Page last updated: 2024-08-16

pyrilamine and cetirizine

pyrilamine has been researched along with cetirizine in 19 studies

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19901 (5.26)18.7374
1990's7 (36.84)18.2507
2000's9 (47.37)29.6817
2010's2 (10.53)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Augert, G; Cottin, M; Demonchaux, P; Dupassieux, P; Jasserand, D; Lenoir, P; Paris, D; Peck, MJ1
Carrupt, PA; Crivori, P; Cruciani, G; Testa, B1
Du, LP; Li, MY; Tsai, KC; Xia, L; You, QD1
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM1
Bakker, RA; Ballesteros, JA; Bruysters, M; Haaksma, E; Jongejan, A; Leurs, R; Pardo, L1
Advenier, C; Candenas, ML; De Vos, C; Naline, E1
Coyle, AJ; Lefort, J; Vargaftig, BB1
Baltes, E; De Vos, C; Gobert, J; Maleux, MR1
Deleuran, B; Jinquan, T; Reimert, CM; Simonsen, C; Thestrup-Pedersen, K; Zachariae, C1
Bach, FW; Kjaer, A; Knigge, U; Madsen, EL; Søe-Jensen, P; Warberg, J1
Andresen, CJ; Smith, WB; Turner, CR; Watson, JW1
Dobashi, K; Houjou, S; Iizuka, K; Mori, M; Nakazawa, T; Sakai, H; Watanabe, K1
Fujii, Y; Harada, C; Hirai, T; Kamei, C; Tanaka, T1
Baerg, K; Rajput, A1
Chatelain, P; Christophe, B; Gillard, M; Gupta, A; Hammarlund-Udenaes, M; Massingham, R1
Al Suleimani, YM; Dong, Y; Walker, MJ1
Aydingöz, IE; Mansur, AT1
Charest-Morin, X; Gera, L; Marceau, F; Roy, C1
Bosma, R; Bouzo-Lorenzo, M; Briddon, SJ; Bushby, N; Fernández-Montalván, A; Georgi, V; Hill, SJ; Inkoom, L; Leurs, R; Sheppard, RJ; Stoddart, LA; Vischer, HF; Waring, MJ1

Trials

1 trial(s) available for pyrilamine and cetirizine

ArticleYear
Cetirizine inhibits the in vitro and ex vivo chemotactic response of T lymphocytes and monocytes.
    The Journal of allergy and clinical immunology, 1995, Volume: 95, Issue:5 Pt 1

    Topics: Anti-Inflammatory Agents, Non-Steroidal; Blood Proteins; Cetirizine; Chemotaxis, Leukocyte; Dermatitis, Atopic; Dose-Response Relationship, Drug; Double-Blind Method; Eosinophil Granule Proteins; Humans; Leukocytes, Mononuclear; Leukotriene B4; Monocytes; N-Formylmethionine Leucyl-Phenylalanine; Placebo Effect; Pyrilamine; Ribonucleases; T-Lymphocytes

1995

Other Studies

18 other study(ies) available for pyrilamine and cetirizine

ArticleYear
Synthesis, structure-activity relationships, and pharmacological evaluation of pyrrolo[3,2,1-ij]quinoline derivatives: potent histamine and platelet activating factor antagonism and 5-lipoxygenase inhibitory properties. Potential therapeutic application i
    Journal of medicinal chemistry, 1995, Feb-17, Volume: 38, Issue:4

    Topics: Animals; Asthma; Female; Guinea Pigs; Histamine Antagonists; In Vitro Techniques; Lipoxygenase Inhibitors; Male; Platelet Activating Factor; Platelet Aggregation Inhibitors; Quinolines; Rabbits; Rats; Rats, Sprague-Dawley; Respiratory Function Tests; Skin Tests; Structure-Activity Relationship

1995
Predicting blood-brain barrier permeation from three-dimensional molecular structure.
    Journal of medicinal chemistry, 2000, Jun-01, Volume: 43, Issue:11

