Page last updated: 2024-08-16

pyrilamine and 4-methylhistamine

pyrilamine has been researched along with 4-methylhistamine in 27 studies

Research

Studies (27)

TimeframeStudies, this research(%)All Research%
pre-199015 (55.56)18.7374
1990's10 (37.04)18.2507
2000's1 (3.70)29.6817
2010's1 (3.70)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Timmerman, H1
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM1
Nowak, JZ; Sek, B1
Akiyama, Y; Kamei, C; Mukai, T; Tasaka, K1
Bugajski, J; Gadek-Michalska, A1
Adaikan, PG; Lau, LC; Ratnam, SS1
Knigge, U; Matzen, S; Warberg, J1
Akahori, H; Kamei, C; Kitazumi, K; Tasaka, K1
Kim, LE; Oudart, N; Sercombe, R; Teste, JF1
Kannisto, P; Owman, C; Schmidt, G; Sjöberg, NO1
Dhawan, BN; Dhawan, KN; Gulati, A; Shukla, R; Srimal, RC1
Joshi, DP; Verma, SC1
Donoso, AO; Zárate, MB1
Ikehara, I; Murakami, M; Saeki, K; Seo, S1
Ikeda, S; Murakami, M; Nishibori, M; Saeki, K; Seo, S1
Donoso, AO; Seltzer, A; Zárate, MB1
Bradley, SL; Russell, JA1
Broadley, KJ; Wilson, C1
Dodds, WJ; Hogan, WJ; Honda, R; Toouli, J1
Kamei, C; Tasaka, K; Tsujimoto, S; Yoshida, T1
Banchelli, G; Buffoni, F; Conforti, L; Ignesti, G; Pirisino, R; Raimondi, L1
Nowak, JZ; Sek, B; Zawilska, JB1
KAMEI, CH1
Ali, AS; Ali, SA; Peter, J2
Jørgensen, H; Kjaer, A; Knigge, U; Warberg, J; Willems, E1
Ebenezer, AJ; Prasad, K; Rajan, S; Thangam, EB1

Reviews

1 review(s) available for pyrilamine and 4-methylhistamine

ArticleYear
Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:1

    Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship

1990

Other Studies

26 other study(ies) available for pyrilamine and 4-methylhistamine

ArticleYear
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4

2005
Cyclic AMP generating systems in vertebrate retina: effects of histamine and an established retinal modulator, dopamine.
    Agents and actions, 1991, Volume: 33, Issue:1-2

    Topics: Adenylyl Cyclases; Animals; Cerebral Cortex; Chickens; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dopamine; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Retina; Thiazoles; Thiourea

1991
Histamine lipolysis I: changes in the free fatty acid levels of dog plasma after intravenous infusion of histamine.
    Methods and findings in experimental and clinical pharmacology, 1990, Volume: 12, Issue:5

    Topics: Aminophylline; Animals; Chromatography, High Pressure Liquid; Diphenhydramine; Dogs; Epinephrine; Fatty Acids, Nonesterified; Female; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Infusions, Intravenous; Lipolysis; Male; Methylhistamines; Pentobarbital; Pyrilamine; Starvation

1990
Antagonistic action of naloxone on central histamine receptors-stimulated corticosterone secretion in rats under stress.
    Agents and actions, 1989, Volume: 28, Issue:3-4

    Topics: Animals; Cimetidine; Corticosterone; Dimaprit; Histamine; Male; Methylhistamines; Naloxone; Pituitary-Adrenal System; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Restraint, Physical; Stress, Physiological; Thiourea

1989
Effect of histamine on human vas deferens in vitro.
    British journal of urology, 1989, Volume: 64, Issue:4

    Topics: Burimamide; Cimetidine; Culture Techniques; Dose-Response Relationship, Drug; Histamine; Humans; Male; Methylhistamines; Muscle Contraction; Pyrilamine; Vas Deferens

1989
Histaminergic stimulation of prolactin secretion mediated via H1- or H2-receptors: dependence on routes of administration.
    Neuroendocrinology, 1986, Volume: 44, Issue:1

    Topics: Animals; Cimetidine; Dimaprit; Histamine; Histamine H1 Antagonists; Male; Methylhistamines; Pituitary Gland, Anterior; Prolactin; Pyrilamine; Pyrimidinones; Rats; Receptors, Histamine; Thiazoles; Thiourea

