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pyridostigmine bromide and physostigmine

pyridostigmine bromide has been researched along with physostigmine in 70 studies

Research

Studies (70)

TimeframeStudies, this research(%)All Research%
pre-199033 (47.14)18.7374
1990's15 (21.43)18.2507
2000's12 (17.14)29.6817
2010's9 (12.86)24.3611
2020's1 (1.43)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ1
Brossi, A; Greig, NH; Holloway, HW; Lahiri, DK; Luo, W; Yu, QS1
Ekins, S; Williams, AJ; Xu, JJ1
Havard, CW; Lange, MJ1
Watts, P; Wilkinson, RG1
Bräunlich, H; Hartwich, R1
Gattenlöhner, W; Rasenack, U1
Landauer, W1
Galli, A; Mori, F1
Fischer, JP; Kewitz, H; Thomsen, T; Zendeh, B1
Anderson, D; Carchman, RA; Carter, WH; Gennings, C; Harris, LW; Lennox, WJ; Solana, RP1
Davis, LH; Kauffman, FC; Whittaker, M1
Dusticier, N; Ebihara, Y; Gauthier, GM; Nieoullon, A; Vercher, JL1
Husain, K; Marjit, DN; Vijayaraghavan, R1
Gross, CL; Kagey-Sobotka, A; Kilduff, JE; Meier, HL; Papirmeister, B1
Finger, AV; McMaster, SB1
Bass, KN; Das Gupta, S; Warnick, JE1
Arndt, H; Sprengard, M1
Riker, WF1
Kewitz, H; Pleul, O; Thomsen, T1
Albuquerque, EX; Aracava, Y; Brossi, A; Cintra, WM; Deshpande, SS; Schönenberger, B1
Beasley, VR; Carmichael, WW; Cook, WO; Dahlem, AM; Dellinger, JA; Harlin, KS1
Birnbaum, SG; Dellinger, JA; Jansen, HT; Zaber, DJ1
Brecht, KM; Lenz, DE; Maxwell, DM; O'Neill, BL1
Annau, Z; Mansour, NA; Shamoo, AE; Valdes, JJ1
Domino, EF1
King, JM; Romano, JA1
Albuquerque, EX; Deshpande, SS; Kauffman, FC; Rickett, DL; Viana, GB1
Bonds, AB; DeBruyn, EJ; Gajewski, YA1
Albuquerque, EX; Eldefrawi, AT; Eldefrawi, ME; Sherby, SM1
Anderson, DR; Harris, LW; Lennox, WJ; Talbot, BG1
Inns, RH; Leadbeater, L; Rylands, JM1
Schneider, R1
Cowan, A; Wray, SR1
Lagerquist, B; Morgan, GM; Stone, CA; Torchiana, ML; Wenger, HC1
Williams, D1
Fuhrmann, M; Gassner, B; Gössinger, H; Hruby, K; Shroff, D1
Akaike, A; Albuquerque, EX; Rickett, DL; Shaw, KP1
Harris, L; Stitcher, D1
Loh, L; Schott, GD1
Anderson, DR; Harris, LW; Lennox, WJ; Swanson, DR; Talbot, BG1
Dawson, RM1
Blick, DW; Brown, GC; Murphy, MR; Weathersby, FR1
Arvat, E; Bellone, J; Boffano, G; Camanni, F; Ghigo, E; Maccario, M; Mazza, E; Müller, EE; Procopio, M; Valetto, M1
Das Gupta, S; Husain, K; Kumar, P; Singh, R; Vijayaraghavan, R1
Blick, DW; Brown, GC; Miller, SA; Murphy, MR1
Friedman, A; Hendler, I; Kaufer, D; Shemer, J; Soreq, H; Tur-Kaspa, I1
Backman, SB; Collier, B; Polosa, C; Stein, RD1
Ariel, N; Barak, D; Bino, T; Ordentlich, A; Shafferman, A; Velan, B1
Hänninen, O; Kaliste-Korhonen, E; Raushel, FM; Tuovinen, K1
Alkalai, D; Cohen, G; Grauer, E; Kapon, J; Raveh, L1
Fitch, TE; Haley, RW; Petty, F; Sinton, CM1
Ben Nathan, D; Danenberg, HD; Grauer, E; Kapon, J; Kobiler, D; Lustig, S1
Aubriot, S; Baubichon, D; Carpentier, P; Dorandeu, F; Foquin, A; Lallement, G1
Baubichon, D; Carpentier, P; Dorandeu, F; Foquin, A; Lallement, G1
Barahona, V; Sánchez-Fortún, S1
Hall, T; Passingham, S; Wetherell, J1
BOUDIN, G; GOULON, M; HAMBURGER, J; LAPRESLE, J; LHERMITTE, F; PEQUIGNOT, H1
Eckert, S; Eyer, P; Mückter, H; Worek, F1
Barahona, MV; Sánchez-Fortún, S1
Bumm, R; Eckert, S; Eyer, P; Herkert, NM; Thiermann, H; Weber, G; Worek, F1
Barak, D; Greig, NH; Ordentlich, A; Shafferman, A; Stein, D; Yu, QS1
Grubbs, RD; Lucot, JB; Mauck, B; Paton, S1
Hasan, MY; Kuča, K; Lorke, DE; Nurulain, SM; Petroianu, GA; Shafiullah, M2
Herkert, NM; Thiermann, H; Worek, F1
Hasan, MY; Kuča, K; Lorke, DE; Nurulain, SM; Petroianu, GA2
Calas, AG; Krejci, E; Nachon, F; Nervo, A1

