Page last updated: 2024-08-18

pyridostigmine bromide and tacrine

pyridostigmine bromide has been researched along with tacrine in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19901 (6.67)18.7374
1990's5 (33.33)18.2507
2000's1 (6.67)29.6817
2010's7 (46.67)24.3611
2020's1 (6.67)2.80

Authors

AuthorsStudies
Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ1
Ekins, S; Williams, AJ; Xu, JJ1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Galli, A; Mori, F1
Fischer, JP; Kewitz, H; Thomsen, T; Zendeh, B1
Arnal, F; Coté, LJ; Ginsburg, S; Lawrence, GD; Naini, A; Sano, M1
Kewitz, H; Pleul, O; Thomsen, T1
Glick, D; Loewenstein-Lichtenstein, Y; Nørgaard-Pedersen, B; Schwarz, M; Soreq, H; Zakut, H1
Ariel, N; Barak, D; Bino, T; Ordentlich, A; Shafferman, A; Velan, B1
Bajgar, J1
Hasan, MY; Kuča, K; Lorke, DE; Nurulain, SM; Petroianu, GA; Shafiullah, M2
Kassa, J; Korabecny, J; Sepsova, V; Tumova, M1
Hasan, MY; Kuča, K; Lorke, DE; Nurulain, SM; Petroianu, GA2

Other Studies

15 other study(ies) available for pyridostigmine bromide and tacrine

ArticleYear
Developing structure-activity relationships for the prediction of hepatotoxicity.
    Chemical research in toxicology, 2010, Jul-19, Volume: 23, Issue:7

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes

2010
A predictive ligand-based Bayesian model for human drug-induced liver injury.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Effectiveness of 1,2,3,4-tetrahydro-9-aminoacridine (THA) as a pretreatment drug for protection of mice from acute diisopropylfluorophosphate (DFP) intoxication.
    Archives of toxicology, 1991, Volume: 65, Issue:4

    Topics: Animals; Brain; Cholinesterase Inhibitors; Diaphragm; Dose-Response Relationship, Drug; Isoflurophate; Male; Mice; Physostigmine; Poisoning; Pyridostigmine Bromide; Tacrine; Time Factors

1991
In vitro effects of various cholinesterase inhibitors on acetyl- and butyrylcholinesterase of healthy volunteers.
    Biochemical pharmacology, 1991, Jan-01, Volume: 41, Issue:1

    Topics: Acetylcholinesterase; Butyrylcholinesterase; Cholinesterase Inhibitors; Erythrocytes; Humans; Physostigmine; Pyridostigmine Bromide; Tacrine; Tetraisopropylpyrophosphamide

1991
Studies on new, centrally active and reversible acetylcholinesterase inhibitors.
    Neurochemical research, 1990, Volume: 15, Issue:6

    Topics: Acetylcholinesterase; Animals; Blood-Brain Barrier; Brain; Cholinesterase Inhibitors; Dopamine; Male; Mice; Neostigmine; Norepinephrine; Pyridostigmine Bromide; Tacrine

1990
Estimation of cholinesterase activity (EC 3.1.1.7; 3.1.1.8) in undiluted plasma and erythrocytes as a tool for measuring in vivo effects of reversible inhibitors.
    Journal of clinical chemistry and clinical biochemistry. Zeitschrift fur klinische Chemie und klinische Biochemie, 1988, Volume: 26, Issue:7

    Topics: Acetylcholinesterase; Butyrylcholinesterase; Carbon Radioisotopes; Cholinesterase Inhibitors; Cholinesterases; Erythrocytes; Female; Humans; Kinetics; Male; Physostigmine; Pyridostigmine Bromide; Radioisotope Dilution Technique; Reference Values; Sex Factors; Tacrine

1988
Genetic predisposition to adverse consequences of anti-cholinesterases in 'atypical' BCHE carriers.
    Nature medicine, 1995, Volume: 1, Issue:10

