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pyrilamine and 2-(2-aminoethyl)pyridine

pyrilamine has been researched along with 2-(2-aminoethyl)pyridine in 33 studies

Research

Studies (33)

TimeframeStudies, this research(%)All Research%
pre-199023 (69.70)18.7374
1990's6 (18.18)18.2507
2000's4 (12.12)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bakker, RA; Elz, S; Govoni, M; Leurs, R; Menge, WM; Schunack, W; Smit, MJ; Timmerman, H; van de Wetering, I1
Bakker, RA; DeGrip, WJ; DeGroot, HJ; Leurs, R; Ratnala, VR; Swarts, HG; VanOostrum, J1
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM1
Phillis, JW; Sastry, BS1
Bast, A; Leurs, R; Smit, MJ; Timmerman, H1
Bani Sacchi, T; Gambassi, F; Giannella, E; Mannaioni, PF; Masini, E; Palmerani, B; Pistelli, A1
Benedito, S; Nielsen, PJ; Nyborg, NC; Prieto, D1
Młynarska, MS1
Matsuki, T; Ohhashi, T1
Edvinsson, L; Jansen, I; Ottosson, A1
Bugajski, J; Gadek-Michalska, A1
Girard, A; Marche, P1
Hutchison, VH; Spriestersbach, KK1
Männistö, PT; Mattila, J; Tuominen, RK2
Donaldson, J; Hill, SJ1
Bugajski, J; Gadek, A1
Fromm, D; Furukawa, T; Olender, EJ; Woods, DJ1
Bohm, U; Falus, A; Fekete, MI; Meretey, K1
Kume, S; Ohashi, T; Ozaki, Y1
Daniel, D; Owen, DA; Poy, E; Woodward, DF1
Joshi, DP; Verma, SC1
Heldsinger, AA; Skoglund, ML; Vinik, AI1
Donoso, AO; Zárate, MB1
Bielkiewicz, B; Cook, DA1
Bugajski, J; Janusz, Z1
Del Soldato, P1
Shah, RJ; Verma, SC1
Broadley, KJ; Wilson, C1
Dodds, WJ; Hogan, WJ; Honda, R; Toouli, J1
Seidler, FJ; Slotkin, TA; Subramanian, N; Whitmore, WL1
Arilla, E; Ocaña Fuentes, A; Puebla, L1
Nakazato, E; Ohno, M; Watanabe, S; Yamamoto, T1

Other Studies

33 other study(ies) available for pyrilamine and 2-(2-aminoethyl)pyridine

ArticleYear
Synthesis and pharmacological identification of neutral histamine H1-receptor antagonists.
    Journal of medicinal chemistry, 2003, Dec-18, Volume: 46, Issue:26

    Topics: Animals; Binding, Competitive; Cell Line; Chlorocebus aethiops; Genes, Reporter; Histamine; Histamine Agonists; Histamine H1 Antagonists; Humans; Inositol Phosphates; Ligands; NF-kappa B; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H4; Structure-Activity Relationship

2003
Large-scale overproduction, functional purification and ligand affinities of the His-tagged human histamine H1 receptor.
    European journal of biochemistry, 2004, Volume: 271, Issue:13

    Topics: Animals; COS Cells; Histidine; Humans; Ligands; Radioligand Assay; Receptors, Histamine H1; Spodoptera

2004
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4

2005
Depression of rat cerebral cortical neurones by H1 and H2 histamine receptor agonists.
    European journal of pharmacology, 1976, Volume: 38, Issue:2

    Topics: Acetylcholine; Animals; Cerebral Cortex; Guanidines; Histamine; Imidazoles; In Vitro Techniques; Male; Metiamide; Neurons; Norepinephrine; Pyridines; Pyrilamine; Rats; Receptors, Drug

1976
Homologous histamine H1 receptor desensitization results in reduction of H1 receptor agonist efficacy.
    European journal of pharmacology, 1991, Apr-24, Volume: 196, Issue:3