Reviews

3 review(s) available for pyridostigmine bromide and physostigmine

ArticleYear
[Myasthenia gravis].
    Recenti progressi in medicina, 1977, Volume: 62, Issue:1

    Topics: Autoimmune Diseases; Cholinesterase Inhibitors; Humans; Myasthenia Gravis; Neostigmine; Physostigmine; Pyridostigmine Bromide; Thymectomy; Thymoma; Thymus Neoplasms

1977
[Tricyclic antidepressive agents: clinical aspects and therapy of poisoning].
    Deutsche medizinische Wochenschrift (1946), 1976, Jul-30, Volume: 101, Issue:31

    Topics: Antidepressive Agents, Tricyclic; Arrhythmias, Cardiac; Brain Diseases; Brain Edema; Diazepam; Gastric Lavage; Humans; Hypotension; Myocardial Infarction; Pacemaker, Artificial; Physostigmine; Pyridostigmine Bromide; Respiration, Artificial; Salicylates

1976
Structure-activity relationship of reversible cholinesterase inhibitors: activation, channel blockade and stereospecificity of the nicotinic acetylcholine receptor-ion channel complex.
    Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas, 1988, Volume: 21, Issue:6

    Topics: Animals; Binding Sites; Chemical Phenomena; Chemistry; Cholinesterase Inhibitors; Edrophonium; Muscle Contraction; Neostigmine; Organophosphate Poisoning; Physostigmine; Pyridostigmine Bromide; Rana pipiens; Receptors, Nicotinic; Sciatic Nerve; Structure-Activity Relationship

1988

Other Studies

67 other study(ies) available for pyridostigmine bromide and physostigmine

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Developing structure-activity relationships for the prediction of hepatotoxicity.
    Chemical research in toxicology, 2010, Jul-19, Volume: 23, Issue:7

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes

2010
Long-acting anticholinesterases for myasthenia gravis: synthesis and activities of quaternary phenylcarbamates of neostigmine, pyridostigmine and physostigmine.
    Bioorganic & medicinal chemistry, 2010, Jul-01, Volume: 18, Issue:13

    Topics: Acetylcholinesterase; Animals; Butyrylcholinesterase; Cholinesterase Inhibitors; Humans; Mice; Myasthenia Gravis; Neostigmine; Phenylcarbamates; Physostigmine; Pyridostigmine Bromide

2010
A predictive ligand-based Bayesian model for human drug-induced liver injury.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands

2010
The interaction of carbamates with acetylcholinesterase.
    Biochemical pharmacology, 1977, Apr-15, Volume: 26, Issue:8

    Topics: Acetylcholinesterase; Animals; Benzofurans; Carbachol; Carbamates; Cattle; Erythrocytes; Insecticides; Kinetics; Physostigmine; Pyridostigmine Bromide

1977
[The use of direct and indirect parasympathomimetics in poisonings with tricyclic antidepressive agents].
    Zeitschrift fur die gesamte innere Medizin und ihre Grenzgebiete, 1978, Oct-15, Volume: 33, Issue:20

    Topics: Amitriptyline; Animals; Antidepressive Agents, Tricyclic; Arecoline; Cholinesterase Inhibitors; Coma; Dibenzocycloheptenes; Imipramine; Paraoxon; Physostigmine; Pyridostigmine Bromide; Rats

1978
Cholinomimetic teratogens: studies with chicken embryos.
    Teratology, 1975, Volume: 12, Issue:2

    Topics: Acetylcholine; Animals; Carbachol; Chick Embryo; Choline; Cholinesterase Inhibitors; Decamethonium Compounds; Drug Synergism; Gallamine Triethiodide; Musculoskeletal System; Neostigmine; Nicotine; Parasympathomimetics; Physostigmine; Pyridostigmine Bromide; Quaternary Ammonium Compounds; Succinylcholine; Teratogens

1975
Effectiveness of 1,2,3,4-tetrahydro-9-aminoacridine (THA) as a pretreatment drug for protection of mice from acute diisopropylfluorophosphate (DFP) intoxication.
    Archives of toxicology, 1991, Volume: 65, Issue:4