    Topics: Blood-Brain Barrier; Databases, Factual; Models, Chemical; Molecular Conformation; Multivariate Analysis; Permeability; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
The pharmacophore hypotheses of I(Kr) potassium channel blockers: novel class III antiarrhythmic agents.
    Bioorganic & medicinal chemistry letters, 2004, Sep-20, Volume: 14, Issue:18

    Topics: Anti-Arrhythmia Agents; Models, Biological; Models, Molecular; Potassium Channel Blockers; Potassium Channels; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2004
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4

2005
Linking agonist binding to histamine H1 receptor activation.
    Nature chemical biology, 2005, Volume: 1, Issue:2

    Topics: Animals; Chlorocebus aethiops; COS Cells; Histamine Agonists; Humans; Models, Molecular; Mutation; Protein Structure, Tertiary; Receptors, Histamine H1; Serine

2005
The effect of cetirizine on the human isolated bronchus: interaction with salbutamol.
    The Journal of allergy and clinical immunology, 1991, Volume: 88, Issue:1

    Topics: Acetylcholine; Albuterol; Bronchi; Bronchoconstriction; Cetirizine; Dose-Response Relationship, Drug; Drug Synergism; Epithelium; Histamine; Histamine H1 Antagonists; Humans; Hydroxyzine; In Vitro Techniques; Pyrilamine

1991
The effect of cetirizine on antigen-dependent leucopenia in the guinea-pig.
    British journal of pharmacology, 1991, Volume: 103, Issue:2

    Topics: Animals; Benzeneacetamides; Benzhydryl Compounds; Blood Platelets; Cetirizine; Female; Guinea Pigs; Histamine H1 Antagonists; Hydroxamic Acids; Hydroxyzine; In Vitro Techniques; Leukocyte Count; Leukopenia; Leukotriene B4; Lipoxygenase Inhibitors; Male; Platelet Activating Factor; Pyrilamine; Terfenadine

1991
Inhibition of histamine and allergen skin wheal by cetirizine in four animal species.
    Annals of allergy, 1987, Volume: 59, Issue:4

    Topics: Allergens; Animals; Benzhydryl Compounds; Cetirizine; Clemastine; Dogs; Female; Guinea Pigs; Histamine; Histamine Antagonists; Hydroxyzine; Hypersensitivity, Immediate; Male; Mice; Mice, Inbred Strains; Pyrilamine; Rats; Rats, Inbred Strains; Skin; Species Specificity; Terfenadine

1987
Insulin/hypoglycemia-induced adrenocorticotropin and beta-endorphin release: involvement of hypothalamic histaminergic neurons.
    Endocrinology, 1993, Volume: 132, Issue:5

    Topics: Adrenocorticotropic Hormone; Animals; beta-Endorphin; Cetirizine; Cimetidine; Histamine; Histamine Agonists; Histamine Antagonists; Hypoglycemia; Hypothalamus; Insulin; Male; Methylhistamines; Neurons; Pyrilamine; Pyrimidinones; Rats; Rats, Wistar

1993
Characterization of a primate model of asthma using anti-allergy/anti-asthma agents.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1996, Volume: 45, Issue:5

    Topics: Albuterol; Animals; Anti-Allergic Agents; Anti-Inflammatory Agents; Antigens; Asthma; Bronchoconstriction; Bronchoconstrictor Agents; Bronchodilator Agents; Cetirizine; Dexamethasone; Disease Models, Animal; Leukocytes; Macaca fascicularis; Male; Methacholine Chloride; Pyrilamine; Salmeterol Xinafoate

1996
Effect of cetirizine on antigen-induced tracheal contraction of passively sensitized guinea pigs.
    Annals of allergy, asthma & immunology : official publication of the American College of Allergy, Asthma, & Immunology, 1996, Volume: 77, Issue:4

    Topics: Animals; Anti-Allergic Agents; Antigens; Calcium; Cells, Cultured; Cetirizine; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine Release; In Vitro Techniques; Lung; Male; Mast Cells; Mice; Mice, Inbred BALB C; Muscle Contraction; Pyrilamine; Trachea

