonary eosinophil migration upon antigen challenge in the actively sensitized guinea pig.
Topics: Animals; Bronchial Hyperreactivity; Cell Movement; Cimetidine; Eosinophils; Guinea Pigs; Indomethacin; Leukotrienes; Male; Ovalbumin; Propionates; Pyrilamine; Quinolines; Receptors, Immunologic; Receptors, Leukotriene | 1991 |
Cyclic AMP generating systems in vertebrate retina: effects of histamine and an established retinal modulator, dopamine.
Topics: Adenylyl Cyclases; Animals; Cerebral Cortex; Chickens; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dopamine; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Retina; Thiazoles; Thiourea | 1991 |
Does intracellular histamine mediate mast cell histamine release?
Topics: Animals; Cell Membrane Permeability; Cimetidine; Concanavalin A; Histamine; Histamine Release; In Vitro Techniques; Male; Mast Cells; Phosphatidylserines; Pyrilamine; Rats; Rats, Inbred Strains; Saponins | 1990 |
Characterization of cardiovascular events mediated by platelet activating factor during systemic anaphylaxis.
Topics: Anaphylaxis; Animals; Arrhythmias, Cardiac; Azepines; Blood Pressure; Cardiac Output; Cimetidine; Electrocardiography; Female; Guinea Pigs; Heart Rate; Hemodynamics; Histamine; Male; Myocardial Contraction; Ovalbumin; Platelet Activating Factor; Pyrilamine; Triazoles | 1990 |
Enhanced prostaglandin synthesis after ultraviolet injury is mediated by endogenous histamine stimulation. A mechanism for irradiation erythema.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Brompheniramine; Cells, Cultured; Chromatography, High Pressure Liquid; Cimetidine; Cycloheximide; Dinoprostone; Dose-Response Relationship, Radiation; Eicosanoids; Epidermis; Erythema; Histamine; Histamine Release; Humans; In Vitro Techniques; Keratinocytes; Prostaglandins; Pyrilamine; Radiation Injuries, Experimental; Time Factors; Ultraviolet Rays | 1990 |
Hypotension induced by growth-hormone-releasing peptide is mediated by mast cell serotonin release in the rat.
Topics: Analysis of Variance; Animals; Cimetidine; Cyproheptadine; Dose-Response Relationship, Drug; Drug Synergism; Growth Hormone-Releasing Hormone; Histamine H2 Antagonists; Histamine Release; Hormones; Hypotension; Injections, Intravenous; Ketanserin; Male; Mast Cells; Naloxone; Oligopeptides; Pyrilamine; Rats; Rats, Inbred Strains; Serotonin | 1990 |
Histamine acts directly on calcitonin gene-related peptide- and substance P-containing trigeminal ganglion neurons as assessed by calcium influx and immunocytochemistry.
Topics: Animals; Calcitonin Gene-Related Peptide; Calcium; Cells, Cultured; Cimetidine; Fura-2; Histamine; Immunohistochemistry; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Substance P; Trigeminal Ganglion | 1990 |
Histamine receptors in the isolated human middle meningeal artery. A comparison with cerebral and temporal arteries.
Topics: Adult; Cerebral Arteries; Cimetidine; Dose-Response Relationship, Drug; Drug Combinations; Female; Histamine; Humans; In Vitro Techniques; Male; Meningeal Arteries; Middle Aged; Osmolar Concentration; Pyrilamine; Receptors, Histamine; Temporal Arteries; Vasodilation | 1991 |
Interleukin-1 (IL-1) stimulates the release of corticotropin-releasing factor (CRF) from superfused rat hypothalamo-neurohypophyseal complexes (HNC) independently of the histaminergic mechanism.
Topics: Animals; Cimetidine; Corticotropin-Releasing Hormone; Histamine; Histamine Antagonists; Hypothalamo-Hypophyseal System; In Vitro Techniques; Interleukin-1; Male; Median Eminence; Perfusion; Pyrilamine; Radioimmunoassay; Rats; Rats, Inbred Strains | 1991 |
Effects of histamine on spontaneous electrical activity of neurons in rat suprachiasmatic nucleus.
Topics: Action Potentials; Animals; Cimetidine; Circadian Rhythm; Histamine; Male; Neurons; Pyrilamine; Rats; Rats, Inbred Strains; Suprachiasmatic Nucleus | 1991 |
Histamine induces endothelium-dependent relaxation of bovine retinal arteries.
Topics: Acetylcholine; Animals; Cattle; Cimetidine; Dimaprit; Endothelium, Vascular; Histamine; Muscle Relaxation; Pyridines; Pyrilamine; Receptors, Histamine; Retinal Artery; Tachyphylaxis; Thiourea | 1991 |
[Evidence for the presence of histamine H2 receptor on poorly differentiated human gastric cancer cell line, MKN45].
Topics: Adenocarcinoma; Cell Line; Cimetidine; Cyclic AMP; Humans; Pyrilamine; Receptors, Histamine H2; Stomach Neoplasms | 1991 |
The intracerebroventricularly administered mast cells degranulator compound 48/80 increases the pituitary-adrenocortical activity in rats.
Topics: Adrenal Cortex; Animals; Brain; Cimetidine; Corticosterone; Cytoplasmic Granules; Histamine; Hypothalamus; Kinetics; Male; Mast Cells; p-Methoxy-N-methylphenethylamine; Pituitary Gland; Pyrilamine; Rats; Rats, Inbred Strains; Thalamus | 1991 |
Effects of antihistamines on wound healing.
Topics: Animals; Cimetidine; Female; Histamine Antagonists; Male; Promethazine; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Wound Healing | 1991 |
Identification and characterization of histamine H1- and H2-receptors in guinea-pig left atrial membranes by [3H]-mepyramine and [3H]-tiotidine binding.
Topics: Animals; Cimetidine; Female; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Guinea Pigs; Heart Atria; In Vitro Techniques; Kinetics; Male; Membranes; Myocardial Contraction; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2 | 1991 |
Histamine augments colonic secretion in guinea pig distal colon.
Topics: 2-Chloroadenosine; Animals; Bradykinin; Bumetanide; Chlorides; Cimetidine; Colon; Dinoprostone; Electric Stimulation; Guinea Pigs; Hexamethonium; Hexamethonium Compounds; Histamine; In Vitro Techniques; Indomethacin; Kinetics; Male; Masoprocol; Muscle, Smooth; Piroxicam; Pyrilamine; Tetrodotoxin; Vasoactive Intestinal Peptide | 1990 |
Histamine stimulation of mucociliary activity in the rabbit maxillary sinus.
Topics: Animals; Atropine; Cilia; Cimetidine; Dimaprit; Female; Histamine; Histamine H2 Antagonists; Male; Maxillary Sinus; Mucociliary Clearance; Pyrilamine; Rabbits; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Muscarinic; Thiourea | 1990 |
Histamine-induced changes in intracellular calcium in undifferentiated N1E-115 cells.
Topics: Animals; Bradykinin; Calcium; Cell Differentiation; Cell Line; Cimetidine; Histamine; Kinetics; Mice; Neuroblastoma; Pyrilamine; Signal Transduction | 1991 |
The significance of brain histamine and its receptors in opioid stimulation of the pituitary-adrenocortical activity.
Topics: Adrenal Cortex; Animals; beta-Endorphin; Brain; Cimetidine; Corticosterone; Endorphins; Enkephalin, Leucine-2-Alanine; Histamine; Histidine Decarboxylase; Male; Morphine; p-Methoxy-N-methylphenethylamine; Pituitary Gland; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine | 1991 |
Role of histamine in pathophysiology of heat stress in rats.
Topics: Animals; Blood-Brain Barrier; Body Water; Brain; Brain Edema; Cimetidine; Histamine; Hot Temperature; Male; Pyrilamine; Rats; Stress, Physiological | 1991 |
Effect of histamine on human placental chorionic veins: interaction with serotonin.
Topics: Chorion; Cimetidine; Drug Interactions; Female; Histamine; Humans; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Placenta; Pregnancy; Pyrilamine; Serotonin; Veins | 1991 |
Modification by some antagonists of the shape changes of venous endothelial cells in response to inflammatory agents in vitro.
Topics: Aminoquinolines; Animals; Bradykinin; Calcimycin; Calcium; Cimetidine; Endothelium, Vascular; Guinea Pigs; Histamine; Histamine Antagonists; Isoproterenol; Platelet Activating Factor; Pyrilamine; Vena Cava, Inferior | 1990 |
H2 receptors mediate cyclical chloride secretion in guinea pig distal colon.
Topics: Animals; Bumetanide; Chlorides; Cimetidine; Colon; Dimaprit; Guinea Pigs; Histamine; In Vitro Techniques; Intestinal Mucosa; Kinetics; Male; Muscle, Smooth; Pyrilamine; Receptors, Histamine H2; Tetrodotoxin; Thiourea | 1990 |
Antagonistic effect of naloxone on the hypertensive response of intraventricularly administered histamine.
Topics: Animals; Blood Pressure; Cimetidine; Dimaprit; Hemodynamics; Histamine; In Vitro Techniques; Injections, Intraventricular; Male; Naloxone; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Thiourea | 1990 |
Histamine stimulation of surfactant secretion from rat type II pneumocytes.
Topics: Adenylyl Cyclases; Alprenolol; Animals; Cells, Cultured; Cimetidine; Cyclic AMP; Histamine; Isoproterenol; Kinetics; Lung; Male; Phosphatidylcholines; Pulmonary Surfactants; Pyrilamine; Rats; Rats, Inbred Strains | 1990 |
Histamine H3 receptors modulate antigen-induced bronchoconstriction in guinea pigs.
Topics: Animals; Antigens; Bronchoconstriction; Cimetidine; Dose-Response Relationship, Drug; Dose-Response Relationship, Immunologic; Guinea Pigs; Histamine; Immunization; Male; Ovalbumin; Piperidines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Skin Tests | 1990 |
Histamine receptors in brain vessels of guinea-pig: in-vitro pharmacology and ligand binding.
Topics: Animals; Basilar Artery; Brain; Calcium; Calcium Channels; Cerebrovascular Circulation; Chlorpheniramine; Cimetidine; Female; Guinea Pigs; Histamine; In Vitro Techniques; Ligands; Nimodipine; Pyrilamine; Receptors, Histamine; Vasoconstriction | 1990 |
Evidence that an atypical beta-adrenoceptor mediates the inhibition of spontaneous rhythmical contractions of rabbit isolated jejunum induced by ritodrine and salbutamol.
Topics: Albuterol; Animals; Cimetidine; Female; In Vitro Techniques; Jejunum; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Pyrilamine; Rabbits; Receptors, Adrenergic, beta; Ritodrine; Yohimbine | 1990 |
Different histamine actions in proximal and distal human coronary arteries in vitro.
Topics: Adolescent; Adult; Aged; Aged, 80 and over; Aging; Child; Cimetidine; Coronary Vessels; Culture Techniques; Endothelium, Vascular; Female; Histamine; Histamine Antagonists; Humans; Male; Middle Aged; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Pyrilamine; Receptors, Histamine | 1990 |
Effect of histamine and 1,4-methylhistamine on gastric vascular resistance in dogs.
Topics: Animals; Cimetidine; Dogs; Female; Histamine; Kinetics; Male; Methylhistamines; Muscle, Smooth; Perfusion; Pyrilamine; Regional Blood Flow; Stomach; Time Factors; Vascular Resistance | 1990 |
Anti-inflammatory activity of bee venom peptide 401 (mast cell degranulating peptide) and compound 48/80 results from mast cell degranulation in vivo.
Topics: Allergens; Animals; Anti-Inflammatory Agents, Non-Steroidal; Bee Venoms; Carrageenan; Cimetidine; Cytoplasmic Granules; Edema; In Vitro Techniques; Irritants; Male; Mast Cells; Methysergide; Nippostrongylus; p-Methoxy-N-methylphenethylamine; Peptides; Pyrilamine; Rats; Rats, Inbred Strains | 1990 |
Inhibition of human skin fibroblast proliferation by histamine and phorbol esters is mediated by protein kinase C.
Topics: Blood; Cell Division; Cell Line; Cimetidine; Dose-Response Relationship, Drug; Down-Regulation; Enzyme Activation; Fibroblasts; Histamine; Humans; Phorbol Esters; Protein Kinase C; Pyrilamine; Receptors, Histamine H1; Thymidine | 1990 |
Effect of histamine on human bronchial arteries in vitro.
Topics: Adult; Bronchial Arteries; Cimetidine; Dinoprost; Histamine; Humans; In Vitro Techniques; Middle Aged; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Pyrilamine | 1990 |
The spinal cord contains multiple factors causing plasma protein extravasation in the skin.
Topics: Adenosine; Animals; Blood Proteins; Cattle; Chromatography, High Pressure Liquid; Cimetidine; Cyclic AMP; Pyrilamine; Skin; Spinal Cord; Substance P; Tissue Extracts | 1985 |
A study on the aetiology of reserpine ulceration and the antiulcer action of solcoseryl in rat stomach.
Topics: Actihaemyl; Animals; Anti-Ulcer Agents; Atropine; Cimetidine; Gastric Acid; Histamine Release; Male; Mast Cells; Pepsin A; Pyrilamine; Rats; Rats, Inbred Strains; Reserpine; Stomach Ulcer; Tissue Extracts | 1985 |
Histamine involvement in the local and systemic microvascular effects produced by intradermal substance P.
Topics: Animals; Body Temperature; Capillary Permeability; Cimetidine; Dose-Response Relationship, Drug; Ear; Guinea Pigs; Histamine; Injections, Intradermal; Male; Pyrilamine; Receptors, Histamine; Skin; Substance P | 1985 |
5-Carboxamidotryptamine: a potent agonist mediating relaxation and elevation of cyclic AMP in the isolated neonatal porcine vena cava.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Animals, Newborn; Atropine; Cimetidine; Cocaine; Cyclic AMP; Dinoprost; Histamine; In Vitro Techniques; Indomethacin; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Propranolol; Prostaglandins F; Pyrilamine; Serotonin; Serotonin Antagonists; Swine; Vena Cava, Inferior | 1986 |
Acute hemodynamic effects of an antitumoral agent: elliptinium. Involvement of histamine release.
Topics: Alkaloids; Animals; Antineoplastic Agents; Aspirin; Atropine; Blood Pressure; Cardiovascular Physiological Phenomena; Cimetidine; Coronary Circulation; Dogs; Ellipticines; Female; Heart Rate; Hemodynamics; Histamine Release; Male; Myocardial Contraction; Propranolol; Pyrilamine | 1986 |
Particle-induced coronary vasoconstriction in the rat heart: pharmacological investigation of underlying mechanisms.
Topics: Animals; Bicarbonates; Calcium Chloride; Cimetidine; Coronary Circulation; Drug Contamination; Filtration; Heart Arrest, Induced; Isoproterenol; Ketanserin; Magnesium; Male; Methysergide; Phenylephrine; Potassium Chloride; Pyrilamine; Rats; Rats, Inbred Strains; Serotonin; Sodium Chloride | 1986 |
A tachykinin antagonist inhibits gastric emptying and gastrointestinal transit in the rat.
Topics: Animals; Bombesin; Cimetidine; Female; Gastric Emptying; Gastrointestinal Motility; Guanethidine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neuropeptides; Pyrilamine; Rats; Rats, Inbred Strains; Substance P; Tachykinins | 1986 |
Experimental renal anaphylaxis: release of histamine and study of its effect on renal perfusion.
Topics: Anaphylaxis; Animals; Cimetidine; Guinea Pigs; Histamine; Histamine Release; Immune Sera; Immunoglobulin G; Kidney; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Renal Circulation | 1987 |
Mechanism of hematocrit increase induced by the combined administration of morphine and adriamycin: role of histamine release.
Topics: Animals; Capillary Permeability; Cimetidine; Doxorubicin; Drug Synergism; Hematocrit; Histamine Release; Liver; Male; Mice; Morphine; Pyrilamine | 1987 |
Autoinhibition of histamine synthesis mediated by presynaptic H3-receptors.
Topics: Animals; Burimamide; Cerebral Cortex; Cimetidine; Histamine; Histamine Release; Hypothalamus; Hypothalamus, Posterior; Imidazoles; Impromidine; Male; Potassium; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H3; Synaptosomes; Thiazoles | 1987 |
The effects of substance P, histamine and histamine antagonists on somatostatin and gastrin release from the isolated perfused rat stomach.