1986
The effects of histamine and some related compounds on conditioned avoidance response in rats.
    Life sciences, 1985, Nov-25, Volume: 37, Issue:21

    Topics: Acetylcholine; Animals; Avoidance Learning; Dimaprit; Diphenhydramine; Dose-Response Relationship, Drug; Histamine; Histamine Antagonists; Hypothalamus; Injections, Intraventricular; Kinetics; Male; Methylhistamines; Pyrilamine; Rats; Rats, Inbred Strains; Scopolamine; Thiazoles; Thiourea

1985
Participation of vascular H1-receptors in histaminergic relaxation of rabbit middle cerebral artery in vitro.
    Archives internationales de pharmacodynamie et de therapie, 1986, Volume: 283, Issue:2

    Topics: Animals; Cerebral Arteries; Cimetidine; Dimaprit; Drug Interactions; Histamine; In Vitro Techniques; Methylhistamines; Muscle Relaxation; Muscle, Smooth, Vascular; Phenethylamines; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Thiourea

1986
Alteration by histamine of the sympathetic nerve-mediated contractions in the bovine ovarian follicle wall in vitro.
    European journal of pharmacology, 1987, Mar-03, Volume: 135, Issue:1

    Topics: Animals; Cattle; Cimetidine; Electrolytes; Female; Glucose; Histamine; In Vitro Techniques; Methylhistamines; Muscle Contraction; Norepinephrine; Ovary; Proteins; Pyrilamine; Sympathetic Nervous System

1987
Evidence for the involvement of histamine in the regulation of blood-brain barrier permeability.
    Pharmacological research communications, 1985, Volume: 17, Issue:4

    Topics: Animals; Blood-Brain Barrier; Colforsin; Diterpenes; Dogs; Female; Fluorescein; Fluoresceins; Histamine; Histamine Antagonists; Male; Methylhistamines; Metiamide; Pyrilamine; Time Factors

1985
Identification and specific blockade of histaminergic receptors in guinea pig vasa deferentia.
    Canadian journal of physiology and pharmacology, 1981, Volume: 59, Issue:10

    Topics: Animals; Dose-Response Relationship, Drug; Guinea Pigs; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Reserpine; Vas Deferens

1981
Release of prolactin and luteinizing hormone by histamine agonists in ovariectomized, steroid-treated rats under ether anesthesia.
    Experimental brain research, 1983, Volume: 52, Issue:2

    Topics: Animals; Castration; Dimaprit; Female; Histamine; Histamine H1 Antagonists; Luteinizing Hormone; Methylhistamines; Metiamide; Pituitary Gland, Anterior; Prolactin; Pyridines; Pyrilamine; Rats; Thiourea

1983
Effect of histamine on cyclic AMP levels in the submandibular gland.
    Agents and actions, 1981, Volume: 11, Issue:1-2

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Cyclic AMP; Female; Guinea Pigs; Histamine; Methylhistamines; Metiamide; Pyrilamine; Submandibular Gland

1981
Amylase secretion induced by histamine from guinea-pig parotid gland.
    Archives internationales de pharmacodynamie et de therapie, 1982, Volume: 255, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Amylases; Animals; Atropine; Guinea Pigs; Histamine; In Vitro Techniques; Male; Methylhistamines; Metiamide; Parotid Gland; Propranolol; Pyrilamine; Stimulation, Chemical; Time Factors

1982
Histamine-induced prolactin release: pharmacological characterization of receptors in male rats.
    Neuroendocrinology, 1983, Volume: 36, Issue:6

    Topics: Anesthesia; Animals; Furans; Histamine; Male; Methylhistamines; Metiamide; Prolactin; Pyrilamine; Ranitidine; Rats; Receptors, Histamine

1983
Distribution of histamine receptors in isolated canine airways.
    Journal of applied physiology: respiratory, environmental and exercise physiology, 1983, Volume: 54, Issue:3

    Topics: Animals; Dogs; Dose-Response Relationship, Drug; Electric Stimulation; Histamine; Methylhistamines; Metiamide; Muscle Contraction; Muscle, Smooth; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Respiratory System; Tissue Distribution

1983
Further characterization of the guinea pig left atrial tension response to histamine by use of selective agonists.
    Agents and actions, 1981, Volume: 11, Issue:3

    Topics: Animals; Female; Guinea Pigs; Heart Atria; Heart Rate; Histamine; In Vitro Techniques; Male; Methylhistamines; Myocardial Contraction; Pyridines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2

