pyrilamine has been researched along with alpha-methylhistamine in 35 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 19 (54.29) | 18.2507 |
| 2000's | 11 (31.43) | 29.6817 |
| 2010's | 5 (14.29) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Clapham, J; Kilpatrick, GJ | 2 |
| Katsoulis, S; Racké, K; Schwörer, H | 1 |
| Anjelkovic, IZ; Collis, CS; Djuric, D; Rosic, M; Segal, MB; Zlokovic, BV | 1 |
| Kohno, S; Nabe, T; Nakao, S; Ogawa, K; Ohata, K; Yamamura, H | 1 |
| Ballabeni, V; Barocelli, E; Chiavarini, M; Impicciatore, M | 1 |
| Kim, CY; Ryu, JH; Sakurai, E; Watanabe, T; Yanai, K | 1 |
| Carson, CC; Davies, MG; Hagen, PO; Kim, YC; Lee, TH | 1 |
| Garbarg, M; Kjaer, A; Knigge, U; Rouleau, A; Warberg, J | 1 |
| Adachi, N; Hirakawa, M; Itano, Y; Oishi, R; Saeki, K; Yamada, T | 1 |
| Kamei, C; Tasaka, K | 1 |
| Bach, FW; Kjaer, A; Knigge, U; Madsen, EL; Søe-Jensen, P; Warberg, J | 1 |
| Assenmacher, I; Barbanel, G; Givalois, L; Ixart, G; Malaval, F; Mekaouche, M; Siaud, P | 1 |
| Davison, JS; Jennings, LJ; Pariente, JA; Salido, GM; Sharkey, KA; Singh, J | 1 |
| Chiyotani, A; Konno, K; Nakata, J; Takeyama, K; Tamaoki, J | 1 |
| Imaizumi, M; Miyazaki, S; Onodera, K; Timmerman, H | 1 |
| Jafri, MS; Moore, KA; Taylor, GE; Weinreich, D | 1 |
| Fu, LW; Longhurst, JC; Pan, HL | 1 |
| Anichtchik, OV; Panula, P; Peitsaro, N | 1 |
| Harasawa, K | 1 |
| Hidaka, Y; Itadani, H; Nakamura, T; Ohta, M; Tanaka, K | 1 |
| Attoub, S; Bado, A; Laigneau, JP; Lewin, MJ; Moizo, L; Sobhani, I | 1 |
| Fogel, WA; Stasiak, A; Wagner, W | 1 |
| Bacon, KB; Center, DM; Cruikshank, WW; Gantner, F; Sakai, K; Tusche, MW | 1 |
| Coppé, MC; Gillardin, JM; Girard, P; Pansart, Y; Verniers, D | 1 |
| Campbell, VC; Katz, JL; Kopajtic, TA; Newman, AH | 1 |
| Eckman, JR; Wagner, MC; Wick, TM | 1 |
| Bakker, RA; Brann, MR; Burstein, ES; Hacksell, U; Leurs, R; Nicholas, MW; Smith, TT; Timmerman, H; Weiner, DM | 1 |
| Miranda, MI; Nuñez-Jaramillo, L; Purón-Sierra, L; Sabath, E | 1 |
| Bahi, A; Kieć-Kononowicz, K; Nurulain, SM; Sadek, B; Łażewska, D | 1 |
| Timmerman, H | 1 |
| Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM | 1 |
| Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K | 1 |
| Carmody, LC; Dandapani, S; Donckele, E; Feng, Y; Fernandez, C; Germain, AR; Gupta, PB; Lander, ES; Morgan, B; Munoz, B; Nag, PP; Palmer, M; Perez, JR; Schreiber, SL; Verplank, L | 1 |
| Adem, A; Kieć-Kononowicz, K; Sadek, B; Shafiullah, M; Shehab, S; Subramanian, D; Więcek, M | 1 |
1 review(s) available for pyrilamine and alpha-methylhistamine
| Article | Year |
|---|---|
Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship | 1990 |
34 other study(ies) available for pyrilamine and alpha-methylhistamine
| Article | Year |
|---|---|
Histamine H3 receptors modulate the release of [3H]-acetylcholine from slices of rat entorhinal cortex: evidence for the possible existence of H3 receptor subtypes.