    Topics: Acetylcholinesterase; Binding Sites; Butyrylcholinesterase; Butyrylthiocholine; Carbamates; Cholinesterase Inhibitors; Homozygote; Humans; Male; Pyridostigmine Bromide; Tacrine

1995
The 'aromatic patch' of three proximal residues in the human acetylcholinesterase active centre allows for versatile interaction modes with inhibitors.
    The Biochemical journal, 1998, Oct-01, Volume: 335 ( Pt 1)

    Topics: Acetylcholinesterase; Alkaloids; Binding Sites; Cholinesterase Inhibitors; Crystallography, X-Ray; Humans; Hydrogen Bonding; Kinetics; Ligands; Models, Chemical; Models, Molecular; Physostigmine; Protein Conformation; Pyridostigmine Bromide; Sesquiterpenes; Structure-Activity Relationship; Tacrine

1998
Protective effect of reversible cholinesterase inhibitors (tacrine, pyridostigmine) and eqbuche against VX poisoning and brain acetylcholinesterase inhibition in rats.
    Acta medica (Hradec Kralove), 2008, Volume: 51, Issue:4

    Topics: Animals; Brain; Chemical Warfare Agents; Cholinesterase Inhibitors; Female; Neurotoxicity Syndromes; Organothiophosphorus Compounds; Pyridostigmine Bromide; Rats; Rats, Wistar; Tacrine

2008
Pretreatment for acute exposure to diisopropylfluorophosphate: in vivo efficacy of various acetylcholinesterase inhibitors.
    Journal of applied toxicology : JAT, 2011, Volume: 31, Issue:6

    Topics: Amiloride; Animals; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Erythrocytes; Female; Humans; Inhibitory Concentration 50; Isoflurophate; Male; Methylene Blue; Metoclopramide; Oximes; Physostigmine; Proportional Hazards Models; Pyridinium Compounds; Pyridostigmine Bromide; Ranitidine; Rats; Tacrine; Tiapride Hydrochloride

2011
Usefulness of administration of non-organophosphate cholinesterase inhibitors before acute exposure to organophosphates: assessment using paraoxon.
    Journal of applied toxicology : JAT, 2013, Volume: 33, Issue:9

    Topics: Animals; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Lethal Dose 50; Male; Organophosphate Poisoning; Oximes; Paraoxon; Physostigmine; Pyridostigmine Bromide; Ranitidine; Rats; Rats, Wistar; Tacrine; Tiapride Hydrochloride

2013
The evaluation of prophylactic efficacy of newly developed reversible inhibitors of acetylcholinesterase in soman-poisoned mice - a comparison with commonly used pyridostigmine.
    Basic & clinical pharmacology & toxicology, 2014, Volume: 115, Issue:6

    Topics: Animals; Antidotes; Cholinesterase Inhibitors; Lethal Dose 50; Male; Mice; Piperazines; Pyridostigmine Bromide; Soman; Tacrine

2014
Reversible cholinesterase inhibitors as pre-treatment for exposure to organophosphates: assessment using azinphos-methyl.
    Journal of applied toxicology : JAT, 2015, Volume: 35, Issue:5

    Topics: Animals; Azinphosmethyl; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Male; Oximes; Physostigmine; Proportional Hazards Models; Pyridinium Compounds; Pyridostigmine Bromide; Ranitidine; Rats; Rats, Wistar; Tacrine

2015
Combined Pre- and Posttreatment of Paraoxon Exposure.
    Molecules (Basel, Switzerland), 2020, Mar-27, Volume: 25, Issue:7

    Topics: Animals; Cholinesterase Inhibitors; Cholinesterase Reactivators; Male; Organophosphates; Oximes; Paraoxon; Physostigmine; Post-Exposure Prophylaxis; Pre-Exposure Prophylaxis; Proportional Hazards Models; Pyridostigmine Bromide; Ranitidine; Rats; Rats, Wistar; Survival Analysis; Tacrine

2020