Topics: Animals; Cimetidine; Gastric Mucosa; Gastrins; Histamine; Histamine Antagonists; In Vitro Techniques; Male; Pyrilamine; Radioimmunoassay; Rats; Rats, Inbred Strains; Somatostatin; Substance P | 1987 |
Changing sensitivity to H1 and H2 receptor antagonists in the growing vasculature.
Topics: Animals; Blood Flow Velocity; Blood Vessels; Capillary Permeability; Cimetidine; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Neovascularization, Pathologic; Prostheses and Implants; Pyrilamine; Rats; Rats, Inbred Strains; Regional Blood Flow | 1988 |
Analysis of the effects of cyclooxygenase and lipoxygenase inhibitors on leukocyte accumulation in the inflammatory site.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Cell Movement; Cimetidine; Cyclooxygenase Inhibitors; Diclofenac; Histamine Release; Indomethacin; Inflammation; Leukocytes; Lipoxygenase Inhibitors; Propionates; Pyrilamine | 1989 |
The effect of cotton bract extract on respiratory glycoconjugate secretion from human airways in vitro.
Topics: Bronchi; Cimetidine; Culture Techniques; Dose-Response Relationship, Drug; Glycoconjugates; Gossypium; Histamine Release; Humans; Indomethacin; Leukotrienes; Lipoxygenase Inhibitors; Mucous Membrane; Plant Extracts; Prostaglandin-Endoperoxide Synthases; Pyrilamine | 1989 |
Hemodynamic side effects of trypanocidal diamidines in rats. Studies on possible antagonisms.
Topics: Amidines; Animals; Blood Pressure; Cell Membrane; Cimetidine; Cromolyn Sodium; Hemodynamics; Male; Pulse; Pyrilamine; Rats; Rats, Inbred Strains; Regional Blood Flow; Trypanocidal Agents | 1989 |
Pharmacological characterization of histamine receptors in the human temporal artery.
Topics: Adult; Cimetidine; Dinoprost; Female; Histamine; Humans; Imidazoles; Impromidine; In Vitro Techniques; Male; Methylhistamines; Middle Aged; Pyridines; Pyrilamine; Receptors, Histamine; Temporal Arteries; Thiazoles; Vasoconstriction; Vasodilation | 1989 |
Role of histamine receptor in mesencephalic nucleus dorsalis raphe in cardiovascular regulation.
Topics: Animals; Cardiovascular Physiological Phenomena; Cats; Cimetidine; Decerebrate State; Female; Fenclonine; Guanethidine; Histamine; Histamine Antagonists; Male; Mesencephalon; Microinjections; Piperoxan; Pyrilamine; Raphe Nuclei; Receptors, Histamine; Vagotomy | 1989 |
Effect of histamine on isolated working guinea pig heart with left ventricular hypertrophy produced by pressure overload.
Topics: Animals; Cardiomegaly; Cimetidine; Dose-Response Relationship, Drug; Guinea Pigs; Heart Function Tests; Histamine; In Vitro Techniques; Male; Norepinephrine; Pyrilamine; Receptors, Histamine H2 | 1989 |
Antagonistic action of naloxone on central histamine receptors-stimulated corticosterone secretion in rats under stress.
Topics: Animals; Cimetidine; Corticosterone; Dimaprit; Histamine; Male; Methylhistamines; Naloxone; Pituitary-Adrenal System; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Restraint, Physical; Stress, Physiological; Thiourea | 1989 |
Demonstration of histamine receptors on the surface of Entamoeba histolytica.
Topics: Animals; Cimetidine; Entamoeba histolytica; Histamine; Pyrilamine; Receptors, Histamine | 1989 |
Neuronal histamine modulates feeding behavior through H1-receptor in rat hypothalamus.
Topics: Animals; Chlorpheniramine; Cimetidine; Drinking Behavior; Famotidine; Feeding Behavior; Histamine; Histamine H2 Antagonists; Hypothalamus; Injections, Intraventricular; Male; Motor Activity; Neurons; Promethazine; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Reference Values; Thiazoles | 1989 |
Involvement of histaminergic neurons in the stress-induced release of pro-opiomelanocortin-derived peptides in rats.
Topics: Adrenocorticotropic Hormone; Animals; beta-Endorphin; beta-Lipotropin; Chromatography, Gel; Cimetidine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Pyrilamine; Pyrimidinones; Rats; Rats, Inbred Strains; Stress, Physiological | 1989 |
Histamine directly acts on beta-adrenoceptors as well as H1-histaminergic receptors, and causes positive inotropic effects in isolated ventricular muscles of carp heart (Cyprinus carpio).
Topics: Animals; Atropine; Carps; Cimetidine; Cyprinidae; Diphenhydramine; Electric Stimulation; Female; Histamine; Histamine Antagonists; In Vitro Techniques; Male; Myocardial Contraction; Propranolol; Pyrilamine; Receptors, Adrenergic, beta; Receptors, Histamine H1; Stereoisomerism | 1989 |
Effect of histamine H2-receptor antagonists on acute inflammatory of the rat paw oedema.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Cimetidine; Edema; Freund's Adjuvant; Histamine; Histamine H2 Antagonists; Male; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Triazoles | 1989 |
Formation of ovarian follicular cysts and corpora lutea after treatment with antihistamine or indomethacin in prepubertal gilts.
Topics: Aging; Animals; Cimetidine; Female; Follicular Phase; Histamine; Histamine H1 Antagonists; Indomethacin; Luteal Phase; Ovarian Cysts; Ovulation; Prostaglandins; Pyrilamine; Swine | 1989 |
HeLa cells have histamine H1-receptors which mediate activation of the K+ conductance.
Topics: Cell Membrane; Cimetidine; Electric Conductivity; Electric Stimulation; HeLa Cells; Histamine; Humans; Ion Channels; Membrane Potentials; Potassium; Pyrilamine; Quinine; Receptors, Histamine; Receptors, Histamine H1 | 1985 |
Role of endogenous opioids and histamine in morphine induced emesis.
Topics: Animals; Cimetidine; Dogs; Endorphins; Histamine; Metiamide; Morphine; Naloxone; Pyrilamine; Vomiting | 1989 |
Role of histamine in traumatic brain edema. An experimental study in the rat.
Topics: Animals; Brain Edema; Brain Injuries; Cimetidine; Histamine; Male; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Wounds, Penetrating | 1989 |
Interactive effects of peptidoleukotrienes and histamine on microvascular permeability and their involvement in experimental cutaneous and conjunctival immediate hypersensitivity.
Topics: Animals; Capillary Permeability; Chromium Radioisotopes; Cimetidine; Conjunctiva; Dicarboxylic Acids; Guinea Pigs; Histamine; Hypersensitivity, Immediate; Iodine Radioisotopes; Leukotrienes; Male; Ovalbumin; Pyrilamine; Skin | 1989 |
Histamine-induced calcium transients in vascular smooth muscle cells: effects of verapamil and diltiazem.
Topics: Aminoquinolines; Animals; Aorta; Calcium; Cell Fractionation; Cells, Cultured; Centrifugation, Density Gradient; Cimetidine; Cytosol; Diltiazem; Fluorescent Dyes; Histamine; Kinetics; Male; Microscopy, Fluorescence; Muscle, Smooth, Vascular; Pyrilamine; Rats; Rats, Inbred Strains; Sarcolemma; Swine; Verapamil | 1989 |
Effects of phorbol esters and forskolin on basal and histamine-induced accumulation of inositol phosphates in cultured bovine adrenal chromaffin cells.
Topics: Adrenal Medulla; Animals; Cattle; Cells, Cultured; Cimetidine; Colforsin; Epinephrine; Histamine; Inositol Phosphates; Kinetics; Norepinephrine; Phorbol Esters; Pyrilamine; Sugar Phosphates; Tetradecanoylphorbol Acetate | 1989 |
Effects of histamine and serotonin on the contractility of isolated pregnant and nonpregnant human myometrium.
Topics: Cimetidine; Dose-Response Relationship, Drug; Drug Interactions; Female; Histamine; Humans; In Vitro Techniques; Ketanserin; Methysergide; Myometrium; Pregnancy; Pyrilamine; Serotonin; Uterine Contraction | 1989 |
Protective effects of histamine H1 and H2 antagonists, adenosine and hydrocortisone on cardiac anaphylaxis.
Topics: Adenosine; Aminopyridines; Anaphylaxis; Animals; Arrhythmias, Cardiac; Cardiac Output; Cimetidine; Guinea Pigs; Heart Rate; Hydrocortisone; In Vitro Techniques; Pyrilamine; Receptors, Histamine | 1989 |
Effect of histamine on human vas deferens in vitro.
Topics: Burimamide; Cimetidine; Culture Techniques; Dose-Response Relationship, Drug; Histamine; Humans; Male; Methylhistamines; Muscle Contraction; Pyrilamine; Vas Deferens | 1989 |
Histamine excites arcuate neurons in vitro through H1 receptors.
Topics: Action Potentials; Animals; Arcuate Nucleus of Hypothalamus; Cimetidine; Female; Histamine; In Vitro Techniques; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine | 1989 |
Effects of histamine on the guinea-pig stomach: excitation of smooth muscle and inhibition of transmitter release.
Topics: Animals; Atropine; Cimetidine; Female; Guinea Pigs; Histamine; In Vitro Techniques; Male; Membrane Potentials; Microelectrodes; Muscle, Smooth; Neuromuscular Junction; Pyrilamine; Stomach; Synaptic Transmission | 1987 |
Angiotensin II-induced relaxation of fowl aorta.
Topics: 5,8,11,14-Eicosatetraynoic Acid; Angiotensin II; Animals; Aorta, Abdominal; Chickens; Cimetidine; Cyclic AMP; Cyclic GMP; In Vitro Techniques; Indomethacin; Methysergide; Microscopy, Electron; Muscle, Smooth, Vascular; Ouabain; Proadifen; Propranolol; Pyrilamine; Vasodilation | 1988 |
Histaminergic systems and sleep. Studies in man with H1 and H2 antagonists.
Topics: Adolescent; Adult; Brompheniramine; Cimetidine; Electroencephalography; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Male; Phenothiazines; Psychomotor Performance; Pyrilamine; Ranitidine; Sleep; Sleep Stages; Sleep, REM; Triprolidine | 1985 |
Synergistic interaction between histamine and ouabain on ventricular fibrillation threshold.
Topics: Animals; Cimetidine; Coronary Circulation; Drug Synergism; Electrocardiography; Guinea Pigs; Heart Rate; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Male; Myocardial Contraction; Ouabain; Pyrilamine; Ventricular Fibrillation | 1985 |
Regulation and actions of gastrointestinal somatostatin.
Topics: Animals; Calcium; Carbachol; Cimetidine; Colon; Egtazic Acid; Feedback; Gastric Mucosa; Gastrins; Histamine; Hydrogen-Ion Concentration; Intestine, Small; Lanthanum; Pimozide; Pyrilamine; Secretory Rate; Somatostatin; Trifluoperazine | 1985 |
Renal vasodilation with ureteral occlusion and prostaglandins: attenuation by histamine H1 antagonists.
Topics: Alprostadil; Animals; Blood Pressure; Bradykinin; Chlorpheniramine; Cimetidine; Dinoprostone; Dogs; Epoprostenol; Female; Glomerular Filtration Rate; Histamine H1 Antagonists; Kidney; Male; Mathematics; Meclofenamic Acid; Methylhistamines; Prostaglandin D2; Prostaglandins; Prostaglandins A; Prostaglandins D; Prostaglandins E; Pyrilamine; Regional Blood Flow; Ureter; Vasodilation | 1985 |
A study of the H2-receptor for histamine stimulating adenylate cyclase in homogenates of guinea-pig lung parenchyma.
Topics: Adenylyl Cyclases; Animals; Cimetidine; Colforsin; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Lung; Male; Propranolol; Pyrilamine; Receptors, Histamine; Receptors, Histamine H2 | 1986 |
Conjunctival eosinophil infiltration evoked by histamine and immediate hypersensitivity. Modification by H1- and H2-receptor blockade.
Topics: Animals; Cell Movement; Cimetidine; Conjunctival Diseases; Eosinophils; Female; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Hypersensitivity, Immediate; Male; Pyrilamine | 1986 |
Histamine and histamine receptors: behavioral thermoregulation in the salamander Necturus maculosus.
Topics: Animals; Body Temperature Regulation; Cimetidine; Dimaprit; Histamine; Histidine; Necturus; Pyridines; Pyrilamine; Receptors, Histamine; Thiourea | 1986 |
Histaminergic stimulation of prolactin secretion mediated via H1- or H2-receptors: dependence on routes of administration.
Topics: Animals; Cimetidine; Dimaprit; Histamine; Histamine H1 Antagonists; Male; Methylhistamines; Pituitary Gland, Anterior; Prolactin; Pyrilamine; Pyrimidinones; Rats; Receptors, Histamine; Thiazoles; Thiourea | 1986 |
Plasmodium berghei-infected mice: lack of effect of meclizine and cimetidine on the development of pulmonary oedema.
Topics: Animals; Capillary Permeability; Cimetidine; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Histamine H1 Antagonists; Malaria; Male; Meclizine; Mice; Plasmodium berghei; Pulmonary Edema; Pyrilamine | 1986 |
[Arrhythmogenic effects of histamine on ischemic hearts of guinea pigs].
Topics: Animals; Arrhythmias, Cardiac; Chlorpheniramine; Cimetidine; Cricetinae; Female; Heart Rate; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Male; Myocardial Infarction; Pyrilamine | 1987 |
Mechanism of histamine-induced epinephrine release in guinea pig.
Topics: Animals; Bronchi; Cimetidine; Decerebrate State; Epinephrine; Guinea Pigs; Hexamethonium; Hexamethonium Compounds; Histamine; Male; Pyrilamine; Sympathectomy, Chemical | 1988 |
Radioautographic characterization of H1 and H2 receptor antagonists. Binding sites in rat gastric mucosal microcirculatory system.
Topics: Animals; Cimetidine; Endothelium, Vascular; Epithelium; Gastric Mucosa; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Microcirculation; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2 | 1988 |
Studies on the site and mechanism of the inhibitory action of intracerebral histamine on the cold-stimulated thyrotropin secretion in male rats.
Topics: Animals; Brain Mapping; Cimetidine; Cold Temperature; Histamine; Hypothalamus; Imidazoles; Impromidine; Injections, Intraventricular; Male; Pyridines; Pyrilamine; Rats; Thyrotropin | 1985 |
Conjunctival immediate hypersensitivity: re-evaluation of histamine involvement in the vasopermeability response.
Topics: Albumins; Animals; Capillary Permeability; Cimetidine; Conjunctiva; Dimaprit; Dose-Response Relationship, Drug; Drug Combinations; Eyelids; Guinea Pigs; Histamine; Histamine Antagonists; Hypersensitivity, Immediate; Imidazoles; Impromidine; Male; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1986 |
Metronidazole and 5-aminosalicylic acid enhance the contractile activity of histaminergic agonists on the guinea-pig isolated ileum.
Topics: Aminosalicylic Acids; Animals; Cimetidine; Computers; Dimaprit; Dose-Response Relationship, Drug; Drug Synergism; Duodenum; Female; Guinea Pigs; Heart; Histamine; Ileum; In Vitro Techniques; Jejunum; Male; Mesalamine; Metronidazole; Muscle Contraction; Myenteric Plexus; Pyrilamine; Receptors, Histamine; Scopolamine; Tetrodotoxin; Thiourea | 1986 |
Participation of vascular H1-receptors in histaminergic relaxation of rabbit middle cerebral artery in vitro.
Topics: Animals; Cerebral Arteries; Cimetidine; Dimaprit; Drug Interactions; Histamine; In Vitro Techniques; Methylhistamines; Muscle Relaxation; Muscle, Smooth, Vascular; Phenethylamines; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Thiourea | 1986 |
Antidromic vasodilatation in the rat hindpaw measured by laser Doppler flowmetry: pharmacological modulation.
Topics: Adrenergic Fibers; Animals; Capsaicin; Cimetidine; Electric Stimulation; Enkephalin, Methionine; Female; Fentanyl; Hindlimb; Lasers; Male; Naloxone; Pyrilamine; Rats; Regional Blood Flow; Rheology; Skin; Vasodilation | 1987 |
Hyperlipemic responses induced by centrally administered histamine H1- and H2-receptor agonists in rats.
Topics: Animals; Brain; Cimetidine; Dimaprit; Fatty Acids, Nonesterified; Hyperlipidemias; Imidazoles; Impromidine; Injections, Intraventricular; Male; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Thiourea | 1987 |
Characterization of histamine receptors in isolated rabbit veins.