    Topics: Animals; Brain; Cholinesterase Inhibitors; Diaphragm; Dose-Response Relationship, Drug; Isoflurophate; Male; Mice; Physostigmine; Poisoning; Pyridostigmine Bromide; Tacrine; Time Factors

1991
In vitro effects of various cholinesterase inhibitors on acetyl- and butyrylcholinesterase of healthy volunteers.
    Biochemical pharmacology, 1991, Jan-01, Volume: 41, Issue:1

    Topics: Acetylcholinesterase; Butyrylcholinesterase; Cholinesterase Inhibitors; Erythrocytes; Humans; Physostigmine; Pyridostigmine Bromide; Tacrine; Tetraisopropylpyrophosphamide

1991
Evaluation of the efficacy of two carbamates, physostigmine and pyridostigmine, when used in conjunction for protection against organophosphate exposure.
    Fundamental and applied toxicology : official journal of the Society of Toxicology, 1990, Volume: 15, Issue:4

    Topics: Acetylcholinesterase; Animals; Cholinesterase Inhibitors; Female; Guinea Pigs; Lethal Dose 50; Male; Models, Biological; Organophosphorus Compounds; Physostigmine; Pyridostigmine Bromide; Regression Analysis; Soman

1990
Activation of glycogen phosphorylase in rat pheochromocytoma PC12 cells and isolated hepatocytes by organophosphates.
    Biochemical pharmacology, 1990, Jan-15, Volume: 39, Issue:2

    Topics: Adenine Nucleotides; Animals; Calcium; Cells, Cultured; Cytosol; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Activation; Hydrogen-Ion Concentration; Liver; Male; Organophosphorus Compounds; Pheochromocytoma; Phosphorylase a; Phosphorylases; Physostigmine; Pyridostigmine Bromide; Rats; Tumor Cells, Cultured; Verapamil

1990
Pyridostigmine-induced inhibition of blood acetylcholinesterase (AChE) and resulting effects on manual ocular tracking performance in the trained baboon.
    Behavioral and neural biology, 1990, Volume: 53, Issue:3

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Attention; Dose-Response Relationship, Drug; Eye Movements; Female; Injections, Intramuscular; Ketamine; Kinesthesis; Male; Papio; Physostigmine; Psychomotor Performance; Pursuit, Smooth; Pyridostigmine Bromide

1990
The effect of pyridostigmine and physostigmine on acute toxicity of diisopropyl fluorophosphate in rats.
    Arhiv za higijenu rada i toksikologiju, 1990, Volume: 41, Issue:1

    Topics: Acetylcholinesterase; Animals; Blood Glucose; Glycogen; Isoflurophate; Male; Physostigmine; Pyridostigmine Bromide; Rats

1990
Histamine release by esterase inhibitors. The regulation of histamine release from human leukocytes of allergic and non-allergic individuals by the serine esterase inhibitors diisopropyl fluorophosphate and pinacolyl methylphosphorofluoridate.
    International archives of allergy and applied immunology, 1985, Volume: 77, Issue:1-2

    Topics: Enzyme Inhibitors; Esterases; Histamine Release; Humans; Hypersensitivity; Isoflurophate; Kinetics; Organophosphorus Compounds; Physostigmine; Pyridostigmine Bromide; Soman; Temperature

1985
Effects of exercise on behavioral sensitivity to carbamate cholinesterase inhibitors.
    Pharmacology, biochemistry, and behavior, 1989, Volume: 33, Issue:4

    Topics: Animals; Behavior, Animal; Conditioning, Operant; Dose-Response Relationship, Drug; Male; Physical Conditioning, Animal; Physical Exertion; Physostigmine; Pyridostigmine Bromide; Random Allocation; Rats; Rats, Inbred Strains; Reinforcement Schedule

1989
Interaction of reversible and irreversible cholinesterase inhibitors on the monosynaptic reflex in neonatal rats.
    Toxicology and applied pharmacology, 1989, Jun-01, Volume: 99, Issue:1

    Topics: Animals; Atropine; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Male; Physostigmine; Pregnancy; Pyridostigmine Bromide; Rats; Rats, Inbred Strains; Reflex, Monosynaptic; Sarin; Spinal Cord

1989
Effects of carbamates upon various behavioural parameters in mice.
    Archives of toxicology. Supplement. = Archiv fur Toxikologie. Supplement, 1989, Volume: 13

    Topics: Animals; Behavior, Animal; Carbamates; Dose-Response Relationship, Drug; Double-Blind Method; Male; Mice; Motor Activity; Physostigmine; Psychomotor Performance; Pyridostigmine Bromide; Respiration

1989
Memory impairment in myasthenia gravis.
    Neurology, 1989, Volume: 39, Issue:4

    Topics: Cognition Disorders; Humans; Memory Disorders; Myasthenia Gravis; Physostigmine; Pyridostigmine Bromide