1996
Epileptogenic activity induced by histamine H(1) antagonists in amygdala-kindled rats.
    Brain research, 2003, Nov-21, Volume: 991, Issue:1-2

    Topics: Amygdala; Animals; Cetirizine; Diphenhydramine; Electroencephalography; Epilepsy; Histamine H1 Antagonists; Injections, Intraperitoneal; Ketotifen; Kindling, Neurologic; Loratadine; Male; Pyrilamine; Rats; Rats, Wistar

2003
Cetirizine-induced dystonic movements.
    Neurology, 2006, Jan-10, Volume: 66, Issue:1

    Topics: Cetirizine; Child, Preschool; Drug Therapy, Combination; Dyskinesia, Drug-Induced; Dystonic Disorders; Female; Histamine H1 Antagonists, Non-Sedating; Humans; Neck Muscles; Nonprescription Drugs; Pyrilamine; Rhinitis, Allergic, Seasonal; Withholding Treatment

2006
Peripheral and central H1 histamine receptor occupancy by levocetirizine, a non-sedating antihistamine; a time course study in the guinea pig.
    British journal of pharmacology, 2007, Volume: 151, Issue:7

    Topics: Administration, Oral; Animals; Anti-Allergic Agents; Blood-Brain Barrier; Brain; Cerebellum; Cetirizine; Chlorpheniramine; Chromatography, Liquid; Dose-Response Relationship, Drug; Guinea Pigs; Half-Life; Histamine H1 Antagonists, Non-Sedating; Ileum; Injections, Intravenous; Male; Muscle Contraction; Muscle, Smooth; Piperazines; Pyrilamine; Receptors, Histamine H1; Tandem Mass Spectrometry; Time Factors; Tritium

2007
Differential responses to various classes of drugs in a model of allergic rhinitis in guinea pigs.
    Pulmonary pharmacology & therapeutics, 2008, Volume: 21, Issue:2

    Topics: Acetates; Acute Disease; Animals; Cetirizine; Cyclopropanes; Dexamethasone; Disease Models, Animal; Guinea Pigs; Heparin; Histamine H1 Antagonists; Male; Nasal Obstruction; NG-Nitroarginine Methyl Ester; Ovalbumin; Pyrilamine; Quinolines; Rhinitis, Allergic, Seasonal; Sneezing; Sulfides

2008
Reverse isotopic response: a rarely reported phenomenon.
    International journal of dermatology, 2009, Volume: 48, Issue:7

    Topics: Adult; Anesthetics, Local; Anti-Allergic Agents; Cetirizine; Dermatitis, Contact; Drug Eruptions; Female; Humans; Insect Bites and Stings; Lidocaine; Pyrilamine

2009
Vasopeptidase-activated latent ligands of the histamine receptor-1.
    International immunopharmacology, 2013, Volume: 17, Issue:3

    Topics: Animals; Arrestins; beta-Arrestins; Bradykinin; Cetirizine; CHO Cells; Cricetulus; HEK293 Cells; Histamine; Histamine Antagonists; Humans; In Vitro Techniques; Ligands; Peptide Hydrolases; Peptides; Prodrugs; Pyrilamine; Radioligand Assay; Receptor, Bradykinin B2; Receptors, Histamine H1; Umbilical Veins; Vasoconstriction

2013
Probe dependency in the determination of ligand binding kinetics at a prototypical G protein-coupled receptor.
    Scientific reports, 2019, 05-27, Volume: 9, Issue:1

    Topics: Binding, Competitive; Cetirizine; Datasets as Topic; Fluorescence Resonance Energy Transfer; Fluorescent Dyes; HEK293 Cells; Histamine H1 Antagonists; Humans; Ligands; Molecular Probes; Olopatadine Hydrochloride; Protein Binding; Pyrilamine; Radioligand Assay; Receptors, Histamine H1; Tritium

2019