Topics: Animals; Cimetidine; Endothelium, Vascular; Female; Histamine; Imidazoles; Impromidine; Male; Pyrilamine; Rabbits; Ranitidine; Receptors, Histamine; Receptors, Histamine H2; Species Specificity; Vasoconstriction; Veins | 1987 |
Endothelium-dependent relaxing effect of histamine on the isolated guinea-pig main pulmonary artery strips.
Topics: Animals; Cimetidine; Endothelium, Vascular; Female; Guinea Pigs; Histamine; Imidazoles; Impromidine; In Vitro Techniques; Male; Muscle Relaxation; Pulmonary Artery; Pyrilamine; Receptors, Histamine H2 | 1987 |
Role of central histaminergic mechanism in behavioural depression (swimming despair) in mice.
Topics: Animals; Atropine; Central Nervous System; Cimetidine; Depression; Desipramine; Disease Models, Animal; Histamine; Imidazoles; Imipramine; Impromidine; Male; Mice; Motor Activity; Pyrilamine; Receptors, Histamine H2 | 1988 |
A highly potent and selective H3 agonist relaxes rabbit middle cerebral artery, in vitro.
Topics: Animals; Cerebral Arteries; Cimetidine; Histamine; Imidazoles; Impromidine; In Vitro Techniques; Male; Methylhistamines; Muscle Relaxation; Muscle, Smooth, Vascular; Potassium; Pyrilamine; Rabbits; Receptors, Histamine | 1988 |
Histamine-induced inositol phospholipid breakdown in the longitudinal smooth muscle of guinea-pig ileum.
Topics: Animals; Cerebellum; Cimetidine; Female; Guinea Pigs; Histamine; Ileum; Imidazoles; Impromidine; In Vitro Techniques; Inositol Phosphates; Kinetics; Male; Muscle Contraction; Phosphatidylinositols; Pyrilamine | 1985 |
Central alpha-2 adrenoceptor-mediated hypertensive response to clonidine in conscious, normotensive rats.
Topics: Animals; Azepines; Blood Pressure; Brain; Cimetidine; Clonidine; Hydroxydopamines; Injections, Intraventricular; Ketanserin; Male; Methoxamine; Oxidopamine; Piperidines; Prazosin; Procaine; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine | 1986 |
Histamine receptor effects on dissipation of an intracellular proton gradient of isolated gastric mucosal surface cells.
Topics: Animals; Bicarbonates; Chlorides; Cimetidine; Dimaprit; Diphenhydramine; Gastric Acid; Gastric Mucosa; Histamine; Protons; Pyridines; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Sodium; Thiourea | 1987 |
Involvement of histamine H1 and H2 receptors in hypothermia induced by ionizing radiation in guinea pigs.
Topics: Animals; Body Temperature; Cimetidine; Cromolyn Sodium; Gamma Rays; Guinea Pigs; Kinetics; Male; Methysergide; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Whole-Body Irradiation | 1988 |
Effect of H1 and H2 agonists on the chemiluminescence of human blood mononuclear cells induced by phytohaemagglutinin.
Topics: Cimetidine; Histamine; Humans; Imidazoles; Impromidine; Luminescent Measurements; Methylhistamines; Monocytes; Phytohemagglutinins; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Structure-Activity Relationship | 1985 |
Characteristics of canine lower esophageal sphincter: a new electrophysiological tool.
Topics: Animals; Carbachol; Cimetidine; Dogs; Electric Stimulation; Electrophysiology; Esophagus; Female; Histamine; In Vitro Techniques; Intercellular Junctions; Male; Microscopy, Electron; Muscle Contraction; Muscle, Smooth; Pirenzepine; Pyrilamine; Reference Values; Tetrodotoxin | 1988 |
Inotropic effect of histamine on papillary muscle of guinea pig with right ventricular hypertrophy.
Topics: Animals; Cardiomyopathy, Hypertrophic; Cimetidine; Epinephrine; Female; Guinea Pigs; Histamine; Male; Myocardial Contraction; Papillary Muscles; Pyrilamine | 1988 |
Changes in the feeding behavior of rats elicited by histamine infusion.
Topics: Animals; Catheterization; Cimetidine; Circadian Rhythm; Dose-Response Relationship, Drug; Feeding Behavior; Histamine; Male; Pyrilamine; Rats; Rats, Inbred Strains; Suprachiasmatic Nucleus | 1988 |
Histaminergic mediation of the stress-induced release of prolactin in male rats.
Topics: Animals; Cimetidine; Ether; Histamine; Injections, Intravenous; Injections, Intraventricular; Male; Prolactin; Pyrilamine; Pyrimidinones; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine; Restraint, Physical; Stress, Physiological | 1988 |
Presynaptic inhibition produced by histamine at nicotinic synapses in enteric ganglia.
Topics: Acetylcholine; Action Potentials; Animals; Cimetidine; Evoked Potentials; Ganglia; Guinea Pigs; Hexamethonium Compounds; Histamine; Intestines; Pyrilamine; Synapses | 1988 |
Mast cell infiltration: a possible mechanism for vein graft vasospasm.
Topics: Animals; Carotid Arteries; Cimetidine; Dose-Response Relationship, Drug; Histamine; Isometric Contraction; Jugular Veins; Male; Mast Cells; Muscle, Smooth, Vascular; Pyrilamine; Rabbits | 1988 |
The influence of histamine at various concentrations on the cell cycle state of hematopoietic stem cells (CFU-s).
Topics: Animals; Bone Marrow; Bone Marrow Cells; Cell Cycle; Cimetidine; Colony-Forming Units Assay; Female; Hematopoietic Stem Cells; Histamine; Male; Mice; Mice, Inbred Strains; Pyrilamine | 1988 |
Electrophysiological and mechanical characteristics of histamine receptors in smooth muscle cells of the guinea-pig ileum.
Topics: Animals; Cimetidine; Electrophysiology; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Membrane Potentials; Microelectrodes; Muscle Contraction; Muscle, Smooth; Potassium Chloride; Pyrilamine; Receptors, Histamine | 1987 |
Is there a prostaglandin involvement in the positive inotropic action of histamine in isolated pregnant rat uterus, apparently mediated via H1-receptors activation?
Topics: Alprostadil; Animals; Aspirin; Chlorpheniramine; Cimetidine; Dinoprost; Dinoprostone; Female; Histamine; Pregnancy; Prostaglandins; Prostaglandins E; Prostaglandins F; Pyrilamine; Quinacrine; Rats; Receptors, Histamine; Receptors, Histamine H1; Stimulation, Chemical; Uterine Contraction | 1987 |
Effect of cimetidine and pyrilamine on histamine-induced ocular surface hyperemia.
Topics: Aminopyridines; Animals; Cimetidine; Drug Therapy, Combination; Eye Diseases; Female; Histamine; Hyperemia; Pyrilamine; Rabbits | 1986 |
Alteration by histamine of the sympathetic nerve-mediated contractions in the bovine ovarian follicle wall in vitro.
Topics: Animals; Cattle; Cimetidine; Electrolytes; Female; Glucose; Histamine; In Vitro Techniques; Methylhistamines; Muscle Contraction; Norepinephrine; Ovary; Proteins; Pyrilamine; Sympathetic Nervous System | 1987 |
Histamine-induced calcium release and phorbol antagonism in cultured airway smooth muscle cells.
Topics: Animals; Benzofurans; Calcium; Cells, Cultured; Cimetidine; Dogs; Dose-Response Relationship, Drug; Fura-2; Histamine; Mathematics; Muscle, Smooth; Nifedipine; Pyrilamine; Receptors, Histamine H1; Tetradecanoylphorbol Acetate; Trachea | 1987 |
Histamine stimulates inositol phosphate accumulation via the H1-receptor in cultured human endothelial cells.
Topics: Cells, Cultured; Cimetidine; Endothelium, Vascular; Female; Histamine; Humans; Inositol; Inositol Phosphates; Kinetics; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Sugar Phosphates; Umbilical Veins | 1987 |
Vasoactive drugs, microvascular permeability, and hemorrhagic pancreatitis in cats.
Topics: Animals; Capillary Permeability; Cats; Cimetidine; Drug Synergism; Female; Hemorrhage; Histamine; Indomethacin; Male; Pancreatitis; Prostaglandins E, Synthetic; Pyrilamine | 1987 |
Histamine affects release and biosynthesis of opioid peptides primarily via H1-receptors in bovine chromaffin cells.
Topics: Adrenal Glands; Animals; Calcium; Cattle; Cells, Cultured; Chromaffin System; Cimetidine; Clemastine; Cobalt; Enkephalin, Leucine; Enkephalin, Methionine; Enkephalins; Gallopamil; Histamine; Histamine Antagonists; Nifedipine; Protein Precursors; Pyrilamine; Ranitidine; Receptors, Histamine; Receptors, Histamine H1; RNA, Messenger | 1987 |
The interaction of ethanol with central histaminergic stimulation of the pituitary-adrenocortical and hyperlipemic activity.
Topics: Animals; Brain; Cimetidine; Corticosterone; Ethanol; Fatty Acids, Nonesterified; Histamine; Male; Pituitary-Adrenal System; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine | 1986 |
Effects of H1- and H2-histamine receptor agonists and antagonists on sleep and wakefulness in the rat.
Topics: Animals; Cimetidine; Diphenhydramine; Electroencephalography; Injections, Intraperitoneal; Injections, Intraventricular; Male; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Sleep, REM; Thiazoles; Wakefulness | 1986 |
Effect of histamine on delayed-type hypersensitivity in mice.
Topics: Adrenalectomy; Animals; Chemotaxis; Cimetidine; Female; Histamine; Hypersensitivity, Delayed; Macrophages; Mice; Mice, Inbred C57BL; Mice, Inbred ICR; Pyrilamine | 1986 |
Histamine induces ovulation in the isolated perfused rat ovary.
Topics: Animals; Cimetidine; Female; Gonadotropins, Equine; Histamine; Luteinizing Hormone; Ovary; Ovulation Induction; Perfusion; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains | 1986 |
Histamine-induced microvascular permeability increases in hamster skin: a response predominantly mediated by H2-receptors.
Topics: Animals; Capillary Permeability; Cimetidine; Cricetinae; Dose-Response Relationship, Drug; Female; Histamine; Kinetics; Male; Mesocricetus; Pyrilamine; Receptors, Histamine H2; Skin | 1986 |
Myocardial and vascular actions of amiloride in spontaneously hypertensive rats.
Topics: Amiloride; Animals; Atropine; Blood Pressure; Cardiovascular System; Cimetidine; Dose-Response Relationship, Drug; Heart Rate; Hypertension; Male; Nephrectomy; Pyrilamine; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Stimulation, Chemical; Sulpiride | 1986 |
Blockade of histamine receptors and thrombin-induced microembolic pulmonary edema in the rat.
Topics: Albumins; Animals; Body Water; Cimetidine; Fibrinolysis; Histamine Antagonists; Male; Microcirculation; Permeability; Pulmonary Edema; Pulmonary Embolism; Pyrilamine; Rats; Rats, Inbred Strains; Thrombin; Tranexamic Acid | 1985 |
Histaminergic regulation of prolactin secretion: dose-response relationship and possible involvement of the dopaminergic system.
Topics: Adult; Cimetidine; Dose-Response Relationship, Drug; Histamine; Humans; Male; Metoclopramide; Prolactin; Pyrilamine; Receptors, Dopamine; Receptors, Histamine H1; Receptors, Histamine H2 | 1986 |
New evidence that the antiestrogen binding site may be a novel growth-promoting histamine receptor (?H3) which mediates the antiestrogenic and antiproliferative effects of tamoxifen.
Topics: Animals; Binding, Competitive; Biological Assay; Cimetidine; Female; Hydroxyzine; Microsomes, Liver; Ovariectomy; Phosphatidylethanolamines; Pyrilamine; Rats; Receptors, Estrogen; Receptors, Histamine; Structure-Activity Relationship; Tamoxifen; Uterus | 1986 |
Binding of 4(5)-[2-(4-azido-2-nitroanilino)ethyl]imidazole to histamine receptors in guinea pig cerebral cortical membranes.
Topics: Animals; Binding, Competitive; Cerebral Cortex; Cimetidine; Guinea Pigs; Histamine; Kinetics; Male; Membranes; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Substrate Specificity; Vas Deferens | 1986 |
Histamine activates H1-receptors to induce cytosolic free calcium transients in cultured vascular smooth muscle cells from rat aorta.
Topics: Aminoquinolines; Animals; Calcium; Cells, Cultured; Cimetidine; Cytosol; Dose-Response Relationship, Drug; Histamine; Kinetics; Muscle, Smooth, Vascular; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H1 | 1986 |
H1-histaminergic activation stimulates inositol-1-phosphate accumulation in chromaffin cells.
Topics: Adrenal Medulla; Animals; Bradykinin; Carbachol; Cattle; Cimetidine; Clemastine; Histamine; Hydrolysis; In Vitro Techniques; Inositol Phosphates; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Sugar Phosphates; Time Factors | 1986 |
A simple technique to simultaneously assess activity at histamine H1- and H2-receptors in vivo.
Topics: Animals; Betahistine; Bronchi; Cimetidine; Female; Guinea Pigs; Heart Rate; Histamine; Male; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2 | 1985 |
Intravenous histamine reduces bombesin-stimulated gastrin release in dogs.
Topics: Animals; Bombesin; Cimetidine; Dogs; Gastric Juice; Gastrins; Histamine; Infusions, Parenteral; Pyrilamine | 1985 |
Involvement of histamine in vascular permeability increase of the rat pleurisy induced by phorbol myristate acetate.
Topics: Animals; Capillary Permeability; Cimetidine; Croton Oil; Drug Interactions; Histamine; Histamine Antagonists; Leukocytes; Male; Methysergide; Phorbols; Pleurisy; Pyrilamine; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Time Factors | 1985 |
Histamine H1- and H2-receptor involvement in eosinophil infiltration and the microvascular changes associated with cutaneous anaphylaxis.
Topics: Animals; Capillary Permeability; Cell Movement; Cimetidine; Drug Combinations; Eosinophils; Guinea Pigs; Male; Passive Cutaneous Anaphylaxis; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Skin | 1985 |
Histamine receptor activation by unsaturated (allyl and propargyl) homologs of histamine.
Topics: Adrenergic Fibers; Animals; Cimetidine; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Muscle Contraction; Myocardial Contraction; Propranolol; Pyrilamine; Receptors, Histamine | 1985 |
Effects of histamine agonists and antagonists on luminol-dependent chemiluminescence of granulocytes.
Topics: Cimetidine; Dimaprit; Granulocytes; Histamine; Histamine Antagonists; Humans; In Vitro Techniques; Luminescent Measurements; Luminol; Pyridazines; Pyridines; Pyrilamine; Ranitidine; Thiourea | 1984 |
Effects of histamine on human isolated heart muscle: comparison with effects of noradrenaline.
Topics: Cimetidine; Dimaprit; Heart; Histamine; Humans; In Vitro Techniques; Myocardial Contraction; Norepinephrine; Propranolol; Pyrilamine; Receptors, Histamine H2; Thiourea | 1980 |
Evaluation of the role of Histamine H1- and H2-receptors in cutaneous inflammation in the guinea-pig produced by histamine and mast cell degranulation.
Topics: Animals; Cimetidine; Dimaprit; Guinea Pigs; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Inflammation; Male; Mast Cells; Mathematics; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Skin; Thiourea; Vasodilation | 1980 |
Effects of histamine receptor antagonists on alkali secretion by lleum.
Topics: Alkalies; Animals; Cimetidine; Histamine; Histamine H1 Antagonists; Ileum; Intestinal Secretions; Pyrilamine; Rabbits; Time Factors | 1981 |
Antagonism of vasodepressor and gastric secretory responses to histamine by the H2-receptor antagonists, ranitidine and cimetidine, in the anaesthetized dog.
Topics: Anesthesia; Animals; Blood Pressure; Cimetidine; Dogs; Dose-Response Relationship, Drug; Female; Furans; Gastric Acid; Guanidines; Histamine; Histamine H2 Antagonists; Male; Pyrilamine; Ranitidine | 1981 |
The effect of ranitidine on gastric acid secretory response curves to histamine, pentagastrin or bethanechol in the dog with a Heidenhain pouch.