1989
Estimation of cholinesterase activity (EC 3.1.1.7; 3.1.1.8) in undiluted plasma and erythrocytes as a tool for measuring in vivo effects of reversible inhibitors.
    Journal of clinical chemistry and clinical biochemistry. Zeitschrift fur klinische Chemie und klinische Biochemie, 1988, Volume: 26, Issue:7

    Topics: Acetylcholinesterase; Butyrylcholinesterase; Carbon Radioisotopes; Cholinesterase Inhibitors; Cholinesterases; Erythrocytes; Female; Humans; Kinetics; Male; Physostigmine; Pyridostigmine Bromide; Radioisotope Dilution Technique; Reference Values; Sex Factors; Tacrine

1988
Comparison of effects of anatoxin-a(s) and paraoxon, physostigmine and pyridostigmine on mouse brain cholinesterase activity.
    Toxicon : official journal of the International Society on Toxinology, 1988, Volume: 26, Issue:8

    Topics: Animals; Bacterial Toxins; Brain; Cholinesterase Inhibitors; Cholinesterases; Cyanobacteria Toxins; Lethal Dose 50; Male; Marine Toxins; Mice; Mice, Inbred BALB C; Microcystins; Paraoxon; Physostigmine; Pyridostigmine Bromide; Rats; Tropanes

1988
Vagal tone monitoring: a potential indicator of anti-cholinesterase exposure in Macaca mulatta.
    Toxicology, 1988, Volume: 49, Issue:2-3

    Topics: Acetylcholinesterase; Animals; Atropine; Cholinesterase Inhibitors; Erythrocytes; Macaca mulatta; Monitoring, Physiologic; Physostigmine; Pyridostigmine Bromide; Vagus Nerve

1988
Effect of carboxylesterase inhibition on carbamate protection against soman toxicity.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 246, Issue:3

    Topics: Acetylcholinesterase; Animals; Carboxylesterase; Carboxylic Ester Hydrolases; Guinea Pigs; Lethal Dose 50; Male; Organophosphorus Compounds; Physostigmine; Pyridostigmine Bromide; Rabbits; Rats; Rats, Inbred Strains; Soman

1988
Biochemical interactions of carbamates and ecothiophate with the activated conformation of nicotinic acetylcholine receptor.
    Journal of biochemical toxicology, 1987,Spring, Volume: 2

    Topics: Biotransformation; Bungarotoxins; Carbamates; Echothiophate Iodide; Neostigmine; Phencyclidine; Physostigmine; Pyridostigmine Bromide; Receptors, Nicotinic

1987
Comparative seizure inducing properties of various cholinesterase inhibitors: antagonism by diazepam and midazolam.
    Neurotoxicology, 1987,Spring, Volume: 8, Issue:1

    Topics: Animals; Atropine; Behavior, Animal; Cholinesterase Inhibitors; Diazepam; Isoflurophate; Male; Midazolam; Neostigmine; Paraoxon; Physostigmine; Pyridostigmine Bromide; Rats; Rats, Inbred Strains; Seizures

1987
Conditioned taste aversion and cholinergic drugs: pharmacological antagonism.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 27, Issue:1

    Topics: Animals; Atropine; Avoidance Learning; Benactyzine; Conditioning, Classical; Male; Parasympathomimetics; Physostigmine; Pyridostigmine Bromide; Rats; Saccharin; Taste

1987
Effectiveness of physostigmine as a pretreatment drug for protection of rats from organophosphate poisoning.
    Fundamental and applied toxicology : official journal of the Society of Toxicology, 1986, Volume: 6, Issue:3

    Topics: Acetylcholinesterase; Action Potentials; Animals; Atropine; Body Weight; Brain; Brain Chemistry; Cholinesterases; Female; gamma-Aminobutyric Acid; Muscle Contraction; Muscles; Neostigmine; Organophosphate Poisoning; Physostigmine; Pyridostigmine Bromide; Rats; Rats, Inbred Strains; Sarin

1986
Anticholinesterase agents affect contrast gain of the cat cortical visual evoked potential.
    Neuroscience letters, 1986, Nov-21, Volume: 71, Issue:3

    Topics: Acetylcholine; Animals; Atropine; Cats; Cholinesterase Inhibitors; Evoked Potentials, Visual; Isoflurophate; Physostigmine; Pyridostigmine Bromide; Soman; Visual Cortex; Visual Perception

1986
Comparison of the actions of carbamate anticholinesterases on the nicotinic acetylcholine receptor.
    Molecular pharmacology, 1985, Volume: 27, Issue:3

    Topics: Acetylcholine; Amphibian Venoms; Animals; Binding, Competitive; Bungarotoxins; Carbachol; Electric Organ; Kinetics; Neostigmine; Physostigmine; Pyridostigmine Bromide; Receptors, Cholinergic; Torpedo