Topics: Acetylcholine; Animals; Dose-Response Relationship, Drug; Hippocampus; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Piperidines; Potassium; Pyrilamine; Ranitidine; Rats; Receptors, Histamine; Receptors, Histamine H3 | 1992 |
Histamine inhibits 5-hydroxytryptamine release from the porcine small intestine: involvement of H3 receptors.
Topics: Animals; Female; Histamine; Hydroxyindoleacetic Acid; In Vitro Techniques; Intestine, Small; Male; Methylhistamines; Pyrilamine; Receptors, Histamine; Serotonin; Swine | 1992 |
The effects of (R) alpha-methyl histamine on the isolated guinea pig aorta.
Topics: Animals; Aorta; Cimetidine; Female; Guanidines; Guinea Pigs; Histamine; Histamine Antagonists; Imidazoles; Impromidine; Male; Methylhistamines; Muscle, Smooth, Vascular; Potassium; Pyrilamine; Receptors, Histamine; Receptors, Histamine H3; Vasoconstriction; Vasodilation | 1991 |
Possible participation of histamine H3-receptors in the regulation of anaphylactic histamine release from isolated rat peritoneal mast cells.
Topics: Anaphylaxis; Animals; Anticonvulsants; Chromatography, High Pressure Liquid; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Histamine; Histamine Agonists; Histamine Antagonists; Histamine Release; In Vitro Techniques; L-Lactate Dehydrogenase; Male; Mast Cells; Methylhistamines; p-Methoxy-N-methylphenethylamine; Peritoneal Cavity; Peritoneum; Piperidines; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H3 | 1994 |
R-alpha-methylhistamine-induced inhibition of gastric acid secretion in pylorus-ligated rats via central histamine H3 receptors.
Topics: Animals; Cimetidine; Female; Gastric Acid; Gastric Mucosa; Histamine Agonists; Histamine Antagonists; Injections, Intraventricular; Methylhistamines; Piperidines; Pylorus; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H3 | 1995 |
Ontogenetic development of histamine receptor subtypes in rat brain demonstrated by quantitative autoradiography.
Topics: Aging; Animals; Autoradiography; Brain; Corpus Striatum; Histamine Agonists; Histidine Decarboxylase; Injections; Methylhistamines; Oxidopamine; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine | 1995 |
Characterization and function of histamine receptors in corpus cavernosum.
Topics: Acetylcholine; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Papaverine; Penis; Piperidines; Pyrilamine; Rabbits; Receptors, Histamine; Thiazoles | 1995 |
Dehydration-induced release of vasopressin involves activation of hypothalamic histaminergic neurons.
Topics: Animals; Arginine Vasopressin; Blood; Cimetidine; Dehydration; Histamine; Hypothalamus; Male; Methylhistamines; Methylhistidines; Neurons; Osmolar Concentration; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Histamine H2 | 1994 |
Aggravation of ischemic neuronal damage in the rat hippocampus by impairment of histaminergic neurotransmission.
Topics: Animals; Benzothiazoles; Brain Ischemia; Cell Death; Hippocampus; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Methylhistidines; Neurons; Phenoxypropanolamines; Piperidines; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine; Synaptic Transmission; Thiazoles | 1993 |
Effect of histamine on memory retrieval in old rats.
Topics: Acetylcholine; Aging; Animals; Anticonvulsants; Avoidance Learning; Cerebrovascular Circulation; Cimetidine; Dose-Response Relationship, Drug; Exploratory Behavior; Histamine; Histamine Agonists; Injections, Intraventricular; Male; Memory; Methylhistamines; Motor Activity; Piperidines; Pyrilamine; Rats; Rats, Wistar | 1993 |
Histamine H3 receptor-mediated modulation of water consumption in the rat.
Topics: Animals; Drinking; Histamine; Histamine Antagonists; Male; Methylhistamines; Nicotinic Acids; Piperidines; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H3; Tetrazoles; Triazoles | 1993 |
Insulin/hypoglycemia-induced adrenocorticotropin and beta-endorphin release: involvement of hypothalamic histaminergic neurons.
Topics: Adrenocorticotropic Hormone; Animals; beta-Endorphin; Cetirizine; Cimetidine; Histamine; Histamine Agonists; Histamine Antagonists; Hypoglycemia; Hypothalamus; Insulin; Male; Methylhistamines; Neurons; Pyrilamine; Pyrimidinones; Rats; Rats, Wistar | 1993 |
Involvement of central histamine in the early phase of ACTH and corticosterone responses to endotoxin in rats.