Topics: Animals; Bethanechol Compounds; Cimetidine; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Furans; Gastric Acid; Histamine; Histamine H2 Antagonists; Male; Pentagastrin; Pyrilamine; Ranitidine | 1981 |
H2-receptor antagonists protect against aspirin-induced gastric lesions in the rat.
Topics: Animals; Aspirin; Cimetidine; Female; Furans; Gastric Mucosa; Histamine H2 Antagonists; Pyrilamine; Ranitidine; Rats; Stomach Ulcer | 1981 |
Slow-reacting substance from alveolar macrophages--a mechanism of asthma?
Topics: Animals; Asthma; Atropine; Autacoids; Chromones; Cimetidine; Ethers; Guinea Pigs; Indomethacin; Macrophages; Methysergide; Muscle Contraction; Muscle, Smooth; Pyrilamine; Trachea | 1981 |
Brain histamine H1- and H2-receptors and histamine-sensitive adenylate cyclase: effects of antipsychotics and antidepressants.
Topics: Adenylyl Cyclases; Animals; Antidepressive Agents; Antipsychotic Agents; Brain; Cimetidine; Female; Guinea Pigs; Histamine; Male; Pyrilamine; Radioligand Assay; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2 | 1981 |
Effect of H1-and H2-receptor antagonists on cutaneous inflammation evoked by histamine analogues and UV radiation.
Topics: Animals; Body Temperature; Cimetidine; Dermatitis; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Pyrilamine; Skin; Ultraviolet Rays; Vasodilation | 1982 |
An inhibitory effect of histamine on the rat anococcygeus muscle.
Topics: Acetylcholine; Animals; Carbachol; Cimetidine; Dimaprit; Drug Interactions; Guanidines; Histamine; Imidazoles; Impromidine; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Pyrilamine; Rats; Thiourea | 1982 |
Carrageenan-induced oedema in the rat paw - histamine participation.
Topics: Animals; Carrageenan; Cimetidine; Edema; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; p-Methoxy-N-methylphenethylamine; Plethysmography; Pyrilamine; Rats; Rats, Inbred Strains; Time Factors | 1982 |
Effect of histamine H1- and H2-receptor antagonists, steroidal and non-steroidal anti-inflammatory agents on carrageenin-induced inflammation of the guinea-pig ear.
Topics: Animals; Anti-Inflammatory Agents; Body Temperature; Carrageenan; Cimetidine; Ear; Glucocorticoids; Guinea Pigs; Histamine H1 Antagonists; Histamine H2 Antagonists; Indomethacin; Inflammation; Male; Pyrilamine; Time Factors | 1982 |
Histamine receptor agonists and antagonists on granulocyte adherence.
Topics: Cimetidine; Clonidine; Granulocytes; Histamine; Histamine Antagonists; Humans; Pyrilamine | 1982 |
[Effect of antihistaminic preparations on gastric secretion in rats].
Topics: Animals; Benzhydryl Compounds; Carbolines; Cimetidine; Cyproheptadine; Diphenhydramine; Gastric Mucosa; Histamine H1 Antagonists; Male; Pyrilamine; Rats | 1983 |
Evidence for histamine H1 and H2 receptors in guinea-pig oxyntic cells.
Topics: Animals; Carbonic Anhydrases; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Impromidine; In Vitro Techniques; Methylhistamines; Parietal Cells, Gastric; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1983 |
Effects of histamine, H1- and H2-receptor antagonists on the activity of serotonergic neurons in the dorsal raphe nucleus.
Topics: Animals; Brain Stem; Cimetidine; Diphenhydramine; gamma-Aminobutyric Acid; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Metiamide; Neurons; Pyrilamine; Ranitidine; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Serotonin; Synaptic Transmission | 1983 |
Effect of histamine receptor antagonists and indomethacin on implantation in the rabbit.
Topics: Aminopyridines; Animals; Capillary Permeability; Cimetidine; Drug Combinations; Drug Interactions; Embryo Implantation; Female; Histamine H1 Antagonists; Indomethacin; Pregnancy; Pyrilamine; Rabbits; Uterus | 1983 |
The effect of antihistaminics on cataleptogenic action of analgesics and haloperidol.
Topics: Analgesics; Analgesics, Opioid; Animals; Catalepsy; Cimetidine; Diphenhydramine; Drug Interactions; Female; Haloperidol; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Male; Piperidines; Pyrilamine; Rats; Rats, Inbred Strains | 1983 |
The effect of histamine, H1 and H2 agonists, and H1 and H2 antagonists on postprandial pancreatic polypeptide release in dogs.
Topics: Animals; Cimetidine; Dimaprit; Dogs; Food; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Pancreatic Polypeptide; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Secretory Rate; Thiazoles; Thiourea | 1983 |
Relaxation and contraction responses to histamine in the human lung parenchymal strip.
Topics: Cimetidine; Dose-Response Relationship, Drug; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; In Vitro Techniques; Indomethacin; Lung; Metiamide; Muscle Contraction; Muscle Relaxation; Potassium Chloride; Pyrilamine | 1984 |
Evidence for the existence of histamine H1- and H2-receptors on astrocytes of cultured rat central nervous system.
Topics: Aminopyridines; Animals; Astrocytes; Brain Stem; Cells, Cultured; Cimetidine; Histamine; Histamine H1 Antagonists; Membrane Potentials; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Spinal Cord; Thiazoles | 1984 |
Intracellular study of effects of histamine on electrical behaviour of myenteric neurones in guinea-pig small intestine.
Topics: Action Potentials; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine Antagonists; In Vitro Techniques; Intestine, Small; Membrane Potentials; Myenteric Plexus; Neurons; Neurotransmitter Agents; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Serotonin; Thiourea | 1984 |
Practical therapeutics: the use of histamine receptor antagonists in contemporary times.
Topics: Astemizole; Benzhydryl Compounds; Benzimidazoles; Child; Cimetidine; Conjunctivitis, Allergic; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Pyrilamine; Rhinitis, Allergic, Seasonal; Terfenadine | 1984 |
Possible role of histamine in rheumatoid arthritis. Treatment with cimetidine and mepyramine.
Topics: Adolescent; Adult; Aminopyridines; Arthritis, Rheumatoid; Cimetidine; Drug Therapy, Combination; Female; Guanidines; Histamine H1 Antagonists; Histamine Release; Humans; Male; Middle Aged; Pyrilamine | 1981 |
Histamine stimulation of digestive enzyme secretion by in vitro rabbit pancreas.
Topics: Amylases; Animals; Chymotrypsinogen; Cimetidine; Drug Combinations; Histamine; Histamine Antagonists; In Vitro Techniques; Lipase; Pancreas; Pancreatin; Pyrilamine; Rabbits; Stimulation, Chemical; Trypsinogen | 1982 |
Alterations in intradental nerve responsiveness induced by electrical stimulation of the inferior alveolar nerve in the cat.
Topics: Alveolar Process; Animals; Cats; Cimetidine; Dental Pulp; Electric Stimulation; Phentolamine; Pyrilamine; Sodium Chloride; Substance P; Trigeminal Nerve | 1983 |
A substance P antagonist inhibits heat-induced oedema in the rat skin.
Topics: Animals; Cimetidine; Edema; Electric Stimulation; Hot Temperature; Male; Nerve Fibers; Peptide Fragments; Pyrilamine; Rats; Skin; Substance P | 1984 |
In vivo characterization of histamine H1- and H2-receptors in the rat stomach microcirculation.
Topics: Animals; Cimetidine; Imidazoles; Impromidine; Kinetics; Male; Microcirculation; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Stomach | 1983 |
Inhibition of the TSH secretion by histamine in male rats.
Topics: Animals; Cimetidine; Cold Temperature; Histamine; Histamine Antagonists; Histidine; Imidazoles; Impromidine; Male; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thyrotropin; Thyrotropin-Releasing Hormone | 1983 |
Central histaminergic stimulation of pituitary--adrenocortical response in the rat.
Topics: Animals; Cimetidine; Corticosterone; Dimaprit; Dose-Response Relationship, Drug; Histamine; Imidazoles; Impromidine; Male; Pituitary-Adrenal System; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1983 |
Studies on cutaneous vascular permeability in the rat: increases caused by histamine and histamine-like agents.
Topics: Animals; Capillary Permeability; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Histamine; Microcirculation; Pyrilamine; Rats; Regional Blood Flow; Skin; Thiourea | 1984 |
Inhibitory histamine H2-receptor in the guinea-pig urinary bladder.
Topics: Acetylcholine; Animals; Calcium; Choline; Cimetidine; Diphenhydramine; Electric Stimulation; Female; Guinea Pigs; Histamine; Imidazoles; Impromidine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nicotine; Norepinephrine; Pyrilamine; Receptors, Histamine; Receptors, Histamine H2; Scopolamine; Tetrodotoxin; Urinary Bladder | 1984 |
Effects of the H2-receptor agonist dimaprit on lymphocyte responsiveness in vitro.
Topics: Animals; Cells, Cultured; Cimetidine; Dimaprit; Ephedrine; Female; Glucosamine; In Vitro Techniques; Lymphocyte Activation; Lymphocytes; Metoprolol; Phagocytosis; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H2; T-Lymphocytes; T-Lymphocytes, Regulatory; Thiourea; Thymidine | 1984 |
Acute systemic anaphylaxis in adult domestic fowl: evidence for the protective role of H2-histaminergic and beta 2-adrenergic receptors.
Topics: Anaphylaxis; Animals; Blood Pressure; Carotid Arteries; Chickens; Chromones; Cimetidine; Dimaprit; Ethers; Heart Rate; Metiamide; Poultry Diseases; Propranolol; Pyrilamine; Receptors, Adrenergic; Receptors, Adrenergic, beta; Receptors, Histamine; Receptors, Histamine H2; Terbutaline; Thiourea | 1980 |
Histamine and human parathyroid adenoma: effect on adenosine 3',5'-monophosphate accumulation in vitro.
Topics: Adenoma; Cimetidine; Cyclic AMP; Female; Histamine; Humans; In Vitro Techniques; Isoproterenol; Male; Parathyroid Hormone; Parathyroid Neoplasms; Propranolol; Pyrilamine | 1981 |
Chick retinal pigment epithelium. A new culture system for studying H2-histamine receptors.
Topics: Animals; Cells, Cultured; Chick Embryo; Cimetidine; Cyclic AMP; Diphenhydramine; Histamine; Methods; Pigment Epithelium of Eye; Pyrilamine; Receptors, Histamine; Receptors, Histamine H2 | 1983 |
Hypothermic and antipyretic effects of ACTH (1-24) and alpha-melanotropin in guinea-pigs.
Topics: Adrenocorticotropic Hormone; Animals; Body Temperature; Bucladesine; Cimetidine; Cosyntropin; Dinoprostone; Guinea Pigs; Injections, Intraventricular; Male; Melanocyte-Stimulating Hormones; Methylhistamines; Methysergide; Norepinephrine; Prostaglandins E; Pyrilamine | 1984 |
Pharmacological prevention of ocular inflammation induced by lens proteins.
Topics: Aminopyridines; Animals; Catechols; Cimetidine; Crystallins; Disease Models, Animal; Drug Therapy, Combination; Endophthalmitis; Female; Indomethacin; Masoprocol; Pyrilamine; Rabbits | 1984 |
Histamine-induced paradoxical growth hormone response to thyrotropin-releasing hormone in normal men.
Topics: Adult; Cimetidine; Growth Hormone; Histamine; Humans; Infusions, Parenteral; Male; Pyrilamine; Thyrotropin; Thyrotropin-Releasing Hormone | 1984 |
Modulation of basal and LRH-stimulated gonadotrophin secretion by histamine in normal men.
Topics: Animals; Cimetidine; Drug Interactions; Follicle Stimulating Hormone; Gonadotropin-Releasing Hormone; Histamine; Luteinizing Hormone; Male; Pituitary Gland, Anterior; Pyrilamine | 1984 |
A method for measuring changes in tracheal mucus gel layer thickness as an indication of an immediate hypersensitivity response.
Topics: Acetylcysteine; Aluminum Hydroxide; Animals; Atropine; Chromones; Cimetidine; Cromolyn Sodium; Dose-Response Relationship, Immunologic; Expectorants; Hypersensitivity, Immediate; Immune Sera; Methods; Methysergide; Mucus; Ovalbumin; Pyrilamine; Rats; Rats, Inbred Strains; Trachea | 1984 |
Further experiments on the pharmacological actions of ergometrine.
Topics: Animals; Cattle; Cimetidine; Coronary Vessels; Dimaprit; Ergonovine; Gastric Acid; Guinea Pigs; Histamine; Muscle Contraction; Pyrilamine; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea | 1981 |
The role of histamine and serotonin in the inflammatory reaction in an experimental model of open wounds in the rat.
Topics: Animals; Capillary Permeability; Cimetidine; Granulation Tissue; Histamine; Histamine Antagonists; Inflammation; Male; Methysergide; Pyrilamine; Rats; Rats, Inbred Strains; Regional Blood Flow; Serotonin Antagonists; Serum Albumin; Wound Healing | 1984 |
Effects of histamine antagonists on noradrenaline-stimulated blood flow and oxygen consumption of brown adipose tissue in the rat.
Topics: Adipose Tissue, Brown; Animals; Body Temperature Regulation; Cimetidine; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Male; Norepinephrine; Oxygen Consumption; Pyrilamine; Rats; Rats, Inbred Strains; Regional Blood Flow | 1984 |
Analgesic effect of histamine induced by intracerebral injection into mice.
Topics: Analgesics; Animals; Benzoquinones; Cimetidine; Diphenhydramine; Electric Stimulation; Enkephalin, Leucine; Histamine; Histamine Antagonists; Male; Mice; Mice, Inbred Strains; Morphine; Naloxone; Promethazine; Pyrilamine; Quinones; Reaction Time | 1984 |
Motor responses to prostaglandin F2 alpha in isolated guinea pig fundus and antrum.
Topics: Animals; Atropine; Cimetidine; Dinoprost; Dose-Response Relationship, Drug; Gastric Fundus; Gastrointestinal Motility; Guinea Pigs; Neural Pathways; Prostaglandins F; Pyloric Antrum; Pyrilamine; Receptors, Cholinergic; Receptors, Histamine | 1983 |
Direct and indirect effects of histamine on the smooth muscle cells of the guinea-pig main pulmonary artery.
Topics: Action Potentials; Animals; Cimetidine; Female; Guinea Pigs; Histamine; Male; Muscle Contraction; Muscle, Smooth, Vascular; Neuromuscular Depolarizing Agents; Neuromuscular Junction; Norepinephrine; Pulmonary Artery; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2 | 1983 |
Effects of histamine and the histamine antagonists mepyramine and cimetidine on human coronary arteries in vitro.
Topics: Adolescent; Adult; Aged; Aminopyridines; Child; Cimetidine; Coronary Vessels; Histamine; Humans; In Vitro Techniques; Middle Aged; Muscle Contraction; Muscle Relaxation; Potassium; Pyrilamine | 1983 |
Action of dimethindene on the electrophysiological and mechanical properties of atrial and ventricular myocardium of guinea-pig.
Topics: Action Potentials; Animals; Cimetidine; Dimethindene; Electrophysiology; Guinea Pigs; In Vitro Techniques; Muscles; Myocardial Contraction; Papillary Muscles; Phentolamine; Pindolol; Pyrilamine; Stimulation, Chemical | 1983 |
Ocular disposition of topically applied histamine, cimetidine, and pyrilamine in the albino rabbit.
Topics: Administration, Topical; Aminopyridines; Animals; Aqueous Humor; Biological Availability; Ciliary Body; Cimetidine; Conjunctiva; Cornea; Eye; Histamine; Iris; Male; Pyrilamine; Rabbits | 1984 |
The influence of age on the distribution and activity of histamine receptors in the rat uterus.
Topics: Aging; Animals; Carbachol; Cimetidine; Electric Stimulation; Female; Histamine; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Uterine Contraction; Uterus | 1984 |
Histamine H2-binding studies in the guinea-pig brain.
Topics: Animals; Brain Chemistry; Cimetidine; Female; Guinea Pigs; Male; Pyrilamine; Radioligand Assay; Receptors, Histamine; Receptors, Histamine H2; Tritium | 1984 |
Effect of histamine on aorta preparations of different species.
Topics: Acetylcholine; Animals; Aorta, Thoracic; Cats; Cimetidine; Guinea Pigs; Histamine; In Vitro Techniques; Mice; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Pyrilamine; Rabbits; Rats; Species Specificity | 1984 |
Histamine antagonists modify systemic digoxin cardiotoxicity by their central action.