1985
Relationship between reversible acetylcholinesterase inhibition and efficacy against soman lethality.
    Life sciences, 1985, Sep-02, Volume: 37, Issue:9

    Topics: Acetylcholinesterase; Animals; Atropine; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Drug Therapy, Combination; Female; Guinea Pigs; Male; Mecamylamine; Organophosphorus Compounds; Physostigmine; Pralidoxime Compounds; Pyridostigmine Bromide; Rats; Soman

1985
Treatment of poisoning by soman.
    Fundamental and applied toxicology : official journal of the Society of Toxicology, 1985, Volume: 5, Issue:6 Pt 2

    Topics: Animals; Antidotes; Atropine; Carbamates; Diazepam; Guinea Pigs; Male; Motor Activity; Organophosphate Poisoning; Parasympatholytics; Phenylpropionates; Physostigmine; Pyridostigmine Bromide; Sarin; Soman; Time Factors

1985
A test for the assessment of the duration of the action of neostigmine and of the relative potencies of various anticholinesterases using the pupil of the mouse.
    The Journal of pharmacy and pharmacology, 1970, Volume: 22, Issue:4

    Topics: Animals; Atropine; Cholinesterase Inhibitors; Edrophonium; Female; Male; Methods; Mice; Miotics; Neostigmine; Physostigmine; Pupil; Pyridostigmine Bromide; Time Factors

1970
Correlation between animal and clinical findings with a psychotomimetic anticholinesterase.
    Neuropharmacology, 1973, Volume: 12, Issue:4

    Topics: Animals; Avoidance Learning; Cholinesterase Inhibitors; Cyclohexanes; Female; Hallucinogens; Lysergic Acid Diethylamide; Physostigmine; Pyridostigmine Bromide; Pyrrolidines; Rats; Time Factors

1973
Pharmacological antagonism of the toxic manifestations of amitriptyline and protriptyline in dogs.
    Toxicology and applied pharmacology, 1972, Volume: 21, Issue:3

    Topics: Amitriptyline; Animals; Antidepressive Agents; Dibenzocycloheptenes; Dogs; Drug Antagonism; Electrocardiography; Heart Rate; Mecamylamine; Methylamines; Physostigmine; Propranolol; Propylamines; Pyridostigmine Bromide

1972
The management of myasthenia.
    Modern trends in neurology, 1967, Volume: 4, Issue:0

    Topics: Adult; Ambenonium Chloride; Carcinoma, Bronchogenic; Ephedrine; Female; Follow-Up Studies; Humans; Hyperthyroidism; Lung Neoplasms; Male; Middle Aged; Muscular Diseases; Myasthenia Gravis; Myositis; Neostigmine; Oculomotor Muscles; Physostigmine; Pyridostigmine Bromide; Thymectomy; Thymoma; Thymus Neoplasms

1967
[Clinical aspects and therapy of acute poisoning by the drug combination melitracen-flupenthixol (Deanxit)].
    Wiener medizinische Wochenschrift (1946), 1983, Jun-15, Volume: 133, Issue:11

    Topics: Adolescent; Adult; Anthracenes; Basal Ganglia Diseases; Biperiden; Cardiac Complexes, Premature; Child, Preschool; Coma; Drug Combinations; Female; Flupenthixol; Gastric Lavage; Humans; Male; Middle Aged; Physostigmine; Pyridostigmine Bromide; Tachycardia; Thioxanthenes

1983
The interaction of anticholinesterase agents with the acetylcholine receptor-ionic channel complex.
    Fundamental and applied toxicology : official journal of the Society of Toxicology, 1984, Volume: 4, Issue:2 Pt 2

    Topics: Action Potentials; Animals; Anura; Cholinesterase Inhibitors; In Vitro Techniques; Ion Channels; Motor Endplate; Muscle Contraction; Physostigmine; Pyridostigmine Bromide; Rats; Receptors, Cholinergic; Receptors, Nicotinic

1984
Protection against diisopropylfluorophosphate intoxication by pyridostigmine and physostigmine in combination with atropine and mecamylamine.
    Naunyn-Schmiedeberg's archives of pharmacology, 1984, Volume: 327, Issue:1

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Antidotes; Atropine; Brain Chemistry; Drug Combinations; Isoflurophate; Male; Mecamylamine; Physostigmine; Pyridostigmine Bromide; Rats

1984
Anticholinesterase drugs in the treatment of chronic pain.
    Pain, 1984, Volume: 20, Issue:2

    Topics: Arm; Cholinesterase Inhibitors; Chronic Disease; Humans; Leg; Male; Middle Aged; Neostigmine; Pain; Physostigmine; Propantheline; Pyridostigmine Bromide; Shoulder; Syndrome

1984
Toxicity of anticholinesterases: interactions of pyridostigmine and physostigmine with soman.
    Drug and chemical toxicology, 1984, Volume: 7, Issue:5