Topics: Adrenocorticotropic Hormone; Animals; Cimetidine; Corticosterone; Escherichia coli; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Kinetics; Lipopolysaccharides; Male; Median Eminence; Methylhistamines; Pyrilamine; Rats; Rats, Sprague-Dawley | 1996 |
Control of exocrine secretion in the guinea-pig pancreas by histamine H3 receptors.
Topics: alpha-Amylases; Animals; Choline; Electric Stimulation; Female; Guinea Pigs; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Pancreas; Piperidines; Pyrilamine; Receptors, Histamine H3; Tritium | 1996 |
Histamine H2 receptor-mediated airway goblet cell secretion and its modulation by histamine-degrading enzymes.
Topics: Amine Oxidase (Copper-Containing); Animals; Asthma; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glycoproteins; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Histamine N-Methyltransferase; Male; Methylhistamines; Mucus; Piperidines; Pyrilamine; Recombinant Proteins; Trachea | 1997 |
Effects of clobenpropit (VUF-9153), a histamine H3-receptor antagonist, on learning and memory, and on cholinergic and monoaminergic systems in mice.
Topics: Acetylcholine; Animals; Avoidance Learning; Benzothiazoles; Biogenic Monoamines; Brain; Drug Interactions; Histamine Antagonists; Histamine H2 Antagonists; Imidazoles; Male; Memory; Methylhistamines; Mice; Mice, Inbred ICR; Phenoxypropanolamines; Piperidines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H3; Scopolamine; Thiazoles; Thiourea | 1997 |
Histamine H1 receptor activation blocks two classes of potassium current, IK(rest) and IAHP, to excite ferret vagal afferents.
Topics: Action Potentials; Animals; Diphenhydramine; Electric Conductivity; Ferrets; Histamine; Histamine Agonists; Histamine H1 Antagonists; Impromidine; Male; Methylhistamines; Neurons, Afferent; Nodose Ganglion; Patch-Clamp Techniques; Potassium; Potassium Channel Blockers; Pyrilamine; Receptors, Histamine H1; Thiazoles; Vagus Nerve | 1997 |
Endogenous histamine stimulates ischemically sensitive abdominal visceral afferents through H1 receptors.
Topics: Abdomen; Afferent Pathways; Animals; Bile Ducts; Blood Pressure; Cats; Chlorpheniramine; Dimaprit; Duodenum; Female; Gallbladder; Histamine; Histamine H1 Antagonists; Indomethacin; Ischemia; Male; Methylhistamines; Nerve Fibers; Neural Conduction; Pancreas; Pyrilamine; Receptors, Histamine H1 | 1997 |
Identification of a histamine H(3)-like receptor in the zebrafish (Danio rerio) brain.
Topics: Animals; Autoradiography; Brain; Cimetidine; Female; Guanosine 5'-O-(3-Thiotriphosphate); Histamine Agonists; Histamine Antagonists; Imidazoles; Kinetics; Male; Methylhistamines; Piperidines; Pyrilamine; Radioligand Assay; Receptors, Histamine H3; Sulfur Radioisotopes; Thiourea; Tritium; Zebrafish | 2000 |
Does the histaminergic system play a role in spinal nociception?
Topics: Animals; Dose-Response Relationship, Drug; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Methylhistamines; Motor Neurons; Pain; Pyrilamine; Ranitidine; Rats; Spinal Cord; Synaptic Transmission | 2000 |
Molecular cloning and characterization of a new human histamine receptor, HH4R.
Topics: Amino Acid Sequence; Binding, Competitive; Cell Line; Cimetidine; Cloning, Molecular; Colforsin; Cyclic AMP; Histamine Agonists; Histamine Antagonists; Humans; Leukocytes; Methylhistamines; Molecular Sequence Data; Pyrilamine; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H3; Receptors, Histamine H4; Recombinant Proteins; Sequence Alignment; Sequence Homology, Amino Acid; Stereoisomerism; Transfection | 2000 |
The H3 receptor is involved in cholecystokinin inhibition of food intake in rats.
Topics: Animals; Brain; Cholecystokinin; Dose-Response Relationship, Drug; Eating; Gastric Mucosa; Histamine; Histamine Agonists; Histamine Antagonists; Injections, Intraperitoneal; Male; Methylhistamines; Piperidines; Pyrilamine; Ranitidine; Rats; Rats, Wistar; Receptors, Histamine H3; Sincalide; Stomach | 2001 |
Mouse mammary epithelial cells bear histamine receptors.