Topics: Aminopyridines; Animals; Arrhythmias, Cardiac; Brain; Cats; Cimetidine; Digoxin; Female; Pyrilamine; Time Factors | 1984 |
Histamine regulation of prolactin secretion through H1- and H2-receptors.
Topics: Cimetidine; Histamine; Humans; Male; Prolactin; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Tachycardia; Thyrotropin-Releasing Hormone | 1982 |
Role of the endothelium in the vasodilator response of rat thoracic aorta to histamine.
Topics: Acetylcholine; Animals; Aorta, Thoracic; Atropine; Cimetidine; Endothelium; Histamine; In Vitro Techniques; Male; Norepinephrine; Pyrilamine; Rats; Vasodilation | 1983 |
Bile salt-induced gastric mucosal damage and histamine receptor antagonists.
Topics: Aminopyridines; Animals; Biological Transport; Cimetidine; Dogs; Gastric Mucosa; Guanidines; Hydrogen-Ion Concentration; Male; Potassium; Pyrilamine; Sodium; Stomach; Taurocholic Acid | 1983 |
Relaxation of isolated rabbit veins mediated by latent histamine H2-receptors.
Topics: Animals; Cimetidine; Dose-Response Relationship, Drug; Histamine; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H2; Veins | 1983 |
The effect of histamine, antihistamines, and a mast cell stabilizer on the growth of cloudman melanoma cells in DBA/2 mice.
Topics: Animals; Chromones; Cimetidine; Histamine; Histamine Antagonists; Immunosuppression Therapy; Male; Mast Cells; Melanoma; Methysergide; Mice; Mice, Inbred DBA; Neoplasms, Experimental; Pyrilamine | 1983 |
Histamine stimulate prostacyclin synthesis in cultured human umbilical vein endothelial cells.
Topics: Cimetidine; Dose-Response Relationship, Drug; Endothelium; Epoprostenol; Female; Histamine; Humans; Kinetics; Pregnancy; Prostaglandins; Pyrilamine; Umbilical Veins | 1980 |
Measurement of canine gastric vascular permeability to plasma proteins in the normal and protein-losing states.
Topics: Animals; Blood Proteins; Capillary Permeability; Cimetidine; Dithiothreitol; Dogs; Fibrinogen; Gastric Mucosa; Histamine; Histamine Antagonists; Papaverine; Protein-Losing Enteropathies; Pyrilamine; Salicylates; Salicylic Acid; Serum Albumin, Radio-Iodinated | 1982 |
Effects of histamine on the resting and stimulation-induced release of [3H]-noradrenaline in guinea-pig isolated atria.
Topics: Animals; Atropine; Cimetidine; Cocaine; Electric Stimulation; Female; Guinea Pigs; Heart Atria; Histamine; In Vitro Techniques; Indomethacin; Male; Myocardium; Norepinephrine; Phentolamine; Propranolol; Pyrilamine | 1982 |
The actions of cimetidine hydrochloride and mepyramine maleate in rat adjuvant arthritis.
Topics: Aminopyridines; Animals; Arthritis; Arthritis, Experimental; Cimetidine; Guanidines; Male; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine H2 | 1982 |
Vascular endothelium and the relaxation effect of histamine on aorta of the rat.
Topics: Acetylcholine; Animals; Aorta, Thoracic; Atropine; Cimetidine; Endothelium; Histamine; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Pyrilamine; Rats | 1982 |
Intracerebroventricular aconitine induced cardiac arrhythmia: involvement of central histaminergic receptors.
Topics: Aconitine; Aconitum; Animals; Arrhythmias, Cardiac; Blood Pressure; Cimetidine; Dogs; Heart; Heart Rate; Injections, Intraventricular; Propranolol; Pyrilamine; Receptors, Histamine | 1982 |
Effects of histamine on the circulatory system.
Topics: Animals; Cardiovascular System; Cats; Chlorpheniramine; Cimetidine; Dogs; Hemodynamics; Histamine; Humans; Pyrilamine; Time Factors | 1982 |
Histamine H-1 receptors on rat peritoneal mast cells.
Topics: Aminopyridines; Animals; Ascitic Fluid; Binding, Competitive; Cimetidine; Diphenhydramine; Histamine; Male; Mast Cells; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1 | 1982 |
Inhibition of electrically induced twitch responses of the guinea-pig ileum by histamine.
Topics: Acetylcholine; Animals; Cimetidine; Electric Stimulation; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Pyrilamine | 1980 |
Temperature dependent receptor interconversion hypothesis: chronotropic histamine receptors in isolated guineapig atria.
Topics: Aminopyridines; Animals; Atrial Function; Cimetidine; Female; Guanidines; Guinea Pigs; Heart; Heart Atria; Heart Rate; Male; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Temperature | 1980 |
The direct excitatory effects of cimetidine on the smooth muscle of guinea pig ileum.
Topics: Acetylcholine; Animals; Atropine; Cimetidine; Female; Guanidines; Guinea Pigs; Ileum; In Vitro Techniques; Magnesium; Male; Muscle Contraction; Muscle, Smooth; Physostigmine; Pyrilamine; Receptors, Muscarinic | 1981 |
[The effect of histamine on smooth muscle cells of the artery of the ear in rabbits].
Topics: Animals; Cimetidine; Female; Histamine; Male; Membrane Potentials; Muscle Contraction; Muscle, Smooth, Vascular; Pyrilamine; Rabbits; Receptors, Histamine H1; Receptors, Histamine H2 | 1981 |
Effect of histamine on the gastric smooth muscles of guinea pig.
Topics: Acetylcholine; Animals; Cimetidine; Guinea Pigs; Histamine; Male; Muscle Contraction; Muscle, Smooth; Papaverine; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Stomach | 1981 |
Quantitation of phototoxic hyperemia and permeability to protein. I. Inhibition by histamine (H1 and H2) and serotonin receptor antagonists in pig skin.
Topics: Animals; Anthracenes; Capillary Permeability; Cimetidine; Erythema; Female; Histamine Antagonists; Male; Methysergide; Photosensitivity Disorders; Pyrilamine; Swine; Ultraviolet Rays | 1980 |
Identification of histamine H1- and H-2-receptors by means of mepyramine, cimetidine and theophylline in the cardiovascular system of the dog.
Topics: Animals; Cardiovascular System; Cimetidine; Dogs; Female; Hemodynamics; Histamine; Male; Organ Specificity; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Theophylline | 1980 |
The effect of histamine and histamine antagonists on gastric acid secretion and mucosal blood flow in man.
Topics: Adult; Cimetidine; Dose-Response Relationship, Drug; Gastric Juice; Gastric Mucosa; Histamine; Histamine Antagonists; Humans; Male; Pyrilamine; Regional Blood Flow; Secretory Rate | 1980 |
Antihistamine effect on synaptosomal uptake of serotonin, norepinephrine and dopamine.
Topics: Animals; Cimetidine; Diphenhydramine; Dopamine; Female; Histamine Antagonists; In Vitro Techniques; Kinetics; Norepinephrine; Promethazine; Pyrilamine; Rats; Serotonin; Synaptosomes | 1980 |
Quantitation of phototoxic hyperemia and permeability to protein: II. Inhibition by histamine (H1 and H2) receptor antagonists in mouse skin.
Topics: Animals; Anthracenes; Blood Circulation; Capillary Permeability; Cimetidine; Female; Hyperemia; Male; Mice; Mice, Nude; Photosensitivity Disorders; Pyrilamine; Skin; Ultraviolet Rays | 1980 |
Histamine stimulates brain phospholipid turnover through a direct, H-1 receptor-mediated mechanism.
Topics: Animals; Brain; Catecholamines; Cimetidine; Histamine; Male; Mast Cells; Methylhistamines; p-Methoxy-N-methylphenethylamine; Phosphates; Phospholipids; Pyridines; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H1; Reserpine | 1980 |
A dual action of histamine on isolated human pulmonary arteries.
Topics: Cimetidine; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Humans; In Vitro Techniques; Muscle Contraction; Muscle Tonus; Muscle, Smooth, Vascular; Pulmonary Artery; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2 | 1980 |
Effects of histamine on porcine isolated myocardium: differentiation from effects on human tissue.
Topics: Adolescent; Adult; Analysis of Variance; Animals; Child; Cimetidine; Dose-Response Relationship, Drug; Female; Heart Atria; Heart Ventricles; Histamine; Humans; In Vitro Techniques; Male; Myocardial Contraction; Norepinephrine; Propranolol; Pyrilamine; Swine | 1993 |
Aminoguanidine selectively inhibits inducible nitric oxide synthase.
Topics: Acetylcholine; Amino Acid Oxidoreductases; Animals; Arginine; Cimetidine; Endothelium, Vascular; Endotoxins; Enzyme Induction; Guanidines; In Vitro Techniques; Indomethacin; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide Synthase; omega-N-Methylarginine; Phenylephrine; Pulmonary Artery; Pyrilamine; Rats; Rats, Wistar | 1993 |
Antihistaminergic pretreatment prevents tissue extravasation of albumin from intra-abdominal trauma in rats.
Topics: Abdominal Injuries; Abdominal Muscles; Anesthesia, General; Animals; Ascitic Fluid; Blood Pressure; Capillary Permeability; Chloralose; Cimetidine; Heart Rate; Hematocrit; Histamine Release; Iodine Radioisotopes; Laparotomy; Mast Cells; Pancreas; Plasma; Plasma Volume; Pyrilamine; Rats; Rats, Wistar; Serum Albumin; Tissue Distribution | 1994 |
Possible participation of histamine H3-receptors in the regulation of anaphylactic histamine release from isolated rat peritoneal mast cells.
Topics: Anaphylaxis; Animals; Anticonvulsants; Chromatography, High Pressure Liquid; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Histamine; Histamine Agonists; Histamine Antagonists; Histamine Release; In Vitro Techniques; L-Lactate Dehydrogenase; Male; Mast Cells; Methylhistamines; p-Methoxy-N-methylphenethylamine; Peritoneal Cavity; Peritoneum; Piperidines; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H3 | 1994 |
Histamine enhances granulocyte-macrophage colony-stimulating factor and interleukin-6 production by human peripheral blood mononuclear cells.
Topics: Antibodies; Cell Adhesion; Cells, Cultured; Cimetidine; Enzyme-Linked Immunosorbent Assay; Granulocyte-Macrophage Colony-Stimulating Factor; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Interleukin-3; Interleukin-6; Kinetics; Leukocytes, Mononuclear; Pyrilamine; Radioimmunoassay; Ranitidine; Stem Cells; Stimulation, Chemical; Terfenadine | 1995 |
R-alpha-methylhistamine-induced inhibition of gastric acid secretion in pylorus-ligated rats via central histamine H3 receptors.
Topics: Animals; Cimetidine; Female; Gastric Acid; Gastric Mucosa; Histamine Agonists; Histamine Antagonists; Injections, Intraventricular; Methylhistamines; Piperidines; Pylorus; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H3 | 1995 |
Recepto-secretory mechanism in histamine-stimulated amylase release from rat parotid gland.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Amylases; Animals; Azepines; Calmodulin; Cimetidine; Culture Techniques; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Isoquinolines; Male; Myosin-Light-Chain Kinase; Parotid Gland; Piperazines; Protein Kinase C; Pyrilamine; Rats; Rats, Wistar; Sulfonamides | 1995 |
Histaminergic modulation of synaptic plasticity in area CA1 of rat hippocampal slices.
Topics: Animals; Cimetidine; Dose-Response Relationship, Drug; Hippocampus; Histamine; Long-Term Potentiation; Male; N-Methylaspartate; Pyrilamine; Rats; Rats, Wistar; Synaptic Transmission; Time Factors | 1995 |
Acute stimulation of glucose transport by histamine in cardiac microvascular endothelial cells.
Topics: Adenosine Diphosphate; Animals; Biological Transport; Cells, Cultured; Cimetidine; Coronary Vessels; Deoxyglucose; Endothelium, Vascular; Glucose; Glucose Transporter Type 1; Glucose Transporter Type 4; Histamine; Insulin; Male; Monosaccharide Transport Proteins; Muscle Proteins; Pyrilamine; Rats; RNA, Messenger; Sulfhydryl Compounds | 1995 |
Posterior hypothalamic control of rabbit tracheal tension and involvement of central histaminergic neurons.
Topics: Animals; Blood Pressure; Cimetidine; Electric Stimulation; Histamine; Hypothalamus, Posterior; Muscle Contraction; Neurons; Pyrilamine; Rabbits; Trachea | 1995 |
Dimaprit, a histamine H2-agonist, inhibits anaphylactic histamine release from mast cells and the decreased release is restored by thioperamide (H3-antagonist), but not by cimetidine (H2-antagonist).
Topics: Anaphylaxis; Animals; Anticonvulsants; Betahistine; Cimetidine; Dimaprit; Histamine H2 Antagonists; Histamine Release; In Vitro Techniques; Indicators and Reagents; Male; Mast Cells; Piperidines; Pyrilamine; Rats; Rats, Wistar | 1993 |
Glucocorticoids enhance histamine-evoked catecholamine secretion from bovine chromaffin cells.
Topics: Androstanols; Animals; Base Sequence; Catecholamines; Cattle; Cells, Cultured; Chromaffin System; Cimetidine; Dexamethasone; Glucocorticoids; Histamine; Molecular Sequence Data; Pyrilamine; Receptors, Histamine H1; RNA, Messenger | 1995 |
Characterization and function of histamine receptors in corpus cavernosum.
Topics: Acetylcholine; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Papaverine; Penis; Piperidines; Pyrilamine; Rabbits; Receptors, Histamine; Thiazoles | 1995 |
Regulation of K+ conductance by histamine H1 and H2 receptors in neurones dissociated from rat neostriatum.
Topics: Animals; Cimetidine; Dose-Response Relationship, Drug; Famotidine; Female; Histamine; Histamine Agonists; Impromidine; In Vitro Techniques; Ion Transport; Male; Membrane Potentials; Methylhistamines; Neostriatum; Potassium; Potassium Channels; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Triprolidine | 1994 |
Histamine-independent modulation of the neuropeptide Y-induced pressor response by alpha-trinositol in the pithed rat.
Topics: Animals; Antihypertensive Agents; Blood Pressure; Cimetidine; Decerebrate State; Diphenhydramine; Electric Stimulation; Heart Rate; Histamine Antagonists; Injections, Intravenous; Inositol Phosphates; Male; Neuropeptide Y; Phenylephrine; Pyrilamine; Rats; Rats, Sprague-Dawley; Vasopressins | 1994 |
Effects of histamine on inositol phosphates and intracellular Ca2+ in human glomerular epithelial cells.
Topics: Calcium; Cells, Cultured; Cimetidine; Cytophotometry; Enzyme Activation; Epithelial Cells; Epithelium; Histamine; Humans; Inositol Phosphates; Kidney Glomerulus; Protein Kinase C; Pyrilamine; Second Messenger Systems | 1994 |
Histamine receptors mediating a positive inotropic effect in guinea pig and rabbit ventricular myocardium: distribution of the receptors and their possible intracellular coupling processes.
Topics: Adenylyl Cyclases; Animals; Cimetidine; Guinea Pigs; Heart Ventricles; Histamine; Hydrolysis; Myocardial Contraction; Myocardium; Papillary Muscles; Phosphatidylinositols; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2 | 1994 |
Mechanisms of antihistamine-induced sedation in the human brain: H1 receptor activation reduces a background leakage potassium current.
Topics: Cerebral Cortex; Cimetidine; Evoked Potentials; Histamine; Histamine Antagonists; Humans; Hypnotics and Sedatives; Membrane Potentials; Neurons; Piperidines; Potassium Channels; Pyrilamine; Receptors, Histamine H1 | 1994 |
Enhancement of cardiac performance of isolated working guinea pig heart by rabbit platelet and involvement of histamine.
Topics: Animals; Blood Platelets; Cimetidine; Guinea Pigs; Heart Rate; Histamine; In Vitro Techniques; Mast Cells; Myocardial Contraction; Pyrilamine; Rabbits | 1993 |
Dehydration-induced release of vasopressin involves activation of hypothalamic histaminergic neurons.
Topics: Animals; Arginine Vasopressin; Blood; Cimetidine; Dehydration; Histamine; Hypothalamus; Male; Methylhistamines; Methylhistidines; Neurons; Osmolar Concentration; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H2 | 1994 |
Central mediation of tracheal pressure through H1 and H2 receptors after histamine administration to the fourth ventricle of anesthetized rabbit.