    Topics: Acetylcholinesterase; Animals; Drug Interactions; Lethal Dose 50; Male; Motor Activity; Organophosphorus Compounds; Physostigmine; Pyridostigmine Bromide; Rats; Rats, Inbred Strains; Soman

1984
Oxime effects on the rate constants of carbamylation and decarbamylation of acetylcholinesterase for pyridostigmine, physostigmine and insecticidal carbamates.
    Neurochemistry international, 1995, Volume: 26, Issue:6

    Topics: Acetylcholinesterase; Animals; Cattle; Erythrocytes; In Vitro Techniques; Insecticides; Kinetics; Oximes; Physostigmine; Pyridostigmine Bromide; Structure-Activity Relationship

1995
Behavioral toxicity of anticholinesterases in primates: effects of daily repeated soman exposure.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 48, Issue:3

    Topics: Animals; Behavior, Animal; Cholinesterase Inhibitors; Cholinesterases; Macaca mulatta; Male; Physostigmine; Postural Balance; Psychomotor Performance; Pyridostigmine Bromide; Soman

1994
Effects of direct and indirect acetylcholine receptor agonists on growth hormone secretion in humans.
    European journal of pharmacology, 1994, Mar-11, Volume: 254, Issue:1-2

    Topics: Adult; Bethanechol Compounds; Cholinergic Antagonists; Cholinesterase Inhibitors; Female; Flushing; Growth Hormone; Growth Hormone-Releasing Hormone; Humans; Injections, Intravenous; Male; Neostigmine; Physostigmine; Pyridostigmine Bromide; Receptors, Cholinergic

1994
Influence of pretreatment of carbamates on dynamic pulmonary mechanics in rats exposed to sarin aerosols.
    Indian journal of physiology and pharmacology, 1993, Volume: 37, Issue:3

    Topics: Aerosols; Animals; Carbamates; Male; Physostigmine; Pyridostigmine Bromide; Rats; Rats, Wistar; Respiratory Mechanics; Sarin

1993
Behavioral toxicity of anticholinesterases in primates: chronic physostigmine and soman interactions.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 45, Issue:3

    Topics: Animals; Behavior, Animal; Cholinesterase Inhibitors; Cholinesterases; Drug Interactions; Injections, Subcutaneous; Macaca mulatta; Male; Physostigmine; Psychomotor Performance; Pyridostigmine Bromide; Soman

1993
Pyridostigmine brain penetration under stress enhances neuronal excitability and induces early immediate transcriptional response.
    Nature medicine, 1996, Volume: 2, Issue:12

    Topics: Acetylthiocholine; Animals; Blood-Brain Barrier; Brain; Cell Membrane Permeability; Cholinesterase Inhibitors; Evoked Potentials; Gene Expression Regulation; Genes, Immediate-Early; Hippocampus; Mice; Molecular Sequence Data; Persian Gulf Syndrome; Physostigmine; Proto-Oncogene Proteins c-fos; Pyridostigmine Bromide; RNA, Messenger; Stress, Physiological; Transcription, Genetic

1996
Bradycardia produced by pyridostigmine and physostigmine.
    Canadian journal of anaesthesia = Journal canadien d'anesthesie, 1997, Volume: 44, Issue:12

    Topics: Animals; Bradycardia; Cats; Cholinesterase Inhibitors; Cholinesterases; Dose-Response Relationship, Drug; Electric Stimulation; Erythrocytes; Heart Rate; Muscarinic Antagonists; Nicotinic Antagonists; Physostigmine; Pyridostigmine Bromide; Vagotomy

1997
The 'aromatic patch' of three proximal residues in the human acetylcholinesterase active centre allows for versatile interaction modes with inhibitors.
    The Biochemical journal, 1998, Oct-01, Volume: 335 ( Pt 1)

    Topics: Acetylcholinesterase; Alkaloids; Binding Sites; Cholinesterase Inhibitors; Crystallography, X-Ray; Humans; Hydrogen Bonding; Kinetics; Ligands; Models, Chemical; Models, Molecular; Physostigmine; Protein Conformation; Pyridostigmine Bromide; Sesquiterpenes; Structure-Activity Relationship; Tacrine

1998
Success of pyridostigmine, physostigmine, eptastigmine and phosphotriesterase treatments in acute sarin intoxication.
    Toxicology, 1999, Jun-15, Volume: 134, Issue:2-3

    Topics: Animals; Antidotes; Aryldialkylphosphatase; Esterases; Lethal Dose 50; Male; Mice; Physostigmine; Pyridostigmine Bromide; Sarin

1999
Stress does not enable pyridostigmine to inhibit brain cholinesterase after parenteral administration.
    Toxicology and applied pharmacology, 2000, May-01, Volume: 164, Issue:3

    Topics: Animals; Brain; Cholinesterase Inhibitors; Cholinesterases; Cold Temperature; Female; Male; Mice; Physostigmine; Pyridostigmine Bromide; Stress, Physiological; Swimming

