Page last updated: 2024-08-21

pyridazine and piperazine

pyridazine has been researched along with piperazine in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fotsch, C; St Jean, DJ1
Biancalani, C; Cesari, N; Cilibrizzi, A; Colucci, M; Dal Piaz, V; Di Gianuario, A; Garrone, B; Giovannoni, MP; Graziano, A; Mangano, G; Pieretti, S; Polenzani, L; Vergelli, C1
Aslanian, RG; Black, TA; Cacciapuoti, A; Herr, RJ; Jenkins, DM; Kim, DW; Kuang, R; Lam, SQ; Lee, JF; McNicholas, PM; Ting, PC; Wainhaus, S; Walker, SS; Wu, H; Xu, Y; Zych, AJ1

Reviews

1 review(s) available for pyridazine and piperazine

ArticleYear
Mitigating heterocycle metabolism in drug discovery.
    Journal of medicinal chemistry, 2012, Jul-12, Volume: 55, Issue:13

    Topics: Animals; Biotransformation; Databases, Factual; Drug Discovery; Drug Interactions; Heterocyclic Compounds, 1-Ring; Heterocyclic Compounds, 4 or More Rings; Humans; Mice; Pharmaceutical Preparations; Rats

2012

Other Studies

2 other study(ies) available for pyridazine and piperazine

ArticleYear
Further studies on arylpiperazinyl alkyl pyridazinones: discovery of an exceptionally potent, orally active, antinociceptive agent in thermally induced pain.
    Journal of medicinal chemistry, 2009, Dec-10, Volume: 52, Issue:23

    Topics: Administration, Oral; Analgesics; Animals; Cell Line; Drug Discovery; Hot Temperature; Humans; Male; Mice; Pain; Piperazine; Piperazines; Pyridazines; Radioligand Assay; Rats; Receptors, Adrenergic; Structure-Activity Relationship

2009
Lead optimization of a sulfonylurea-based piperazine pyridazinone series of glucan synthase inhibitors.
    Bioorganic & medicinal chemistry letters, 2012, Jul-15, Volume: 22, Issue:14

    Topics: Animals; Antifungal Agents; Candida; Cell Line; Enzyme Inhibitors; Glucosyltransferases; Humans; Lead; Molecular Structure; Piperazine; Piperazines; Pyridazines; Rats; Structure-Activity Relationship; Sulfonylurea Compounds

2012