Topics: Animals; Atropine; Blood Pressure; Cimetidine; Histamine; Injections, Intraventricular; Phentolamine; Pressure; Pyrilamine; Rabbits; Receptors, Histamine H1; Receptors, Histamine H2; Trachea | 1994 |
Exposure to heavy charged particles affects thermoregulation in rats.
Topics: Alpha Particles; Animals; Argon; Body Temperature Regulation; Cimetidine; Helium; Indomethacin; Iron Radioisotopes; Male; Neon; Pyrilamine; Rats; Rats, Sprague-Dawley | 1994 |
A neuroprotective effect of histamine H1 receptor antagonist on ischemia-induced decrease in 2-deoxyglucose uptake in rat hippocampal slices.
Topics: Animals; Brain Ischemia; Cimetidine; Deoxyglucose; Hippocampus; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Male; Pyrilamine; Rats; Rats, Wistar | 1993 |
Changes in plasma adrenocorticotropic hormone and cortisol levels induced by intracerebroventricular injection of histamine and its related compounds in dogs.
Topics: Adrenocorticotropic Hormone; Animals; Cimetidine; Dogs; Hexamethonium; Hexamethonium Compounds; Histamine; Hydrocortisone; Hypophysectomy; Injections, Intraventricular; Male; Methylhistamines; Pyrilamine | 1993 |
The study of histamine H1- and H2-receptors in human lung cancer.
Topics: Adenocarcinoma; Adult; Airway Obstruction; Chronic Disease; Cimetidine; Humans; Lung Neoplasms; Middle Aged; Neoplasm Proteins; Pneumonia; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Tuberculoma; Tuberculosis, Pulmonary | 1993 |
Role of mast cell histamine in brown adipose tissue thermogenic response to VMH stimulation.
Topics: Adipocytes; Adipose Tissue, Brown; Animals; Body Temperature Regulation; Cimetidine; Electric Stimulation; Female; Histamine; Male; Mast Cells; Norepinephrine; Oxygen Consumption; Pyrilamine; Rats; Rats, Inbred Strains; Tissue Distribution; Ventromedial Hypothalamic Nucleus | 1994 |
Histamine lipolytic activity and semicarbazide-sensitive amine oxidase (SSAO) of rat white adipose tissue (WAT).
Topics: Adipose Tissue; Amine Oxidase (Copper-Containing); Animals; Benzylamines; Cimetidine; Histamine; Isoproterenol; Kinetics; Lipolysis; Male; Methylhistamines; Pyrilamine; Rats; Rats, Wistar; Semicarbazides | 1993 |
Histamine stimulates normal human melanocytes in vitro: one of the possible inducers of hyperpigmentation in urticaria pigmentosa.
Topics: Adult; Cells, Cultured; Cimetidine; Glycoproteins; Histamine; Humans; Hyperpigmentation; Imidazoles; Male; Melanocytes; Membrane Glycoproteins; Monophenol Monooxygenase; Oxidoreductases; Pyrilamine; Reference Values; Urticaria Pigmentosa | 1993 |
Effect of histamine on memory retrieval in old rats.
Topics: Acetylcholine; Aging; Animals; Anticonvulsants; Avoidance Learning; Cerebrovascular Circulation; Cimetidine; Dose-Response Relationship, Drug; Exploratory Behavior; Histamine; Histamine Agonists; Injections, Intraventricular; Male; Memory; Methylhistamines; Motor Activity; Piperidines; Pyrilamine; Rats; Rats, Wistar | 1993 |
Insulin/hypoglycemia-induced adrenocorticotropin and beta-endorphin release: involvement of hypothalamic histaminergic neurons.
Topics: Adrenocorticotropic Hormone; Animals; beta-Endorphin; Cetirizine; Cimetidine; Histamine; Histamine Agonists; Histamine Antagonists; Hypoglycemia; Hypothalamus; Insulin; Male; Methylhistamines; Neurons; Pyrilamine; Pyrimidinones; Rats; Rats, Wistar | 1993 |
Cis-urocanic acid stimulates human peripheral blood monocyte prostaglandin E2 production and suppresses indirectly tumor necrosis factor-alpha levels.
Topics: Brompheniramine; Cells, Cultured; Cimetidine; Cyclic AMP; Dinoprostone; Diphenhydramine; Histamine; Humans; In Vitro Techniques; Interleukin-1; Interleukin-6; Lipopolysaccharides; Monocytes; Pyrilamine; Second Messenger Systems; Stereoisomerism; Tumor Necrosis Factor-alpha; Urocanic Acid | 1993 |
Altered response to histamine in brain tumor vessels: the selective increase of regional cerebral blood flow in transplanted rat brain tumor.
Topics: Animals; Blood Pressure; Blood-Brain Barrier; Brain Neoplasms; Capillary Permeability; Cerebral Arteries; Cerebrovascular Circulation; Cimetidine; Glioma; Histamine; Infusions, Intra-Arterial; Male; Neoplasm Transplantation; Pyrilamine; Rats; Rats, Wistar | 1993 |
Characterization of histamine receptors in isolated pig basilar artery by functional and radioligand binding studies.
Topics: Animals; Basilar Artery; Cimetidine; Histamine; In Vitro Techniques; Pyrilamine; Radioligand Assay; Receptors, Histamine H1; Receptors, Histamine H2; Vasoconstriction | 1993 |
Adenosine is a mediator of ethanol-induced gastric vasodilation in dogs.
Topics: Adenosine; Animals; Cimetidine; Dogs; Ethanol; Histamine; Indomethacin; Male; Muscle, Smooth; Purinergic Antagonists; Pyrilamine; Regional Blood Flow; Stomach; Theophylline; Vascular Resistance; Vasodilation | 1993 |
Histamine H1 receptor binding sites in mouse uterine horns.
Topics: Animals; Cimetidine; Estrus; Female; Gonadal Steroid Hormones; Histamine; In Vitro Techniques; Kinetics; Membranes; Mice; Ovariectomy; Pregnancy; Pyrilamine; Receptors, Histamine H1; Uterus | 1993 |
Characterization of neurogenic inflammation in the airways of two highly inbred rat strains.
Topics: Animals; Benzamides; Blood Pressure; Bronchi; Capillary Permeability; Capsaicin; Cimetidine; Coloring Agents; Dose-Response Relationship, Drug; Evans Blue; Histamine Antagonists; Indoles; Inflammation; Isoindoles; Methysergide; Neurokinin-1 Receptor Antagonists; Piperidines; Pyrilamine; Rats; Rats, Inbred F344; Rats, Inbred Strains; Receptors, Neurokinin-1; Serotonin; Serotonin Antagonists; Substance P; Trachea | 1995 |
Increases in cyclic AMP levels couple to H1 receptors in atria from autoimmune myocarditis mice.
Topics: Animals; Autoimmune Diseases; Cimetidine; Cyclic AMP; Heart Atria; Histamine; Histamine Agonists; Histamine Antagonists; Male; Mice; Myocarditis; Phosphatidylinositols; Pyrilamine; Receptors, Histamine H1; Signal Transduction; Thiazoles | 1995 |
Parathyroid hormone induces a rapid increase in the number of active osteoclasts by releasing histamine from mast cells.
Topics: Animals; Cell Degranulation; Cimetidine; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine Release; Mast Cells; Microscopy, Fluorescence; Osteoclasts; Parathyroid Hormone; Pyrilamine; Rats; Rats, Wistar | 1996 |
Involvement of central histamine in the early phase of ACTH and corticosterone responses to endotoxin in rats.
Topics: Adrenocorticotropic Hormone; Animals; Cimetidine; Corticosterone; Escherichia coli; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Kinetics; Lipopolysaccharides; Male; Median Eminence; Methylhistamines; Pyrilamine; Rats; Rats, Sprague-Dawley | 1996 |
Effect of oxitropium bromide on histamine-induced airway goblet cell secretion.
Topics: Administration, Inhalation; Aerosols; Animals; Atropine; Cimetidine; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine Antagonists; Histocytochemistry; Injections, Intravenous; Male; Mucus; Muscarinic Antagonists; Piperidines; Pyrilamine; Receptors, Histamine; Scopolamine Derivatives; Trachea; Vagus Nerve | 1996 |
Hippocampal somatostatin receptors and modulation of adenylyl cyclase activity in histamine-treated rats.
Topics: Adenylyl Cyclases; Animals; Cerebral Ventricles; Cimetidine; Colforsin; Dose-Response Relationship, Drug; Guanylyl Imidodiphosphate; Hippocampus; Histamine; Injections, Intraperitoneal; Injections, Intraventricular; Kinetics; Pyrilamine; Rats; Rats, Wistar; Receptors, Somatostatin; Somatostatin; Time Factors | 1996 |
EFFECTS OF HISTAMINE AND RELATED COMPOUNDS ON THE BOVINE IRIS DILATOR.
Topics: Analysis of Variance; Animals; Cattle; Chlorpheniramine; Cimetidine; Diphenhydramine; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Ileum; Iris; Lethal Dose 50; Male; Methylhistamines; Muscle Contraction; Muscle, Smooth; p-Methoxy-N-methylphenethylamine; Piperidines; Potassium; Pyrilamine; Ranitidine; Receptors, Histamine H1; Substance P | 1996 |
Sensitivity of histamine H3 receptor agonist-stimulated [35S]GTP gamma[S] binding to pertussis toxin.
Topics: Animals; Cerebral Cortex; Cimetidine; Guanosine 5'-O-(3-Thiotriphosphate); Histamine Agonists; Histamine H2 Antagonists; In Vitro Techniques; Male; Methylhistamines; Pertussis Toxin; Protein Binding; Pyrilamine; Radioligand Assay; Rats; Receptors, Histamine H3; Sulfur Radioisotopes; Virulence Factors, Bordetella | 1996 |
Histamine augments VCAM-1 expression on IL-4- and TNF-alpha-stimulated human umbilical vein endothelial cells.
Topics: Amanitins; Antibodies, Blocking; Antigens, CD; Cell Adhesion; Cells, Cultured; Cimetidine; Eosinophils; Histamine; Histamine Antagonists; Humans; Immunohistochemistry; Integrin alpha4; Interleukin-4; Piperidines; Platelet Activating Factor; Pyrilamine; Tumor Necrosis Factor-alpha; Umbilical Veins; Vascular Cell Adhesion Molecule-1 | 1996 |
Histamine activates phospholipase C in human airway epithelial cells via a phorbol ester-sensitive pathway.
Topics: Calcium; Calcium-Transporting ATPases; Cell Line; Cimetidine; Cystic Fibrosis; Enzyme Activation; Enzyme Inhibitors; Epithelium; GTP-Binding Proteins; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Inositol Phosphates; Pertussis Toxin; Protein Kinase C; Pyrilamine; Receptors, Histamine H1; Signal Transduction; Thapsigargin; Trachea; Type C Phospholipases; Virulence Factors, Bordetella | 1996 |
Decrease in plasma volume from intra-abdominal trauma in rats is prevented by H1 but not by H2 histaminergic blockade.
Topics: Abdomen; Animals; Cimetidine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Plasma Volume; Pyrilamine; Rats; Rats, Wistar | 1996 |
Circadian rhythm photic phase shifts are not altered by histamine receptor antagonists.
Topics: Animals; Benzothiazoles; Cimetidine; Circadian Rhythm; Cricetinae; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Mesocricetus; Phenoxypropanolamines; Photoperiod; Piperidines; Pyrilamine; Receptors, Histamine H3; Thiazoles | 1996 |
"In vivo" and "in vitro" antitumoral action of Larrea divaricata Cav.
Topics: Analysis of Variance; Animals; Antineoplastic Agents, Phytogenic; Carcinoma; Cell Division; Cimetidine; Cyclic AMP; Female; Histamine; Lymphoma, T-Cell; Mammary Neoplasms, Animal; Phytotherapy; Plant Extracts; Plants, Medicinal; Pregnancy; Propranolol; Pyrilamine; Rats; Thymidine | 1996 |
Stimulation of formation of adenosine 3',5'-phosphate by histamine in myenteric ganglia isolated from guinea-pig small intestine.
Topics: Animals; Cimetidine; Cyclic AMP; Ganglia; Guinea Pigs; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Intestine, Small; Male; Myenteric Plexus; Pyrilamine; Signal Transduction; Stimulation, Chemical; Tripelennamine | 1996 |
Histamine H2 receptor-mediated airway goblet cell secretion and its modulation by histamine-degrading enzymes.
Topics: Amine Oxidase (Copper-Containing); Animals; Asthma; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glycoproteins; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine N-Methyltransferase; Male; Methylhistamines; Mucus; Piperidines; Pyrilamine; Recombinant Proteins; Trachea | 1997 |
Release of calcitonin gene-related peptide in cardiac anaphylaxis.
Topics: 6-Ketoprostaglandin F1 alpha; Anaphylaxis; Animals; Calcitonin Gene-Related Peptide; Cimetidine; Coronary Circulation; Cyclooxygenase Inhibitors; Guinea Pigs; Heart; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Indomethacin; Leukotriene C4; Lipoxygenase Inhibitors; Myocardium; Ovalbumin; Pyrilamine; Quinolines; Thromboxane B2 | 1997 |
Neuropeptides, radiation, and thermoregulation.
Topics: Adrenocorticotropic Hormone; Animals; Body Temperature; Body Temperature Regulation; Cimetidine; Dinoprostone; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Histamine H1 Antagonists; Histamine H2 Antagonists; Methysergide; Neurotensin; Pyrilamine; Pyrogens; Radiation, Ionizing; Rats; Serotonin Antagonists | 1997 |
Human mast cell tryptase: a stimulus of microvascular leakage and mast cell activation.
Topics: Animals; Capillary Permeability; Chromatography, Affinity; Chymases; Cimetidine; Dose-Response Relationship, Drug; Drug Interactions; Evans Blue; Extravasation of Diagnostic and Therapeutic Materials; Guinea Pigs; Heparin; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Hot Temperature; Humans; Inflammation Mediators; Injections, Intravenous; Lung; Mast Cells; Protease Inhibitors; Pyrilamine; Serine Endopeptidases; Skin; Tryptases | 1997 |
Action of ebrotidine, ranitidine and cimetidine on the specific binding to histamine H1- and H2-receptors.
Topics: Animals; Benzenesulfonates; Cell Membrane; Cerebellum; Cerebral Cortex; Cimetidine; Depression, Chemical; Guinea Pigs; Histamine H2 Antagonists; In Vitro Techniques; Isotope Labeling; Male; Protein Binding; Pyrilamine; Ranitidine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Tritium | 1997 |
Evidence for the involvement of histaminergic neurones in the regulation of the rat oxytocinergic system during pregnancy and parturition.
Topics: Afferent Pathways; Animals; Cimetidine; Female; Histamine; Histamine Antagonists; Histidine Decarboxylase; In Situ Hybridization; Labor, Obstetric; Lactation; Mammillary Bodies; Neurons; Oxytocin; Paraventricular Hypothalamic Nucleus; Pregnancy; Pregnancy, Animal; Pyrilamine; Rats; Rats, Wistar; RNA, Messenger | 1997 |
The effects of neurotransmitter antagonists and glucose on luteinizing hormone secretion in growth-restricted wethers.
Topics: Animals; Cimetidine; Cyproheptadine; Food Deprivation; Glucose; Luteinizing Hormone; Male; Neurotransmitter Agents; Pimozide; Propranolol; Pyrilamine; Sheep | 1997 |
Atypical association of H1 and H2 histamine receptors with signal transduction pathways during multistage mouse skin carcinogenesis.
Topics: 9,10-Dimethyl-1,2-benzanthracene; Animals; Cell Count; Cimetidine; Cyclic AMP; Female; Histamine H1 Antagonists; Histamine H2 Antagonists; Hydrolysis; Mast Cells; Mice; Phosphatidylinositols; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Second Messenger Systems; Signal Transduction; Skin Neoplasms; Tetradecanoylphorbol Acetate | 1997 |
H1 and H2 histamine receptors modulate osteoclastic resorption by different pathways: evidence obtained by using receptor antagonists in a rat synchronized resorption model.
Topics: Animals; Bone Resorption; Carboxylesterase; Carboxylic Ester Hydrolases; Cell Degranulation; Cimetidine; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Histocytochemistry; Male; Mast Cells; Microcirculation; Osteoclasts; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H2 | 1997 |
[Possible involvement of histamine in humoral regulation of the spontaneous contractile activity of the chick embryo amnion].