    Topics: Animals; Guinea Pigs; Histamine; In Vitro Techniques; Inositol Phosphates; Jejunum; Male; Membranes; Muscle Contraction; Muscle, Smooth; Phosphatidylinositols; Pyridines; Pyrilamine; Receptors, Histamine H1; Tritium

1991
Histamine release by platelet aggregation.
    Agents and actions, 1990, Volume: 30, Issue:1-2

    Topics: Animals; Arachidonic Acids; Blood Platelets; Histamine Release; In Vitro Techniques; L-Lactate Dehydrogenase; Male; Mast Cells; Platelet Aggregation; Pyridines; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains

1990
Histamine induces endothelium-dependent relaxation of bovine retinal arteries.
    Investigative ophthalmology & visual science, 1991, Volume: 32, Issue:1

    Topics: Acetylcholine; Animals; Cattle; Cimetidine; Dimaprit; Endothelium, Vascular; Histamine; Muscle Relaxation; Pyridines; Pyrilamine; Receptors, Histamine; Retinal Artery; Tachyphylaxis; Thiourea

1991
Antagonistic effect of naloxone on the hypertensive response of intraventricularly administered histamine.
    Agents and actions, 1990, Volume: 30, Issue:1-2

    Topics: Animals; Blood Pressure; Cimetidine; Dimaprit; Hemodynamics; Histamine; In Vitro Techniques; Injections, Intraventricular; Male; Naloxone; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Thiourea

1990
Endothelium and mechanical responses of isolated monkey pulmonary veins to histamine.
    The American journal of physiology, 1990, Volume: 259, Issue:4 Pt 2

    Topics: Animals; Dimaprit; Endothelium, Vascular; Famotidine; Hemoglobins; Histamine; In Vitro Techniques; Macaca; Methylene Blue; Pulmonary Veins; Pyridines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea; Vasoconstriction; Vasodilation

1990
Pharmacological characterization of histamine receptors in the human temporal artery.
    British journal of clinical pharmacology, 1989, Volume: 27, Issue:2

    Topics: Adult; Cimetidine; Dinoprost; Female; Histamine; Humans; Imidazoles; Impromidine; In Vitro Techniques; Male; Methylhistamines; Middle Aged; Pyridines; Pyrilamine; Receptors, Histamine; Temporal Arteries; Thiazoles; Vasoconstriction; Vasodilation

1989
Antagonistic action of naloxone on central histamine receptors-stimulated corticosterone secretion in rats under stress.
    Agents and actions, 1989, Volume: 28, Issue:3-4

    Topics: Animals; Cimetidine; Corticosterone; Dimaprit; Histamine; Male; Methylhistamines; Naloxone; Pituitary-Adrenal System; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Restraint, Physical; Stress, Physiological; Thiourea

1989
Phosphoinositides and cicletanine.
    Drugs under experimental and clinical research, 1988, Volume: 14, Issue:2-3

    Topics: Angiotensin II; Animals; Antihypertensive Agents; Aorta, Thoracic; Cells, Cultured; Dimaprit; Diuretics; Guinea Pigs; Histamine; Male; Muscle, Smooth, Vascular; Phenylephrine; Phosphatidylinositols; Pyridines; Pyrilamine; Thiourea

1988
Histamine and histamine receptors: behavioral thermoregulation in the salamander Necturus maculosus.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1986, Volume: 85, Issue:1

    Topics: Animals; Body Temperature Regulation; Cimetidine; Dimaprit; Histamine; Histidine; Necturus; Pyridines; Pyrilamine; Receptors, Histamine; Thiourea

1986
Studies on the site and mechanism of the inhibitory action of intracerebral histamine on the cold-stimulated thyrotropin secretion in male rats.
    Brain research, 1985, Sep-23, Volume: 343, Issue:2

    Topics: Animals; Brain Mapping; Cimetidine; Cold Temperature; Histamine; Hypothalamus; Imidazoles; Impromidine; Injections, Intraventricular; Male; Pyridines; Pyrilamine; Rats; Thyrotropin