Topics: Animals; Binding Sites; Cimetidine; Epithelial Cells; Female; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Mammary Glands, Animal; Methylhistamines; Mice; Mice, Inbred BALB C; Pyrilamine; Radiopharmaceuticals; Receptors, Histamine | 2002 |
Histamine h(4) and h(2) receptors control histamine-induced interleukin-16 release from human CD8(+) T cells.
Topics: Base Sequence; CD4-Positive T-Lymphocytes; CD8-Positive T-Lymphocytes; Cells, Cultured; Cimetidine; Dimaprit; DNA Primers; Female; Gene Expression Regulation; Histamine; Humans; Interleukin-16; Male; Methylhistamines; Polymerase Chain Reaction; Pyrilamine; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H2; Receptors, Histamine H4 | 2002 |
Role of the histamine system in nefopam-induced antinociception in mice.
Topics: Acetic Acid; Analgesics, Non-Narcotic; Animals; Enzyme Inhibitors; Formaldehyde; Guinea Pigs; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Male; Methylhistamines; Methylhistidines; Mice; Mice, Inbred ICR; Nefopam; Pain Measurement; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3 | 2004 |
Assessment of the influence of histaminergic actions on cocaine-like effects of 3alpha-diphenylmethoxytropane analogs.
Topics: Animals; Benztropine; Binding, Competitive; Brain; Cocaine; Discrimination Learning; Dopamine Uptake Inhibitors; Guanidines; Histamine; Histamine Agonists; Histamine H1 Antagonists; In Vitro Techniques; Male; Methylhistamines; Motor Activity; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine H3; Tropanes | 2005 |
Histamine increases sickle erythrocyte adherence to endothelium.
Topics: Analysis of Variance; Anemia, Sickle Cell; Cell Adhesion; Cells, Cultured; Endothelial Cells; Endothelium, Vascular; Erythrocytes; Famotidine; Histamine; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Imidazoles; Methylhistamines; P-Selectin; Piperidines; Pyrilamine; Stimulation, Chemical; Thiazoles; Thiourea; Venules | 2006 |
In vitro pharmacology of clinically used central nervous system-active drugs as inverse H(1) receptor agonists.
Topics: Animals; Central Nervous System Agents; Chlorocebus aethiops; Cloning, Molecular; COS Cells; Histamine Agonists; Histamine H1 Antagonists; Humans; Methylhistamines; Mice; NIH 3T3 Cells; Pyrilamine; Receptors, Histamine H1 | 2007 |
Blockade of nucleus basalis magnocellularis or activation of insular cortex histamine receptors disrupts formation but not retrieval of aversive taste memory.
Topics: Animals; Basal Nucleus of Meynert; Conditioning, Classical; Histamine Agonists; Histamine H1 Antagonists; Male; Mental Recall; Methylhistamines; Pyrilamine; Rats; Rats, Sprague-Dawley; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H3; Taste Perception; Temporal Lobe; Time Factors | 2010 |
The novel non-imidazole histamine H3 receptor antagonist DL77 reduces voluntary alcohol intake and ethanol-induced conditioned place preference in mice.
Topics: Alcohol Deterrents; Alcohol Drinking; Animals; Central Nervous System Depressants; Choice Behavior; Conditioning, Psychological; Dose-Response Relationship, Drug; Ethanol; Histamine Agonists; Histamine H1 Antagonists; Histamine H3 Antagonists; Male; Methylhistamines; Mice, Inbred C57BL; Phenyl Ethers; Piperidines; Pyrilamine; Spatial Behavior; Taste Perception; Volition | 2015 |
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4 | 2005 |
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship | 2010 |
Cinnamides as selective small-molecule inhibitors of a cellular model of breast cancer stem cells.
Topics: Amides; Breast Neoplasms; Cell Line, Tumor; Drug Screening Assays, Antitumor; Female; Humans; Neoplastic Stem Cells; Small Molecule Libraries; Structure-Activity Relationship | 2013 |
Anticonvulsant properties of histamine H3 receptor ligands belonging to N-substituted carbamates of imidazopropanol.
Topics: 1-Propanol; Animals; Anticonvulsants; Carbamates; Electroshock; Histamine Agonists; Histamine Antagonists; Imidazoles; Ligands; Rats; Rats, Wistar; Receptors, Histamine H3; Seizures | 2013 |