Topics: Amnion; Animals; Chick Embryo; Cimetidine; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Muscle Contraction; Muscle, Smooth; Promethazine; Pyrilamine | 1997 |
Effect of histamine on human fibroblast in vitro.
Topics: Cell Division; Cells, Cultured; Cimetidine; Collagen; DNA; Fibroblasts; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Pyrilamine | 1997 |
Two components of blood-brain barrier disruption in the rat.
Topics: Animals; Arachidonic Acid; Blood-Brain Barrier; Bucladesine; Calcitonin Gene-Related Peptide; Cerebrovascular Circulation; Cimetidine; Cyclic AMP; Dura Mater; Female; Fluorescent Dyes; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Hydrogen-Ion Concentration; Isoproterenol; Isoquinolines; Male; Pia Mater; Pyrilamine; Rats; Rats, Wistar; Sympathomimetics; Time Factors | 1997 |
Comparison of responses to T-kinin and bradykinin in the mesenteric vascular bed of the cat.
Topics: Adamantane; Analysis of Variance; Animals; Bradykinin; Bradykinin Receptor Antagonists; Cats; Cimetidine; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Female; Histamine Antagonists; Male; Meclofenamic Acid; Mesentery; Morpholines; NG-Nitroarginine Methyl Ester; Piperidines; Potassium Channels; Pyrilamine | 1997 |
PACAP-induced plasma extravasation in rat skin.
Topics: Albuterol; Animals; Bucladesine; Capillary Permeability; Cimetidine; Dose-Response Relationship, Drug; Histamine Antagonists; Neuropeptides; Pituitary Adenylate Cyclase-Activating Polypeptide; Pyrilamine; Rats; Rats, Inbred F344; Skin; Specific Pathogen-Free Organisms; Substance P; Vasoactive Intestinal Peptide; Vasodilator Agents | 1997 |
Effects of acute glucose overload on histamine H2 receptor-mediated Ca2+ mobilization in bovine cerebral endothelial cells.
Topics: Animals; Bradykinin; Brain; Bucladesine; Calcium; Cattle; Cells, Cultured; Cimetidine; Cyclic AMP; Dose-Response Relationship, Drug; Endothelium, Vascular; Glucose; Histamine; Histamine Antagonists; Homeostasis; Microcirculation; Neomycin; Neurotransmitter Agents; Protein Kinase C; Pyrilamine; Ranitidine; Receptors, Histamine H2; Staurosporine | 1998 |
Regulation of cerebral microvascular permeability by histamine in the anaesthetized rat.
Topics: Anesthesia, General; Animals; Capillary Permeability; Cerebrovascular Circulation; Cimetidine; Dimaprit; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Muscle, Smooth, Vascular; Pia Mater; Pyrilamine; Rats; Venules | 1998 |
Regulation of H1-receptor coupling and H1-receptor mRNA by histamine in bovine tracheal smooth muscle.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Cattle; Cimetidine; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Indoles; Indomethacin; Maleimides; Muscle, Smooth; Pyrilamine; Receptors, Histamine H1; RNA, Messenger; Trachea | 1998 |
Substituted pyrido[3,2-b]oxazin-3(4H)-ones: synthesis and evaluation of antinociceptive activity.
Topics: Analgesics; Animals; Benzeneacetamides; Cimetidine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Guinea Pigs; Histamine Antagonists; Male; Mice; Models, Chemical; Nociceptors; Oxazines; Pyridines; Pyrilamine; Pyrrolidines; Receptors, Opioid; Structure-Activity Relationship | 1998 |
Histamine-induced synthesis and secretion of nerve growth factor from astrocytes.
Topics: Animals; Animals, Newborn; Astrocytes; Cells, Cultured; Cimetidine; Dose-Response Relationship, Drug; Enzyme-Linked Immunosorbent Assay; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Interleukin-1; Nerve Growth Factors; Pyrilamine; Rats; Rats, Wistar | 1998 |
Histamine receptors in human epithelial cells--characterization of the receptor G-protein-effector system.
Topics: Breast; Cell Line; Cimetidine; Epithelial Cells; Female; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Inositol; Models, Theoretical; Phosphatidylinositols; Pyrilamine; Radioligand Assay; Receptors, Cell Surface; Receptors, Histamine | 1998 |
Histamine receptors signalling in epidermal tumor cell lines with H-ras gene alterations.
Topics: 9,10-Dimethyl-1,2-benzanthracene; Animals; Carcinogens; Cimetidine; Cyclic AMP; Gene Expression Regulation, Neoplastic; Genes, ras; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Inositol Phosphates; Keratinocytes; Mice; Mutation; Oncogene Protein p21(ras); Pyrilamine; Receptors, Histamine; Second Messenger Systems; Signal Transduction; Tumor Cells, Cultured | 1998 |
Thioperamide, a histamine H3-receptor blocker, facilitates vasopressor response to footshocks.
Topics: Animals; Antihypertensive Agents; Blood Pressure; Cimetidine; Electric Stimulation; Enzyme Inhibitors; Heart Rate; Hindlimb; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistidines; Norepinephrine; Phentolamine; Piperidines; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Vasoconstrictor Agents | 1998 |
Roles of histamine receptor in a guinea pig asthma model.
Topics: Animals; Asthma; Cimetidine; Disease Models, Animal; Guinea Pigs; Histamine Antagonists; Lung; Male; Pyrilamine; Radioligand Assay; Receptors, Histamine H1; Receptors, Histamine H2 | 1998 |
Analysis of an H1 receptor-mediated, zinc-potentiated vasoconstrictor action of the histidyl dipeptide carnosine in rabbit saphenous vein.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Carnosine; Cimetidine; Drug Interactions; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Indomethacin; Ketanserin; Methiothepin; Muscle Contraction; Muscle Relaxation; Pyrilamine; Rabbits; Radioligand Assay; Receptors, Histamine H1; Receptors, Histamine H2; Saphenous Vein; Serotonin Antagonists; Vasoconstrictor Agents; Zinc | 1998 |
The role of histamine H1, H2 and H3 receptors on enteric ascending synaptic transmission in the guinea pig ileum.
Topics: Animals; Cimetidine; Dimaprit; Electric Stimulation; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Ileum; Male; Motor Neurons; Muscle Contraction; Muscle, Smooth; Pyrilamine; Receptors, Histamine; Synaptic Transmission | 1998 |
Role of the endothelium in the vasorelaxing influence of histamine on isolated human subcutaneous resistance arteries.
Topics: Adipose Tissue; Arteries; Cimetidine; Endothelium, Vascular; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Muscle Relaxation; Nitric Oxide; Pyrilamine | 1999 |
Histaminergic and catecholaminergic interactions in the central regulation of vasopressin and oxytocin secretion.
Topics: Animals; Arginine Vasopressin; Blood Pressure; Cerebral Ventricles; Cimetidine; Epinephrine; Histamine; Histamine Agonists; Hypothalamus; Imidazoles; Infusions, Parenteral; Male; Methylhistamines; Norepinephrine; Oxytocin; Pituitary Gland, Posterior; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H2; Thiazoles; Thiourea | 1999 |
Molecular properties of central and peripheral histamine H1 and H2 receptors.
Topics: Animals; Astrocytes; Binding, Competitive; Cattle; Cells, Cultured; Cerebral Cortex; Cimetidine; Endothelium, Vascular; Histamine H1 Antagonists; Histamine H2 Antagonists; Muscle, Smooth, Vascular; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H2 | 2000 |
Mepyramine but not cimetidine or clobenpropit blocks pertussis toxin-induced histamine sensitization in rats.
Topics: Animals; Blood Gas Analysis; Blood Pressure; Cimetidine; Drug Interactions; Histamine; Histamine Antagonists; Imidazoles; Male; Pertussis Toxin; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine; Thiourea; Virulence Factors, Bordetella | 2000 |
Involvement of tyrosine phosphorylation in the positive inotropic effect produced by H(1)-receptors with histamine in guinea-pig left atrium.
Topics: Animals; Atrial Function; Chlorpheniramine; Cimetidine; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Genistein; Guinea Pigs; Heart Atria; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Isoflavones; Isoproterenol; Male; Myocardial Contraction; Phosphorylation; Protein-Tyrosine Kinases; Pyrilamine; Receptors, Histamine H1; Time Factors; Tyrosine; Tyrphostins | 2000 |
Identification of a histamine H(3)-like receptor in the zebrafish (Danio rerio) brain.
Topics: Animals; Autoradiography; Brain; Cimetidine; Female; Guanosine 5'-O-(3-Thiotriphosphate); Histamine Agonists; Histamine Antagonists; Imidazoles; Kinetics; Male; Methylhistamines; Piperidines; Pyrilamine; Radioligand Assay; Receptors, Histamine H3; Sulfur Radioisotopes; Thiourea; Tritium; Zebrafish | 2000 |
Cholinergic and glutamatergic activation reverses working memory failure by hippocampal histamine H1 receptor blockade in rats.
Topics: Acetylcholine; Animals; Cholinesterase Inhibitors; Cimetidine; Cycloserine; Drug Interactions; Glutamic Acid; Hippocampus; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Memory; Memory Disorders; Neurons; Physostigmine; Pyridines; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, N-Methyl-D-Aspartate | 2000 |
Effects of drugs acting as histamine releasers or histamine receptor blockers on an experimental anxiety model in mice.
Topics: Animals; Anxiety; Cimetidine; Disease Models, Animal; Histamine Antagonists; Histamine Release; Injections, Intraperitoneal; Injections, Intraventricular; Male; Mice; p-Methoxy-N-methylphenethylamine; Piperidines; Pyrilamine | 2000 |
Molecular cloning and characterization of a new human histamine receptor, HH4R.
Topics: Amino Acid Sequence; Binding, Competitive; Cell Line; Cimetidine; Cloning, Molecular; Colforsin; Cyclic AMP; Histamine Agonists; Histamine Antagonists; Humans; Leukocytes; Methylhistamines; Molecular Sequence Data; Pyrilamine; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H3; Receptors, Histamine H4; Recombinant Proteins; Sequence Alignment; Sequence Homology, Amino Acid; Stereoisomerism; Transfection | 2000 |
The major role of peripheral release of histamine and 5-hydroxytryptamine in formalin-induced nociception.
Topics: Animals; Anti-Asthmatic Agents; Cimetidine; Cromolyn Sodium; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Indoles; Male; Meclizine; Neurons, Afferent; Nociceptors; p-Methoxy-N-methylphenethylamine; Pain; Pain Measurement; Piperazines; Pyrilamine; Rats; Rats, Wistar; Serotonin; Serotonin Antagonists; Tropisetron | 2001 |
Role of mast cells in zymosan-induced peritoneal inflammation in Balb/c and mast cell-deficient WBB6F1 mice.
Topics: Animals; Anti-Asthmatic Agents; Cimetidine; Cromolyn Sodium; Histamine Antagonists; Hypoglycemic Agents; Mast Cells; Mice; Mice, Inbred BALB C; Mice, Knockout; Peritonitis; Pyrilamine; Ranitidine; Receptors, Histamine; Triprolidine; Zymosan | 2001 |
Regulation of parasympathetic neurons by mast cells and histamine in the guinea pig heart.
Topics: Action Potentials; Animals; Cimetidine; Female; Ganglia, Parasympathetic; Guinea Pigs; Heart; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Immunohistochemistry; Male; Mast Cells; Microtubule-Associated Proteins; Neurons; Ovalbumin; Pyrilamine; Receptors, Histamine; Vagus Nerve | 2001 |
Histamine-Induced increases in intracellular free Ca2+ levels in hepatoma cells.
Topics: Biological Transport; Calcium; Carcinoma, Hepatocellular; Cimetidine; Cytosol; Extracellular Space; Fluorescent Dyes; Fura-2; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Inositol 1,4,5-Trisphosphate; Liver Neoplasms; Pyrilamine; Tumor Cells, Cultured | 2000 |
The effects of histamine and its antagonists on the cochlear microphonic and the compound action potential of the guinea pig.
Topics: Administration, Topical; Animals; Cimetidine; Cochlea; Dose-Response Relationship, Drug; Evoked Potentials; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Pyrilamine; Tympanic Membrane | 2001 |
Characterization of histamine-induced increases in intracellular free Ca2+ concentrations in Chang liver cells.
Topics: Calcium; Calcium Signaling; Calcium-Transporting ATPases; Cell Line; Cimetidine; Extracellular Space; Fluorescent Dyes; Fura-2; Hepatocytes; Histamine; Humans; Inositol 1,4,5-Trisphosphate; Intracellular Fluid; Kinetics; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Spectrometry, Fluorescence; Thapsigargin | 2001 |
Enhancement by histamine of vascular endothelial growth factor production in granulation tissue via H(2) receptors.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Cells, Cultured; Cimetidine; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Endothelial Growth Factors; Enzyme Inhibitors; Fibroblasts; Gene Expression Regulation; Granulation Tissue; Histamine; Histamine Antagonists; Immunohistochemistry; Indoles; Indomethacin; Inflammation; Isoquinolines; Lymphokines; Macrophages, Peritoneal; Male; Maleimides; Naphthalenes; Neovascularization, Pathologic; Piperidines; Protein Kinase C; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine H2; RNA, Messenger; Specific Pathogen-Free Organisms; Sulfonamides; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors | 2001 |
Histamine-induced IL-6 and IL-8 production are differentially modulated by IFN-gamma and IL-4 in human keratinocytes.
Topics: Benzimidazoles; Cells, Cultured; Cimetidine; Dose-Response Relationship, Drug; Drug Combinations; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Interferon-gamma; Interleukin-4; Interleukin-6; Interleukin-8; Keratinocytes; Pyrilamine | 2002 |
Mouse mammary epithelial cells bear histamine receptors.
Topics: Animals; Binding Sites; Cimetidine; Epithelial Cells; Female; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Mammary Glands, Animal; Methylhistamines; Mice; Mice, Inbred BALB C; Pyrilamine; Radiopharmaceuticals; Receptors, Histamine | 2002 |
The initial inositol 1,4,5-trisphosphate response induced by histamine is strongly amplified by Ca(2+) release from internal stores in smooth muscle.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Androstadienes; Animals; Calcium; Carbachol; Cimetidine; Extracellular Space; Guinea Pigs; Histamine; Histamine Agonists; Inositol 1,4,5-Trisphosphate; Kinetics; Lithium; Muscle, Smooth; Pyrilamine; Ryanodine; Thapsigargin; Type C Phospholipases; Urinary Bladder; Wortmannin | 2002 |
The control effect of histamine on body temperature and respiratory function in IgE-dependent systemic anaphylaxis.
Topics: Allergens; Anaphylaxis; Animals; Blood Pressure; Body Temperature; Cimetidine; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine Decarboxylase; Immunization, Passive; Immunoglobulin E; Mast Cells; Mice; Mice, Knockout; Pyrilamine; Respiratory Function Tests; Tidal Volume; Trinitrobenzenes | 2002 |
Histamine h(4) and h(2) receptors control histamine-induced interleukin-16 release from human CD8(+) T cells.
Topics: Base Sequence; CD4-Positive T-Lymphocytes; CD8-Positive T-Lymphocytes; Cells, Cultured; Cimetidine; Dimaprit; DNA Primers; Female; Gene Expression Regulation; Histamine; Humans; Interleukin-16; Male; Methylhistamines; Polymerase Chain Reaction; Pyrilamine; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H2; Receptors, Histamine H4 | 2002 |
Histamine H1 receptors in rat dorsal raphe nucleus: pharmacological characterisation and linking to increased neuronal activity.
Topics: Action Potentials; Animals; Brain Stem; Cimetidine; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Inositol Phosphates; Male; Neurons; Pyrilamine; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Histamine H1; Serotonin | 2002 |
Murine tumor necrosis factor-alpha sensitizes plasma corticosterone activity and the manifestation of shock: modulation by histamine.
Topics: Animals; Anti-Inflammatory Agents; Biogenic Monoamines; Cimetidine; Corticosterone; Dexamethasone; Diphenhydramine; Histamine; Histamine Antagonists; Hypothalamus; Male; Mice; Pyrilamine; Receptors, Histamine; Shock; Tumor Necrosis Factor-alpha | 2002 |
Histaminergic modulation of the intact respiratory network of adult mice.
Topics: Animals; Cimetidine; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Hypoxia; Medulla Oblongata; Mice; Mice, Inbred C57BL; Nerve Net; Neurons; Phrenic Nerve; Piperidines; Pons; Pyrilamine; Receptors, Histamine H3; Respiratory System | 2003 |
Effects of histamine and cholinergic systems on memory retention of passive avoidance learning in rats.