2000
Stressful manipulations that elevate corticosterone reduce blood-brain barrier permeability to pyridostigmine in the Rat.
    Toxicology and applied pharmacology, 2000, May-15, Volume: 165, Issue:1

    Topics: Acetylcholinesterase; Anesthetics, Inhalation; Animals; Anti-Inflammatory Agents; Blood-Brain Barrier; Brain; Central Nervous System; Cholinesterase Inhibitors; Corticosterone; Halothane; Male; Mice; Permeability; Physostigmine; Pyridostigmine Bromide; Rats; Rats, Long-Evans; Rats, Wistar; Stress, Physiological

2000
Viral neuroinvasion as a marker for BBB integrity following exposure to cholinesterase inhibitors.
    Life sciences, 2001, Jan-19, Volume: 68, Issue:9

    Topics: Alphavirus Infections; Animals; Blood-Brain Barrier; Brain; Central Nervous System Diseases; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Female; Lethal Dose 50; Mice; Mice, Inbred ICR; Permeability; Physostigmine; Pyridostigmine Bromide; Sindbis Virus; Soman; Viremia

2001
Subchronic administration of various pretreatments of nerve agent poisoning. I. Protection of blood and central cholinesterases, innocuousness towards blood-brain barrier permeability.
    Drug and chemical toxicology, 2001, Volume: 24, Issue:2

    Topics: Alkaloids; Animals; Blood-Brain Barrier; Brain; Cholinesterase Inhibitors; Cholinesterases; Erythrocytes; Evans Blue; Guinea Pigs; Male; Microscopy, Fluorescence; Neuroprotective Agents; Physostigmine; Pyridostigmine Bromide; Serum Albumin; Sesquiterpenes

2001
Subchronic administration of various pretreatments of nerve agent poisoning. II. Compared efficacy against soman toxicity.
    Drug and chemical toxicology, 2001, Volume: 24, Issue:2

    Topics: Alkaloids; Animals; Cholinesterase Inhibitors; Electroencephalography; Guinea Pigs; Male; Neuroprotective Agents; Physostigmine; Pyridostigmine Bromide; Scopolamine; Seizures; Sesquiterpenes; Soman; Time Factors

2001
The use of carbamates, atropine, and 2-pyridine aldoxime methoiodide in the protection of Artemia salina against poisoning by carbophenothion.
    Environmental toxicology and chemistry, 2001, Volume: 20, Issue:9

    Topics: Animals; Artemia; Atropine; Cholinesterase Inhibitors; Cholinesterase Reactivators; Dose-Response Relationship, Drug; Drug Interactions; Insecticides; Lethal Dose 50; Muscarinic Antagonists; Organothiophosphorus Compounds; Physostigmine; Pralidoxime Compounds; Pyridostigmine Bromide; Water Pollutants, Chemical

2001
Physostigmine and hyoscine improves protection against the lethal and incapacitating effects of nerve agent poisoning in the guinea-pig.
    Neurotoxicology, 2002, Volume: 23, Issue:3

    Topics: Animals; Antidotes; Body Temperature; Chemical Warfare Agents; Cholinesterase Inhibitors; Cholinesterases; Drug Implants; Guinea Pigs; Male; Muscarinic Antagonists; Organothiophosphorus Compounds; Physostigmine; Pyridostigmine Bromide; Scopolamine; Weight Gain

2002
[HOW TO TREAT MYASTHENIA].
    La Presse medicale, 1964, Oct-10, Volume: 72

    Topics: Ambenonium Chloride; Ephedrine; Humans; Muscle Weakness; Myasthenia Gravis; Neostigmine; Physostigmine; Prognosis; Pyridostigmine Bromide; Respiratory Insufficiency; Spironolactone; Surgical Procedures, Operative; Thymus Neoplasms

1964
Kinetic analysis of the protection afforded by reversible inhibitors against irreversible inhibition of acetylcholinesterase by highly toxic organophosphorus compounds.
    Biochemical pharmacology, 2006, Jul-28, Volume: 72, Issue:3

    Topics: Acetylcholinesterase; Algorithms; Alkaloids; Carbamates; Cholinesterase Inhibitors; Cholinesterase Reactivators; Dose-Response Relationship, Drug; Erythrocytes; Humans; Kinetics; Organophosphorus Compounds; Paraoxon; Physostigmine; Pyridostigmine Bromide; Sesquiterpenes; Time Factors

2006
Toxicity and characterization of cholinesterase-inhibition induced by diisopropyl fluorophosphate in Artemia salina larvae.
    Ecotoxicology and environmental safety, 2009, Volume: 72, Issue:3

    Topics: Animals; Artemia; Atropine; Cholinesterase Inhibitors; Cholinesterase Reactivators; Drug Therapy, Combination; Isoflurophate; Larva; Longevity; Muscarinic Antagonists; Physostigmine; Pralidoxime Compounds; Pyridostigmine Bromide; Toxicity Tests, Acute; Water Pollutants, Chemical