1985
Selective enhancement of histamine H1-receptor responses in guinea-pig ileal smooth muscle by 1,4-dithiothreitol.
    British journal of pharmacology, 1986, Volume: 87, Issue:1

    Topics: Acetylcholine; Animals; Dimaprit; Dithionitrobenzoic Acid; Dithiothreitol; Dose-Response Relationship, Drug; Female; Guanidines; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Thiourea

1986
Hyperlipemic responses induced by centrally administered histamine H1- and H2-receptor agonists in rats.
    Agents and actions, 1987, Volume: 20, Issue:3-4

    Topics: Animals; Brain; Cimetidine; Dimaprit; Fatty Acids, Nonesterified; Hyperlipidemias; Imidazoles; Impromidine; Injections, Intraventricular; Male; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Thiourea

1987
Histamine receptor effects on dissipation of an intracellular proton gradient of isolated gastric mucosal surface cells.
    Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), 1987, Volume: 185, Issue:4

    Topics: Animals; Bicarbonates; Chlorides; Cimetidine; Dimaprit; Diphenhydramine; Gastric Acid; Gastric Mucosa; Histamine; Protons; Pyridines; Pyrilamine; Rabbits; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Sodium; Thiourea

1987
Effect of H1 and H2 agonists on the chemiluminescence of human blood mononuclear cells induced by phytohaemagglutinin.
    Immunopharmacology, 1985, Volume: 9, Issue:3

    Topics: Cimetidine; Histamine; Humans; Imidazoles; Impromidine; Luminescent Measurements; Methylhistamines; Monocytes; Phytohemagglutinins; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Structure-Activity Relationship

1985
Effects of histamine agonists and antagonists on luminol-dependent chemiluminescence of granulocytes.
    Agents and actions, 1984, Volume: 15, Issue:3-4

    Topics: Cimetidine; Dimaprit; Granulocytes; Histamine; Histamine Antagonists; Humans; In Vitro Techniques; Luminescent Measurements; Luminol; Pyridazines; Pyridines; Pyrilamine; Ranitidine; Thiourea

1984
Evaluation of the role of Histamine H1- and H2-receptors in cutaneous inflammation in the guinea-pig produced by histamine and mast cell degranulation.
    British journal of pharmacology, 1980, Volume: 69, Issue:4

    Topics: Animals; Cimetidine; Dimaprit; Guinea Pigs; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Inflammation; Male; Mast Cells; Mathematics; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Skin; Thiourea; Vasodilation

1980
Identification and specific blockade of histaminergic receptors in guinea pig vasa deferentia.
    Canadian journal of physiology and pharmacology, 1981, Volume: 59, Issue:10

    Topics: Animals; Dose-Response Relationship, Drug; Guinea Pigs; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Reserpine; Vas Deferens

1981
Evidence for histamine H1 and H2 receptors in guinea-pig oxyntic cells.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:1

    Topics: Animals; Carbonic Anhydrases; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Female; Guinea Pigs; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; Impromidine; In Vitro Techniques; Methylhistamines; Parietal Cells, Gastric; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1983
Release of prolactin and luteinizing hormone by histamine agonists in ovariectomized, steroid-treated rats under ether anesthesia.
    Experimental brain research, 1983, Volume: 52, Issue:2

    Topics: Animals; Castration; Dimaprit; Female; Histamine; Histamine H1 Antagonists; Luteinizing Hormone; Methylhistamines; Metiamide; Pituitary Gland, Anterior; Prolactin; Pyridines; Pyrilamine; Rats; Thiourea

1983
The mechanism of the histamine-induced desensitization of guinea-pig ileum.
    General pharmacology, 1984, Volume: 15, Issue:1

    Topics: Animals; Guinea Pigs; Histamine; Histamine H1 Antagonists; Ileum; In Vitro Techniques; Male; Methylhistamines; Pyridines; Pyrilamine; Receptors, Histamine; Receptors, Histamine H1