Topics: Acetylcholine; Animals; Avoidance Learning; Cimetidine; Dose-Response Relationship, Drug; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Memory; Muscarinic Antagonists; Nicotine; Pyrilamine; Rats; Rats, Wistar; Reaction Time; Receptors, Cholinergic; Receptors, Histamine; Retention, Psychology; Scopolamine | 2003 |
Abolition of arteriolar dilation but not constriction to histamine in cremaster muscle of eNOS-/- mice.
Topics: Animals; Arterioles; Cimetidine; Endothelium, Vascular; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Mice; Mice, Inbred C57BL; Mice, Inbred Strains; Muscle, Skeletal; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Nitric Oxide Synthase Type III; Platelet Endothelial Cell Adhesion Molecule-1; Pyrilamine; Receptors, Histamine; Signal Transduction; Vasoconstriction; Vasodilation | 2003 |
Influence of histamine, cimetidine and pyrilamine on naloxone-induced jumping in morphine-dependent mice.
Topics: Animals; Atropine; Cimetidine; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Combinations; Drug Interactions; Histamine; Histamine H2 Antagonists; Injections, Intraperitoneal; Injections, Intraventricular; Injections, Subcutaneous; Mice; Morphine; Morphine Dependence; Motor Activity; Naloxone; Prazosin; Propranolol; Pyrilamine; Receptors, Histamine H2; Yohimbine | 2003 |
The histamine H2-receptor antagonist, cimetidine, inhibits the articular osteopenia in rats with adjuvant-induced arthritis by suppressing the osteoclast differentiation induced by histamine.
Topics: Animals; Arthritis, Experimental; Bone Density; Bone Resorption; Cartilage, Articular; Cell Differentiation; Cimetidine; Dimaprit; Female; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Osteoclasts; Pyrilamine; Rats; Rats, Inbred Lew | 2003 |
The effects of pyrilamine and cimetidine on mRNA C-fos expression and nociceptive flinching behavior in rats.
Topics: Animals; Behavior, Animal; Blotting, Northern; Cimetidine; Dose-Response Relationship, Drug; Formaldehyde; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Pain; Pain Measurement; Pain Threshold; Proto-Oncogene Proteins c-fos; Pyrilamine; Rats; Rats, Wistar; RNA, Messenger; Spinal Cord | 2003 |
Histamine and prostaglandin interaction in regulation of oxytocin and vasopressin secretion.
Topics: Animals; Cimetidine; Cyclooxygenase Inhibitors; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Hypothalamus; Indomethacin; Lipopolysaccharides; Male; Oxytocin; Prostaglandin Antagonists; Prostaglandins; Pyrilamine; Rats; Rats, Wistar; Vasopressins | 2003 |
Critical role of histamine H4 receptor in leukotriene B4 production and mast cell-dependent neutrophil recruitment induced by zymosan in vivo.
Topics: Animals; Bone Marrow Cells; Carrageenan; Cimetidine; Cytokines; Dose-Response Relationship, Drug; Enzyme-Linked Immunosorbent Assay; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine Release; Leukotriene B4; Mast Cells; Mice; Mice, Inbred BALB C; Neutrophil Infiltration; Piperidines; Pleurisy; Pyrilamine; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H3; Receptors, Histamine H4; Zymosan | 2003 |
Cardiovascular effects of the toxin(s) of the Australian paralysis tick, Ixodes holocyclus, in the rat.
Topics: Action Potentials; Animals; Anti-Arrhythmia Agents; Antitoxins; Cimetidine; Dose-Response Relationship, Drug; Electrophysiology; Histological Techniques; Ixodes; Male; Metoprolol; Microelectrodes; Microscopy, Electron; Myocardial Contraction; Myocardium; Pinacidil; Pyrilamine; Rats; Rats, Wistar; Spider Venoms; Tetrodotoxin; Verapamil | 2004 |
Histaminergic H1 and H2 receptors located within the ventromedial hypothalamus regulate food and water intake in rats.
Topics: Animals; Avoidance Learning; Cimetidine; Drinking; Eating; Histamine H1 Antagonists; Histamine H2 Antagonists; Injections; Male; Motor Activity; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H2; Sodium; Sodium Chloride; Ventromedial Hypothalamic Nucleus; Water Deprivation | 2004 |
Central H1 and H2 receptor participation in the control of water and salt intake in rats.
Topics: Animals; Avoidance Learning; Behavior, Animal; Brain; Cimetidine; Drinking; Eating; Histamine H1 Antagonists; Histamine H2 Antagonists; Injections, Intraventricular; Lithium; Male; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H2; Salts; Time Factors; Water Deprivation | 2005 |
Orally administered FPRL1 receptor agonist peptide MMK-1 inhibits etoposide-induced alopecia by a mechanism different from intraperitoneally administered MMK-1.
Topics: Administration, Oral; Alopecia; Animals; Cimetidine; Disease Models, Animal; Etoposide; Female; Indomethacin; Injections, Intraperitoneal; Male; Peptides; Pyrilamine; Rats; Receptors, Formyl Peptide; Receptors, Lipoxin | 2006 |
Mechanisms of the vasorelaxant effect of Danshen (Salvia miltiorrhiza) in rat knee joints.
Topics: Adrenergic beta-Antagonists; Animals; Atropine; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Capsaicin; Cimetidine; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Drugs, Chinese Herbal; Flurbiprofen; Hindlimb; Histamine Antagonists; Joints; Muscarinic Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Peptide Fragments; Propranolol; Prostaglandins; Pyrilamine; Rats; Rats, Sprague-Dawley; Salvia miltiorrhiza; Vasodilator Agents | 2006 |
Enhanced histamine-mediated contraction of rabbit penile dorsal artery in diet-induced hypercholesterolemia.
Topics: Animals; Arteries; Cholesterol, Dietary; Cimetidine; Dose-Response Relationship, Drug; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Hypercholesterolemia; Male; Muscle, Smooth, Vascular; Norepinephrine; Penis; Pyrilamine; Rabbits; Vasoconstriction; Vasoconstrictor Agents | 2006 |
Histamine ameliorates spatial memory deficits induced by MK-801 infusion into ventral hippocampus as evaluated by radial maze task in rats.
Topics: Animals; Cimetidine; Dizocilpine Maleate; Dose-Response Relationship, Drug; Hippocampus; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Injections, Intraventricular; Male; Maze Learning; Memory Disorders; Pyrilamine; Rats; Rats, Sprague-Dawley | 2005 |
Differential modulation of cell recruitment and acute edema in a model of Polybia paulista venom-induced inflammation.
Topics: Acute Disease; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cimetidine; Dose-Response Relationship, Drug; Edema; Eosinophils; Histamine H1 Antagonists; Histamine H2 Antagonists; Indoles; Indomethacin; Leukocytes; Male; Neutrophil Infiltration; Peritoneal Cavity; Pyrilamine; Rats; Rats, Wistar; Wasp Venoms | 2006 |
Histamine-induced enhancement of vasopressin and oxytocin secretion in rat neurohypophyseal tissue cultures.
Topics: Animals; Cimetidine; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Kinetics; Male; Oxytocin; Piperidines; Pituitary Gland, Posterior; Pyrilamine; Rats; Tissue Culture Techniques; Vasopressins | 2006 |
Histamine modulates mast cell degranulation through an indirect mechanism in a model IgE-mediated reaction.
Topics: Animals; beta-N-Acetylhexosaminidases; Cell Degranulation; Cimetidine; Female; Flow Cytometry; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Immunoglobulin E; Immunohistochemistry; Macrophages; Mast Cells; Nitric Oxide; p-Methoxy-N-methylphenethylamine; Peritoneal Cavity; Pyrilamine; Rats; Rats, Wistar; Toxocara canis; Toxocariasis; Tumor Necrosis Factor-alpha | 2006 |
Histamine signaling through the H(2) receptor in the Peyer's patch is important for controlling Yersinia enterocolitica infection.
Topics: Animals; Anti-Allergic Agents; Anti-Ulcer Agents; Cimetidine; Dimaprit; Female; Gene Expression Profiling; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine Decarboxylase; Mice; Mice, Inbred C57BL; Oligonucleotide Array Sequence Analysis; Omeprazole; Peyer's Patches; Pyrilamine; Receptors, Histamine H2; Signal Transduction; Survival Rate; Yersinia enterocolitica; Yersinia Infections | 2006 |
A comparison between the cardiovascular actions of urocortin 1 and urocortin 2 (stresscopin-related peptide) in conscious rats.
Topics: Adrenergic beta-Antagonists; Animals; Atropine; Cardiovascular Agents; Cimetidine; Corticotropin-Releasing Hormone; Heart Rate; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Muscarinic Antagonists; Peptide Fragments; Propranolol; Pyrilamine; Rats; Rats, Sprague-Dawley; Urocortins | 2007 |
Degranulation of mast cells and histamine release involved in rat pain-related behaviors and edema induced by scorpion Buthus martensi Karch venom.
Topics: Animals; Chlorpheniramine; Cimetidine; Dose-Response Relationship, Drug; Edema; Histamine Antagonists; Histamine Release; Hyperalgesia; Inflammation; Mast Cells; Pain; Proto-Oncogene Proteins c-fos; Pyrilamine; Rats; Rats, Sprague-Dawley; Scorpion Venoms; Scorpions; Spinal Cord; Time Factors | 2007 |
Compound 48/80 induces endothelium-dependent and histamine release-independent relaxation in rabbit aorta.
Topics: Animals; Aorta; Cimetidine; Endothelium, Vascular; Estrenes; Histamine H1 Antagonists; Histamine Release; In Vitro Techniques; Male; Muscle Relaxation; NG-Nitroarginine Methyl Ester; Nitric Oxide; p-Methoxy-N-methylphenethylamine; Pyrilamine; Pyrrolidinones; Rabbits | 2008 |
A comparative study of histamine activities on differentiation of osteoblasts and osteoclasts.
Topics: Alkaline Phosphatase; Animals; Bone Marrow Cells; Bone Morphogenetic Protein 2; Bone Morphogenetic Proteins; Cell Differentiation; Cell Line; Cells, Cultured; Cimetidine; Core Binding Factor Alpha 1 Subunit; Dose-Response Relationship, Drug; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Mice; Mice, Inbred C57BL; Osteoblasts; Osteoclasts; Pyrilamine; RANK Ligand; Receptors, Histamine H1; Receptors, Histamine H2; RNA, Messenger; Transforming Growth Factor beta | 2007 |
Characterization of the effect of histamine on mouse corpus cavernosum.
Topics: Animals; Cimetidine; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Male; Mice; Penile Erection; Penis; Pyrilamine | 2008 |
[Role of histamine H(1) and H(2) receptors in the modulation of respiratory rhythmical discharge in medulla oblongata slice preparation of neonatal rats].
Topics: Animals; Animals, Newborn; Cimetidine; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Hypoglossal Nerve; In Vitro Techniques; Male; Medulla Oblongata; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine H1; Receptors, Histamine H2; Respiration | 2008 |
Modification of the picryl chloride-induced allergic dermatitis model in mouse ear lobes by 12-O-tetradecanoylphorbol 13-acetate, and analysis of the role of histamine in the modified model.
Topics: Animals; Cell Count; Cimetidine; Cyclophosphamide; Cyclosporine; Cytokines; Dermatitis, Allergic Contact; Disease Models, Animal; Ear Auricle; Eosinophil Peroxidase; Eosinophils; Gene Expression; Histamine; Histamine Antagonists; Immunoglobulin E; Interferon-gamma; Interleukin-4; Male; Mast Cells; Mice; Mice, Inbred BALB C; Picryl Chloride; Piperidines; Pyrilamine; Tetradecanoylphorbol Acetate; Thymic Stromal Lymphopoietin | 2009 |
Ameliorative effects of histamine on spatial memory deficits induced by scopolamine infusion into bilateral dorsal or ventral hippocampus as evaluated by the radial arm maze task.
Topics: Animals; Cimetidine; Dose-Response Relationship, Drug; Hippocampus; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Male; Maze Learning; Memory Disorders; Memory, Short-Term; Pyrilamine; Rats; Rats, Sprague-Dawley; Scopolamine; Spatial Behavior | 2009 |
Concurrent blockade of platelet-activating factor and histamine prevents life-threatening peanut-induced anaphylactic reactions.
Topics: Allergens; Anaphylaxis; Animals; Arachis; Cholera Toxin; Cimetidine; Disease Models, Animal; Drug Therapy, Combination; Enzyme Inhibitors; Female; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Hydroxyurea; Immunoglobulin E; Immunoglobulin G; Lipoxygenase Inhibitors; Mice; Mice, Inbred C57BL; Peanut Hypersensitivity; Platelet Membrane Glycoproteins; Pyrilamine; Receptors, G-Protein-Coupled; Receptors, Histamine | 2009 |
Involvement of histamine and histamine H2 receptors in nicotinamide-induced differentiation of human amniotic epithelial cells into insulin-producing cells.
Topics: Adult; Amniotic Fluid; C-Peptide; Cell Differentiation; Cells, Cultured; Cimetidine; Epithelial Cells; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Insulin; Insulin-Secreting Cells; Niacinamide; Nicotinic Agonists; Pregnancy; Pyrilamine; Receptors, Histamine H2 | 2010 |
Synthesis and dual histamine H₁ and H₂ receptor antagonist activity of cyanoguanidine derivatives.
Topics: Animals; Cimetidine; Guanidines; Guinea Pigs; Histamine H1 Antagonists; Histamine H2 Antagonists; Magnetic Resonance Spectroscopy; Male; Molecular Structure; Piperidines; Pyrilamine | 2013 |
Involvement of H1 and H2 receptors and soluble guanylate cyclase in histamine-induced relaxation of rat mesenteric collecting lymphatics.
Topics: Animals; Cimetidine; Endothelium, Lymphatic; Guanylate Cyclase; Histamine H1 Antagonists; Histamine H2 Antagonists; Lymphatic Vessels; Male; Mesentery; Muscle Relaxation; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; Oxadiazoles; Pyrilamine; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Cytoplasmic and Nuclear; Receptors, Histamine H1; Receptors, Histamine H2; Soluble Guanylyl Cyclase | 2014 |
Histamine deficiency exacerbates myocardial injury in acute myocardial infarction through impaired macrophage infiltration and increased cardiomyocyte apoptosis.
Topics: Acute Disease; Animals; Apoptosis; Cell Line; Cimetidine; Creatine Kinase, MB Form; Disease Models, Animal; Heart Injuries; Histamine; Histidine Decarboxylase; Humans; Macrophages; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Knockout; Mice, Transgenic; Myocardial Infarction; Myocytes, Cardiac; Promoter Regions, Genetic; Pyrilamine | 2015 |
A critical time window for the analgesic effect of central histamine in the partial sciatic ligation model of neuropathic pain.
Topics: Analgesics; Animals; Central Nervous System; Cimetidine; Disease Models, Animal; Drug Administration Routes; Histamine H1 Antagonists; Histamine H2 Antagonists; Histidine; Histidine Decarboxylase; Hyperalgesia; Mice; Mice, Inbred C57BL; Mice, Knockout; Pain Threshold; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Interleukin-1; Sciatic Neuropathy | 2016 |
The histaminergic system is involved in psychological stress-induced hyperthermia in rats.
Topics: Animals; Body Temperature Regulation; Cimetidine; Fever; Histamine; Histamine Agonists; Imidazoles; Male; Pyrilamine; Rats; Rats, Wistar; Stress, Physiological | 2017 |
Histaminergic Receptors Modulate Spinal Cord Injury-Induced Neuronal Nitric Oxide Synthase Upregulation and Cord Pathology: New Roles of Nanowired Drug Delivery for Neuroprotection.
Topics: Animals; Cimetidine; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Delivery Systems; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Male; Nanowires; Nitric Oxide Synthase Type I; Pyrilamine; Rats; Receptors, Histamine; Regional Blood Flow; Spinal Cord Injuries; Up-Regulation | 2017 |
Histamine receptors mediate contraction of reticular groove smooth muscle of adult goats.
Topics: Animals; Blotting, Western; Cimetidine; Cyproheptadine; Dose-Response Relationship, Drug; Goats; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Immunohistochemistry; Muscle Contraction; Muscle, Smooth; Pyrilamine; Receptors, Histamine; Stomach, Ruminant | 2020 |