1981
Effect of histamine on motor function of opossum sphincter of Oddi.
    The American journal of physiology, 1981, Volume: 241, Issue:2

    Topics: Ampulla of Vater; Animals; Female; Histamine; Male; Methylhistamines; Metiamide; Motor Activity; Opossums; Pyridines; Pyrilamine; Receptors, Histamine H1; Sphincter of Oddi; Sympatholytics; Tetrodotoxin

1981
Changes in plasma adrenocorticotropic hormone and cortisol levels induced by intracerebroventricular injection of histamine and its related compounds in dogs.
    Pharmacology, 1993, Volume: 47, Issue:2

    Topics: Adrenocorticotropic Hormone; Animals; Cimetidine; Dogs; Hexamethonium; Hexamethonium Compounds; Histamine; Hydrocortisone; Hypophysectomy; Injections, Intraventricular; Male; Methylhistamines; Pyrilamine

1993
Histamine lipolytic activity and semicarbazide-sensitive amine oxidase (SSAO) of rat white adipose tissue (WAT).
    Biochemical pharmacology, 1993, Oct-19, Volume: 46, Issue:8

    Topics: Adipose Tissue; Amine Oxidase (Copper-Containing); Animals; Benzylamines; Cimetidine; Histamine; Isoproterenol; Kinetics; Lipolysis; Male; Methylhistamines; Pyrilamine; Rats; Rats, Wistar; Semicarbazides

1993
A bizarre receptor mediating stimulatory effect of histamine on cyclic AMP formation in duck pineal gland.
    Neuroscience letters, 1995, Dec-29, Volume: 202, Issue:1-2

    Topics: Animals; Cyclic AMP; Ducks; Histamine; Histamine Agonists; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Methylhistamines; Pineal Gland; Pyrilamine; Ranitidine; Receptors, Histamine

1995
EFFECTS OF HISTAMINE AND RELATED COMPOUNDS ON THE BOVINE IRIS DILATOR.
    Methods and findings in experimental and clinical pharmacology, 1996, Volume: 18, Issue:4

    Topics: Analysis of Variance; Animals; Cattle; Chlorpheniramine; Cimetidine; Diphenhydramine; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Ileum; Iris; Lethal Dose 50; Male; Methylhistamines; Muscle Contraction; Muscle, Smooth; p-Methoxy-N-methylphenethylamine; Piperidines; Potassium; Pyrilamine; Ranitidine; Receptors, Histamine H1; Substance P

1996
Effect of histaminergic drugs on integumental melanophores of adult Bufo melanostictus.
    Indian journal of experimental biology, 1996, Volume: 34, Issue:5

    Topics: Animals; Bufonidae; Cell Aggregation; Histamine; Histamine Agents; In Vitro Techniques; Melanophores; Methylhistamines; Metiamide; Pyrilamine

1996
Histamine receptors in the skin melanophores of Indian bullfrog Rana tigerina.
    Comparative biochemistry and physiology. Part A, Molecular & integrative physiology, 1998, Volume: 121, Issue:3

    Topics: Animals; Edetic Acid; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Melanins; Melanophores; Methylhistamines; Metiamide; p-Methoxy-N-methylphenethylamine; Pyrilamine; Ranidae; Receptors, Histamine; Skin; Skin Pigmentation

1998
Histaminergic and catecholaminergic interactions in the central regulation of vasopressin and oxytocin secretion.
    Endocrinology, 1999, Volume: 140, Issue:8

    Topics: Animals; Arginine Vasopressin; Blood Pressure; Cerebral Ventricles; Cimetidine; Epinephrine; Histamine; Histamine Agonists; Hypothalamus; Imidazoles; Infusions, Parenteral; Male; Methylhistamines; Norepinephrine; Oxytocin; Pituitary Gland, Posterior; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H2; Thiazoles; Thiourea

1999
Silencing of H4R inhibits the production of IL-1β through SAPK/JNK signaling in human mast cells.
    Journal of receptor and signal transduction research, 2018, Volume: 38, Issue:3

    Topics: Calcium; Cell Line; Gene Expression Regulation; Gene Silencing; Histamine; Humans; Indoles; Interleukin-1beta; MAP Kinase Kinase 4; MAP Kinase Signaling System; Mast Cells; Methylhistamines; Piperazines; Pyrilamine; Receptors, Histamine H4; RNA, Small Interfering

2018