1984
Inhibition of the TSH secretion by histamine in male rats.
    Acta endocrinologica, 1983, Volume: 103, Issue:1

    Topics: Animals; Cimetidine; Cold Temperature; Histamine; Histamine Antagonists; Histidine; Imidazoles; Impromidine; Male; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thyrotropin; Thyrotropin-Releasing Hormone

1983
Central histaminergic stimulation of pituitary--adrenocortical response in the rat.
    Life sciences, 1983, Sep-19, Volume: 33, Issue:12

    Topics: Animals; Cimetidine; Corticosterone; Dimaprit; Dose-Response Relationship, Drug; Histamine; Imidazoles; Impromidine; Male; Pituitary-Adrenal System; Pyridines; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiourea

1983
Studies with specific agonists and antagonists of the role of histamine H1- and H2-receptor activation in the pathogenesis of gastric lesions in rats.
    Agents and actions, 1984, Volume: 14, Issue:2

    Topics: Aminopyridines; Animals; Atropine; Dimaprit; Drug Interactions; Female; Histamine; Pyridines; Pyrilamine; Ranitidine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Stomach Ulcer; Thiourea

1984
Influence of temperature on sensitivity of histamine & its analogues in guinea pig tracheal chain.
    Indian journal of experimental biology, 1982, Volume: 20, Issue:1

    Topics: Animals; Female; Guinea Pigs; Histamine; In Vitro Techniques; Male; Pyridines; Pyrilamine; Receptors, Histamine; Temperature; Trachea

1982
Further characterization of the guinea pig left atrial tension response to histamine by use of selective agonists.
    Agents and actions, 1981, Volume: 11, Issue:3

    Topics: Animals; Female; Guinea Pigs; Heart Atria; Heart Rate; Histamine; In Vitro Techniques; Male; Methylhistamines; Myocardial Contraction; Pyridines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2

1981
Effect of histamine on motor function of opossum sphincter of Oddi.
    The American journal of physiology, 1981, Volume: 241, Issue:2

    Topics: Ampulla of Vater; Animals; Female; Histamine; Male; Methylhistamines; Metiamide; Motor Activity; Opossums; Pyridines; Pyrilamine; Receptors, Histamine H1; Sphincter of Oddi; Sympatholytics; Tetrodotoxin

1981
Histamine stimulates brain phospholipid turnover through a direct, H-1 receptor-mediated mechanism.
    Life sciences, 1980, Oct-06, Volume: 27, Issue:14

    Topics: Animals; Brain; Catecholamines; Cimetidine; Histamine; Male; Mast Cells; Methylhistamines; p-Methoxy-N-methylphenethylamine; Phosphates; Phospholipids; Pyridines; Pyrilamine; Rats; Receptors, Histamine; Receptors, Histamine H1; Reserpine

1980
Histamine H1-receptors modulate somatostatin receptors coupled to the inhibition of adenylyl cyclase in the rat frontoparietal cortex.
    Peptides, 1997, Volume: 18, Issue:10

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Binding, Competitive; Cell Membrane; Colforsin; Frontal Lobe; Guanylyl Imidodiphosphate; Histamine Antagonists; Parietal Lobe; Protein Binding; Pyridines; Pyrilamine; Radioimmunoassay; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, Somatostatin; Somatostatin

1997
Cholinergic and glutamatergic activation reverses working memory failure by hippocampal histamine H1 receptor blockade in rats.
    Life sciences, 2000, Volume: 67, Issue:10

    Topics: Acetylcholine; Animals; Cholinesterase Inhibitors; Cimetidine; Cycloserine; Drug Interactions; Glutamic Acid; Hippocampus; Histamine Agonists; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Memory; Memory Disorders; Neurons; Physostigmine; Pyridines; Pyrilamine; Rats; Rats, Wistar; Receptors, Histamine H1; Receptors, N-Methyl-D-Aspartate

2000