pyridine has been researched along with chloroquine in 5 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 3 (60.00) | 29.6817 |
2010's | 2 (40.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bambal, RB; Bates, M; Berry, N; Biagini, GA; Bonar-Law, R; Bray, PG; Brigandi, RA; Davis, CB; Gargallo, DV; Gibbons, P; Gomez-delas-Heras, FM; Gresham, SL; Hart, TK; Hindley, S; Lawrence, RM; Maggs, JL; Mukhtar, A; O'Neill, PM; Park, BK; Roberts, P; Shone, AE; Stocks, PA; Ward, SA; Winstanley, PA | 1 |
Asadollahy, E; Bambal, RB; Bates, M; Berry, N; Biagini, G; Bray, PG; Brigandi, RA; Davies, J; Davis, CB; Gargallo, DV; Gomez-de-Las-Heras, FM; Gresham, SL; Hall, C; Hindley, S; Lander, H; Maggs, JL; Nixon, G; O'Neill, PM; Parapini, S; Park, BK; Rimmer, K; Roberts, P; Shone, AE; Stanford, D; Stocks, PA; Taramelli, D; Vivas, L; Ward, SA; Winstanley, PA | 1 |
Egan, TJ; Ncokazi, KK | 1 |
El Kaïm, L; Grimaud, L; Pravin, P | 1 |
Abramo, C; Budu, A; Butera, AP; Carmona, AK; da Silva, GR; da Silva, MG; de Almeida, HG; de Brito, CFA; de Castro, WV; de Miranda Martins, NR; de Pilla Varotti, F; de Sousa Luz, LS; de Souza Reis, V; do Nascimento, SB; Dos Santos, FV; Gazarini, ML; Guimarães, DSM; Guimarães, L; Júnior, CSN; Kemmer, VM; Maluf, SEC; Marinho, JA; Ribeiro-Viana, RM; Silva, LR; Viana, GHR | 1 |
5 other study(ies) available for pyridine and chloroquine
Article | Year |
---|---|
Candidate selection and preclinical evaluation of N-tert-butyl isoquine (GSK369796), an affordable and effective 4-aminoquinoline antimalarial for the 21st century.
Topics: Aminoquinolines; Amodiaquine; Animals; Antimalarials; Benzylamines; Cytochrome P-450 Enzyme Inhibitors; Dogs; Drug Evaluation, Preclinical; Drug Resistance; Female; Haplorhini; Heme; Humans; Malaria; Mice; Models, Molecular; Plasmodium berghei; Plasmodium falciparum; Plasmodium yoelii; Rats; Structure-Activity Relationship | 2009 |
Synthesis, antimalarial activity, and preclinical pharmacology of a novel series of 4'-fluoro and 4'-chloro analogues of amodiaquine. Identification of a suitable "back-up" compound for N-tert-butyl isoquine.
Topics: Aminoquinolines; Amodiaquine; Animals; Antimalarials; Cell Survival; Chloroquine; Dogs; Drug Resistance; Female; Haplorhini; Hepatocytes; Humans; In Vitro Techniques; Malaria; Male; Mice; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Plasmodium yoelii; Rats; Rats, Wistar; Structure-Activity Relationship | 2009 |
A colorimetric high-throughput beta-hematin inhibition screening assay for use in the search for antimalarial compounds.
Topics: Animals; Antimalarials; Chloroquine; Colorimetry; Drug Evaluation, Preclinical; Hemeproteins; Inhibitory Concentration 50; Pyridines | 2005 |
Ugi-Smiles couplings of 4-substituted pyridine derivatives: a fast access to chloroquine analogues.
Topics: Antimalarials; Chloroquine; Molecular Structure; Pyridines; Time Factors | 2012 |
Improvement of antimalarial activity of a 3-alkylpiridine alkaloid analog by replacing the pyridine ring to a thiazole-containing heterocycle: Mode of action, mutagenicity profile, and Caco-2 cell-based permeability.
Topics: Alkaloids; Animals; Antimalarials; Caco-2 Cells; Cell Line; Cell Line, Tumor; Chloroquine; Female; Hemeproteins; Humans; Malaria; Mice; Mutagens; Permeability; Plasmodium berghei; Plasmodium falciparum; Pyridines; Thiazoles | 2019 |