2009
Identical kinetics of human erythrocyte and muscle acetylcholinesterase with respect to carbamate pre-treatment, residual activity upon soman challenge and spontaneous reactivation after withdrawal of the inhibitors.
    Toxicology, 2008, Apr-18, Volume: 246, Issue:2-3

    Topics: Acetylcholinesterase; Carbamates; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Enzyme Activation; Erythrocytes; Humans; Kinetics; Muscle, Skeletal; Physostigmine; Pyridostigmine Bromide; Soman

2008
Accommodation of physostigmine and its analogues by acetylcholinesterase is dominated by hydrophobic interactions.
    The Biochemical journal, 2009, Jan-01, Volume: 417, Issue:1

    Topics: Acetylcholinesterase; Binding Sites; Catalysis; Cholinesterase Inhibitors; Humans; Hydrophobic and Hydrophilic Interactions; Kinetics; Models, Molecular; Molecular Structure; Mutation; Phenylcarbamates; Physostigmine; Protein Binding; Pyridostigmine Bromide; Rivastigmine; Structure-Activity Relationship

2009
Cholinesterase inhibitors and stress: effects on brain muscarinic receptor density in mice.
    Neurotoxicology, 2010, Volume: 31, Issue:5

    Topics: Animals; Brain; Cholinesterase Inhibitors; Cholinesterases; Disease Models, Animal; Dose-Response Relationship, Drug; Male; Mice; Mice, Inbred C57BL; Physostigmine; Protein Binding; Pyridostigmine Bromide; Receptors, Muscarinic; Stress, Psychological

2010
Pretreatment for acute exposure to diisopropylfluorophosphate: in vivo efficacy of various acetylcholinesterase inhibitors.
    Journal of applied toxicology : JAT, 2011, Volume: 31, Issue:6

    Topics: Amiloride; Animals; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Erythrocytes; Female; Humans; Inhibitory Concentration 50; Isoflurophate; Male; Methylene Blue; Metoclopramide; Oximes; Physostigmine; Proportional Hazards Models; Pyridinium Compounds; Pyridostigmine Bromide; Ranitidine; Rats; Tacrine; Tiapride Hydrochloride

2011
In vitro kinetic interactions of pyridostigmine, physostigmine and soman with erythrocyte and muscle acetylcholinesterase from different species.
    Toxicology letters, 2011, Sep-25, Volume: 206, Issue:1

    Topics: Acetylcholinesterase; Animals; Carbamates; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Drug Interactions; Erythrocytes; Female; Guinea Pigs; Humans; In Vitro Techniques; Kinetics; Macaca mulatta; Male; Muscle, Skeletal; Physostigmine; Pyridostigmine Bromide; Soman; Species Specificity; Swine

2011
Usefulness of administration of non-organophosphate cholinesterase inhibitors before acute exposure to organophosphates: assessment using paraoxon.
    Journal of applied toxicology : JAT, 2013, Volume: 33, Issue:9

    Topics: Animals; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Lethal Dose 50; Male; Organophosphate Poisoning; Oximes; Paraoxon; Physostigmine; Pyridostigmine Bromide; Ranitidine; Rats; Rats, Wistar; Tacrine; Tiapride Hydrochloride

2013
Reversible cholinesterase inhibitors as pre-treatment for exposure to organophosphates: assessment using azinphos-methyl.
    Journal of applied toxicology : JAT, 2015, Volume: 35, Issue:5

    Topics: Animals; Azinphosmethyl; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Male; Oximes; Physostigmine; Proportional Hazards Models; Pyridinium Compounds; Pyridostigmine Bromide; Ranitidine; Rats; Rats, Wistar; Tacrine

2015
Respiratory failure triggered by cholinesterase inhibitors may involve activation of a reflex sensory pathway by acetylcholine spillover.
    Toxicology, 2019, 08-01, Volume: 424

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Cholinesterase Inhibitors; Collagen; Female; Irritants; Male; Mice; Mice, Knockout; Muscle Proteins; Neuromuscular Junction; Physostigmine; Pyridostigmine Bromide; Reflex; Respiration; Respiratory Insufficiency; Sensory Receptor Cells; Signal Transduction

2019
Combined Pre- and Posttreatment of Paraoxon Exposure.
    Molecules (Basel, Switzerland), 2020, Mar-27, Volume: 25, Issue:7

    Topics: Animals; Cholinesterase Inhibitors; Cholinesterase Reactivators; Male; Organophosphates; Oximes; Paraoxon; Physostigmine; Post-Exposure Prophylaxis; Pre-Exposure Prophylaxis; Proportional Hazards Models; Pyridostigmine Bromide; Ranitidine; Rats; Rats, Wistar; Survival Analysis; Tacrine

2020